BDBM50653653 CHEMBL6151096

SMILES O=C1CCC(c2ccnc3[nH]ncc23)C(=O)N1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50653653   

TargetProtein cereblon(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653653BDBM50653653(CHEMBL6151096)
Affinity DataKd:  510nMAssay Description:Inhibition of TPA-induced AP-1 activation in cells expressing beta-lactamase after 18 hrs using FRET substrate by cell-based high-throughput screenin...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetProtein cereblon(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653653BDBM50653653(CHEMBL6151096)
Affinity DataIC50: 720nMAssay Description:Antagonist activity at CGRP receptor assessed as inhibition of CGRP-stimulated cAMP production by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed