BDBM50654794 CHEMBL6150573

SMILES Cc1cc(NC(=O)Cc2ccc(-n3cnc4cc(-c5cn[nH]c5)ccc43)cc2)sn1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50654794   

TargetVascular endothelial growth factor receptor 3(Human)
Arromax Pharmatech Co. Ltd.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654794BDBM50654794(CHEMBL6150573)
Affinity DataIC50: 87nMAssay Description:Inhibition of MPS1 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Arromax Pharmatech Co. Ltd.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654794BDBM50654794(CHEMBL6150573)
Affinity DataIC50: 129nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Arromax Pharmatech Co. Ltd.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654794BDBM50654794(CHEMBL6150573)
Affinity DataIC50: 304nMAssay Description:Inhibition of BACE1 (unknown origin) by cell-based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Arromax Pharmatech Co. Ltd.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654794BDBM50654794(CHEMBL6150573)
Affinity DataIC50: 805nMAssay Description:Inhibition of human Nav1.5 at -50 mV holding potential by cell-based IonWorks barracuda automated electrophysiology methodMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed