BDBM170081 US9073940, 439
SMILES COC1CCN(CCN2CCC[C@@H](C2)n2nc(C(=O)N3CCOCC3)c3CS(=O)(=O)c4ccccc4-c23)C1
InChI Key InChIKey=LUKHPIFOJUBBBW-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 170081
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha/alpha [E542K,E545K,H1047R]/beta/gamma/delta isoform(Human)
Merck Serono
US Patent
Merck Serono
US Patent
Affinity DataIC50: 25nMAssay Description:The efficacy of compounds of the invention in inhibiting the PI3K induced-lipid phosphorylation may be tested in the following binding assay. The ass...More data for this Ligand-Target Pair
