BDBM50314514 5-(2,3-dimethylphenyl)-N-(2-methoxyethyl)-N-(6-methoxypyridin-3-yl)pyrazine-2-carboxamide::CHEMBL1093599
SMILES CCN1CCN(CCC(=O)Nc2ccc(S(=O)(=O)N(CC(N)=O)c3ccc(N(CC(N)=O)S(=O)(=O)c4ccccc4)c4ccccc34)cc2)CC1
InChI Key InChIKey=YWIMUONNODRZHD-UHFFFAOYSA-N
Data 3 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 50314514
TargetNuclear factor erythroid 2-related factor 2(Human)
Henan University of Chinese Medicine
Curated by ChEMBL
Henan University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Antagonist activity at human recombinant TRPV1 assessed as inhibition of capsaicin-induced in intracellular calcium levels by cell-based FLIPR assayMore data for this Ligand-Target Pair
