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Synthesis, screening and validation of cysteine-reactive fragments as chikungunya virus protease inhibitors.
Bioorg Med Chem Lett 122: 0-0 (0)
Australian National University
Design, synthesis, and biological evaluation of novel aminopyrimidine derivatives as EGFR inhibitors.
Bioorg Med Chem Lett 122: 0-0 (0)
Jiangnan University
Discovery of ATP competitive PDHK1/2 dual inhibitors.
Bioorg Med Chem Lett 122: 0-0 (0)
China Innovation Center of Roche
Design, synthesis, molecular docking and ADME of novel phenylalanine derivatives as mushroom tyrosinase inhibitors.
Bioorg Med Chem Lett 122: 0-0 (0)
Sun Yat-sen University
Discovery of 4-((quinolin-8-ylthio)methyl)benzamide derivatives as a new class of SARS-CoV-2 nsp13 inhibitors.
Bioorg Med Chem Lett 122: 0-0 (0)
Sichuan University