BDBM50654789 CHEMBL6114929

SMILES CC(C)(C)c1cc(NC(=O)Cc2ccc(-n3cnc4cc(-c5cccnc5)ccc43)cc2)on1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50654789   

TargetPlatelet-derived growth factor receptor alpha(Human)
Arromax Pharmatech Co. Ltd.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654789BDBM50654789(CHEMBL6114929)
Affinity DataIC50: 0.280nMAssay Description:Inhibition of 20S immunoproteasome beta 2 (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Arromax Pharmatech Co. Ltd.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654789BDBM50654789(CHEMBL6114929)
Affinity DataIC50: 0.730nMAssay Description:Agonist activity at human A2B adenosine receptor by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetPlatelet-derived growth factor receptor beta(Human)
Arromax Pharmatech Co. Ltd.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654789BDBM50654789(CHEMBL6114929)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of 20S immunoproteasome beta 2 (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetVascular endothelial growth factor receptor 3(Human)
Arromax Pharmatech Co. Ltd.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654789BDBM50654789(CHEMBL6114929)
Affinity DataIC50: 2.60nMAssay Description:Agonist activity at TAS2R1 (unknown origin) by stably expressed cell-based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Arromax Pharmatech Co. Ltd.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654789BDBM50654789(CHEMBL6114929)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of BACE1 (unknown origin) by cell-based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Arromax Pharmatech Co. Ltd.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654789BDBM50654789(CHEMBL6114929)
Affinity DataIC50: 5.80nMAssay Description:Inhibition of human Nav1.5 at -50 mV holding potential by cell-based IonWorks barracuda automated electrophysiology methodMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed