19 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
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Design, synthesis, and biological characterization of proteolysis targeting chimera (PROTACs) for the ataxia telangiectasia and RAD3-related (ATR) kinase.

Martin-Luther-University of Halle-Wittenberg
Discovery of Preclinical Candidate AD1058 as a Highly Potent, Selective, and Brain-Penetrant ATR Inhibitor for the Treatment of Advanced Malignancies.

Shanghai Institute of Materia Medica
Discovery of the Potent and Selective ATR Inhibitor Camonsertib (RP-3500).

Repare Therapeutics, Inc.
Recent advances in DDR (DNA damage response) inhibitors for cancer therapy.

Hubei Polytechnic University
BAY-8400: A Novel Potent and Selective DNA-PK Inhibitor which Shows Synergistic Efficacy in Combination with Targeted Alpha Therapies.

Bayer
Synthetic Lethality through the Lens of Medicinal Chemistry.

Istituto Italiano Di Tecnologia
ATR Inhibitors as Potential Treatment for Cancers.

Therachem Research Medilab
1,3,4-oxadiazole homophthalimide derivative compounds as histone deacetylase 6 inhibitor, and the pharmaceutical composition comprising the same

Chong Kun Dang Pharmaceutical
2,3-DIHYDROBENZO[B][1,4]DIOXIN-6-YL CONTAINING COMPOUNDS USEFUL AS IMMUNOMODULATORS

Bristol-Myers Squibb
Crystalline succinate salt of 6-(6-aminopyrazin-2-yl)-n-(4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)imidazo[1,2-a]pyrazin-8-amine

Kronos Bio
Cycloalkyl-diamines for the treatment of inflammation

Medisynergics
Pyrazole derivatives as MALT1 inhibitors

Janssen Pharmaceutica
Bicyclic heterocyclic compound

Mitsubishi Tanabe Pharma
Substituted pyrazoloazepin-8-ones and their use as phosphodiesterase inhibitors

Leo Pharma
Substituted [5,6]cyclic-4(3H)-pyrimidinones as anticancer agents

Zenji Research Laboratories
Compounds and their use for reducing uric acid levels

Acquist
Sulfur-containing compounds targeting vesicular acetylcholine transporter

Washington University
3-amino-pyridines as GPBAR1 agonists

Hoffmann-La Roche
Compounds useful as inhibitors of ATR kinase

Vertex Pharmaceuticals