BDBM169948 US9073940, 298

SMILES Fc1cccc2-c3c(CS(=O)(=O)c12)c(nn3C1CCN(C1)C1CCOCC1)C(=O)N1CCOCC1

InChI Key InChIKey=GXTWTBFETNXESR-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 169948   

TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha/alpha [E542K,E545K,H1047R]/beta/gamma/delta isoform(Human)
Merck Serono

US Patent

LigandBDBM169948(US9073940, 298)Copy SMILESCopy InChI

Affinity DataIC50: 29nMAssay Description:The efficacy of compounds of the invention in inhibiting the PI3K induced-lipid phosphorylation may be tested in the following binding assay. The ass...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
3/9/2016
Entry Details
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