BindingDB Reactant_set_id	Ligand SMILES	Ligand InChI	Ligand InChI Key	BindingDB MonomerID	BindingDB Ligand Name	Target Name	Target Source Organism According to Curator or DataSource	Ki (nM)	IC50 (nM)	Kd (nM)	EC50 (nM)	kon (M-1-s-1)	koff (s-1)	pH	Temp (C)	Curation/DataSource	Article DOI	BindingDB Entry DOI	PMID	PubChem AID	Patent Number	Authors	Date of publication	Date in BindingDB	Institution	Link to Ligand in BindingDB	Link to Target in BindingDB	Link to Ligand-Target Pair in BindingDB	Ligand HET ID in PDB	PDB ID(s) for Ligand-Target Complex	PubChem CID	PubChem SID	ChEBI ID of Ligand	ChEMBL ID of Ligand	DrugBank ID of Ligand	IUPHAR_GRAC ID of Ligand	KEGG ID of Ligand	ZINC ID of Ligand	Number of Protein Chains in Target (>1 implies a multichain complex)	BindingDB Target Chain Sequence 1	PDB ID(s) of Target Chain 1	UniProt (SwissProt) Recommended Name of Target Chain 1	UniProt (SwissProt) Entry Name of Target Chain 1	UniProt (SwissProt) Primary ID of Target Chain 1	UniProt (SwissProt) Secondary ID(s) of Target Chain 1	UniProt (SwissProt) Alternative ID(s) of Target Chain 1	UniProt (TrEMBL) Submitted Name of Target Chain 1	UniProt (TrEMBL) Entry Name of Target Chain 1	UniProt (TrEMBL) Primary ID of Target Chain 1	UniProt (TrEMBL) Secondary ID(s) of Target Chain 1	UniProt (TrEMBL) Alternative ID(s) of Target Chain 1	BindingDB Target Chain Sequence 2	PDB ID(s) of Target Chain 2	UniProt (SwissProt) Recommended Name of Target Chain 2	UniProt (SwissProt) Entry Name of Target Chain 2	UniProt (SwissProt) Primary ID of Target Chain 2	UniProt (SwissProt) Secondary ID(s) of Target Chain 2	UniProt (SwissProt) Alternative ID(s) of Target Chain 2	UniProt (TrEMBL) Submitted Name of Target Chain 2	UniProt (TrEMBL) Entry Name of Target Chain 2	UniProt (TrEMBL) Primary ID of Target Chain 2	UniProt (TrEMBL) Secondary ID(s) of Target Chain 2	UniProt (TrEMBL) Alternative ID(s) of Target Chain 2	BindingDB Target Chain Sequence 3	PDB ID(s) of Target Chain 3	UniProt (SwissProt) Recommended Name of Target Chain 3	UniProt (SwissProt) Entry Name of Target Chain 3	UniProt (SwissProt) Primary ID of Target Chain 3	UniProt (SwissProt) Secondary ID(s) of Target Chain 3	UniProt (SwissProt) Alternative ID(s) of Target Chain 3	UniProt (TrEMBL) Submitted Name of Target Chain 3	UniProt (TrEMBL) Entry Name of Target Chain 3	UniProt (TrEMBL) Primary ID of Target Chain 3	UniProt (TrEMBL) Secondary ID(s) of Target Chain 3	UniProt (TrEMBL) Alternative ID(s) of Target Chain 3	BindingDB Target Chain Sequence 4	PDB ID(s) of Target Chain 4	UniProt (SwissProt) Recommended Name of Target Chain 4	UniProt (SwissProt) Entry Name of Target Chain 4	UniProt (SwissProt) Primary ID of Target Chain 4	UniProt (SwissProt) Secondary ID(s) of Target Chain 4	UniProt (SwissProt) Alternative ID(s) of Target Chain 4	UniProt (TrEMBL) Submitted Name of Target Chain 4	UniProt (TrEMBL) Entry Name of Target Chain 4	UniProt (TrEMBL) Primary ID of Target Chain 4	UniProt (TrEMBL) Secondary ID(s) of Target Chain 4	UniProt (TrEMBL) Alternative ID(s) of Target Chain 4	BindingDB Target Chain Sequence 5	PDB ID(s) of Target Chain 5	UniProt (SwissProt) Recommended Name of Target Chain 5	UniProt (SwissProt) Entry Name of Target Chain 5	UniProt (SwissProt) Primary ID of Target Chain 5	UniProt (SwissProt) Secondary ID(s) of Target Chain 5	UniProt (SwissProt) Alternative ID(s) of Target Chain 5	UniProt (TrEMBL) Submitted Name of Target Chain 5	UniProt (TrEMBL) Entry Name of Target Chain 5	UniProt (TrEMBL) Primary ID of Target Chain 5	UniProt (TrEMBL) Secondary ID(s) of Target Chain 5	UniProt (TrEMBL) Alternative ID(s) of Target Chain 5	BindingDB Target Chain Sequence 6	PDB ID(s) of Target Chain 6	UniProt (SwissProt) Recommended Name of Target Chain 6	UniProt (SwissProt) Entry Name of Target Chain 6	UniProt (SwissProt) Primary ID of Target Chain 6	UniProt (SwissProt) Secondary ID(s) of Target Chain 6	UniProt (SwissProt) Alternative ID(s) of Target Chain 6	UniProt (TrEMBL) Submitted Name of Target Chain 6	UniProt (TrEMBL) Entry Name of Target Chain 6	UniProt (TrEMBL) Primary ID of Target Chain 6	UniProt (TrEMBL) Secondary ID(s) of Target Chain 6	UniProt (TrEMBL) Alternative ID(s) of Target Chain 6	BindingDB Target Chain Sequence 7	PDB ID(s) of Target Chain 7	UniProt (SwissProt) Recommended Name of Target Chain 7	UniProt (SwissProt) Entry Name of Target Chain 7	UniProt (SwissProt) Primary ID of Target Chain 7	UniProt (SwissProt) Secondary ID(s) of Target Chain 7	UniProt (SwissProt) Alternative ID(s) of Target Chain 7	UniProt (TrEMBL) Submitted Name of Target Chain 7	UniProt (TrEMBL) Entry Name of Target Chain 7	UniProt (TrEMBL) Primary ID of Target Chain 7	UniProt (TrEMBL) Secondary ID(s) of Target Chain 7	UniProt (TrEMBL) Alternative ID(s) of Target Chain 7	BindingDB Target Chain Sequence 8	PDB ID(s) of Target Chain 8	UniProt (SwissProt) Recommended Name of Target Chain 8	UniProt (SwissProt) Entry Name of Target Chain 8	UniProt (SwissProt) Primary ID of Target Chain 8	UniProt (SwissProt) Secondary ID(s) of Target Chain 8	UniProt (SwissProt) Alternative ID(s) of Target Chain 8	UniProt (TrEMBL) Submitted Name of Target Chain 8	UniProt (TrEMBL) Entry Name of Target Chain 8	UniProt (TrEMBL) Primary ID of Target Chain 8	UniProt (TrEMBL) Secondary ID(s) of Target Chain 8	UniProt (TrEMBL) Alternative ID(s) of Target Chain 8	BindingDB Target Chain Sequence 9	PDB ID(s) of Target Chain 9	UniProt (SwissProt) Recommended Name of Target Chain 9	UniProt (SwissProt) Entry Name of Target Chain 9	UniProt (SwissProt) Primary ID of Target Chain 9	UniProt (SwissProt) Secondary ID(s) of Target Chain 9	UniProt (SwissProt) Alternative ID(s) of Target Chain 9	UniProt (TrEMBL) Submitted Name of Target Chain 9	UniProt (TrEMBL) Entry Name of Target Chain 9	UniProt (TrEMBL) Primary ID of Target Chain 9	UniProt (TrEMBL) Secondary ID(s) of Target Chain 9	UniProt (TrEMBL) Alternative ID(s) of Target Chain 9	BindingDB Target Chain Sequence 10	PDB ID(s) of Target Chain 10	UniProt (SwissProt) Recommended Name of Target Chain 10	UniProt (SwissProt) Entry Name of Target Chain 10	UniProt (SwissProt) Primary ID of Target Chain 10	UniProt (SwissProt) Secondary ID(s) of Target Chain 10	UniProt (SwissProt) Alternative ID(s) of Target Chain 10	UniProt (TrEMBL) Submitted Name of Target Chain 10	UniProt (TrEMBL) Entry Name of Target Chain 10	UniProt (TrEMBL) Primary ID of Target Chain 10	UniProt (TrEMBL) Secondary ID(s) of Target Chain 10	UniProt (TrEMBL) Alternative ID(s) of Target Chain 10	BindingDB Target Chain Sequence 11	PDB ID(s) of Target Chain 11	UniProt (SwissProt) Recommended Name of Target Chain 11	UniProt (SwissProt) Entry Name of Target Chain 11	UniProt (SwissProt) Primary ID of Target Chain 11	UniProt (SwissProt) Secondary ID(s) of Target Chain 11	UniProt (SwissProt) Alternative ID(s) of Target Chain 11	UniProt (TrEMBL) Submitted Name of Target Chain 11	UniProt (TrEMBL) Entry Name of Target Chain 11	UniProt (TrEMBL) Primary ID of Target Chain 11	UniProt (TrEMBL) Secondary ID(s) of Target Chain 11	UniProt (TrEMBL) Alternative ID(s) of Target Chain 11	BindingDB Target Chain Sequence 12	PDB ID(s) of Target Chain 12	UniProt (SwissProt) Recommended Name of Target Chain 12	UniProt (SwissProt) Entry Name of Target Chain 12	UniProt (SwissProt) Primary ID of Target Chain 12	UniProt (SwissProt) Secondary ID(s) of Target Chain 12	UniProt (SwissProt) Alternative ID(s) of Target Chain 12	UniProt (TrEMBL) Submitted Name of Target Chain 12	UniProt (TrEMBL) Entry Name of Target Chain 12	UniProt (TrEMBL) Primary ID of Target Chain 12	UniProt (TrEMBL) Secondary ID(s) of Target Chain 12	UniProt (TrEMBL) Alternative ID(s) of Target Chain 12	BindingDB Target Chain Sequence 13	PDB ID(s) of Target Chain 13	UniProt (SwissProt) Recommended Name of Target Chain 13	UniProt (SwissProt) Entry Name of Target Chain 13	UniProt (SwissProt) Primary ID of Target Chain 13	UniProt (SwissProt) Secondary ID(s) of Target Chain 13	UniProt (SwissProt) Alternative ID(s) of Target Chain 13	UniProt (TrEMBL) Submitted Name of Target Chain 13	UniProt (TrEMBL) Entry Name of Target Chain 13	UniProt (TrEMBL) Primary ID of Target Chain 13	UniProt (TrEMBL) Secondary ID(s) of Target Chain 13	UniProt (TrEMBL) Alternative ID(s) of Target Chain 13	BindingDB Target Chain Sequence 14	PDB ID(s) of Target Chain 14	UniProt (SwissProt) Recommended Name of Target Chain 14	UniProt (SwissProt) Entry Name of Target Chain 14	UniProt (SwissProt) Primary ID of Target Chain 14	UniProt (SwissProt) Secondary ID(s) of Target Chain 14	UniProt (SwissProt) Alternative ID(s) of Target Chain 14	UniProt (TrEMBL) Submitted Name of Target Chain 14	UniProt (TrEMBL) Entry Name of Target Chain 14	UniProt (TrEMBL) Primary ID of Target Chain 14	UniProt (TrEMBL) Secondary ID(s) of Target Chain 14	UniProt (TrEMBL) Alternative ID(s) of Target Chain 14	BindingDB Target Chain Sequence 15	PDB ID(s) of Target Chain 15	UniProt (SwissProt) Recommended Name of Target Chain 15	UniProt (SwissProt) Entry Name of Target Chain 15	UniProt (SwissProt) Primary ID of Target Chain 15	UniProt (SwissProt) Secondary ID(s) of Target Chain 15	UniProt (SwissProt) Alternative ID(s) of Target Chain 15	UniProt (TrEMBL) Submitted Name of Target Chain 15	UniProt (TrEMBL) Entry Name of Target Chain 15	UniProt (TrEMBL) Primary ID of Target Chain 15	UniProt (TrEMBL) Secondary ID(s) of Target Chain 15	UniProt (TrEMBL) Alternative ID(s) of Target Chain 15	BindingDB Target Chain Sequence 16	PDB ID(s) of Target Chain 16	UniProt (SwissProt) Recommended Name of Target Chain 16	UniProt (SwissProt) Entry Name of Target Chain 16	UniProt (SwissProt) Primary ID of Target Chain 16	UniProt (SwissProt) Secondary ID(s) of Target Chain 16	UniProt (SwissProt) Alternative ID(s) of Target Chain 16	UniProt (TrEMBL) Submitted Name of Target Chain 16	UniProt (TrEMBL) Entry Name of Target Chain 16	UniProt (TrEMBL) Primary ID of Target Chain 16	UniProt (TrEMBL) Secondary ID(s) of Target Chain 16	UniProt (TrEMBL) Alternative ID(s) of Target Chain 16	BindingDB Target Chain Sequence 17	PDB ID(s) of Target Chain 17	UniProt (SwissProt) Recommended Name of Target Chain 17	UniProt (SwissProt) Entry Name of Target Chain 17	UniProt (SwissProt) Primary ID of Target Chain 17	UniProt (SwissProt) Secondary ID(s) of Target Chain 17	UniProt (SwissProt) Alternative ID(s) of Target Chain 17	UniProt (TrEMBL) Submitted Name of Target Chain 17	UniProt (TrEMBL) Entry Name of Target Chain 17	UniProt (TrEMBL) Primary ID of Target Chain 17	UniProt (TrEMBL) Secondary ID(s) of Target Chain 17	UniProt (TrEMBL) Alternative ID(s) of Target Chain 17	BindingDB Target Chain Sequence 18	PDB ID(s) of Target Chain 18	UniProt (SwissProt) Recommended Name of Target Chain 18	UniProt (SwissProt) Entry Name of Target Chain 18	UniProt (SwissProt) Primary ID of Target Chain 18	UniProt (SwissProt) Secondary ID(s) of Target Chain 18	UniProt (SwissProt) Alternative ID(s) of Target Chain 18	UniProt (TrEMBL) Submitted Name of Target Chain 18	UniProt (TrEMBL) Entry Name of Target Chain 18	UniProt (TrEMBL) Primary ID of Target Chain 18	UniProt (TrEMBL) Secondary ID(s) of Target Chain 18	UniProt (TrEMBL) Alternative ID(s) of Target Chain 18	BindingDB Target Chain Sequence 19	PDB ID(s) of Target Chain 19	UniProt (SwissProt) Recommended Name of Target Chain 19	UniProt (SwissProt) Entry Name of Target Chain 19	UniProt (SwissProt) Primary ID of Target Chain 19	UniProt (SwissProt) Secondary ID(s) of Target Chain 19	UniProt (SwissProt) Alternative ID(s) of Target Chain 19	UniProt (TrEMBL) Submitted Name of Target Chain 19	UniProt (TrEMBL) Entry Name of Target Chain 19	UniProt (TrEMBL) Primary ID of Target Chain 19	UniProt (TrEMBL) Secondary ID(s) of Target Chain 19	UniProt (TrEMBL) Alternative ID(s) of Target Chain 19	BindingDB Target Chain Sequence 20	PDB ID(s) of Target Chain 20	UniProt (SwissProt) Recommended Name of Target Chain 20	UniProt (SwissProt) Entry Name of Target Chain 20	UniProt (SwissProt) Primary ID of Target Chain 20	UniProt (SwissProt) Secondary ID(s) of Target Chain 20	UniProt (SwissProt) Alternative ID(s) of Target Chain 20	UniProt (TrEMBL) Submitted Name of Target Chain 20	UniProt (TrEMBL) Entry Name of Target Chain 20	UniProt (TrEMBL) Primary ID of Target Chain 20	UniProt (TrEMBL) Secondary ID(s) of Target Chain 20	UniProt (TrEMBL) Alternative ID(s) of Target Chain 20	BindingDB Target Chain Sequence 21	PDB ID(s) of Target Chain 21	UniProt (SwissProt) Recommended Name of Target Chain 21	UniProt (SwissProt) Entry Name of Target Chain 21	UniProt (SwissProt) Primary ID of Target Chain 21	UniProt (SwissProt) Secondary ID(s) of Target Chain 21	UniProt (SwissProt) Alternative ID(s) of Target Chain 21	UniProt (TrEMBL) Submitted Name of Target Chain 21	UniProt (TrEMBL) Entry Name of Target Chain 21	UniProt (TrEMBL) Primary ID of Target Chain 21	UniProt (TrEMBL) Secondary ID(s) of Target Chain 21	UniProt (TrEMBL) Alternative ID(s) of Target Chain 21	BindingDB Target Chain Sequence 22	PDB ID(s) of Target Chain 22	UniProt (SwissProt) Recommended Name of Target Chain 22	UniProt (SwissProt) Entry Name of Target Chain 22	UniProt (SwissProt) Primary ID of Target Chain 22	UniProt (SwissProt) Secondary ID(s) of Target Chain 22	UniProt (SwissProt) Alternative ID(s) of Target Chain 22	UniProt (TrEMBL) Submitted Name of Target Chain 22	UniProt (TrEMBL) Entry Name of Target Chain 22	UniProt (TrEMBL) Primary ID of Target Chain 22	UniProt (TrEMBL) Secondary ID(s) of Target Chain 22	UniProt (TrEMBL) Alternative ID(s) of Target Chain 22	BindingDB Target Chain Sequence 23	PDB ID(s) of Target Chain 23	UniProt (SwissProt) Recommended Name of Target Chain 23	UniProt (SwissProt) Entry Name of Target Chain 23	UniProt (SwissProt) Primary ID of Target Chain 23	UniProt (SwissProt) Secondary ID(s) of Target Chain 23	UniProt (SwissProt) Alternative ID(s) of Target Chain 23	UniProt (TrEMBL) Submitted Name of Target Chain 23	UniProt (TrEMBL) Entry Name of Target Chain 23	UniProt (TrEMBL) Primary ID of Target Chain 23	UniProt (TrEMBL) Secondary ID(s) of Target Chain 23	UniProt (TrEMBL) Alternative ID(s) of Target Chain 23	BindingDB Target Chain Sequence 24	PDB ID(s) of Target Chain 24	UniProt (SwissProt) Recommended Name of Target Chain 24	UniProt (SwissProt) Entry Name of Target Chain 24	UniProt (SwissProt) Primary ID of Target Chain 24	UniProt (SwissProt) Secondary ID(s) of Target Chain 24	UniProt (SwissProt) Alternative ID(s) of Target Chain 24	UniProt (TrEMBL) Submitted Name of Target Chain 24	UniProt (TrEMBL) Entry Name of Target Chain 24	UniProt (TrEMBL) Primary ID of Target Chain 24	UniProt (TrEMBL) Secondary ID(s) of Target Chain 24	UniProt (TrEMBL) Alternative ID(s) of Target Chain 24	BindingDB Target Chain Sequence 25	PDB ID(s) of Target Chain 25	UniProt (SwissProt) Recommended Name of Target Chain 25	UniProt (SwissProt) Entry Name of Target Chain 25	UniProt (SwissProt) Primary ID of Target Chain 25	UniProt (SwissProt) Secondary ID(s) of Target Chain 25	UniProt (SwissProt) Alternative ID(s) of Target Chain 25	UniProt (TrEMBL) Submitted Name of Target Chain 25	UniProt (TrEMBL) Entry Name of Target Chain 25	UniProt (TrEMBL) Primary ID of Target Chain 25	UniProt (TrEMBL) Secondary ID(s) of Target Chain 25	UniProt (TrEMBL) Alternative ID(s) of Target Chain 25	BindingDB Target Chain Sequence 26	PDB ID(s) of Target Chain 26	UniProt (SwissProt) Recommended Name of Target Chain 26	UniProt (SwissProt) Entry Name of Target Chain 26	UniProt (SwissProt) Primary ID of Target Chain 26	UniProt (SwissProt) Secondary ID(s) of Target Chain 26	UniProt (SwissProt) Alternative ID(s) of Target Chain 26	UniProt (TrEMBL) Submitted Name of Target Chain 26	UniProt (TrEMBL) Entry Name of Target Chain 26	UniProt (TrEMBL) Primary ID of Target Chain 26	UniProt (TrEMBL) Secondary ID(s) of Target Chain 26	UniProt (TrEMBL) Alternative ID(s) of Target Chain 26	BindingDB Target Chain Sequence 27	PDB ID(s) of Target Chain 27	UniProt (SwissProt) Recommended Name of Target Chain 27	UniProt (SwissProt) Entry Name of Target Chain 27	UniProt (SwissProt) Primary ID of Target Chain 27	UniProt (SwissProt) Secondary ID(s) of Target Chain 27	UniProt (SwissProt) Alternative ID(s) of Target Chain 27	UniProt (TrEMBL) Submitted Name of Target Chain 27	UniProt (TrEMBL) Entry Name of Target Chain 27	UniProt (TrEMBL) Primary ID of Target Chain 27	UniProt (TrEMBL) Secondary ID(s) of Target Chain 27	UniProt (TrEMBL) Alternative ID(s) of Target Chain 27	BindingDB Target Chain Sequence 28	PDB ID(s) of Target Chain 28	UniProt (SwissProt) Recommended Name of Target Chain 28	UniProt (SwissProt) Entry Name of Target Chain 28	UniProt (SwissProt) Primary ID of Target Chain 28	UniProt (SwissProt) Secondary ID(s) of Target Chain 28	UniProt (SwissProt) Alternative ID(s) of Target Chain 28	UniProt (TrEMBL) Submitted Name of Target Chain 28	UniProt (TrEMBL) Entry Name of Target Chain 28	UniProt (TrEMBL) Primary ID of Target Chain 28	UniProt (TrEMBL) Secondary ID(s) of Target Chain 28	UniProt (TrEMBL) Alternative ID(s) of Target Chain 28	BindingDB Target Chain Sequence 29	PDB ID(s) of Target Chain 29	UniProt (SwissProt) Recommended Name of Target Chain 29	UniProt (SwissProt) Entry Name of Target Chain 29	UniProt (SwissProt) Primary ID of Target Chain 29	UniProt (SwissProt) Secondary ID(s) of Target Chain 29	UniProt (SwissProt) Alternative ID(s) of Target Chain 29	UniProt (TrEMBL) Submitted Name of Target Chain 29	UniProt (TrEMBL) Entry Name of Target Chain 29	UniProt (TrEMBL) Primary ID of Target Chain 29	UniProt (TrEMBL) Secondary ID(s) of Target Chain 29	UniProt (TrEMBL) Alternative ID(s) of Target Chain 29	BindingDB Target Chain Sequence 30	PDB ID(s) of Target Chain 30	UniProt (SwissProt) Recommended Name of Target Chain 30	UniProt (SwissProt) Entry Name of Target Chain 30	UniProt (SwissProt) Primary ID of Target Chain 30	UniProt (SwissProt) Secondary ID(s) of Target Chain 30	UniProt (SwissProt) Alternative ID(s) of Target Chain 30	UniProt (TrEMBL) Submitted Name of Target Chain 30	UniProt (TrEMBL) Entry Name of Target Chain 30	UniProt (TrEMBL) Primary ID of Target Chain 30	UniProt (TrEMBL) Secondary ID(s) of Target Chain 30	UniProt (TrEMBL) Alternative ID(s) of Target Chain 30	BindingDB Target Chain Sequence 31	PDB ID(s) of Target Chain 31	UniProt (SwissProt) Recommended Name of Target Chain 31	UniProt (SwissProt) Entry Name of Target Chain 31	UniProt (SwissProt) Primary ID of Target Chain 31	UniProt (SwissProt) Secondary ID(s) of Target Chain 31	UniProt (SwissProt) Alternative ID(s) of Target Chain 31	UniProt (TrEMBL) Submitted Name of Target Chain 31	UniProt (TrEMBL) Entry Name of Target Chain 31	UniProt (TrEMBL) Primary ID of Target Chain 31	UniProt (TrEMBL) Secondary ID(s) of Target Chain 31	UniProt (TrEMBL) Alternative ID(s) of Target Chain 31	BindingDB Target Chain Sequence 32	PDB ID(s) of Target Chain 32	UniProt (SwissProt) Recommended Name of Target Chain 32	UniProt (SwissProt) Entry Name of Target Chain 32	UniProt (SwissProt) Primary ID of Target Chain 32	UniProt (SwissProt) Secondary ID(s) of Target Chain 32	UniProt (SwissProt) Alternative ID(s) of Target Chain 32	UniProt (TrEMBL) Submitted Name of Target Chain 32	UniProt (TrEMBL) Entry Name of Target Chain 32	UniProt (TrEMBL) Primary ID of Target Chain 32	UniProt (TrEMBL) Secondary ID(s) of Target Chain 32	UniProt (TrEMBL) Alternative ID(s) of Target Chain 32	BindingDB Target Chain Sequence 33	PDB ID(s) of Target Chain 33	UniProt (SwissProt) Recommended Name of Target Chain 33	UniProt (SwissProt) Entry Name of Target Chain 33	UniProt (SwissProt) Primary ID of Target Chain 33	UniProt (SwissProt) Secondary ID(s) of Target Chain 33	UniProt (SwissProt) Alternative ID(s) of Target Chain 33	UniProt (TrEMBL) Submitted Name of Target Chain 33	UniProt (TrEMBL) Entry Name of Target Chain 33	UniProt (TrEMBL) Primary ID of Target Chain 33	UniProt (TrEMBL) Secondary ID(s) of Target Chain 33	UniProt (TrEMBL) Alternative ID(s) of Target Chain 33	BindingDB Target Chain Sequence 34	PDB ID(s) of Target Chain 34	UniProt (SwissProt) Recommended Name of Target Chain 34	UniProt (SwissProt) Entry Name of Target Chain 34	UniProt (SwissProt) Primary ID of Target Chain 34	UniProt (SwissProt) Secondary ID(s) of Target Chain 34	UniProt (SwissProt) Alternative ID(s) of Target Chain 34	UniProt (TrEMBL) Submitted Name of Target Chain 34	UniProt (TrEMBL) Entry Name of Target Chain 34	UniProt (TrEMBL) Primary ID of Target Chain 34	UniProt (TrEMBL) Secondary ID(s) of Target Chain 34	UniProt (TrEMBL) Alternative ID(s) of Target Chain 34	BindingDB Target Chain Sequence 35	PDB ID(s) of Target Chain 35	UniProt (SwissProt) Recommended Name of Target Chain 35	UniProt (SwissProt) Entry Name of Target Chain 35	UniProt (SwissProt) Primary ID of Target Chain 35	UniProt (SwissProt) Secondary ID(s) of Target Chain 35	UniProt (SwissProt) Alternative ID(s) of Target Chain 35	UniProt (TrEMBL) Submitted Name of Target Chain 35	UniProt (TrEMBL) Entry Name of Target Chain 35	UniProt (TrEMBL) Primary ID of Target Chain 35	UniProt (TrEMBL) Secondary ID(s) of Target Chain 35	UniProt (TrEMBL) Alternative ID(s) of Target Chain 35	BindingDB Target Chain Sequence 36	PDB ID(s) of Target Chain 36	UniProt (SwissProt) Recommended Name of Target Chain 36	UniProt (SwissProt) Entry Name of Target Chain 36	UniProt (SwissProt) Primary ID of Target Chain 36	UniProt (SwissProt) Secondary ID(s) of Target Chain 36	UniProt (SwissProt) Alternative ID(s) of Target Chain 36	UniProt (TrEMBL) Submitted Name of Target Chain 36	UniProt (TrEMBL) Entry Name of Target Chain 36	UniProt (TrEMBL) Primary ID of Target Chain 36	UniProt (TrEMBL) Secondary ID(s) of Target Chain 36	UniProt (TrEMBL) Alternative ID(s) of Target Chain 36	BindingDB Target Chain Sequence 37	PDB ID(s) of Target Chain 37	UniProt (SwissProt) Recommended Name of Target Chain 37	UniProt (SwissProt) Entry Name of Target Chain 37	UniProt (SwissProt) Primary ID of Target Chain 37	UniProt (SwissProt) Secondary ID(s) of Target Chain 37	UniProt (SwissProt) Alternative ID(s) of Target Chain 37	UniProt (TrEMBL) Submitted Name of Target Chain 37	UniProt (TrEMBL) Entry Name of Target Chain 37	UniProt (TrEMBL) Primary ID of Target Chain 37	UniProt (TrEMBL) Secondary ID(s) of Target Chain 37	UniProt (TrEMBL) Alternative ID(s) of Target Chain 37	BindingDB Target Chain Sequence 38	PDB ID(s) of Target Chain 38	UniProt (SwissProt) Recommended Name of Target Chain 38	UniProt (SwissProt) Entry Name of Target Chain 38	UniProt (SwissProt) Primary ID of Target Chain 38	UniProt (SwissProt) Secondary ID(s) of Target Chain 38	UniProt (SwissProt) Alternative ID(s) of Target Chain 38	UniProt (TrEMBL) Submitted Name of Target Chain 38	UniProt (TrEMBL) Entry Name of Target Chain 38	UniProt (TrEMBL) Primary ID of Target Chain 38	UniProt (TrEMBL) Secondary ID(s) of Target Chain 38	UniProt (TrEMBL) Alternative ID(s) of Target Chain 38	BindingDB Target Chain Sequence 39	PDB ID(s) of Target Chain 39	UniProt (SwissProt) Recommended Name of Target Chain 39	UniProt (SwissProt) Entry Name of Target Chain 39	UniProt (SwissProt) Primary ID of Target Chain 39	UniProt (SwissProt) Secondary ID(s) of Target Chain 39	UniProt (SwissProt) Alternative ID(s) of Target Chain 39	UniProt (TrEMBL) Submitted Name of Target Chain 39	UniProt (TrEMBL) Entry Name of Target Chain 39	UniProt (TrEMBL) Primary ID of Target Chain 39	UniProt (TrEMBL) Secondary ID(s) of Target Chain 39	UniProt (TrEMBL) Alternative ID(s) of Target Chain 39	BindingDB Target Chain Sequence 40	PDB ID(s) of Target Chain 40	UniProt (SwissProt) Recommended Name of Target Chain 40	UniProt (SwissProt) Entry Name of Target Chain 40	UniProt (SwissProt) Primary ID of Target Chain 40	UniProt (SwissProt) Secondary ID(s) of Target Chain 40	UniProt (SwissProt) Alternative ID(s) of Target Chain 40	UniProt (TrEMBL) Submitted Name of Target Chain 40	UniProt (TrEMBL) Entry Name of Target Chain 40	UniProt (TrEMBL) Primary ID of Target Chain 40	UniProt (TrEMBL) Secondary ID(s) of Target Chain 40	UniProt (TrEMBL) Alternative ID(s) of Target Chain 40	BindingDB Target Chain Sequence 41	PDB ID(s) of Target Chain 41	UniProt (SwissProt) Recommended Name of Target Chain 41	UniProt (SwissProt) Entry Name of Target Chain 41	UniProt (SwissProt) Primary ID of Target Chain 41	UniProt (SwissProt) Secondary ID(s) of Target Chain 41	UniProt (SwissProt) Alternative ID(s) of Target Chain 41	UniProt (TrEMBL) Submitted Name of Target Chain 41	UniProt (TrEMBL) Entry Name of Target Chain 41	UniProt (TrEMBL) Primary ID of Target Chain 41	UniProt (TrEMBL) Secondary ID(s) of Target Chain 41	UniProt (TrEMBL) Alternative ID(s) of Target Chain 41	BindingDB Target Chain Sequence 42	PDB ID(s) of Target Chain 42	UniProt (SwissProt) Recommended Name of Target Chain 42	UniProt (SwissProt) Entry Name of Target Chain 42	UniProt (SwissProt) Primary ID of Target Chain 42	UniProt (SwissProt) Secondary ID(s) of Target Chain 42	UniProt (SwissProt) Alternative ID(s) of Target Chain 42	UniProt (TrEMBL) Submitted Name of Target Chain 42	UniProt (TrEMBL) Entry Name of Target Chain 42	UniProt (TrEMBL) Primary ID of Target Chain 42	UniProt (TrEMBL) Secondary ID(s) of Target Chain 42	UniProt (TrEMBL) Alternative ID(s) of Target Chain 42	BindingDB Target Chain Sequence 43	PDB ID(s) of Target Chain 43	UniProt (SwissProt) Recommended Name of Target Chain 43	UniProt (SwissProt) Entry Name of Target Chain 43	UniProt (SwissProt) Primary ID of Target Chain 43	UniProt (SwissProt) Secondary ID(s) of Target Chain 43	UniProt (SwissProt) Alternative ID(s) of Target Chain 43	UniProt (TrEMBL) Submitted Name of Target Chain 43	UniProt (TrEMBL) Entry Name of Target Chain 43	UniProt (TrEMBL) Primary ID of Target Chain 43	UniProt (TrEMBL) Secondary ID(s) of Target Chain 43	UniProt (TrEMBL) Alternative ID(s) of Target Chain 43	BindingDB Target Chain Sequence 44	PDB ID(s) of Target Chain 44	UniProt (SwissProt) Recommended Name of Target Chain 44	UniProt (SwissProt) Entry Name of Target Chain 44	UniProt (SwissProt) Primary ID of Target Chain 44	UniProt (SwissProt) Secondary ID(s) of Target Chain 44	UniProt (SwissProt) Alternative ID(s) of Target Chain 44	UniProt (TrEMBL) Submitted Name of Target Chain 44	UniProt (TrEMBL) Entry Name of Target Chain 44	UniProt (TrEMBL) Primary ID of Target Chain 44	UniProt (TrEMBL) Secondary ID(s) of Target Chain 44	UniProt (TrEMBL) Alternative ID(s) of Target Chain 44	BindingDB Target Chain Sequence 45	PDB ID(s) of Target Chain 45	UniProt (SwissProt) Recommended Name of Target Chain 45	UniProt (SwissProt) Entry Name of Target Chain 45	UniProt (SwissProt) Primary ID of Target Chain 45	UniProt (SwissProt) Secondary ID(s) of Target Chain 45	UniProt (SwissProt) Alternative ID(s) of Target Chain 45	UniProt (TrEMBL) Submitted Name of Target Chain 45	UniProt (TrEMBL) Entry Name of Target Chain 45	UniProt (TrEMBL) Primary ID of Target Chain 45	UniProt (TrEMBL) Secondary ID(s) of Target Chain 45	UniProt (TrEMBL) Alternative ID(s) of Target Chain 45	BindingDB Target Chain Sequence 46	PDB ID(s) of Target Chain 46	UniProt (SwissProt) Recommended Name of Target Chain 46	UniProt (SwissProt) Entry Name of Target Chain 46	UniProt (SwissProt) Primary ID of Target Chain 46	UniProt (SwissProt) Secondary ID(s) of Target Chain 46	UniProt (SwissProt) Alternative ID(s) of Target Chain 46	UniProt (TrEMBL) Submitted Name of Target Chain 46	UniProt (TrEMBL) Entry Name of Target Chain 46	UniProt (TrEMBL) Primary ID of Target Chain 46	UniProt (TrEMBL) Secondary ID(s) of Target Chain 46	UniProt (TrEMBL) Alternative ID(s) of Target Chain 46	BindingDB Target Chain Sequence 47	PDB ID(s) of Target Chain 47	UniProt (SwissProt) Recommended Name of Target Chain 47	UniProt (SwissProt) Entry Name of Target Chain 47	UniProt (SwissProt) Primary ID of Target Chain 47	UniProt (SwissProt) Secondary ID(s) of Target Chain 47	UniProt (SwissProt) Alternative ID(s) of Target Chain 47	UniProt (TrEMBL) Submitted Name of Target Chain 47	UniProt (TrEMBL) Entry Name of Target Chain 47	UniProt (TrEMBL) Primary ID of Target Chain 47	UniProt (TrEMBL) Secondary ID(s) of Target Chain 47	UniProt (TrEMBL) Alternative ID(s) of Target Chain 47	BindingDB Target Chain Sequence 48	PDB ID(s) of Target Chain 48	UniProt (SwissProt) Recommended Name of Target Chain 48	UniProt (SwissProt) Entry Name of Target Chain 48	UniProt (SwissProt) Primary ID of Target Chain 48	UniProt (SwissProt) Secondary ID(s) of Target Chain 48	UniProt (SwissProt) Alternative ID(s) of Target Chain 48	UniProt (TrEMBL) Submitted Name of Target Chain 48	UniProt (TrEMBL) Entry Name of Target Chain 48	UniProt (TrEMBL) Primary ID of Target Chain 48	UniProt (TrEMBL) Secondary ID(s) of Target Chain 48	UniProt (TrEMBL) Alternative ID(s) of Target Chain 48	BindingDB Target Chain Sequence 49	PDB ID(s) of Target Chain 49	UniProt (SwissProt) Recommended Name of Target Chain 49	UniProt (SwissProt) Entry Name of Target Chain 49	UniProt (SwissProt) Primary ID of Target Chain 49	UniProt (SwissProt) Secondary ID(s) of Target Chain 49	UniProt (SwissProt) Alternative ID(s) of Target Chain 49	UniProt (TrEMBL) Submitted Name of Target Chain 49	UniProt (TrEMBL) Entry Name of Target Chain 49	UniProt (TrEMBL) Primary ID of Target Chain 49	UniProt (TrEMBL) Secondary ID(s) of Target Chain 49	UniProt (TrEMBL) Alternative ID(s) of Target Chain 49	BindingDB Target Chain Sequence 50	PDB ID(s) of Target Chain 50	UniProt (SwissProt) Recommended Name of Target Chain 50	UniProt (SwissProt) Entry Name of Target Chain 50	UniProt (SwissProt) Primary ID of Target Chain 50	UniProt (SwissProt) Secondary ID(s) of Target Chain 50	UniProt (SwissProt) Alternative ID(s) of Target Chain 50	UniProt (TrEMBL) Submitted Name of Target Chain 50	UniProt (TrEMBL) Entry Name of Target Chain 50	UniProt (TrEMBL) Primary ID of Target Chain 50	UniProt (TrEMBL) Secondary ID(s) of Target Chain 50	UniProt (TrEMBL) Alternative ID(s) of Target Chain 50
558549	COCCN1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C26H28Cl2F3N3O2/c1-16-12-17(26(29,30)31)13-23-20(16)14-18(32(23)2)15-21-22(27)5-4-19(24(21)28)25(35)34-8-6-33(7-9-34)10-11-36-3/h4-5,12-14H,6-11,15H2,1-3H3	NVYIMYFBPUMFNN-UHFFFAOYSA-N	292711	US10106501, Example A	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292711	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292711&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122982	381613000							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558550	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCN(CC4)C4COC4)c3Cl)cc12)C(F)(F)F	InChI=1S/C26H26Cl2F3N3O2/c1-15-9-16(26(29,30)31)10-23-20(15)11-17(32(23)2)12-21-22(27)4-3-19(24(21)28)25(35)34-7-5-33(6-8-34)18-13-36-14-18/h3-4,9-11,18H,5-8,12-14H2,1-2H3	YOLONXDHSMBQTJ-UHFFFAOYSA-N	292717	US10106501, Example A1	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292717	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292717&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123920	381613006							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558551	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC4)S(C)(=O)=O)c3Cl)cc12)C(F)(F)F	InChI=1S/C25H25Cl2F3N2O3S/c1-14-10-15(25(28,29)30)11-22-19(14)12-16(31(22)2)13-20-21(26)5-4-18(23(20)27)24(33)32-8-6-17(7-9-32)36(3,34)35/h4-5,10-12,17H,6-9,13H2,1-3H3	PMEHDBLITJSZNF-UHFFFAOYSA-N	292718	US10106501, Example A1-11	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292718	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292718&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123342	381613007							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558552	Cc1cc(cc2n(C)c(cc12)C(=O)c1c(Cl)ccc(C(=O)N2CCC(CC2)C2COC2)c1Cl)C(F)(F)F	InChI=1S/C27H25Cl2F3N2O3/c1-14-9-17(27(30,31)32)10-21-19(14)11-22(33(21)2)25(35)23-20(28)4-3-18(24(23)29)26(36)34-7-5-15(6-8-34)16-12-37-13-16/h3-4,9-11,15-16H,5-8,12-13H2,1-2H3	WIPGALGNRKVTRZ-UHFFFAOYSA-N	292719	US10106501, Example AP-6	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292719	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292719&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123066	381613008							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558553	C[C@@H]1CN(CC[C@@H]1C(O)=O)C(=O)c1ccc(Cl)c(C(=O)c2cc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl |r|	InChI=1S/C26H23Cl2F3N2O4/c1-12-8-14(26(29,30)31)9-19-17(12)10-20(32(19)3)23(34)21-18(27)5-4-16(22(21)28)24(35)33-7-6-15(25(36)37)13(2)11-33/h4-5,8-10,13,15H,6-7,11H2,1-3H3,(H,36,37)	YSBUXVMUHRACRG-UHFFFAOYSA-N	292720	US10106501, Example AQ-4::US10106501, Example AQ-3	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292720	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292720&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123555	381613009							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558554	C[C@@H]1CN(CC[C@@H]1C(O)=O)C(=O)c1ccc(Cl)c(C(=O)c2cc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl |r|	InChI=1S/C26H23Cl2F3N2O4/c1-12-8-14(26(29,30)31)9-19-17(12)10-20(32(19)3)23(34)21-18(27)5-4-16(22(21)28)24(35)33-7-6-15(25(36)37)13(2)11-33/h4-5,8-10,13,15H,6-7,11H2,1-3H3,(H,36,37)	YSBUXVMUHRACRG-UHFFFAOYSA-N	292720	US10106501, Example AQ-4::US10106501, Example AQ-3	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292720	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292720&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123555	381613009							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558555	C[C@H]1CN(CC[C@H]1C(O)=O)C(=O)c1ccc(Cl)c(C(=O)c2cc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl |r|	InChI=1S/C26H23Cl2F3N2O4/c1-12-8-14(26(29,30)31)9-19-17(12)10-20(32(19)3)23(34)21-18(27)5-4-16(22(21)28)24(35)33-7-6-15(25(36)37)13(2)11-33/h4-5,8-10,13,15H,6-7,11H2,1-3H3,(H,36,37)	YSBUXVMUHRACRG-UHFFFAOYSA-N	292722	US10106501, Example AQ-5	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292722	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292722&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122899	381613010							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558556	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC4)C(O)=O)c3Cl)cc12)C(F)(F)F	InChI=1S/C25H23Cl2F3N2O3/c1-13-9-15(25(28,29)30)10-21-18(13)11-16(31(21)2)12-19-20(26)4-3-17(22(19)27)23(33)32-7-5-14(6-8-32)24(34)35/h3-4,9-11,14H,5-8,12H2,1-2H3,(H,34,35)	NVDKGFYFKVWJLJ-UHFFFAOYSA-N	292723	US10106501, Example B	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292723	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292723&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123531	381613011							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558557	CC1CN(CCC1C(O)=O)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C26H25Cl2F3N2O3/c1-13-8-15(26(29,30)31)9-22-19(13)10-16(32(22)3)11-20-21(27)5-4-18(23(20)28)24(34)33-7-6-17(25(35)36)14(2)12-33/h4-5,8-10,14,17H,6-7,11-12H2,1-3H3,(H,35,36)	OSLRVFJRYRWWCB-UHFFFAOYSA-N	292724	US10106501, Example B-1	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292724	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292724&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123634	381613012							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558558	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC4)OCC(O)=O)c3Cl)cc12)C(F)(F)F	InChI=1S/C26H25Cl2F3N2O4/c1-14-9-15(26(29,30)31)10-22-19(14)11-16(32(22)2)12-20-21(27)4-3-18(24(20)28)25(36)33-7-5-17(6-8-33)37-13-23(34)35/h3-4,9-11,17H,5-8,12-13H2,1-2H3,(H,34,35)	VRHYDLLTXRRGLH-UHFFFAOYSA-N	292725	US10106501, Example B-2	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292725	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292725&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123855	381613013							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558559	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(C4)C(O)=O)c3Cl)cc12)C(F)(F)F	InChI=1S/C24H21Cl2F3N2O3/c1-12-7-14(24(27,28)29)8-20-17(12)9-15(30(20)2)10-18-19(25)4-3-16(21(18)26)22(32)31-6-5-13(11-31)23(33)34/h3-4,7-9,13H,5-6,10-11H2,1-2H3,(H,33,34)	HMUIDHAZDMXORD-UHFFFAOYSA-N	292726	US10106501, Example B-3	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292726	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292726&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123306	381613014							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558560	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CC(C4)C(O)=O)c3Cl)cc12)C(F)(F)F	InChI=1S/C23H19Cl2F3N2O3/c1-11-5-13(23(26,27)28)6-19-16(11)7-14(29(19)2)8-17-18(24)4-3-15(20(17)25)21(31)30-9-12(10-30)22(32)33/h3-7,12H,8-10H2,1-2H3,(H,32,33)	WBHBWIDGMPCPHH-UHFFFAOYSA-N	292727	US10106501, Example B-4	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292727	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292727&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123660	381613015							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558561	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CC(C)(C4)C(O)=O)c3Cl)cc12)C(F)(F)F	InChI=1S/C24H21Cl2F3N2O3/c1-12-6-13(24(27,28)29)7-19-16(12)8-14(30(19)3)9-17-18(25)5-4-15(20(17)26)21(32)31-10-23(2,11-31)22(33)34/h4-8H,9-11H2,1-3H3,(H,33,34)	MNEYTVQVSLFUCE-UHFFFAOYSA-N	292728	US10106501, Example B-5	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292728	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292728&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123659	381613016							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558562	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC(O)=O)C4)c3Cl)cc12)C(F)(F)F	InChI=1S/C25H23Cl2F3N2O3/c1-13-7-15(25(28,29)30)9-21-18(13)10-16(31(21)2)11-19-20(26)4-3-17(23(19)27)24(35)32-6-5-14(12-32)8-22(33)34/h3-4,7,9-10,14H,5-6,8,11-12H2,1-2H3,(H,33,34)	QHBIYPNFBINASK-UHFFFAOYSA-N	292729	US10106501, Example B-6	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292729	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292729&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123480	381613017							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558563	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)cc12)C(F)(F)F	InChI=1S/C26H25Cl2F3N2O3/c1-14-9-16(26(29,30)31)11-22-19(14)12-17(32(22)2)13-20-21(27)4-3-18(24(20)28)25(36)33-7-5-15(6-8-33)10-23(34)35/h3-4,9,11-12,15H,5-8,10,13H2,1-2H3,(H,34,35)	MSIBFBGRCUGKLK-UHFFFAOYSA-N	292730	US10106501, Example B-7	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292730	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292730&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123714	381613018							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558564	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4C[C@H]5[C@@H](C4)C5C(O)=O)c3Cl)cc12)C(F)(F)F |r|	InChI=1S/C25H21Cl2F3N2O3/c1-11-5-12(25(28,29)30)6-20-15(11)7-13(31(20)2)8-16-19(26)4-3-14(22(16)27)23(33)32-9-17-18(10-32)21(17)24(34)35/h3-7,17-18,21H,8-10H2,1-2H3,(H,34,35)	MQMIYNFKAWASSW-UHFFFAOYSA-N	292731	US10106501, Example B-8	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292731	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292731&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123300	381613019							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558565	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CC(CC(O)=O)C4)c3Cl)cc12)C(F)(F)F	InChI=1S/C24H21Cl2F3N2O3/c1-12-5-14(24(27,28)29)7-20-17(12)8-15(30(20)2)9-18-19(25)4-3-16(22(18)26)23(34)31-10-13(11-31)6-21(32)33/h3-5,7-8,13H,6,9-11H2,1-2H3,(H,32,33)	QXJBVMZDEVSQLX-UHFFFAOYSA-N	292732	US10106501, Example B-9	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292732	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292732&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123488	381613020							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558566	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(O)C(C4)C(O)=O)c3Cl)cc12)C(F)(F)F	InChI=1S/C25H23Cl2F3N2O4/c1-12-7-13(25(28,29)30)8-20-16(12)9-14(31(20)2)10-17-19(26)4-3-15(22(17)27)23(34)32-6-5-21(33)18(11-32)24(35)36/h3-4,7-9,18,21,33H,5-6,10-11H2,1-2H3,(H,35,36)	HUICEALSYFBLEN-UHFFFAOYSA-N	292733	US10106501, Example B-10	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292733	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292733&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123406	381613021							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558567	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCCC(C4)C(O)=O)c3Cl)cc12)C(F)(F)F	InChI=1S/C25H23Cl2F3N2O3/c1-13-8-15(25(28,29)30)9-21-18(13)10-16(31(21)2)11-19-20(26)6-5-17(22(19)27)23(33)32-7-3-4-14(12-32)24(34)35/h5-6,8-10,14H,3-4,7,11-12H2,1-2H3,(H,34,35)	LNZQOBLCYQFJGE-UHFFFAOYSA-N	292734	US10106501, Example B-11	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292734	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292734&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123775	381613022							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558568	COC1(CN(C1)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl)C(O)=O	InChI=1S/C24H21Cl2F3N2O4/c1-12-6-13(24(27,28)29)7-19-16(12)8-14(30(19)2)9-17-18(25)5-4-15(20(17)26)21(32)31-10-23(11-31,35-3)22(33)34/h4-8H,9-11H2,1-3H3,(H,33,34)	ACQJPBFQKQKBSD-UHFFFAOYSA-N	292735	US10106501, Example B-12	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292735	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292735&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123419	381613023							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558569	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(C)(CC4)C(O)=O)c3Cl)cc12)C(F)(F)F	InChI=1S/C26H25Cl2F3N2O3/c1-14-10-15(26(29,30)31)11-21-18(14)12-16(32(21)3)13-19-20(27)5-4-17(22(19)28)23(34)33-8-6-25(2,7-9-33)24(35)36/h4-5,10-12H,6-9,13H2,1-3H3,(H,35,36)	RIUVXTJCXSALNU-UHFFFAOYSA-N	292736	US10106501, Example B-13	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292736	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292736&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123954	381613024							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558570	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(F)(CC4)C(O)=O)c3Cl)cc12)C(F)(F)F	InChI=1S/C25H22Cl2F4N2O3/c1-13-9-14(25(29,30)31)10-20-17(13)11-15(32(20)2)12-18-19(26)4-3-16(21(18)27)22(34)33-7-5-24(28,6-8-33)23(35)36/h3-4,9-11H,5-8,12H2,1-2H3,(H,35,36)	MITALCPHFSUDAY-UHFFFAOYSA-N	292737	US10106501, Example B-14	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292737	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292737&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123627	381613025							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558571	COC[C@@H]1CN(C[C@H]1C(O)=O)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl |r|	InChI=1S/C26H25Cl2F3N2O4/c1-13-6-15(26(29,30)31)7-22-18(13)8-16(32(22)2)9-19-21(27)5-4-17(23(19)28)24(34)33-10-14(12-37-3)20(11-33)25(35)36/h4-8,14,20H,9-12H2,1-3H3,(H,35,36)	WJIOGGXIAJEHJZ-UHFFFAOYSA-N	292738	US10106501, Example B-15	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292738	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292738&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123597	381613026							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558572	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4C[C@]5(CC[C@@H]4C5)C(O)=O)c3Cl)cc12)C(F)(F)F |r|	InChI=1S/C26H23Cl2F3N2O3/c1-13-7-14(26(29,30)31)8-21-18(13)9-16(32(21)2)10-19-20(27)4-3-17(22(19)28)23(34)33-12-25(24(35)36)6-5-15(33)11-25/h3-4,7-9,15H,5-6,10-12H2,1-2H3,(H,35,36)	WNUKAQFGQCCRKO-UHFFFAOYSA-N	292739	US10106501, Example B-16	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292739	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292739&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123514	381613027							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558573	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CC5(CC(CC(O)=O)C5)C4)c3Cl)cc12)C(F)(F)F	InChI=1S/C27H25Cl2F3N2O3/c1-14-5-16(27(30,31)32)7-22-19(14)8-17(33(22)2)9-20-21(28)4-3-18(24(20)29)25(37)34-12-26(13-34)10-15(11-26)6-23(35)36/h3-5,7-8,15H,6,9-13H2,1-2H3,(H,35,36)	HZQVQSYHKFSYGV-UHFFFAOYSA-N	292740	US10106501, Example B-17	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292740	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292740&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123486	381613028							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558574	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CC5(CC(C5)C(O)=O)C4)c3Cl)cc12)C(F)(F)F	InChI=1S/C26H23Cl2F3N2O3/c1-13-5-15(26(29,30)31)6-21-18(13)7-16(32(21)2)8-19-20(27)4-3-17(22(19)28)23(34)33-11-25(12-33)9-14(10-25)24(35)36/h3-7,14H,8-12H2,1-2H3,(H,35,36)	SZEWMEBFWNQVPK-UHFFFAOYSA-N	292741	US10106501, Example B-18	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292741	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292741&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123040	381613029							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558575	CC(C1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl)C(O)=O	InChI=1S/C27H27Cl2F3N2O3/c1-14-10-17(27(30,31)32)11-23-20(14)12-18(33(23)3)13-21-22(28)5-4-19(24(21)29)25(35)34-8-6-16(7-9-34)15(2)26(36)37/h4-5,10-12,15-16H,6-9,13H2,1-3H3,(H,36,37)	QWTBSGNEIWJVHH-UHFFFAOYSA-N	292742	US10106501, Example B-19	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292742	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292742&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123815	381613030							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558576	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC4)C(O)C(O)=O)c3Cl)cc12)C(F)(F)F	InChI=1S/C26H25Cl2F3N2O4/c1-13-9-15(26(29,30)31)10-21-18(13)11-16(32(21)2)12-19-20(27)4-3-17(22(19)28)24(35)33-7-5-14(6-8-33)23(34)25(36)37/h3-4,9-11,14,23,34H,5-8,12H2,1-2H3,(H,36,37)	IZDUHYXDAPGFQI-UHFFFAOYSA-N	292743	US10106501, Example B-20	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292743	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292743&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124129491	381613031					C02929		1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558577	CC1CN(CCC1CC(O)=O)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C27H27Cl2F3N2O3/c1-14-8-17(27(30,31)32)10-23-20(14)11-18(33(23)3)12-21-22(28)5-4-19(25(21)29)26(37)34-7-6-16(9-24(35)36)15(2)13-34/h4-5,8,10-11,15-16H,6-7,9,12-13H2,1-3H3,(H,35,36)	AYLGDDUTJUCSPB-UHFFFAOYSA-N	292744	US10106501, Example B-21	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292744	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292744&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122943	381613032							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558578	Cc1cc(cc2n(C)c(Cc3c(Cl)ncc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)cc12)C(F)(F)F	InChI=1S/C25H24Cl2F3N3O3/c1-13-7-15(25(28,29)30)9-20-17(13)10-16(32(20)2)11-18-22(26)19(12-31-23(18)27)24(36)33-5-3-14(4-6-33)8-21(34)35/h7,9-10,12,14H,3-6,8,11H2,1-2H3,(H,34,35)	JASFBIUNBYREPV-UHFFFAOYSA-N	292745	US10106501, Example B-22	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292745	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292745&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123777	381613033							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558579	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC4)C(C)(C)C(O)=O)c3Cl)cc12)C(F)(F)F	InChI=1S/C28H29Cl2F3N2O3/c1-15-11-17(28(31,32)33)12-23-20(15)13-18(34(23)4)14-21-22(29)6-5-19(24(21)30)25(36)35-9-7-16(8-10-35)27(2,3)26(37)38/h5-6,11-13,16H,7-10,14H2,1-4H3,(H,37,38)	FNYHXAITGYZSDG-UHFFFAOYSA-N	292746	US10106501, Example B-23	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292746	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292746&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123934	381613034							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558580	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CCC(O)=O)CC4)c3Cl)cc12)C(F)(F)F	InChI=1S/C27H27Cl2F3N2O3/c1-15-11-17(27(30,31)32)12-23-20(15)13-18(33(23)2)14-21-22(28)5-4-19(25(21)29)26(37)34-9-7-16(8-10-34)3-6-24(35)36/h4-5,11-13,16H,3,6-10,14H2,1-2H3,(H,35,36)	FXVGCYYSKUYPAK-UHFFFAOYSA-N	292747	US10106501, Example B-24	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292747	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292747&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123559	381613035							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558581	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N[C@H]4CC[C@H](CC4)C(O)=O)c3Cl)cc12)C(F)(F)F |r,wU:19.18,22.25,(2.08,.88,;1.31,2.21,;2.08,3.55,;1.31,4.88,;-.23,4.88,;-1,3.55,;-2.51,3.23,;-3.84,4,;-2.67,1.69,;-4,.92,;-4,-.62,;-5.33,-1.39,;-6.67,-.62,;-5.33,-2.93,;-4,-3.7,;-2.67,-2.93,;-1.33,-3.7,;-1.33,-5.24,;,-2.93,;1.33,-3.7,;2.67,-2.93,;4,-3.7,;4,-5.24,;2.67,-6.01,;1.33,-5.24,;5.33,-6.01,;6.67,-5.24,;5.33,-7.55,;-2.67,-1.39,;-1.33,-.62,;-1.26,1.07,;-.23,2.21,;2.08,6.21,;3.62,6.21,;1.31,7.55,;2.85,7.55,)|	InChI=1S/C26H25Cl2F3N2O3/c1-13-9-15(26(29,30)31)10-22-19(13)11-17(33(22)2)12-20-21(27)8-7-18(23(20)28)24(34)32-16-5-3-14(4-6-16)25(35)36/h7-11,14,16H,3-6,12H2,1-2H3,(H,32,34)(H,35,36)	AZDFVUILZYVTKM-UHFFFAOYSA-N	292748	US10106501, Example B-25	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292748	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292748&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122884	381613036							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558582	C[C@H]1CN(CC[C@@H]1C(O)=O)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl |r|	InChI=1S/C26H25Cl2F3N2O3/c1-13-8-15(26(29,30)31)9-22-19(13)10-16(32(22)3)11-20-21(27)5-4-18(23(20)28)24(34)33-7-6-17(25(35)36)14(2)12-33/h4-5,8-10,14,17H,6-7,11-12H2,1-3H3,(H,35,36)	OSLRVFJRYRWWCB-UHFFFAOYSA-N	292749	US10106501, Example B-26	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292749	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292749&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124129016	381613037							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558583	Cc1cc(nc2n(C)c(Cc3c(Cl)cnc(C(=O)N4CCOCC4)c3Cl)cc12)C(F)(F)F	InChI=1S/C21H19Cl2F3N4O2/c1-11-7-16(21(24,25)26)28-19-13(11)8-12(29(19)2)9-14-15(22)10-27-18(17(14)23)20(31)30-3-5-32-6-4-30/h7-8,10H,3-6,9H2,1-2H3	VGRKWALWCULKOZ-UHFFFAOYSA-N	292750	US10106501, Example GH	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292750	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292750&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123452	381613038							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558584	Cc1cc(cc2n(C)c(Cc3c(Cl)ncc(C(=O)N4CCC(O)(CCO)CC4)c3Cl)cc12)C(F)(F)F	InChI=1S/C25H26Cl2F3N3O3/c1-14-9-15(25(28,29)30)10-20-17(14)11-16(32(20)2)12-18-21(26)19(13-31-22(18)27)23(35)33-6-3-24(36,4-7-33)5-8-34/h9-11,13,34,36H,3-8,12H2,1-2H3	HYSCAPQAWANYCJ-UHFFFAOYSA-N	292751	US10106501, Example BH-2	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292751	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292751&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123330	381613039							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558585	Cc1cc(cc2[nH]c(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)cc12)C(F)(F)F	InChI=1S/C22H19Cl2F3N2O2/c1-12-8-13(22(25,26)27)9-19-16(12)10-14(28-19)11-17-18(23)3-2-15(20(17)24)21(30)29-4-6-31-7-5-29/h2-3,8-10,28H,4-7,11H2,1H3	SKCIUTDOKGNNGB-UHFFFAOYSA-N	292752	US10106501, Example C	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292752	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292752&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123336	381613040							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558586	Cc1c(Cc2c(Cl)ccc(C(=O)N3CCN(CC3)C3COC3)c2Cl)nc2c(C)cc(nn12)C(F)(F)F	InChI=1S/C24H24Cl2F3N5O2/c1-13-9-20(24(27,28)29)31-34-14(2)19(30-22(13)34)10-17-18(25)4-3-16(21(17)26)23(35)33-7-5-32(6-8-33)15-11-36-12-15/h3-4,9,15H,5-8,10-12H2,1-2H3	ZCLZXWZISNFATP-UHFFFAOYSA-N	292753	US10106501, Example CZ-1	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292753	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292753&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122924	381613041							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558587	Cc1c(nc2c(C)cc(nn12)C(F)(F)F)C(=O)c1c(Cl)ccc(C(=O)N2CCC(CC(O)=O)CC2)c1Cl	InChI=1S/C24H21Cl2F3N4O4/c1-11-9-16(24(27,28)29)31-33-12(2)20(30-22(11)33)21(36)18-15(25)4-3-14(19(18)26)23(37)32-7-5-13(6-8-32)10-17(34)35/h3-4,9,13H,5-8,10H2,1-2H3,(H,34,35)	ZHKFCHGUAAKOMM-UHFFFAOYSA-N	292754	US10106501, Example CZ-1A	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292754	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292754&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123049	381613042							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558588	Cc1c(Cc2c(Cl)ccc(C(=O)N3CCC(CC3)C3COC3)c2Cl)nc2c(C)cc(nn12)C(F)(F)F	InChI=1S/C25H25Cl2F3N4O2/c1-13-9-21(25(28,29)30)32-34-14(2)20(31-23(13)34)10-18-19(26)4-3-17(22(18)27)24(35)33-7-5-15(6-8-33)16-11-36-12-16/h3-4,9,15-16H,5-8,10-12H2,1-2H3	UMVLBXNKAQACCY-UHFFFAOYSA-N	292755	US10106501, Example CZ-2	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292755	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292755&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122908	381613043							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558589	C[C@@H]1CN(CCN1S(C)(=O)=O)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(nn3c2C)C(F)(F)F)c1Cl |r|	InChI=1S/C23H24Cl2F3N5O3S/c1-12-9-19(23(26,27)28)30-33-14(3)18(29-21(12)33)10-16-17(24)6-5-15(20(16)25)22(34)31-7-8-32(13(2)11-31)37(4,35)36/h5-6,9,13H,7-8,10-11H2,1-4H3	MVLGCGNIUURKKQ-UHFFFAOYSA-N	292756	US10106501, Example CZ-3	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292756	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292756&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122839	381613044							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558590	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)cc12)C(F)(F)F	InChI=1S/C23H21Cl2F3N2O2/c1-13-9-14(23(26,27)28)10-20-17(13)11-15(29(20)2)12-18-19(24)4-3-16(21(18)25)22(31)30-5-7-32-8-6-30/h3-4,9-11H,5-8,12H2,1-2H3	YGYIEBMYABQRGD-UHFFFAOYSA-N	292757	US10106501, Example D	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292757	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292757&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122932	381613045							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558591	CCn1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)cc2c(C)cc(cc12)C(F)(F)F	InChI=1S/C24H23Cl2F3N2O2/c1-3-31-16(12-18-14(2)10-15(11-21(18)31)24(27,28)29)13-19-20(25)5-4-17(22(19)26)23(32)30-6-8-33-9-7-30/h4-5,10-12H,3,6-9,13H2,1-2H3	MIMAAXIVEWOPCR-UHFFFAOYSA-N	292758	US10106501, Example D-1	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292758	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292758&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123670	381613046							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558592	CC(=O)n1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)cc2c(C)cc(cc12)C(F)(F)F	InChI=1S/C24H21Cl2F3N2O3/c1-13-9-15(24(27,28)29)10-21-18(13)11-16(31(21)14(2)32)12-19-20(25)4-3-17(22(19)26)23(33)30-5-7-34-8-6-30/h3-4,9-11H,5-8,12H2,1-2H3	VNBJAJRWUHABJF-UHFFFAOYSA-N	292759	US10106501, Example D-2	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292759	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292759&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123160	381613047							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558593	CC(C)Cn1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)cc2c(C)cc(cc12)C(F)(F)F	InChI=1S/C26H27Cl2F3N2O2/c1-15(2)14-33-18(12-20-16(3)10-17(11-23(20)33)26(29,30)31)13-21-22(27)5-4-19(24(21)28)25(34)32-6-8-35-9-7-32/h4-5,10-12,15H,6-9,13-14H2,1-3H3	FOJURYOFHWSLMR-UHFFFAOYSA-N	292760	US10106501, Example D-3	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292760	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292760&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123478	381613048							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558594	Cc1nn(Cc2c(Cl)ccc(C(=O)N3CCC(CC3)C3COC3)c2Cl)c2c(C)cc(cc12)C(F)(F)F	InChI=1S/C26H26Cl2F3N3O2/c1-14-9-18(26(29,30)31)10-20-15(2)32-34(24(14)20)11-21-22(27)4-3-19(23(21)28)25(35)33-7-5-16(6-8-33)17-12-36-13-17/h3-4,9-10,16-17H,5-8,11-13H2,1-2H3	DYBNUJKKDSSNEH-UHFFFAOYSA-N	292761	(2,4-dichloro-3-((3,7-dimethyl-5-(trifluoromethyl)-1H-indazol-1-yl)methyl)phenyl)(4-(oxetan-3-yl)piperidin-1-yl)methanone::US10106501, Example DD-1	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292761	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292761&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123214	381613049							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558595	C[C@@H]1CN(CC[C@@H]1C(O)=O)C(=O)c1ccc(Cl)c(Cn2cc(C)c3cc(cc(C)c23)C(F)(F)F)c1Cl |r|	InChI=1S/C26H25Cl2F3N2O3/c1-13-8-16(26(29,30)31)9-19-15(3)11-33(23(13)19)12-20-21(27)5-4-18(22(20)28)24(34)32-7-6-17(25(35)36)14(2)10-32/h4-5,8-9,11,14,17H,6-7,10,12H2,1-3H3,(H,35,36)	YUVITFLKAVYHMK-UHFFFAOYSA-N	292762	US10106501, Example DH1-1	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292762	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292762&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122875	381613050							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558596	C[C@H]1CN(CC[C@H]1C(O)=O)C(=O)c1ccc(Cl)c(Cn2cc(C)c3cc(cc(C)c23)C(F)(F)F)c1Cl |r|	InChI=1S/C26H25Cl2F3N2O3/c1-13-8-16(26(29,30)31)9-19-15(3)11-33(23(13)19)12-20-21(27)5-4-18(22(20)28)24(34)32-7-6-17(25(35)36)14(2)10-32/h4-5,8-9,11,14,17H,6-7,10,12H2,1-3H3,(H,35,36)	YUVITFLKAVYHMK-UHFFFAOYSA-N	292763	US10106501, Example DH1-2	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292763	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292763&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123321	381613051							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558597	Cc1cn(C(=O)c2c(Cl)ccc(C(=O)N3CCC(CC3)C(O)=O)c2Cl)c2c(C)cc(cc12)C(F)(F)F	InChI=1S/C25H21Cl2F3N2O4/c1-12-9-15(25(28,29)30)10-17-13(2)11-32(21(12)17)23(34)19-18(26)4-3-16(20(19)27)22(33)31-7-5-14(6-8-31)24(35)36/h3-4,9-11,14H,5-8H2,1-2H3,(H,35,36)	FOPRDSZNQDJPIG-UHFFFAOYSA-N	292764	US10106501, Example DJ1-1	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292764	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292764&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123770	381613052							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558598	C[C@@H]1CN(CC[C@@H]1C(O)=O)C(=O)c1ccc(Cl)c(C(=O)n2cc(C)c3cc(cc(C)c23)C(F)(F)F)c1Cl |r|	InChI=1S/C26H23Cl2F3N2O4/c1-12-8-15(26(29,30)31)9-18-14(3)11-33(22(12)18)24(35)20-19(27)5-4-17(21(20)28)23(34)32-7-6-16(25(36)37)13(2)10-32/h4-5,8-9,11,13,16H,6-7,10H2,1-3H3,(H,36,37)	NEAOTPQCWMDIAB-UHFFFAOYSA-N	292765	US10106501, Example DJ1-2	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292765	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292765&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123051	381613053							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558599	C[C@H]1CN(CC[C@H]1C(O)=O)C(=O)c1ccc(Cl)c(C(=O)n2cc(C)c3cc(cc(C)c23)C(F)(F)F)c1Cl |r|	InChI=1S/C26H23Cl2F3N2O4/c1-12-8-15(26(29,30)31)9-18-14(3)11-33(22(12)18)24(35)20-19(27)5-4-17(21(20)28)23(34)32-7-6-16(25(36)37)13(2)10-32/h4-5,8-9,11,13,16H,6-7,10H2,1-3H3,(H,36,37)	NEAOTPQCWMDIAB-UHFFFAOYSA-N	292766	US10106501, Example DJ1-3	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292766	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292766&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123825	381613054							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558600	Cc1cc(OC(F)(F)F)cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)cc12	InChI=1S/C23H21Cl2F3N2O3/c1-13-9-15(33-23(26,27)28)12-20-17(13)10-14(29(20)2)11-18-19(24)4-3-16(21(18)25)22(31)30-5-7-32-8-6-30/h3-4,9-10,12H,5-8,11H2,1-2H3	FIQMWEHWEFDOOF-UHFFFAOYSA-N	292767	US10106501, Example DP-1	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292767	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292767&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123576	381613055							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558601	CC1CN(CCC1C(O)=O)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(OC(F)(F)F)cc3n2C)c1Cl	InChI=1S/C26H25Cl2F3N2O4/c1-13-8-16(37-26(29,30)31)11-22-19(13)9-15(32(22)3)10-20-21(27)5-4-18(23(20)28)24(34)33-7-6-17(25(35)36)14(2)12-33/h4-5,8-9,11,14,17H,6-7,10,12H2,1-3H3,(H,35,36)	FBCFWLPBMMUOTI-UHFFFAOYSA-N	292768	US10106501, Example DP-2	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292768	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292768&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123885	381613056							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558602	C[C@H]1CN(CC[C@H]1C(O)=O)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(OC(F)(F)F)cc3n2C)c1Cl |r|	InChI=1S/C26H25Cl2F3N2O4/c1-13-8-16(37-26(29,30)31)11-22-19(13)9-15(32(22)3)10-20-21(27)5-4-18(23(20)28)24(34)33-7-6-17(25(35)36)14(2)12-33/h4-5,8-9,11,14,17H,6-7,10,12H2,1-3H3,(H,35,36)	FBCFWLPBMMUOTI-UHFFFAOYSA-N	292769	US10106501, Example DP-3	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292769	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292769&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122873	381613057							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558603	Cc1cc(OC(F)(F)F)cc2n(C)cc(Cc3c(Cl)ccc(C(=O)N4CCC(CC4)C(O)=O)c3Cl)c12	InChI=1S/C25H23Cl2F3N2O4/c1-13-9-16(36-25(28,29)30)11-20-21(13)15(12-31(20)2)10-18-19(26)4-3-17(22(18)27)23(33)32-7-5-14(6-8-32)24(34)35/h3-4,9,11-12,14H,5-8,10H2,1-2H3,(H,34,35)	VEFZTTLTOCPAAR-UHFFFAOYSA-N	292770	US10106501, Example DU	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292770	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292770&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123436	381613058							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558604	Cc1cc(OC(F)(F)F)cc2n(C)cc(Cc3c(Cl)ccc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)c12	InChI=1S/C26H25Cl2F3N2O4/c1-14-9-17(37-26(29,30)31)12-21-23(14)16(13-32(21)2)11-19-20(27)4-3-18(24(19)28)25(36)33-7-5-15(6-8-33)10-22(34)35/h3-4,9,12-13,15H,5-8,10-11H2,1-2H3,(H,34,35)	BIYFFUYJLYYTIO-UHFFFAOYSA-N	292771	US10106501, Example DU1-1	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292771	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292771&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123149	381613059							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558605	CC1CN(CCC1C(O)=O)C(=O)c1ccc(Cl)c(Cc2cn(C)c3cc(OC(F)(F)F)cc(C)c23)c1Cl	InChI=1S/C26H25Cl2F3N2O4/c1-13-8-16(37-26(29,30)31)10-21-22(13)15(12-32(21)3)9-19-20(27)5-4-18(23(19)28)24(34)33-7-6-17(25(35)36)14(2)11-33/h4-5,8,10,12,14,17H,6-7,9,11H2,1-3H3,(H,35,36)	XWGGYKIWUHKVDK-UHFFFAOYSA-N	292772	US10106501, Example DU1-2	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292772	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292772&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123395	381613060							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558606	Cc1cc(cc2n(C)cc(Cc3c(Cl)ncc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)c12)C(F)(F)F	InChI=1S/C25H24Cl2F3N3O3/c1-13-7-16(25(28,29)30)10-19-21(13)15(12-32(19)2)9-17-22(26)18(11-31-23(17)27)24(36)33-5-3-14(4-6-33)8-20(34)35/h7,10-12,14H,3-6,8-9H2,1-2H3,(H,34,35)	NVDGKVMJPGNXBW-UHFFFAOYSA-N	292773	US10106501, Example DV	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292773	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292773&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123012	381613061							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558607	Cc1cc(cc2n(C)cc(Cc3c(Cl)cnc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)c12)C(F)(F)F	InChI=1S/C25H24Cl2F3N3O3/c1-13-7-16(25(28,29)30)10-19-21(13)15(12-32(19)2)9-17-18(26)11-31-23(22(17)27)24(36)33-5-3-14(4-6-33)8-20(34)35/h7,10-12,14H,3-6,8-9H2,1-2H3,(H,34,35)	CILHTKBVCASUJE-UHFFFAOYSA-N	292774	US10106501, Example DW	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292774	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292774&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123638	381613062							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558608	Cc1cc(OC(F)(F)F)cc2n(C)cc(Cc3c(Cl)cnc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)c12	InChI=1S/C25H24Cl2F3N3O4/c1-13-7-16(37-25(28,29)30)10-19-21(13)15(12-32(19)2)9-17-18(26)11-31-23(22(17)27)24(36)33-5-3-14(4-6-33)8-20(34)35/h7,10-12,14H,3-6,8-9H2,1-2H3,(H,34,35)	PLVLLWWKXBSBDY-UHFFFAOYSA-N	292775	US10106501, Example DX	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292775	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292775&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123068	381613063							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558609	Cc1cc(OC(F)(F)F)cc2n(C)cc(Cc3c(Cl)ncc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)c12	InChI=1S/C25H24Cl2F3N3O4/c1-13-7-16(37-25(28,29)30)10-19-21(13)15(12-32(19)2)9-17-22(26)18(11-31-23(17)27)24(36)33-5-3-14(4-6-33)8-20(34)35/h7,10-12,14H,3-6,8-9H2,1-2H3,(H,34,35)	AXLCPZVTECLMPV-UHFFFAOYSA-N	292776	US10106501, Example DY	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292776	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292776&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123069	381613064							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558610	Cc1cc(cc2occ(Cc3c(Cl)ccc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)c12)C(F)(F)F	InChI=1S/C25H22Cl2F3NO4/c1-13-8-16(25(28,29)30)11-20-22(13)15(12-35-20)10-18-19(26)3-2-17(23(18)27)24(34)31-6-4-14(5-7-31)9-21(32)33/h2-3,8,11-12,14H,4-7,9-10H2,1H3,(H,32,33)	NZGFAFJCLIWOAL-UHFFFAOYSA-N	292777	US10106501, Example DZ	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292777	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292777&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123102	381613065							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558611	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)cc2ccc(cc12)C(F)(F)F	InChI=1S/C22H19Cl2F3N2O2/c1-28-15(10-13-2-3-14(11-19(13)28)22(25,26)27)12-17-18(23)5-4-16(20(17)24)21(30)29-6-8-31-9-7-29/h2-5,10-11H,6-9,12H2,1H3	CWBSCPVTABVSEI-UHFFFAOYSA-N	292778	US10106501, Example E	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292778	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292778&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123092	381613066							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558612	Cc1nn(C(=O)c2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)c2c(C)cc(cc12)C(F)(F)F	InChI=1S/C25H22Cl2F3N3O4/c1-12-9-15(25(28,29)30)11-17-13(2)31-33(22(12)17)24(37)20-18(26)4-3-16(21(20)27)23(36)32-7-5-14(6-8-32)10-19(34)35/h3-4,9,11,14H,5-8,10H2,1-2H3,(H,34,35)	BWSXRKXMYVQOGJ-UHFFFAOYSA-N	292779	US10106501, Example EA	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292779	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292779&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122848	381613067							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558613	Cc1n(nc2c(C)cc(cc12)C(F)(F)F)C(=O)c1c(Cl)ccc(C(=O)N2CCC(CC(O)=O)CC2)c1Cl	InChI=1S/C25H22Cl2F3N3O4/c1-12-9-15(25(28,29)30)11-17-13(2)33(31-22(12)17)24(37)20-18(26)4-3-16(21(20)27)23(36)32-7-5-14(6-8-32)10-19(34)35/h3-4,9,11,14H,5-8,10H2,1-2H3,(H,34,35)	BTJUUYVXNAIHNL-UHFFFAOYSA-N	292780	US10106501, Example EB	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292780	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292780&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122824	381613068							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558614	Cc1cc(cc2cnn(C(=O)c3c(Cl)ccc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)c12)C(F)(F)F	InChI=1S/C24H20Cl2F3N3O4/c1-12-8-15(24(27,28)29)10-14-11-30-32(21(12)14)23(36)19-17(25)3-2-16(20(19)26)22(35)31-6-4-13(5-7-31)9-18(33)34/h2-3,8,10-11,13H,4-7,9H2,1H3,(H,33,34)	PQGVIMZCRYQSHB-UHFFFAOYSA-N	292781	US10106501, Example EC	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292781	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292781&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124129621	381613069							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558615	Cc1cc(cc2cn(Cc3c(Cl)ccc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C24H22Cl2F3N3O3/c1-13-8-16(24(27,28)29)10-15-11-32(30-22(13)15)12-18-19(25)3-2-17(21(18)26)23(35)31-6-4-14(5-7-31)9-20(33)34/h2-3,8,10-11,14H,4-7,9,12H2,1H3,(H,33,34)	ZDWNSPBEKZNESW-UHFFFAOYSA-N	292782	US10106501, Example ED	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292782	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292782&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123109	381613070							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558616	Cc1cc(cc2n(C)nc(Cc3c(Cl)ccc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)c12)C(F)(F)F	InChI=1S/C25H24Cl2F3N3O3/c1-13-9-15(25(28,29)30)11-20-22(13)19(31-32(20)2)12-17-18(26)4-3-16(23(17)27)24(36)33-7-5-14(6-8-33)10-21(34)35/h3-4,9,11,14H,5-8,10,12H2,1-2H3,(H,34,35)	JVRSMTNVMPVDAZ-UHFFFAOYSA-N	292783	US10106501, Example EE	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292783	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292783&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123168	381613071							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558617	Cc1nn(Cc2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)c2ccc(cc12)C(F)(F)F	InChI=1S/C24H22Cl2F3N3O3/c1-13-17-11-15(24(27,28)29)2-5-20(17)32(30-13)12-18-19(25)4-3-16(22(18)26)23(35)31-8-6-14(7-9-31)10-21(33)34/h2-5,11,14H,6-10,12H2,1H3,(H,33,34)	FXDUKZFOQUCZEM-UHFFFAOYSA-N	292784	US10106501, Example EF	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292784	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292784&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122964	381613072							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558618	Cc1cn(Cc2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)c2c(C)cc(OC(F)(F)F)cc12	InChI=1S/C26H25Cl2F3N2O4/c1-14-9-17(37-26(29,30)31)11-19-15(2)12-33(24(14)19)13-20-21(27)4-3-18(23(20)28)25(36)32-7-5-16(6-8-32)10-22(34)35/h3-4,9,11-12,16H,5-8,10,13H2,1-2H3,(H,34,35)	HGXLAEQMHUMJET-UHFFFAOYSA-N	292785	US10106501, Example EG	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292785	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292785&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122916	381613073							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558619	Cc1cn(Cc2c(Cl)ccc(C(=O)N3CCC(CC3)C(O)=O)c2Cl)c2c(C)cc(OC(F)(F)F)cc12	InChI=1S/C25H23Cl2F3N2O4/c1-13-9-16(36-25(28,29)30)10-18-14(2)11-32(22(13)18)12-19-20(26)4-3-17(21(19)27)23(33)31-7-5-15(6-8-31)24(34)35/h3-4,9-11,15H,5-8,12H2,1-2H3,(H,34,35)	IHYRUJNTHWJRAQ-UHFFFAOYSA-N	292786	US10106501, Example EG-1	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292786	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292786&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124129624	381613074							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558620	C[C@H]1CN(CC[C@H]1C(O)=O)C(=O)c1ccc(Cl)c(Cn2cc(C)c3cc(OC(F)(F)F)cc(C)c23)c1Cl |r|	InChI=1S/C26H25Cl2F3N2O4/c1-13-8-16(37-26(29,30)31)9-19-15(3)11-33(23(13)19)12-20-21(27)5-4-18(22(20)28)24(34)32-7-6-17(25(35)36)14(2)10-32/h4-5,8-9,11,14,17H,6-7,10,12H2,1-3H3,(H,35,36)	OFQPJQDCAUICAI-UHFFFAOYSA-N	292787	US10106501, Example EG-2	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292787	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292787&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124129625	381613075							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558621	Cc1cn(C(=O)c2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)c2c(C)cc(OC(F)(F)F)cc12	InChI=1S/C26H23Cl2F3N2O5/c1-13-9-16(38-26(29,30)31)11-18-14(2)12-33(23(13)18)25(37)21-19(27)4-3-17(22(21)28)24(36)32-7-5-15(6-8-32)10-20(34)35/h3-4,9,11-12,15H,5-8,10H2,1-2H3,(H,34,35)	ISPYRNPMXAFLAF-UHFFFAOYSA-N	292788	US10106501, Example EH	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292788	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292788&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122931	381613076							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558622	Cc1cn(C(=O)c2c(Cl)ccc(C(=O)N3CCC(CC3)C(O)=O)c2Cl)c2c(C)cc(OC(F)(F)F)cc12	InChI=1S/C25H21Cl2F3N2O5/c1-12-9-15(37-25(28,29)30)10-17-13(2)11-32(21(12)17)23(34)19-18(26)4-3-16(20(19)27)22(33)31-7-5-14(6-8-31)24(35)36/h3-4,9-11,14H,5-8H2,1-2H3,(H,35,36)	ONYFLSUKTFIHND-UHFFFAOYSA-N	292789	US10106501, Example EH-1	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292789	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292789&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122990	381613077							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558623	OC(=O)CC1CCN(CC1)C(=O)c1ccc(Cl)c(Cn2ccc3cc(OC(F)(F)F)ccc23)c1Cl	InChI=1S/C24H21Cl2F3N2O4/c25-19-3-2-17(23(34)30-8-5-14(6-9-30)11-21(32)33)22(26)18(19)13-31-10-7-15-12-16(1-4-20(15)31)35-24(27,28)29/h1-4,7,10,12,14H,5-6,8-9,11,13H2,(H,32,33)	XNCKCCABPNKZGI-UHFFFAOYSA-N	292790	US10106501, Example EI	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292790	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292790&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123056	381613078							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558624	CC(C)c1ccc2n(Cc3c(Cl)ccc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)ccc2c1	InChI=1S/C26H28Cl2N2O3/c1-16(2)18-3-6-23-19(14-18)9-12-30(23)15-21-22(27)5-4-20(25(21)28)26(33)29-10-7-17(8-11-29)13-24(31)32/h3-6,9,12,14,16-17H,7-8,10-11,13,15H2,1-2H3,(H,31,32)	KIWCJWPCEOHKFK-UHFFFAOYSA-N	292791	US10106501, Example EI-1	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292791	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292791&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124129626	381613079							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558625	CSc1ccc2n(Cc3c(Cl)ccc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)ccc2c1	InChI=1S/C24H24Cl2N2O3S/c1-32-17-2-5-21-16(13-17)8-11-28(21)14-19-20(25)4-3-18(23(19)26)24(31)27-9-6-15(7-10-27)12-22(29)30/h2-5,8,11,13,15H,6-7,9-10,12,14H2,1H3,(H,29,30)	OUICKGGDUCCGJK-UHFFFAOYSA-N	292792	US10106501, Example EI-2	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292792	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292792&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124129627	381613080							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558626	OC(=O)CC1CCN(CC1)C(=O)c1ccc(Cl)c(Cn2ccc3cccc(Cl)c23)c1Cl	InChI=1S/C23H21Cl3N2O3/c24-18-5-4-16(23(31)27-9-6-14(7-10-27)12-20(29)30)21(26)17(18)13-28-11-8-15-2-1-3-19(25)22(15)28/h1-5,8,11,14H,6-7,9-10,12-13H2,(H,29,30)	MERMIZMUERYVOT-UHFFFAOYSA-N	292793	US10106501, Example EI-3	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292793	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292793&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124129628	381613081							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558627	OC(=O)CC1CCN(CC1)C(=O)c1ccc(Cl)c(Cn2ccc3cc(ccc23)C(F)(F)F)c1Cl	InChI=1S/C24H21Cl2F3N2O3/c25-19-3-2-17(23(34)30-8-5-14(6-9-30)11-21(32)33)22(26)18(19)13-31-10-7-15-12-16(24(27,28)29)1-4-20(15)31/h1-4,7,10,12,14H,5-6,8-9,11,13H2,(H,32,33)	HJOCTANPXRBJQP-UHFFFAOYSA-N	292794	US10106501, Example EI-4	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292794	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292794&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124129234	381613082							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558628	OC(=O)CC1CCN(CC1)C(=O)c1ccc(Cl)c(Cn2ccc3cc(cc(Cl)c23)C(F)(F)F)c1Cl	InChI=1S/C24H20Cl3F3N2O3/c25-18-2-1-16(23(35)31-6-3-13(4-7-31)9-20(33)34)21(27)17(18)12-32-8-5-14-10-15(24(28,29)30)11-19(26)22(14)32/h1-2,5,8,10-11,13H,3-4,6-7,9,12H2,(H,33,34)	MNEOHCYSHVKLIC-UHFFFAOYSA-N	292795	US10106501, Example EI-6::US10106501, Example EI-5	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292795	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292795&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123797	381613083							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558629	OC(=O)CC1CCN(CC1)C(=O)c1ccc(Cl)c(Cn2ccc3cc(cc(Cl)c23)C(F)(F)F)c1Cl	InChI=1S/C24H20Cl3F3N2O3/c25-18-2-1-16(23(35)31-6-3-13(4-7-31)9-20(33)34)21(27)17(18)12-32-8-5-14-10-15(24(28,29)30)11-19(26)22(14)32/h1-2,5,8,10-11,13H,3-4,6-7,9,12H2,(H,33,34)	MNEOHCYSHVKLIC-UHFFFAOYSA-N	292795	US10106501, Example EI-6::US10106501, Example EI-5	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292795	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292795&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123797	381613083							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558630	OC(=O)CC1CCN(CC1)C(=O)c1ccc(Cl)c(Cn2ccc3c(cccc23)C(F)(F)F)c1Cl	InChI=1S/C24H21Cl2F3N2O3/c25-19-5-4-16(23(34)30-9-6-14(7-10-30)12-21(32)33)22(26)17(19)13-31-11-8-15-18(24(27,28)29)2-1-3-20(15)31/h1-5,8,11,14H,6-7,9-10,12-13H2,(H,32,33)	ULJFHCBDXHUADF-UHFFFAOYSA-N	292798	US10106501, Example EI-7	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292798	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292798&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123418	381613085							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558631	Cc1cc(OC(F)(F)F)cc2ccn(Cc3c(Cl)ccc(C(=O)N4CCC(CCC(O)=O)CC4)c3Cl)c12	InChI=1S/C26H25Cl2F3N2O4/c1-15-12-18(37-26(29,30)31)13-17-8-11-33(24(15)17)14-20-21(27)4-3-19(23(20)28)25(36)32-9-6-16(7-10-32)2-5-22(34)35/h3-4,8,11-13,16H,2,5-7,9-10,14H2,1H3,(H,34,35)	AFDWEWFEENHJIB-UHFFFAOYSA-N	292799	US10106501, Example EJ-2	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292799	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292799&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124129630	381613086							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558632	Cc1cc(OC(F)(F)F)cc2ccn(Cc3c(Cl)ccc(C(=O)N4CC5(CC(CC(O)=O)C5)C4)c3Cl)c12	InChI=1S/C26H23Cl2F3N2O4/c1-14-6-17(37-26(29,30)31)8-16-4-5-32(23(14)16)11-19-20(27)3-2-18(22(19)28)24(36)33-12-25(13-33)9-15(10-25)7-21(34)35/h2-6,8,15H,7,9-13H2,1H3,(H,34,35)	OFPDKILKHWNOCL-UHFFFAOYSA-N	292800	US10106501, Example EJ-1	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292800	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292800&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124129629	381613087							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558633	Cc1ccc(C(=O)N2CCC(CC(O)=O)CC2)c(C)c1Cn1ccc2cc(OC(F)(F)F)cc(C)c12	InChI=1S/C27H29F3N2O4/c1-16-4-5-22(26(35)31-9-6-19(7-10-31)13-24(33)34)18(3)23(16)15-32-11-8-20-14-21(36-27(28,29)30)12-17(2)25(20)32/h4-5,8,11-12,14,19H,6-7,9-10,13,15H2,1-3H3,(H,33,34)	PBCZWAPFABNLCQ-UHFFFAOYSA-N	292801	US10106501, Example EK	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292801	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292801&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122892	381613088							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558634	Cc1cc(OC(F)(F)F)cc2ccn(C(=O)c3c(Cl)ccc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)c12	InChI=1S/C25H21Cl2F3N2O5/c1-13-10-16(37-25(28,29)30)12-15-6-9-32(22(13)15)24(36)20-18(26)3-2-17(21(20)27)23(35)31-7-4-14(5-8-31)11-19(33)34/h2-3,6,9-10,12,14H,4-5,7-8,11H2,1H3,(H,33,34)	YMVJKDIALKFKBM-UHFFFAOYSA-N	292802	US10106501, Example EL	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292802	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292802&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123673	381613089							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558635	Cc1cc(OC(F)(F)F)cc2ccn(C(=O)c3c(Cl)ccc(C(=O)N4CC5(CC(CC(O)=O)C5)C4)c3Cl)c12	InChI=1S/C26H21Cl2F3N2O5/c1-13-6-16(38-26(29,30)31)8-15-4-5-33(22(13)15)24(37)20-18(27)3-2-17(21(20)28)23(36)32-11-25(12-32)9-14(10-25)7-19(34)35/h2-6,8,14H,7,9-12H2,1H3,(H,34,35)	RQRGEANPZLKCNT-UHFFFAOYSA-N	292803	US10106501, Example EL-1	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292803	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292803&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124129218	381613090							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558636	Cc1cc(OC(F)F)cc2ccn(Cc3c(Cl)ccc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)c12	InChI=1S/C25H24Cl2F2N2O4/c1-14-10-17(35-25(28)29)12-16-6-9-31(23(14)16)13-19-20(26)3-2-18(22(19)27)24(34)30-7-4-15(5-8-30)11-21(32)33/h2-3,6,9-10,12,15,25H,4-5,7-8,11,13H2,1H3,(H,32,33)	LFLUTKCZQVVZKM-UHFFFAOYSA-N	292804	US10106501, Example EM	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292804	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292804&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122856	381613091							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558637	OC(=O)CC1CCN(CC1)C(=O)c1ccc(Cl)c(Cn2ccc3cc(cc(F)c23)C2CC2)c1Cl	InChI=1S/C26H25Cl2FN2O3/c27-21-4-3-19(26(34)30-8-5-15(6-9-30)11-23(32)33)24(28)20(21)14-31-10-7-17-12-18(16-1-2-16)13-22(29)25(17)31/h3-4,7,10,12-13,15-16H,1-2,5-6,8-9,11,14H2,(H,32,33)	HJHIDPUZFDBIFV-UHFFFAOYSA-N	292805	US10106501, Example EO::US10106501, Example EN	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292805	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292805&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123392	381613092							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558638	OC(=O)CC1CCN(CC1)C(=O)c1ccc(Cl)c(Cn2ccc3cc(cc(F)c23)C2CC2)c1Cl	InChI=1S/C26H25Cl2FN2O3/c27-21-4-3-19(26(34)30-8-5-15(6-9-30)11-23(32)33)24(28)20(21)14-31-10-7-17-12-18(16-1-2-16)13-22(29)25(17)31/h3-4,7,10,12-13,15-16H,1-2,5-6,8-9,11,14H2,(H,32,33)	HJHIDPUZFDBIFV-UHFFFAOYSA-N	292805	US10106501, Example EO::US10106501, Example EN	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292805	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292805&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123392	381613092							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558639	OC(=O)CC1CCN(CC1)C(=O)c1ccc(Cl)c(Cn2ccc3cc(cc(F)c23)C(F)(F)F)c1Cl	InChI=1S/C24H20Cl2F4N2O3/c25-18-2-1-16(23(35)31-6-3-13(4-7-31)9-20(33)34)21(26)17(18)12-32-8-5-14-10-15(24(28,29)30)11-19(27)22(14)32/h1-2,5,8,10-11,13H,3-4,6-7,9,12H2,(H,33,34)	HLEGBALKBSGPGV-UHFFFAOYSA-N	292807	US10106501, Example EP	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292807	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292807&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123060	381613093							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558640	Cc1cn(C(=O)c2c(Cl)ncc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)c2c(C)cc(cc12)C(F)(F)F	InChI=1S/C25H22Cl2F3N3O4/c1-12-7-15(25(28,29)30)9-16-13(2)11-33(21(12)16)24(37)19-20(26)17(10-31-22(19)27)23(36)32-5-3-14(4-6-32)8-18(34)35/h7,9-11,14H,3-6,8H2,1-2H3,(H,34,35)	NRQUQNYNZDWJHD-UHFFFAOYSA-N	292808	US10106501, Example EQ	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292808	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292808&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123680	381613094							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558641	Cc1cn(Cc2c(Cl)ncc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)c2c(C)cc(cc12)C(F)(F)F	InChI=1S/C25H24Cl2F3N3O3/c1-13-7-16(25(28,29)30)9-17-14(2)11-33(22(13)17)12-19-21(26)18(10-31-23(19)27)24(36)32-5-3-15(4-6-32)8-20(34)35/h7,9-11,15H,3-6,8,12H2,1-2H3,(H,34,35)	YRBJRFJSESZNTP-UHFFFAOYSA-N	292809	US10106501, Example ER	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292809	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292809&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122847	381613095							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558642	Cc1cc(cc2ccn(C(=O)c3c(Cl)ccc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)c12)C(F)(F)F	InChI=1S/C25H21Cl2F3N2O4/c1-13-10-16(25(28,29)30)12-15-6-9-32(22(13)15)24(36)20-18(26)3-2-17(21(20)27)23(35)31-7-4-14(5-8-31)11-19(33)34/h2-3,6,9-10,12,14H,4-5,7-8,11H2,1H3,(H,33,34)	CIUPEQBZTMBVLP-UHFFFAOYSA-N	292810	US10106501, Example ES	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292810	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292810&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123456	381613096							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558643	Cc1cn(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)c2c(C)nc(cc12)C(F)(F)F	InChI=1S/C22H20Cl2F3N3O2/c1-12-10-30(20-13(2)28-18(9-15(12)20)22(25,26)27)11-16-17(23)4-3-14(19(16)24)21(31)29-5-7-32-8-6-29/h3-4,9-10H,5-8,11H2,1-2H3	JLMYCGAXXUXCQC-UHFFFAOYSA-N	292811	US10106501, Example ET	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292811	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292811&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123252	381613097							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558644	Cc1cn(Cc2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)c2c(C)nc(cc12)C(F)(F)F	InChI=1S/C25H24Cl2F3N3O3/c1-13-11-33(23-14(2)31-20(10-17(13)23)25(28,29)30)12-18-19(26)4-3-16(22(18)27)24(36)32-7-5-15(6-8-32)9-21(34)35/h3-4,10-11,15H,5-9,12H2,1-2H3,(H,34,35)	KKNNECJYBLUQAR-UHFFFAOYSA-N	292812	US10106501, Example EU	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292812	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292812&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123037	381613098							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558645	Cc1cn(C(=O)c2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)c2c(C)nc(cc12)C(F)(F)F	InChI=1S/C25H22Cl2F3N3O4/c1-12-11-33(22-13(2)31-18(10-16(12)22)25(28,29)30)24(37)20-17(26)4-3-15(21(20)27)23(36)32-7-5-14(6-8-32)9-19(34)35/h3-4,10-11,14H,5-9H2,1-2H3,(H,34,35)	YMLWDVWVYPCIFL-UHFFFAOYSA-N	292813	US10106501, Example EV	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292813	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292813&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123145	381613099							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558646	Cc1cn(Cc2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)c2c(C)cc(nc12)C(F)(F)F	InChI=1S/C25H24Cl2F3N3O3/c1-13-9-19(25(28,29)30)31-22-14(2)11-33(23(13)22)12-17-18(26)4-3-16(21(17)27)24(36)32-7-5-15(6-8-32)10-20(34)35/h3-4,9,11,15H,5-8,10,12H2,1-2H3,(H,34,35)	KPICWCQMJHRIQZ-UHFFFAOYSA-N	292814	US10106501, Example EW	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292814	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292814&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122877	381613100							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558647	Cc1c(ccc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)cc12)C#N	InChI=1S/C23H21Cl2N3O2/c1-14-15(13-26)3-6-21-18(14)11-16(27(21)2)12-19-20(24)5-4-17(22(19)25)23(29)28-7-9-30-10-8-28/h3-6,11H,7-10,12H2,1-2H3	XRTQBXCVBUSQSM-UHFFFAOYSA-N	292815	US10106501, Example EX	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292815	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292815&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123820	381613101							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558648	Cc1c(ccc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)cc12)C#N	InChI=1S/C26H25Cl2N3O3/c1-15-17(14-29)3-6-23-20(15)12-18(30(23)2)13-21-22(27)5-4-19(25(21)28)26(34)31-9-7-16(8-10-31)11-24(32)33/h3-6,12,16H,7-11,13H2,1-2H3,(H,32,33)	NVPHGOZFJWJSLC-UHFFFAOYSA-N	292816	US10106501, Example EY	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292816	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292816&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122949	381613102							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558649	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)cc2c(Cl)cc(Cl)cc12	InChI=1S/C21H18Cl4N2O2/c1-26-13(10-15-18(24)8-12(22)9-19(15)26)11-16-17(23)3-2-14(20(16)25)21(28)27-4-6-29-7-5-27/h2-3,8-10H,4-7,11H2,1H3	MUVKBENYCIOXEU-UHFFFAOYSA-N	292817	US10106501, Example EZ	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292817	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292817&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123106	381613103							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558650	Cc1cc(cc2n(C)cc(Cc3c(Cl)ccc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)c12)C(F)(F)F	InChI=1S/C26H25Cl2F3N2O3/c1-14-9-17(26(29,30)31)12-21-23(14)16(13-32(21)2)11-19-20(27)4-3-18(24(19)28)25(36)33-7-5-15(6-8-33)10-22(34)35/h3-4,9,12-13,15H,5-8,10-11H2,1-2H3,(H,34,35)	SFUWMXGVJMCIBN-UHFFFAOYSA-N	292818	US10106501, Example F	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292818	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292818&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123712	381613104							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558651	Cc1cc(cc2n(C)cc(Cc3c(Cl)ccc(C(=O)N4C[C@H]5[C@@H](C4)[C@@H]5C(O)=O)c3Cl)c12)C(F)(F)F |r|	InChI=1S/C25H21Cl2F3N2O3/c1-11-5-13(25(28,29)30)7-19-20(11)12(8-31(19)2)6-15-18(26)4-3-14(22(15)27)23(33)32-9-16-17(10-32)21(16)24(34)35/h3-5,7-8,16-17,21H,6,9-10H2,1-2H3,(H,34,35)	YGLXLBLOPZIOLA-UHFFFAOYSA-N	292819	US10106501, Example F1-1	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292819	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292819&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123370	381613105							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558652	C[C@@H]1CN(CC[C@@H]1C(O)=O)C(=O)c1ccc(Cl)c(Cc2cn(C)c3cc(cc(C)c23)C(F)(F)F)c1Cl |r|	InChI=1S/C26H25Cl2F3N2O3/c1-13-8-16(26(29,30)31)10-21-22(13)15(12-32(21)3)9-19-20(27)5-4-18(23(19)28)24(34)33-7-6-17(25(35)36)14(2)11-33/h4-5,8,10,12,14,17H,6-7,9,11H2,1-3H3,(H,35,36)	AVEZWISTIIOEEB-UHFFFAOYSA-N	292820	US10106501, Example F1-2	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292820	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292820&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123915	381613106							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558653	C[C@H]1CN(CC[C@H]1C(O)=O)C(=O)c1ccc(Cl)c(Cc2cn(C)c3cc(cc(C)c23)C(F)(F)F)c1Cl |r|	InChI=1S/C26H25Cl2F3N2O3/c1-13-8-16(26(29,30)31)10-21-22(13)15(12-32(21)3)9-19-20(27)5-4-18(23(19)28)24(34)33-7-6-17(25(35)36)14(2)11-33/h4-5,8,10,12,14,17H,6-7,9,11H2,1-3H3,(H,35,36)	AVEZWISTIIOEEB-UHFFFAOYSA-N	292821	US10106501, Example F1-3	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292821	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292821&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123923	381613107							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558654	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)cc2c(Cl)cc(Cl)cc12	InChI=1S/C24H22Cl4N2O3/c1-29-15(11-17-20(27)9-14(25)10-21(17)29)12-18-19(26)3-2-16(23(18)28)24(33)30-6-4-13(5-7-30)8-22(31)32/h2-3,9-11,13H,4-8,12H2,1H3,(H,31,32)	UEIHPKUXECDEKQ-UHFFFAOYSA-N	292822	US10106501, Example FA	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292822	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292822&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123541	381613108							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558655	Cc1cc(cc2n(C)c(Cc3c(Cl)ncc(C(=O)N4CCC5(CCOC5)CC4)c3Cl)cc12)C#N	InChI=1S/C26H26Cl2N4O2/c1-16-9-17(13-29)10-22-19(16)11-18(31(22)2)12-20-23(27)21(14-30-24(20)28)25(33)32-6-3-26(4-7-32)5-8-34-15-26/h9-11,14H,3-8,12,15H2,1-2H3	SEFADELPCXLLBV-UHFFFAOYSA-N	292823	US10106501, Example FB	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292823	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292823&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123147	381613109							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558656	Cc1cc(cc2n(C)c(Cc3c(Cl)ncc(C(=O)N4CCC(CC4)C4COC4)c3Cl)cc12)C#N	InChI=1S/C26H26Cl2N4O2/c1-15-7-16(11-29)8-23-20(15)9-19(31(23)2)10-21-24(27)22(12-30-25(21)28)26(33)32-5-3-17(4-6-32)18-13-34-14-18/h7-9,12,17-18H,3-6,10,13-14H2,1-2H3	ASLIORWYTAGLPH-UHFFFAOYSA-N	292824	US10106501, Example FC	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292824	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292824&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122840	381613110							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558657	COc1cc(C)c2cc(Cc3c(Cl)ccc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)n(C)c2c1	InChI=1S/C26H28Cl2N2O4/c1-15-10-18(34-3)14-23-20(15)12-17(29(23)2)13-21-22(27)5-4-19(25(21)28)26(33)30-8-6-16(7-9-30)11-24(31)32/h4-5,10,12,14,16H,6-9,11,13H2,1-3H3,(H,31,32)	SUJMEXATQSIBEY-UHFFFAOYSA-N	292825	US10106501, Example FD	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292825	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292825&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122955	381613111							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558658	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)cc2c(F)cc(cc12)C(F)(F)F	InChI=1S/C25H22Cl2F4N2O3/c1-32-15(12-18-20(28)9-14(10-21(18)32)25(29,30)31)11-17-19(26)3-2-16(23(17)27)24(36)33-6-4-13(5-7-33)8-22(34)35/h2-3,9-10,12-13H,4-8,11H2,1H3,(H,34,35)	KLGFFKGIDCNTCD-UHFFFAOYSA-N	292826	US10106501, Example FE	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292826	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292826&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123367	381613112							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558659	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCC(CC3)C(O)=O)c2Cl)cc2c(F)cc(cc12)C(F)(F)F	InChI=1S/C24H20Cl2F4N2O3/c1-31-14(11-17-19(27)8-13(9-20(17)31)24(28,29)30)10-16-18(25)3-2-15(21(16)26)22(33)32-6-4-12(5-7-32)23(34)35/h2-3,8-9,11-12H,4-7,10H2,1H3,(H,34,35)	MCNZCRAYJBCMKR-UHFFFAOYSA-N	292827	US10106501, Example FE-2	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292827	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292827&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124129210	381613113							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558660	C[C@@H]1CN(CC[C@@H]1C(O)=O)C(=O)c1ccc(Cl)c(Cc2cc3c(F)cc(cc3n2C)C(F)(F)F)c1Cl |r|	InChI=1S/C25H22Cl2F4N2O3/c1-12-11-33(6-5-15(12)24(35)36)23(34)16-3-4-19(26)17(22(16)27)9-14-10-18-20(28)7-13(25(29,30)31)8-21(18)32(14)2/h3-4,7-8,10,12,15H,5-6,9,11H2,1-2H3,(H,35,36)	WXGXZJWPGFSTFS-UHFFFAOYSA-N	292828	US10106501, Example FE-3	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292828	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292828&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124129212	381613114							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558661	C[C@H]1CN(CC[C@H]1C(O)=O)C(=O)c1ccc(Cl)c(Cc2cc3c(F)cc(cc3n2C)C(F)(F)F)c1Cl |r|	InChI=1S/C25H22Cl2F4N2O3/c1-12-11-33(6-5-15(12)24(35)36)23(34)16-3-4-19(26)17(22(16)27)9-14-10-18-20(28)7-13(25(29,30)31)8-21(18)32(14)2/h3-4,7-8,10,12,15H,5-6,9,11H2,1-2H3,(H,35,36)	WXGXZJWPGFSTFS-UHFFFAOYSA-N	292829	US10106501, Example FE-4	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292829	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292829&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124129213	381613115							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558662	Cc1cc(OC(F)F)cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)cc12	InChI=1S/C26H26Cl2F2N2O4/c1-14-9-17(36-26(29)30)13-22-19(14)11-16(31(22)2)12-20-21(27)4-3-18(24(20)28)25(35)32-7-5-15(6-8-32)10-23(33)34/h3-4,9,11,13,15,26H,5-8,10,12H2,1-2H3,(H,33,34)	LACKLUVZEJUYFO-UHFFFAOYSA-N	292830	US10106501, Example FF	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292830	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292830&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123164	381613116							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558663	CC1CN(CCC1C(O)=O)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(OC(F)F)cc3n2C)c1Cl	InChI=1S/C26H26Cl2F2N2O4/c1-13-8-16(36-26(29)30)11-22-19(13)9-15(31(22)3)10-20-21(27)5-4-18(23(20)28)24(33)32-7-6-17(25(34)35)14(2)12-32/h4-5,8-9,11,14,17,26H,6-7,10,12H2,1-3H3,(H,34,35)	VTODGFSQFNMEJE-UHFFFAOYSA-N	292831	US10106501, Example FF-1	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292831	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292831&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124129632	381613117							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558664	Cc1cc(OC(F)F)cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC4)C(O)=O)c3Cl)cc12	InChI=1S/C25H24Cl2F2N2O4/c1-13-9-16(35-25(28)29)12-21-18(13)10-15(30(21)2)11-19-20(26)4-3-17(22(19)27)23(32)31-7-5-14(6-8-31)24(33)34/h3-4,9-10,12,14,25H,5-8,11H2,1-2H3,(H,33,34)	VHZCVSBHAMIDJT-UHFFFAOYSA-N	292832	US10106501, Example FF-2	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292832	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292832&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124129633	381613118							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558665	Cc1cc(cc2n(C)c(cc12)C(=O)c1c(Cl)ncc(C(=O)N2CCC(CC(O)=O)CC2)c1Cl)C(F)(F)F	InChI=1S/C25H22Cl2F3N3O4/c1-12-7-14(25(28,29)30)9-17-15(12)10-18(32(17)2)22(36)20-21(26)16(11-31-23(20)27)24(37)33-5-3-13(4-6-33)8-19(34)35/h7,9-11,13H,3-6,8H2,1-2H3,(H,34,35)	MFPZQDMMWAJJPL-UHFFFAOYSA-N	292833	US10106501, Example FG	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292833	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292833&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123494	381613119							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558666	Cc1cc(cc2n(C)c(Cc3c(Cl)cnc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)cc12)C(F)(F)F	InChI=1S/C25H24Cl2F3N3O3/c1-13-7-15(25(28,29)30)9-20-17(13)10-16(32(20)2)11-18-19(26)12-31-23(22(18)27)24(36)33-5-3-14(4-6-33)8-21(34)35/h7,9-10,12,14H,3-6,8,11H2,1-2H3,(H,34,35)	AQKBJIRLXOMBKI-UHFFFAOYSA-N	292834	US10106501, Example FH	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292834	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292834&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123439	381613120							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558667	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)cc2ccc(OC(F)(F)F)cc12	InChI=1S/C25H23Cl2F3N2O4/c1-31-16(11-15-2-3-17(13-21(15)31)36-25(28,29)30)12-19-20(26)5-4-18(23(19)27)24(35)32-8-6-14(7-9-32)10-22(33)34/h2-5,11,13-14H,6-10,12H2,1H3,(H,33,34)	RHILDZGPZYBDSH-UHFFFAOYSA-N	292835	US10106501, Example FI	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292835	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292835&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123298	381613121							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558668	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCC(CC3)C(O)=O)c2Cl)cc2ccc(OC(F)(F)F)cc12	InChI=1S/C24H21Cl2F3N2O4/c1-30-15(10-14-2-3-16(12-20(14)30)35-24(27,28)29)11-18-19(25)5-4-17(21(18)26)22(32)31-8-6-13(7-9-31)23(33)34/h2-5,10,12-13H,6-9,11H2,1H3,(H,33,34)	HLLPGNUHMAJIEO-UHFFFAOYSA-N	292836	US10106501, Example FI-1	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292836	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292836&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124129634	381613122							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558669	CC1CN(CCC1C(O)=O)C(=O)c1ccc(Cl)c(Cc2cc3ccc(OC(F)(F)F)cc3n2C)c1Cl	InChI=1S/C25H23Cl2F3N2O4/c1-13-12-32(8-7-17(13)24(34)35)23(33)18-5-6-20(26)19(22(18)27)10-15-9-14-3-4-16(36-25(28,29)30)11-21(14)31(15)2/h3-6,9,11,13,17H,7-8,10,12H2,1-2H3,(H,34,35)	RGXQNYDDDJOOHR-UHFFFAOYSA-N	292837	US10106501, Example FI-2::US10106501, Example FI-3	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292837	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292837&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124129239	381613123							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558670	CC1CN(CCC1C(O)=O)C(=O)c1ccc(Cl)c(Cc2cc3ccc(OC(F)(F)F)cc3n2C)c1Cl	InChI=1S/C25H23Cl2F3N2O4/c1-13-12-32(8-7-17(13)24(34)35)23(33)18-5-6-20(26)19(22(18)27)10-15-9-14-3-4-16(36-25(28,29)30)11-21(14)31(15)2/h3-6,9,11,13,17H,7-8,10,12H2,1-2H3,(H,34,35)	RGXQNYDDDJOOHR-UHFFFAOYSA-N	292837	US10106501, Example FI-2::US10106501, Example FI-3	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292837	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292837&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124129239	381613123							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558671	Cc1nc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCN(CC4)C4COC4)c3Cl)cc12)C(F)(F)F	InChI=1S/C25H25Cl2F3N4O2/c1-14-18-9-15(32(2)21(18)11-22(31-14)25(28,29)30)10-19-20(26)4-3-17(23(19)27)24(35)34-7-5-33(6-8-34)16-12-36-13-16/h3-4,9,11,16H,5-8,10,12-13H2,1-2H3	ZNLRHSAYWCZMLB-UHFFFAOYSA-N	292839	US10106501, Example FJ	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292839	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292839&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122983	381613124							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558672	CC(=O)Nc1cc(C)c2cc(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)n(C)c2c1	InChI=1S/C24H25Cl2N3O3/c1-14-10-16(27-15(2)30)11-22-19(14)12-17(28(22)3)13-20-21(25)5-4-18(23(20)26)24(31)29-6-8-32-9-7-29/h4-5,10-12H,6-9,13H2,1-3H3,(H,27,30)	FZFFKUULKPTJFT-UHFFFAOYSA-N	292840	US10106501, Example FK	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292840	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292840&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123297	381613125							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558673	Cn1c(Cc2c(Cl)c(ccc2C2CC2)C(=O)N2CCC(CC(O)=O)CC2)cc2ccc(OC(F)(F)F)cc12	InChI=1S/C28H28ClF3N2O4/c1-33-19(13-18-4-5-20(15-24(18)33)38-28(30,31)32)14-23-21(17-2-3-17)6-7-22(26(23)29)27(37)34-10-8-16(9-11-34)12-25(35)36/h4-7,13,15-17H,2-3,8-12,14H2,1H3,(H,35,36)	VOZBLWCMNUOPLQ-UHFFFAOYSA-N	292841	US10106501, Example FL	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292841	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292841&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123424	381613126							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558674	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)cc2c(F)cc(cc12)C1CC1	InChI=1S/C27H27Cl2FN2O3/c1-31-18(14-21-23(30)11-17(12-24(21)31)16-2-3-16)13-20-22(28)5-4-19(26(20)29)27(35)32-8-6-15(7-9-32)10-25(33)34/h4-5,11-12,14-16H,2-3,6-10,13H2,1H3,(H,33,34)	QXDZXBJAYLGDMJ-UHFFFAOYSA-N	292842	US10106501, Example FM	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292842	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292842&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123236	381613127							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558675	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCC(CC3)C(O)=O)c2Cl)cc2c(F)cc(cc12)C1CC1	InChI=1S/C26H25Cl2FN2O3/c1-30-17(13-20-22(29)10-16(11-23(20)30)14-2-3-14)12-19-21(27)5-4-18(24(19)28)25(32)31-8-6-15(7-9-31)26(33)34/h4-5,10-11,13-15H,2-3,6-9,12H2,1H3,(H,33,34)	TWTRRYLNKZCMCT-UHFFFAOYSA-N	292843	US10106501, Example FN	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292843	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292843&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123146	381613128							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558676	CN(C)C(=O)c1cc(C)c2cc(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)n(C)c2c1	InChI=1S/C25H27Cl2N3O3/c1-15-11-16(24(31)28(2)3)12-22-19(15)13-17(29(22)4)14-20-21(26)6-5-18(23(20)27)25(32)30-7-9-33-10-8-30/h5-6,11-13H,7-10,14H2,1-4H3	WTLUFONYBICOEE-UHFFFAOYSA-N	292844	US10106501, Example FO	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292844	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292844&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123761	381613129							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558677	CNC(=O)c1cc(C)c2cc(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)n(C)c2c1	InChI=1S/C24H25Cl2N3O3/c1-14-10-15(23(30)27-2)11-21-18(14)12-16(28(21)3)13-19-20(25)5-4-17(22(19)26)24(31)29-6-8-32-9-7-29/h4-5,10-12H,6-9,13H2,1-3H3,(H,27,30)	VLIXTVPVWYUJCY-UHFFFAOYSA-N	292845	US10106501, Example FP	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292845	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292845&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123563	381613130							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558678	Cc1cc(cc2n(C)cc(Cc3c(Cl)ccc(C(=O)N4CCC(CC4)C(O)=O)c3Cl)c12)C(F)(F)F	InChI=1S/C25H23Cl2F3N2O3/c1-13-9-16(25(28,29)30)11-20-21(13)15(12-31(20)2)10-18-19(26)4-3-17(22(18)27)23(33)32-7-5-14(6-8-32)24(34)35/h3-4,9,11-12,14H,5-8,10H2,1-2H3,(H,34,35)	MGIUBYDSGZRDSY-UHFFFAOYSA-N	292846	US10106501, Example FQ	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292846	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292846&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122907	381613131							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558679	Cc1cn(Cc2c(Cl)cnc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)c2c(C)cc(cc12)C(F)(F)F	InChI=1S/C25H24Cl2F3N3O3/c1-13-7-16(25(28,29)30)9-17-14(2)11-33(23(13)17)12-18-19(26)10-31-22(21(18)27)24(36)32-5-3-15(4-6-32)8-20(34)35/h7,9-11,15H,3-6,8,12H2,1-2H3,(H,34,35)	ZZRVMXKMGKZHDI-UHFFFAOYSA-N	292847	US10106501, Example FR	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292847	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292847&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122893	381613132							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558680	Cc1cc(nc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC4)C(O)=O)c3Cl)cc12)C(F)(F)F	InChI=1S/C24H22Cl2F3N3O3/c1-12-9-19(24(27,28)29)30-21-16(12)10-14(31(21)2)11-17-18(25)4-3-15(20(17)26)22(33)32-7-5-13(6-8-32)23(34)35/h3-4,9-10,13H,5-8,11H2,1-2H3,(H,34,35)	DMWMQDLGWODIJV-UHFFFAOYSA-N	292848	US10106501, Example FS	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292848	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292848&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123357	381613133							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558681	COCCC1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(nc3n2C)C(F)(F)F)c1Cl	InChI=1S/C26H28Cl2F3N3O2/c1-15-12-22(26(29,30)31)32-24-19(15)13-17(33(24)2)14-20-21(27)5-4-18(23(20)28)25(35)34-9-6-16(7-10-34)8-11-36-3/h4-5,12-13,16H,6-11,14H2,1-3H3	NJEBCAKTQLXBCO-UHFFFAOYSA-N	292849	US10106501, Example FT	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292849	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292849&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123755	381613134							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558682	Cc1cc(nc2n(C)c(cc12)C(=O)c1c(Cl)ccc(C(=O)N2CCC(CC(O)=O)CC2)c1Cl)C(F)(F)F	InChI=1S/C25H22Cl2F3N3O4/c1-12-9-18(25(28,29)30)31-23-15(12)11-17(32(23)2)22(36)20-16(26)4-3-14(21(20)27)24(37)33-7-5-13(6-8-33)10-19(34)35/h3-4,9,11,13H,5-8,10H2,1-2H3,(H,34,35)	HQKYBKZRKJLBHZ-UHFFFAOYSA-N	292850	US10106501, Example FU	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292850	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292850&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123271	381613135							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558683	Cc1cc(nc2n(C)c(cc12)C(=O)c1c(Cl)ccc(C(=O)N2CCC(CC2)C#N)c1Cl)C(F)(F)F	InChI=1S/C24H19Cl2F3N4O2/c1-12-9-18(24(27,28)29)31-22-15(12)10-17(32(22)2)21(34)19-16(25)4-3-14(20(19)26)23(35)33-7-5-13(11-30)6-8-33/h3-4,9-10,13H,5-8H2,1-2H3	SIMRAMNMSOIQHQ-UHFFFAOYSA-N	292851	US10106501, Example FV	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292851	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292851&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123401	381613136							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558684	C[C@H]1CN(CC[C@@H]1O)C(=O)c1ccc(Cl)c(C(=O)c2cc3c(C)cc(nc3n2C)C(F)(F)F)c1Cl |r|	InChI=1S/C24H22Cl2F3N3O3/c1-11-8-18(24(27,28)29)30-22-14(11)9-16(31(22)3)21(34)19-15(25)5-4-13(20(19)26)23(35)32-7-6-17(33)12(2)10-32/h4-5,8-9,12,17,33H,6-7,10H2,1-3H3	MNHROSSQGZBREQ-UHFFFAOYSA-N	292852	US10106501, Example FW	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292852	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292852&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123795	381613137							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558685	C[C@H]1CN(CC[C@H]1C(O)=O)C(=O)c1ccc(Cl)c(C(=O)c2cc3c(C)cc(nc3n2C)C(F)(F)F)c1Cl |r|	InChI=1S/C25H22Cl2F3N3O4/c1-11-8-18(25(28,29)30)31-22-15(11)9-17(32(22)3)21(34)19-16(26)5-4-14(20(19)27)23(35)33-7-6-13(24(36)37)12(2)10-33/h4-5,8-9,12-13H,6-7,10H2,1-3H3,(H,36,37)	OBYGZJPIKCLJFK-UHFFFAOYSA-N	292853	US10106501, Example FX	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292853	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292853&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123416	381613138							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558686	COCCC1CCN(CC1)C(=O)c1ccc(Cl)c(C(=O)c2cc3c(C)cc(nc3n2C)C(F)(F)F)c1Cl	InChI=1S/C26H26Cl2F3N3O3/c1-14-12-20(26(29,30)31)32-24-17(14)13-19(33(24)2)23(35)21-18(27)5-4-16(22(21)28)25(36)34-9-6-15(7-10-34)8-11-37-3/h4-5,12-13,15H,6-11H2,1-3H3	PEOOGPKLIIUWDL-UHFFFAOYSA-N	292854	US10106501, Example FY	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292854	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292854&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123916	381613139							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558687	Cc1cc(nc2n(C)c(cc12)C(=O)c1c(Cl)ccc(C(=O)N2CCC(O)CC2)c1Cl)C(F)(F)F	InChI=1S/C23H20Cl2F3N3O3/c1-11-9-17(23(26,27)28)29-21-14(11)10-16(30(21)2)20(33)18-15(24)4-3-13(19(18)25)22(34)31-7-5-12(32)6-8-31/h3-4,9-10,12,32H,5-8H2,1-2H3	LBYSKYZGSJZYCY-UHFFFAOYSA-N	292855	US10106501, Example FZ	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292855	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292855&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123845	381613140							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558688	Cc1ccc(C(=O)N2CCOCC2)c(C)c1Cc1cc2c(C)cc(cc2n1C)C(F)(F)F	InChI=1S/C25H27F3N2O2/c1-15-5-6-20(24(31)30-7-9-32-10-8-30)17(3)21(15)13-19-14-22-16(2)11-18(25(26,27)28)12-23(22)29(19)4/h5-6,11-12,14H,7-10,13H2,1-4H3	IOJVIJSTROAGAR-UHFFFAOYSA-N	292856	US10106501, Example G	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292856	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292856&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123144	381613141							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558689	C[C@H]1CN(CC[C@H]1CC(O)=O)C(=O)c1ccc(Cl)c(C(=O)c2cc3c(C)cc(nc3n2C)C(F)(F)F)c1Cl |r|	InChI=1S/C26H24Cl2F3N3O4/c1-12-8-19(26(29,30)31)32-24-16(12)10-18(33(24)3)23(37)21-17(27)5-4-15(22(21)28)25(38)34-7-6-14(9-20(35)36)13(2)11-34/h4-5,8,10,13-14H,6-7,9,11H2,1-3H3,(H,35,36)	MYBRBMDHVWNSJC-UHFFFAOYSA-N	292857	US10106501, Example GA	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292857	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292857&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123620	381613142							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558690	Cc1cc(nc2n(C)c(cc12)C(=O)c1c(Cl)ccc(C(=O)N2CCC(CC2)S(C)(=O)=O)c1Cl)C(F)(F)F	InChI=1S/C24H22Cl2F3N3O4S/c1-12-10-18(24(27,28)29)30-22-15(12)11-17(31(22)2)21(33)19-16(25)5-4-14(20(19)26)23(34)32-8-6-13(7-9-32)37(3,35)36/h4-5,10-11,13H,6-9H2,1-3H3	VCRQIFDICPPVKF-UHFFFAOYSA-N	292858	US10106501, Example GB	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292858	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292858&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123824	381613143							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558691	C[C@H]1CN(CC[C@H]1CC(O)=O)C(=O)c1cnc(Cl)c(Cc2cc3c(C)cc(nc3n2C)C(F)(F)F)c1Cl |r|	InChI=1S/C25H25Cl2F3N4O3/c1-12-6-19(25(28,29)30)32-23-16(12)8-15(33(23)3)9-17-21(26)18(10-31-22(17)27)24(37)34-5-4-14(7-20(35)36)13(2)11-34/h6,8,10,13-14H,4-5,7,9,11H2,1-3H3,(H,35,36)	JHLFCHSRGKFNML-UHFFFAOYSA-N	292859	US10106501, Example GC	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292859	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292859&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123650	381613144							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558692	Cc1cc(nc2n(C)c(Cc3c(Cl)ncc(C(=O)N4CCN(CC4)S(C)(=O)=O)c3Cl)cc12)C(F)(F)F	InChI=1S/C22H22Cl2F3N5O3S/c1-12-8-17(22(25,26)27)29-20-14(12)9-13(30(20)2)10-15-18(23)16(11-28-19(15)24)21(33)31-4-6-32(7-5-31)36(3,34)35/h8-9,11H,4-7,10H2,1-3H3	NMOXBZUZTWMYIZ-UHFFFAOYSA-N	292860	US10106501, Example GE	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292860	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292860&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123153	381613145							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558693	Cc1cc(nc2n(C)c(Cc3c(Cl)ncc(C(=O)N4CCOCC4)c3Cl)cc12)C(F)(F)F	InChI=1S/C21H19Cl2F3N4O2/c1-11-7-16(21(24,25)26)28-19-13(11)8-12(29(19)2)9-14-17(22)15(10-27-18(14)23)20(31)30-3-5-32-6-4-30/h7-8,10H,3-6,9H2,1-2H3	QEGUFLZLFOLHGE-UHFFFAOYSA-N	292861	US10106501, Example GF	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292861	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292861&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123504	381613146							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558694	Cc1cc(nc2n(C)c(Cc3c(Cl)ncc(C(=O)N4CCC(CC4)S(C)(=O)=O)c3Cl)cc12)C(F)(F)F	InChI=1S/C23H23Cl2F3N4O3S/c1-12-8-18(23(26,27)28)30-21-15(12)9-13(31(21)2)10-16-19(24)17(11-29-20(16)25)22(33)32-6-4-14(5-7-32)36(3,34)35/h8-9,11,14H,4-7,10H2,1-3H3	MPSFXJNANLAXFK-UHFFFAOYSA-N	292862	US10106501, Example GG	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292862	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292862&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123240	381613147							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558695	Cn1c(cc2ccc(OC(F)(F)F)cc12)C(=O)c1c(Cl)ccc(C(=O)N2CCC(CC(O)=O)CC2)c1Cl	InChI=1S/C25H21Cl2F3N2O5/c1-31-18-12-15(37-25(28,29)30)3-2-14(18)11-19(31)23(35)21-17(26)5-4-16(22(21)27)24(36)32-8-6-13(7-9-32)10-20(33)34/h2-5,11-13H,6-10H2,1H3,(H,33,34)	JFISMWULRLPYAQ-UHFFFAOYSA-N	292863	US10106501, Example GI	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292863	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292863&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123123	381613148							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558696	Cn1c(Cc2c(Cl)cnc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)cc2ccc(OC(F)(F)F)cc12	InChI=1S/C24H22Cl2F3N3O4/c1-31-15(9-14-2-3-16(11-19(14)31)36-24(27,28)29)10-17-18(25)12-30-22(21(17)26)23(35)32-6-4-13(5-7-32)8-20(33)34/h2-3,9,11-13H,4-8,10H2,1H3,(H,33,34)	WWIKSFMFZFAELS-UHFFFAOYSA-N	292864	US10106501, Example GK	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292864	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292864&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123162	381613149							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558697	Cn1c(Cc2c(Cl)ncc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)cc2c(F)cc(cc12)C1CC1	InChI=1S/C26H26Cl2FN3O3/c1-31-17(11-18-21(29)9-16(10-22(18)31)15-2-3-15)12-19-24(27)20(13-30-25(19)28)26(35)32-6-4-14(5-7-32)8-23(33)34/h9-11,13-15H,2-8,12H2,1H3,(H,33,34)	DXHUJHAGTASXAO-UHFFFAOYSA-N	292865	US10106501, Example GN	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292865	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292865&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123547	381613150							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558698	Cc1ccc(C(=O)N2CCOCC2)c(C)c1C(=O)c1cc2c(C)cc(cc2n1C)C(F)(F)F	InChI=1S/C25H25F3N2O3/c1-14-5-6-18(24(32)30-7-9-33-10-8-30)16(3)22(14)23(31)21-13-19-15(2)11-17(25(26,27)28)12-20(19)29(21)4/h5-6,11-13H,7-10H2,1-4H3	FNNYJRBYDQFIFG-UHFFFAOYSA-N	292866	US10106501, Example G1	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292866	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292866&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123860	381613151							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558699	CN(C)C1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3[nH]2)C(F)(F)F)c1Cl	InChI=1S/C25H26Cl2F3N3O/c1-14-10-15(25(28,29)30)11-22-19(14)12-16(31-22)13-20-21(26)5-4-18(23(20)27)24(34)33-8-6-17(7-9-33)32(2)3/h4-5,10-12,17,31H,6-9,13H2,1-3H3	NHDQEJUGJPGBEB-UHFFFAOYSA-N	292867	US10106501, Example H	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292867	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292867&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123836	381613152							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558700	CN(C)C1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C26H28Cl2F3N3O/c1-15-11-16(26(29,30)31)12-23-20(15)13-18(33(23)4)14-21-22(27)6-5-19(24(21)28)25(35)34-9-7-17(8-10-34)32(2)3/h5-6,11-13,17H,7-10,14H2,1-4H3	LYZLYLHDBZCUIX-UHFFFAOYSA-N	292868	US10106501, Example I	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292868	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292868&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123234	381613153							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558701	Cc1cc(cc2ccn(Cc3c(Cl)ccc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)c12)C(F)(F)F	InChI=1S/C25H23Cl2F3N2O3/c1-14-10-17(25(28,29)30)12-16-6-9-32(23(14)16)13-19-20(26)3-2-18(22(19)27)24(35)31-7-4-15(5-8-31)11-21(33)34/h2-3,6,9-10,12,15H,4-5,7-8,11,13H2,1H3,(H,33,34)	PGISETOBANJZCF-UHFFFAOYSA-N	292869	US10106501, Example DS::US10106501, Example J	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292869	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292869&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122941	381613154							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558702	Cc1ccc(C(=O)N2CCOCC2)c(C)c1C(O)c1cc2c(C)cc(cc2n1C)C(F)(F)F	InChI=1S/C25H27F3N2O3/c1-14-5-6-18(24(32)30-7-9-33-10-8-30)16(3)22(14)23(31)21-13-19-15(2)11-17(25(26,27)28)12-20(19)29(21)4/h5-6,11-13,23,31H,7-10H2,1-4H3	ISXGAWOYEFNKJC-UHFFFAOYSA-N	292870	US10106501, Example K	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292870	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292870&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123157	381613155							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558703	COC(c1cc2c(C)cc(cc2n1C)C(F)(F)F)c1c(C)ccc(C(=O)N2CCOCC2)c1C	InChI=1S/C26H29F3N2O3/c1-15-6-7-19(25(32)31-8-10-34-11-9-31)17(3)23(15)24(33-5)22-14-20-16(2)12-18(26(27,28)29)13-21(20)30(22)4/h6-7,12-14,24H,8-11H2,1-5H3	TYJMVUHXOUMCAW-UHFFFAOYSA-N	292871	US10106501, Example K1	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292871	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292871&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123129	381613156							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558704	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCC(O)CC3)c2Cl)cc2ccc(cc12)C(F)(F)F	InChI=1S/C23H21Cl2F3N2O2/c1-29-15(10-13-2-3-14(11-20(13)29)23(26,27)28)12-18-19(24)5-4-17(21(18)25)22(32)30-8-6-16(31)7-9-30/h2-5,10-11,16,31H,6-9,12H2,1H3	WLDOGNDGQJAZAQ-UHFFFAOYSA-N	292872	US10106501, Example L	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292872	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292872&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123322	381613157							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558705	CN(C)C1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2cc3ccc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C25H26Cl2F3N3O/c1-31(2)17-8-10-33(11-9-17)24(34)19-6-7-21(26)20(23(19)27)14-18-12-15-4-5-16(25(28,29)30)13-22(15)32(18)3/h4-7,12-13,17H,8-11,14H2,1-3H3	QZESUTWSNVLNII-UHFFFAOYSA-N	292873	US10106501, Example L-1	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292873	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292873&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123757	381613158							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558706	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCC(CO)CC3)c2Cl)cc2ccc(cc12)C(F)(F)F	InChI=1S/C24H23Cl2F3N2O2/c1-30-17(10-15-2-3-16(11-21(15)30)24(27,28)29)12-19-20(25)5-4-18(22(19)26)23(33)31-8-6-14(13-32)7-9-31/h2-5,10-11,14,32H,6-9,12-13H2,1H3	NEBBGXSQDAIJES-UHFFFAOYSA-N	292874	US10106501, Example L-2	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292874	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292874&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123577	381613159							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558707	CC(=O)N1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2cc3ccc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C24H22Cl2F3N3O2/c1-14(33)31-7-9-32(10-8-31)23(34)18-5-6-20(25)19(22(18)26)13-17-11-15-3-4-16(24(27,28)29)12-21(15)30(17)2/h3-6,11-12H,7-10,13H2,1-2H3	GAYOMEIWFNMSNQ-UHFFFAOYSA-N	292875	US10106501, Example L-3	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292875	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292875&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122986	381613160							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558708	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCCC(O)C3)c2Cl)cc2ccc(cc12)C(F)(F)F	InChI=1S/C23H21Cl2F3N2O2/c1-29-15(9-13-4-5-14(10-20(13)29)23(26,27)28)11-18-19(24)7-6-17(21(18)25)22(32)30-8-2-3-16(31)12-30/h4-7,9-10,16,31H,2-3,8,11-12H2,1H3	JMBBPHCFIXAYFB-UHFFFAOYSA-N	292876	US10106501, Example L-4	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292876	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292876&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123476	381613161							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558709	Cn1c(Cc2c(Cl)ccc(C(=O)N3CC[C@@H](F)[C@H](O)C3)c2Cl)cc2ccc(cc12)C(F)(F)F |r|	InChI=1S/C23H20Cl2F4N2O2/c1-30-14(8-12-2-3-13(9-19(12)30)23(27,28)29)10-16-17(24)5-4-15(21(16)25)22(33)31-7-6-18(26)20(32)11-31/h2-5,8-9,18,20,32H,6-7,10-11H2,1H3	GVKNNVSEOWKOKY-UHFFFAOYSA-N	292877	US10106501, Example L-5	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292877	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292877&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123173	381613162							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558710	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCC(CC3)C(O)=O)c2Cl)cc2ccc(cc12)C(F)(F)F	InChI=1S/C24H21Cl2F3N2O3/c1-30-16(10-14-2-3-15(11-20(14)30)24(27,28)29)12-18-19(25)5-4-17(21(18)26)22(32)31-8-6-13(7-9-31)23(33)34/h2-5,10-11,13H,6-9,12H2,1H3,(H,33,34)	QZGCUISVDJUNLI-UHFFFAOYSA-N	292878	US10106501, Example M	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292878	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292878&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123583	381613163							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558711	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCC(C(O)C3)C(O)=O)c2Cl)cc2ccc(cc12)C(F)(F)F	InChI=1S/C24H21Cl2F3N2O4/c1-30-14(8-12-2-3-13(9-19(12)30)24(27,28)29)10-17-18(25)5-4-16(21(17)26)22(33)31-7-6-15(23(34)35)20(32)11-31/h2-5,8-9,15,20,32H,6-7,10-11H2,1H3,(H,34,35)	INSNNSYIZXCEPS-UHFFFAOYSA-N	292879	US10106501, Example N	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292879	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292879&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123871	381613164							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558712	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCN(CC3)C3CC(C3)C(O)=O)c2Cl)cc2ccc(cc12)C(F)(F)F |(-4.54,3.16,;-3.45,2.07,;-3.61,.54,;-4.94,-.23,;-4.94,-1.77,;-6.28,-2.54,;-7.61,-1.77,;-6.28,-4.08,;-4.94,-4.85,;-3.61,-4.08,;-2.28,-4.85,;-2.28,-6.39,;-.94,-4.08,;.39,-4.85,;1.72,-4.08,;1.72,-2.54,;.39,-1.77,;-.94,-2.54,;3.06,-1.77,;4.55,-2.17,;4.94,-.68,;3.46,-.28,;6.28,.09,;7.61,-.68,;6.28,1.63,;-3.61,-2.54,;-2.28,-1.77,;-2.2,-.09,;-1.17,1.06,;.37,1.06,;1.14,2.39,;.37,3.72,;-1.17,3.72,;-1.94,2.39,;1.14,5.06,;1.91,6.39,;2.68,5.06,;.37,6.39,)|	InChI=1S/C27H26Cl2F3N3O3/c1-33-18(10-15-2-3-17(13-23(15)33)27(30,31)32)14-21-22(28)5-4-20(24(21)29)25(36)35-8-6-34(7-9-35)19-11-16(12-19)26(37)38/h2-5,10,13,16,19H,6-9,11-12,14H2,1H3,(H,37,38)	WOVVDILGIQXWFZ-UHFFFAOYSA-N	292880	US10106501, Example O	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292880	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292880&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123307	381613165							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558713	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)cc2cc(ccc12)C(F)(F)F	InChI=1S/C22H19Cl2F3N2O2/c1-28-15(11-13-10-14(22(25,26)27)2-5-19(13)28)12-17-18(23)4-3-16(20(17)24)21(30)29-6-8-31-9-7-29/h2-5,10-11H,6-9,12H2,1H3	PZNSVUAFPRSOAD-UHFFFAOYSA-N	292881	US10106501, Example P	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292881	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292881&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123088	381613166							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558714	CN1C(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)Cc2c1cc(cc2C)C(F)(F)F	InChI=1S/C23H23Cl2F3N2O2/c1-13-9-14(23(26,27)28)10-20-17(13)11-15(29(20)2)12-18-19(24)4-3-16(21(18)25)22(31)30-5-7-32-8-6-30/h3-4,9-10,15H,5-8,11-12H2,1-2H3	XRSWLDPJVQOQAB-UHFFFAOYSA-N	292882	US10106501, Example Q	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292882	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292882&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123466	381613167							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558715	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)cc2c(Cl)cc(cc12)C#N	InChI=1S/C25H22Cl3N3O3/c1-30-16(11-18-21(27)8-15(13-29)9-22(18)30)12-19-20(26)3-2-17(24(19)28)25(34)31-6-4-14(5-7-31)10-23(32)33/h2-3,8-9,11,14H,4-7,10,12H2,1H3,(H,32,33)	CMFWAERHCPREOM-UHFFFAOYSA-N	292883	US10106501, Example DR::US10106501, Example R	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292883	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292883&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123405	381613168							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558716	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCN(CC4)C4CC(C4)C(O)=O)c3Cl)cc12)C(F)(F)F |(1.14,-.28,;.37,1.06,;1.14,2.39,;.37,3.72,;-1.17,3.72,;-1.94,2.39,;-3.45,2.07,;-4.54,3.16,;-3.61,.54,;-4.94,-.23,;-4.94,-1.77,;-6.28,-2.54,;-7.61,-1.77,;-6.28,-4.08,;-4.94,-4.85,;-3.61,-4.08,;-2.28,-4.85,;-2.28,-6.39,;-.94,-4.08,;.39,-4.85,;1.72,-4.08,;1.72,-2.54,;.39,-1.77,;-.94,-2.54,;3.06,-1.77,;4.55,-2.17,;4.94,-.68,;3.46,-.28,;6.28,.09,;7.61,-.68,;6.28,1.63,;-3.61,-2.54,;-2.28,-1.77,;-2.2,-.09,;-1.17,1.06,;1.14,5.06,;1.91,6.39,;2.47,4.29,;-.2,5.83,)|	InChI=1S/C28H28Cl2F3N3O3/c1-15-9-17(28(31,32)33)12-24-21(15)13-18(34(24)2)14-22-23(29)4-3-20(25(22)30)26(37)36-7-5-35(6-8-36)19-10-16(11-19)27(38)39/h3-4,9,12-13,16,19H,5-8,10-11,14H2,1-2H3,(H,38,39)	HYNKNSXEAHAGBN-UHFFFAOYSA-N	292884	US10106501, Example S	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292884	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292884&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123925	381613169							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558717	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCN(CC4)C(C)(C)C(O)=O)c3Cl)cc12)C(F)(F)F	InChI=1S/C27H28Cl2F3N3O3/c1-15-11-16(27(30,31)32)12-22-19(15)13-17(33(22)4)14-20-21(28)6-5-18(23(20)29)24(36)34-7-9-35(10-8-34)26(2,3)25(37)38/h5-6,11-13H,7-10,14H2,1-4H3,(H,37,38)	LSLYUFVRWCYVGH-UHFFFAOYSA-N	292885	US10106501, Example T	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292885	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292885&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123631	381613170							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558718	CC(N1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl)C(O)=O	InChI=1S/C26H26Cl2F3N3O3/c1-14-10-16(26(29,30)31)11-22-19(14)12-17(32(22)3)13-20-21(27)5-4-18(23(20)28)24(35)34-8-6-33(7-9-34)15(2)25(36)37/h4-5,10-12,15H,6-9,13H2,1-3H3,(H,36,37)	JCFKKUGXZJJYJE-UHFFFAOYSA-N	292886	US10106501, Example U	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292886	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292886&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123059	381613171							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558719	Cc1cc2cc(Cc3c(Cl)ccc(C(=O)N4CCC(CC4)C(O)=O)c3Cl)n(C)c2cc1C(F)(F)F	InChI=1S/C25H23Cl2F3N2O3/c1-13-9-15-10-16(31(2)21(15)12-19(13)25(28,29)30)11-18-20(26)4-3-17(22(18)27)23(33)32-7-5-14(6-8-32)24(34)35/h3-4,9-10,12,14H,5-8,11H2,1-2H3,(H,34,35)	KOQAZOFAOWDWGM-UHFFFAOYSA-N	292887	US10106501, Example V	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292887	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292887&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123731	381613172							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558720	COc1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C19H16Cl2F3NO/c1-10-6-11(19(22,23)24)7-16-13(10)8-12(25(16)2)9-14-15(20)4-5-17(26-3)18(14)21/h4-8H,9H2,1-3H3	TUKWZYPATDWWHS-UHFFFAOYSA-N	292888	US10106501, Example W	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292888	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292888&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123063	381613173							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558721	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(O)c3Cl)cc12)C(F)(F)F	InChI=1S/C18H14Cl2F3NO/c1-9-5-10(18(21,22)23)6-15-12(9)7-11(24(15)2)8-13-14(19)3-4-16(25)17(13)20/h3-7,25H,8H2,1-2H3	LBHAUZRXQCMKBP-UHFFFAOYSA-N	292889	US10106501, Example X	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292889	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292889&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123762	381613174							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558722	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(OCC(O)=O)c3Cl)cc12)C(F)(F)F	InChI=1S/C20H16Cl2F3NO3/c1-10-5-11(20(23,24)25)6-16-13(10)7-12(26(16)2)8-14-15(21)3-4-17(19(14)22)29-9-18(27)28/h3-7H,8-9H2,1-2H3,(H,27,28)	KSEQDNPKKLRWKF-UHFFFAOYSA-N	292890	US10106501, Example Y	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292890	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292890&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123372	381613175							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558723	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(OCCC(O)=O)c3Cl)cc12)C(F)(F)F	InChI=1S/C21H18Cl2F3NO3/c1-11-7-12(21(24,25)26)8-17-14(11)9-13(27(17)2)10-15-16(22)3-4-18(20(15)23)30-6-5-19(28)29/h3-4,7-9H,5-6,10H2,1-2H3,(H,28,29)	QIJLKJFNSFBXFS-UHFFFAOYSA-N	292891	US10106501, Example Y1	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292891	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292891&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123701	381613176							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558724	COc1ncc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C18H15Cl2F3N2O/c1-9-4-10(18(21,22)23)5-15-12(9)6-11(25(15)2)7-13-14(19)8-24-17(26-3)16(13)20/h4-6,8H,7H2,1-3H3	CRCVVHASIDFEQC-UHFFFAOYSA-N	292892	US10106501, Example Z	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292892	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292892&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123485	381613177							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558725	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCN(CC4)C4COC4)c3Cl)cc12)C#N	InChI=1S/C26H26Cl2N4O2/c1-16-9-17(13-29)10-24-21(16)11-18(30(24)2)12-22-23(27)4-3-20(25(22)28)26(33)32-7-5-31(6-8-32)19-14-34-15-19/h3-4,9-11,19H,5-8,12,14-15H2,1-2H3	ZTHHWVAQJFDGJY-UHFFFAOYSA-N	292893	US10106501, Example AA	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292893	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292893&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123388	381613178							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558726	CC(O)C1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C#N)c1Cl	InChI=1S/C26H27Cl2N3O2/c1-15-10-17(14-29)11-24-21(15)12-19(30(24)3)13-22-23(27)5-4-20(25(22)28)26(33)31-8-6-18(7-9-31)16(2)32/h4-5,10-12,16,18,32H,6-9,13H2,1-3H3	SQZSPIJCLSAQFF-UHFFFAOYSA-N	292894	US10106501, Example AA-1	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292894	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292894&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123001	381613179							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558727	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC4)C(C)(C)O)c3Cl)cc12)C#N	InChI=1S/C27H29Cl2N3O2/c1-16-11-17(15-30)12-24-21(16)13-19(31(24)4)14-22-23(28)6-5-20(25(22)29)26(33)32-9-7-18(8-10-32)27(2,3)34/h5-6,11-13,18,34H,7-10,14H2,1-4H3	ZWZQCSDGLNNAMU-UHFFFAOYSA-N	292895	US10106501, Example AA-2	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292895	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292895&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123484	381613180							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558728	COC1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C#N)c1Cl	InChI=1S/C25H25Cl2N3O2/c1-15-10-16(14-28)11-23-20(15)12-17(29(23)2)13-21-22(26)5-4-19(24(21)27)25(31)30-8-6-18(32-3)7-9-30/h4-5,10-12,18H,6-9,13H2,1-3H3	ITTWGIADNNXLGM-UHFFFAOYSA-N	292896	US10106501, Example AA-3	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292896	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292896&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123717	381613181							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558729	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(O)CC4)c3Cl)cc12)C#N	InChI=1S/C24H23Cl2N3O2/c1-14-9-15(13-27)10-22-19(14)11-16(28(22)2)12-20-21(25)4-3-18(23(20)26)24(31)29-7-5-17(30)6-8-29/h3-4,9-11,17,30H,5-8,12H2,1-2H3	GIDRUOUNAIXTPO-UHFFFAOYSA-N	292897	US10106501, Example AA-4	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292897	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292897&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123833	381613182							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558730	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCCC(O)C4)c3Cl)cc12)C#N	InChI=1S/C24H23Cl2N3O2/c1-14-8-15(12-27)9-22-19(14)10-16(28(22)2)11-20-21(25)6-5-18(23(20)26)24(31)29-7-3-4-17(30)13-29/h5-6,8-10,17,30H,3-4,7,11,13H2,1-2H3	MVIRJSPCLSXXLM-UHFFFAOYSA-N	292898	US10106501, Example AA-5	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292898	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292898&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123050	381613183							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558731	CN(C)C1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C#N)c1Cl	InChI=1S/C26H28Cl2N4O/c1-16-11-17(15-29)12-24-21(16)13-19(31(24)4)14-22-23(27)6-5-20(25(22)28)26(33)32-9-7-18(8-10-32)30(2)3/h5-6,11-13,18H,7-10,14H2,1-4H3	FMJFRTUBUSZHNN-UHFFFAOYSA-N	293019	US10106501, Example AA-6	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293019	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293019&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123448	381613304							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558732	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CO)CC4)c3Cl)cc12)C#N	InChI=1S/C25H25Cl2N3O2/c1-15-9-17(13-28)10-23-20(15)11-18(29(23)2)12-21-22(26)4-3-19(24(21)27)25(32)30-7-5-16(14-31)6-8-30/h3-4,9-11,16,31H,5-8,12,14H2,1-2H3	LOOIWKXYYQHPGQ-UHFFFAOYSA-N	293020	US10106501, Example AA-7	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293020	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293020&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123369	381613305							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558733	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC4)C(C)(C)CO)c3Cl)cc12)C#N	InChI=1S/C28H31Cl2N3O2/c1-17-11-18(15-31)12-25-22(17)13-20(32(25)4)14-23-24(29)6-5-21(26(23)30)27(35)33-9-7-19(8-10-33)28(2,3)16-34/h5-6,11-13,19,34H,7-10,14,16H2,1-4H3	SXALKUXESKEORZ-UHFFFAOYSA-N	293021	US10106501, Example AA-8	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293021	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293021&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123396	381613306							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558734	CN1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C#N)c1Cl	InChI=1S/C24H24Cl2N4O/c1-15-10-16(14-27)11-22-19(15)12-17(29(22)3)13-20-21(25)5-4-18(23(20)26)24(31)30-8-6-28(2)7-9-30/h4-5,10-12H,6-9,13H2,1-3H3	LLNUWYOKDDBBPP-UHFFFAOYSA-N	293022	US10106501, Example AA-9	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293022	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293022&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123431	381613307							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558735	CC1CN(CCN1C)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C#N)c1Cl	InChI=1S/C25H26Cl2N4O/c1-15-9-17(13-28)10-23-20(15)11-18(30(23)4)12-21-22(26)6-5-19(24(21)27)25(32)31-8-7-29(3)16(2)14-31/h5-6,9-11,16H,7-8,12,14H2,1-4H3	ZNKGHBADDFCFBA-UHFFFAOYSA-N	293023	US10106501, Example AA-10	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293023	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293023&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123492	381613308							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558736	CC(C)N1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C#N)c1Cl	InChI=1S/C26H28Cl2N4O/c1-16(2)31-7-9-32(10-8-31)26(33)20-5-6-23(27)22(25(20)28)14-19-13-21-17(3)11-18(15-29)12-24(21)30(19)4/h5-6,11-13,16H,7-10,14H2,1-4H3	MVRVFRWAAMJPGQ-UHFFFAOYSA-N	293024	US10106501, Example AA-11	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293024	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293024&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123191	381613309							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558737	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCN(CCO)CC4)c3Cl)cc12)C#N	InChI=1S/C25H26Cl2N4O2/c1-16-11-17(15-28)12-23-20(16)13-18(29(23)2)14-21-22(26)4-3-19(24(21)27)25(33)31-7-5-30(6-8-31)9-10-32/h3-4,11-13,32H,5-10,14H2,1-2H3	FGFARKLKSOVFTM-UHFFFAOYSA-N	293025	US10106501, Example AA-12	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293025	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293025&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123534	381613310							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558738	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCCN(CCO)CC4)c3Cl)cc12)C#N	InChI=1S/C26H28Cl2N4O2/c1-17-12-18(16-29)13-24-21(17)14-19(30(24)2)15-22-23(27)5-4-20(25(22)28)26(34)32-7-3-6-31(8-9-32)10-11-33/h4-5,12-14,33H,3,6-11,15H2,1-2H3	NJPPUQFSNBKWDC-UHFFFAOYSA-N	293026	US10106501, Example AA-13	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293026	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293026&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123715	381613311							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558739	CN(C)C1CCN(C1)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C#N)c1Cl	InChI=1S/C25H26Cl2N4O/c1-15-9-16(13-28)10-23-20(15)11-18(30(23)4)12-21-22(26)6-5-19(24(21)27)25(32)31-8-7-17(14-31)29(2)3/h5-6,9-11,17H,7-8,12,14H2,1-4H3	HYBMRLPXULHKKJ-UHFFFAOYSA-N	293027	US10106501, Example AA-14	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293027	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293027&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123610	381613312							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558740	COCCN1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C#N)c1Cl	InChI=1S/C26H28Cl2N4O2/c1-17-12-18(16-29)13-24-21(17)14-19(30(24)2)15-22-23(27)5-4-20(25(22)28)26(33)32-8-6-31(7-9-32)10-11-34-3/h4-5,12-14H,6-11,15H2,1-3H3	IWEZKAPDRMSLMQ-UHFFFAOYSA-N	293028	US10106501, Example AA-15	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293028	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293028&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123489	381613313							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558741	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CC(C4)N4CCCC4)c3Cl)cc12)C#N	InChI=1S/C26H26Cl2N4O/c1-16-9-17(13-29)10-24-21(16)11-18(30(24)2)12-22-23(27)6-5-20(25(22)28)26(33)32-14-19(15-32)31-7-3-4-8-31/h5-6,9-11,19H,3-4,7-8,12,14-15H2,1-2H3	UTCLRDMHDQNQHP-UHFFFAOYSA-N	293029	US10106501, Example AA-16	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293029	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293029&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123303	381613314							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558742	CC(F)CN1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C#N)c1Cl	InChI=1S/C26H27Cl2FN4O/c1-16-10-18(14-30)11-24-21(16)12-19(31(24)3)13-22-23(27)5-4-20(25(22)28)26(34)33-8-6-32(7-9-33)15-17(2)29/h4-5,10-12,17H,6-9,13,15H2,1-3H3	USYAMKPGZGXQBX-UHFFFAOYSA-N	293030	US10106501, Example AA-17	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293030	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293030&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123507	381613315							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558743	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(O)C4)c3Cl)cc12)C#N	InChI=1S/C23H21Cl2N3O2/c1-13-7-14(11-26)8-21-18(13)9-15(27(21)2)10-19-20(24)4-3-17(22(19)25)23(30)28-6-5-16(29)12-28/h3-4,7-9,16,29H,5-6,10,12H2,1-2H3	WREILYWGIFNOPC-UHFFFAOYSA-N	293031	US10106501, Example AA-18	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293031	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293031&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123572	381613316							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558744	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CO)C4)c3Cl)cc12)C#N	InChI=1S/C24H23Cl2N3O2/c1-14-7-16(11-27)8-22-19(14)9-17(28(22)2)10-20-21(25)4-3-18(23(20)26)24(31)29-6-5-15(12-29)13-30/h3-4,7-9,15,30H,5-6,10,12-13H2,1-2H3	MDDMJXSBCRVTTL-UHFFFAOYSA-N	293032	US10106501, Example AA-19	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293032	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293032&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123908	381613317							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558745	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CC(O)C4)c3Cl)cc12)C#N	InChI=1S/C22H19Cl2N3O2/c1-12-5-13(9-25)6-20-17(12)7-14(26(20)2)8-18-19(23)4-3-16(21(18)24)22(29)27-10-15(28)11-27/h3-7,15,28H,8,10-11H2,1-2H3	LVXFKDKKCSUABS-UHFFFAOYSA-N	293033	US10106501, Example AA-20	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293033	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293033&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123441	381613318							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558746	COC1CN(C1)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C#N)c1Cl	InChI=1S/C23H21Cl2N3O2/c1-13-6-14(10-26)7-21-18(13)8-15(27(21)2)9-19-20(24)5-4-17(22(19)25)23(29)28-11-16(12-28)30-3/h4-8,16H,9,11-12H2,1-3H3	UZOPJFMWHNBISM-UHFFFAOYSA-N	293034	US10106501, Example AA-21	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293034	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293034&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123542	381613319							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558747	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)NC4CCC(O)CC4)c3Cl)cc12)C#N |(2.75,.11,;1.98,1.44,;2.75,2.78,;1.98,4.11,;.44,4.11,;-.33,2.78,;-1.84,2.46,;-3.17,3.23,;-2,.92,;-3.33,.15,;-3.33,-1.39,;-4.67,-2.16,;-6,-1.39,;-4.67,-3.7,;-3.33,-4.47,;-2,-3.7,;-.67,-4.47,;-.67,-6.01,;.67,-3.7,;2,-4.47,;2,-6.01,;3.33,-6.78,;4.67,-6.01,;6,-6.78,;4.67,-4.47,;3.33,-3.7,;-2,-2.16,;-.67,-1.39,;-.59,.3,;.44,1.44,;2.75,5.44,;3.52,6.78,)|	InChI=1S/C25H25Cl2N3O2/c1-14-9-15(13-28)10-23-20(14)11-17(30(23)2)12-21-22(26)8-7-19(24(21)27)25(32)29-16-3-5-18(31)6-4-16/h7-11,16,18,31H,3-6,12H2,1-2H3,(H,29,32)	WDLSZTUHBOIQCI-UHFFFAOYSA-N	293035	US10106501, Example AA-22	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293035	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293035&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123409	381613320							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558748	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)NC4CCOCC4)c3Cl)cc12)C#N	InChI=1S/C24H23Cl2N3O2/c1-14-9-15(13-27)10-22-19(14)11-17(29(22)2)12-20-21(25)4-3-18(23(20)26)24(30)28-16-5-7-31-8-6-16/h3-4,9-11,16H,5-8,12H2,1-2H3,(H,28,30)	CTTSWECVWBYKMZ-UHFFFAOYSA-N	293036	US10106501, Example AA-23	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293036	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293036&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123411	381613321							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558749	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)NC4COC4)c3Cl)cc12)C#N	InChI=1S/C22H19Cl2N3O2/c1-12-5-13(9-25)6-20-17(12)7-15(27(20)2)8-18-19(23)4-3-16(21(18)24)22(28)26-14-10-29-11-14/h3-7,14H,8,10-11H2,1-2H3,(H,26,28)	DQDYTCGODBILGH-UHFFFAOYSA-N	293037	US10106501, Example AA-24	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293037	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293037&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122937	381613322							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558750	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC5(COC5)CC4)c3Cl)cc12)C#N	InChI=1S/C26H25Cl2N3O2/c1-16-9-17(13-29)10-23-20(16)11-18(30(23)2)12-21-22(27)4-3-19(24(21)28)25(32)31-7-5-26(6-8-31)14-33-15-26/h3-4,9-11H,5-8,12,14-15H2,1-2H3	SRXNMNYOPKROLT-UHFFFAOYSA-N	293038	US10106501, Example AA-25	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293038	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293038&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123819	381613323							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558751	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CC5(COC5)C4)c3Cl)cc12)C#N	InChI=1S/C24H21Cl2N3O2/c1-14-5-15(9-27)6-21-18(14)7-16(28(21)2)8-19-20(25)4-3-17(22(19)26)23(30)29-10-24(11-29)12-31-13-24/h3-7H,8,10-13H2,1-2H3	QGVJGURRAZEHEE-UHFFFAOYSA-N	293039	US10106501, Example AA-26	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293039	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293039&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123352	381613324							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558752	COCCC1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C#N)c1Cl	InChI=1S/C27H29Cl2N3O2/c1-17-12-19(16-30)13-25-22(17)14-20(31(25)2)15-23-24(28)5-4-21(26(23)29)27(33)32-9-6-18(7-10-32)8-11-34-3/h4-5,12-14,18H,6-11,15H2,1-3H3	XUOXNWAVUBTIRJ-UHFFFAOYSA-N	293040	US10106501, Example AA-27	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293040	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293040&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122970	381613325							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558753	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC4)C4COC4)c3Cl)cc12)C#N	InChI=1S/C27H27Cl2N3O2/c1-16-9-17(13-30)10-25-22(16)11-20(31(25)2)12-23-24(28)4-3-21(26(23)29)27(33)32-7-5-18(6-8-32)19-14-34-15-19/h3-4,9-11,18-19H,5-8,12,14-15H2,1-2H3	XUGNMKWCPOVJCN-UHFFFAOYSA-N	293041	US10106501, Example AA-28	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293041	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293041&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123763	381613326							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558754	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CCO)CC4)c3Cl)cc12)C#N	InChI=1S/C26H27Cl2N3O2/c1-16-11-18(15-29)12-24-21(16)13-19(30(24)2)14-22-23(27)4-3-20(25(22)28)26(33)31-8-5-17(6-9-31)7-10-32/h3-4,11-13,17,32H,5-10,14H2,1-2H3	MIYBHFKXVIIMAA-UHFFFAOYSA-N	293042	US10106501, Example AA-29	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293042	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293042&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123927	381613327							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558755	COCC1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C#N)c1Cl	InChI=1S/C26H27Cl2N3O2/c1-16-10-18(14-29)11-24-21(16)12-19(30(24)2)13-22-23(27)5-4-20(25(22)28)26(32)31-8-6-17(7-9-31)15-33-3/h4-5,10-12,17H,6-9,13,15H2,1-3H3	WFDAONAOIFDLDQ-UHFFFAOYSA-N	293043	US10106501, Example AA-30	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293043	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293043&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123524	381613328							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558756	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC(C)(C)O)CC4)c3Cl)cc12)C#N	InChI=1S/C28H31Cl2N3O2/c1-17-11-19(16-31)12-25-22(17)13-20(32(25)4)14-23-24(29)6-5-21(26(23)30)27(34)33-9-7-18(8-10-33)15-28(2,3)35/h5-6,11-13,18,35H,7-10,14-15H2,1-4H3	UMDBFDZQAHGLCT-UHFFFAOYSA-N	293044	US10106501, Example AA-31	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293044	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293044&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122914	381613329							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558757	CNC(=O)[C@@H]1CCCN1C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C#N)c1Cl |r|	InChI=1S/C25H24Cl2N4O2/c1-14-9-15(13-28)10-22-18(14)11-16(30(22)3)12-19-20(26)7-6-17(23(19)27)25(33)31-8-4-5-21(31)24(32)29-2/h6-7,9-11,21H,4-5,8,12H2,1-3H3,(H,29,32)	QWGPEECIWYISRL-UHFFFAOYSA-N	293045	US10106501, Example AA-32	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293045	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293045&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123199	381613330							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558758	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)cc12)C#N	InChI=1S/C23H21Cl2N3O2/c1-14-9-15(13-26)10-21-18(14)11-16(27(21)2)12-19-20(24)4-3-17(22(19)25)23(29)28-5-7-30-8-6-28/h3-4,9-11H,5-8,12H2,1-2H3	ZKASOECVISRZCR-UHFFFAOYSA-N	293046	US10106501, Example AA-35	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293046	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293046&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123317	381613331							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558759	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC5(CCOC5)CC4)c3Cl)cc12)C#N	InChI=1S/C27H27Cl2N3O2/c1-17-11-18(15-30)12-24-21(17)13-19(31(24)2)14-22-23(28)4-3-20(25(22)29)26(33)32-8-5-27(6-9-32)7-10-34-16-27/h3-4,11-13H,5-10,14,16H2,1-2H3	MSTZBSJZCOSDAK-UHFFFAOYSA-N	293047	US10106501, Example AA-36	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293047	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293047&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123177	381613332							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558760	CC(O)CC1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C#N)c1Cl	InChI=1S/C27H29Cl2N3O2/c1-16-10-19(15-30)12-25-22(16)13-20(31(25)3)14-23-24(28)5-4-21(26(23)29)27(34)32-8-6-18(7-9-32)11-17(2)33/h4-5,10,12-13,17-18,33H,6-9,11,14H2,1-3H3	VKOIVPISVYEKSH-UHFFFAOYSA-N	293048	US10106501, Example AA-37	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293048	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293048&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122936	381613333							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558761	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CC[C@@H](O)C4)c3Cl)cc12)C#N |r|	InChI=1S/C23H21Cl2N3O2/c1-13-7-14(11-26)8-21-18(13)9-15(27(21)2)10-19-20(24)4-3-17(22(19)25)23(30)28-6-5-16(29)12-28/h3-4,7-9,16,29H,5-6,10,12H2,1-2H3	WREILYWGIFNOPC-UHFFFAOYSA-N	293049	US10106501, Example AA-40::US10106501, Example AA-39	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293049	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293049&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123603	381613334							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558762	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CC[C@@H](O)C4)c3Cl)cc12)C#N |r|	InChI=1S/C23H21Cl2N3O2/c1-13-7-14(11-26)8-21-18(13)9-15(27(21)2)10-19-20(24)4-3-17(22(19)25)23(30)28-6-5-16(29)12-28/h3-4,7-9,16,29H,5-6,10,12H2,1-2H3	WREILYWGIFNOPC-UHFFFAOYSA-N	293049	US10106501, Example AA-40::US10106501, Example AA-39	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293049	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293049&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123603	381613334							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558763	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)cc2cc(ccc12)C#N	InChI=1S/C22H19Cl2N3O2/c1-26-16(11-15-10-14(13-25)2-5-20(15)26)12-18-19(23)4-3-17(21(18)24)22(28)27-6-8-29-9-7-27/h2-5,10-11H,6-9,12H2,1H3	XYHMHVTZCILHOH-UHFFFAOYSA-N	293051	US10106501, Example AB	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293051	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293051&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123477	381613335							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558764	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)cc2ccc(cc12)C#N	InChI=1S/C22H19Cl2N3O2/c1-26-16(11-15-3-2-14(13-25)10-20(15)26)12-18-19(23)5-4-17(21(18)24)22(28)27-6-8-29-9-7-27/h2-5,10-11H,6-9,12H2,1H3	WGXVGTXGWBCKBU-UHFFFAOYSA-N	293052	US10106501, Example AC	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293052	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293052&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123079	381613336							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558765	Cc1cc(cc2n(C)c(cc12)C(=O)c1c(Cl)ccc(C(=O)N2CCOCC2)c1Cl)C#N	InChI=1S/C23H19Cl2N3O3/c1-13-9-14(12-26)10-18-16(13)11-19(27(18)2)22(29)20-17(24)4-3-15(21(20)25)23(30)28-5-7-31-8-6-28/h3-4,9-11H,5-8H2,1-2H3	REOSQSWUYVWADO-UHFFFAOYSA-N	293053	US10106501, Example AD	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293053	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293053&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122952	381613337							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558766	Cc1ccc(C(=O)N2CCOCC2)c(C)c1Cc1cc2c(C)cc(cc2n1C)C#N	InChI=1S/C25H27N3O2/c1-16-5-6-21(25(29)28-7-9-30-10-8-28)18(3)22(16)13-20-14-23-17(2)11-19(15-26)12-24(23)27(20)4/h5-6,11-12,14H,7-10,13H2,1-4H3	KNTDNGPOBVPGLY-UHFFFAOYSA-N	293054	US10106501, Example AE	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293054	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293054&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123585	381613338							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558767	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(O[C@H]4CC[C@@H](CC4)C(O)=O)c3Cl)cc12)C#N |r,wU:20.23,wD:17.16,(2.75,-8.28,;1.98,-6.95,;2.75,-5.62,;1.98,-4.28,;.44,-4.28,;-.33,-5.62,;-1.84,-5.94,;-2.98,-4.91,;-2,-7.47,;-3.33,-8.24,;-3.33,-9.78,;-4.67,-10.55,;-6,-9.78,;-4.67,-12.09,;-3.33,-12.86,;-2,-12.09,;-.67,-12.86,;.67,-12.09,;2,-12.86,;3.33,-12.09,;3.33,-10.55,;2,-9.78,;.67,-10.55,;4.67,-9.78,;6,-10.55,;4.67,-8.24,;-2,-10.55,;-.67,-9.78,;-.59,-8.09,;.44,-6.95,;2.75,-2.95,;3.52,-1.62,)|	InChI=1S/C25H24Cl2N2O3/c1-14-9-15(13-28)10-22-19(14)11-17(29(22)2)12-20-21(26)7-8-23(24(20)27)32-18-5-3-16(4-6-18)25(30)31/h7-11,16,18H,3-6,12H2,1-2H3,(H,30,31)	YQJUKJFVQYFRAK-UHFFFAOYSA-N	293055	trans-4-(2,4-dichloro-3-((6-cyano-1,4-dimethyl-1H-indol-2-yl)methyl)phenoxy)cyclohexanecarboxylic acid::US10106501, Example AF	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293055	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293055&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123077	381613339							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558768	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(O[C@H]4CC[C@H](CC4)C(O)=O)c3Cl)cc12)C#N |r,wU:17.16,20.23,(2.75,-8.28,;1.98,-6.95,;2.75,-5.62,;1.98,-4.28,;.44,-4.28,;-.33,-5.62,;-1.84,-5.94,;-2.98,-4.91,;-2,-7.47,;-3.33,-8.24,;-3.33,-9.78,;-4.67,-10.55,;-6,-9.78,;-4.67,-12.09,;-3.33,-12.86,;-2,-12.09,;-.67,-12.86,;.67,-12.09,;.67,-10.55,;2,-9.78,;3.33,-10.55,;3.33,-12.09,;2,-12.86,;4.67,-9.78,;6,-10.55,;4.67,-8.24,;-2,-10.55,;-.67,-9.78,;-.59,-8.09,;.44,-6.95,;2.75,-2.95,;3.52,-1.62,)|	InChI=1S/C25H24Cl2N2O3/c1-14-9-15(13-28)10-22-19(14)11-17(29(22)2)12-20-21(26)7-8-23(24(20)27)32-18-5-3-16(4-6-18)25(30)31/h7-11,16,18H,3-6,12H2,1-2H3,(H,30,31)	YQJUKJFVQYFRAK-UHFFFAOYSA-N	293056	cis-4-(2,4-dichloro-3-((6-cyano-1,4-dimethyl-1H-indol-2-yl)methyl)phenoxy)cyclohexanecarboxylic acid::US10106501, Example AF1	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293056	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293056&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123077	381613340							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558769	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(O[C@H]4CC[C@@H](C4)C(O)=O)c3Cl)cc12)C#N |r|	InChI=1S/C24H22Cl2N2O3/c1-13-7-14(12-27)8-21-18(13)10-16(28(21)2)11-19-20(25)5-6-22(23(19)26)31-17-4-3-15(9-17)24(29)30/h5-8,10,15,17H,3-4,9,11H2,1-2H3,(H,29,30)	GWMOUDSPJATIPF-UHFFFAOYSA-N	293057	trans-3-(2,4-dichloro-3-((6-cyano-1,4-dimethyl-1H-indol-2-yl)methyl)phenoxy)cyclopentanecarboxylic acid::US10106501, Example AG	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293057	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293057&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123501	381613341							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558770	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(O[C@H]4CC[C@H](C4)C(O)=O)c3Cl)cc12)C#N |r|	InChI=1S/C24H22Cl2N2O3/c1-13-7-14(12-27)8-21-18(13)10-16(28(21)2)11-19-20(25)5-6-22(23(19)26)31-17-4-3-15(9-17)24(29)30/h5-8,10,15,17H,3-4,9,11H2,1-2H3,(H,29,30)	GWMOUDSPJATIPF-UHFFFAOYSA-N	293058	cis-3-(2,4-dichloro-3-((6-cyano-1,4-dimethyl-1H-indol-2-yl)methyl)phenoxy)cyclopentanecarboxylic acid::US10106501, Example AG1	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293058	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293058&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123498	381613342							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558771	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(O[C@H]4C[C@@H](C4)C(O)=O)c3Cl)cc12)C#N |r,wU:17.16,wD:19.21,(3.14,-8.11,;2.37,-6.77,;3.14,-5.44,;2.37,-4.1,;.83,-4.1,;.06,-5.44,;-1.45,-5.76,;-2.59,-4.73,;-1.61,-7.29,;-2.94,-8.06,;-2.94,-9.6,;-4.28,-10.37,;-5.61,-9.6,;-4.28,-11.91,;-2.94,-12.68,;-1.61,-11.91,;-.28,-12.68,;1.06,-11.91,;1.46,-10.42,;2.94,-10.82,;2.55,-12.31,;4.28,-10.05,;5.61,-10.82,;4.28,-8.51,;-1.61,-10.37,;-.28,-9.6,;-.2,-7.92,;.83,-6.77,;3.14,-2.77,;3.91,-1.44,)|	InChI=1S/C23H20Cl2N2O3/c1-12-5-13(11-26)6-20-17(12)9-15(27(20)2)10-18-19(24)3-4-21(22(18)25)30-16-7-14(8-16)23(28)29/h3-6,9,14,16H,7-8,10H2,1-2H3,(H,28,29)	SZDYHGOLVVDOKY-UHFFFAOYSA-N	293059	trans-3-(2,4-dichloro-3-((6-cyano-1,4-dimethyl-1H-indol-2-yl)methyl)phenoxy)cyclobutanecarboxylic acid::US10106501, Example AH	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293059	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293059&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123691	381613343							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558772	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(O[C@H]4C[C@H](C4)C(O)=O)c3Cl)cc12)C#N |r,wU:17.16,19.21,(3.14,-8.11,;2.37,-6.77,;3.14,-5.44,;2.37,-4.1,;.83,-4.1,;.06,-5.44,;-1.45,-5.76,;-2.59,-4.73,;-1.61,-7.29,;-2.94,-8.06,;-2.94,-9.6,;-4.28,-10.37,;-5.61,-9.6,;-4.28,-11.91,;-2.94,-12.68,;-1.61,-11.91,;-.28,-12.68,;1.06,-11.91,;1.46,-10.42,;2.94,-10.82,;2.55,-12.31,;4.28,-10.05,;5.61,-10.82,;4.28,-8.51,;-1.61,-10.37,;-.28,-9.6,;-.2,-7.92,;.83,-6.77,;3.14,-2.77,;3.91,-1.44,)|	InChI=1S/C23H20Cl2N2O3/c1-12-5-13(11-26)6-20-17(12)9-15(27(20)2)10-18-19(24)3-4-21(22(18)25)30-16-7-14(8-16)23(28)29/h3-6,9,14,16H,7-8,10H2,1-2H3,(H,28,29)	SZDYHGOLVVDOKY-UHFFFAOYSA-N	293060	cis-3-(2,4-dichloro-3-((6-cyano-1,4-dimethyl-1H-indol-2-yl)methyl)phenoxy)cyclobutanecarboxylic acid::US10106501, Example AH1	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293060	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293060&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123691	381613344							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558773	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(O[C@H]4C[C@@H](C4)C(O)=O)c3Cl)cc12)C(F)(F)F |r,wU:17.16,wD:19.21,(3.14,-8.45,;2.37,-7.11,;3.14,-5.78,;2.37,-4.45,;.83,-4.45,;.06,-5.78,;-1.45,-6.1,;-2.59,-5.07,;-1.61,-7.63,;-2.94,-8.4,;-2.94,-9.94,;-4.28,-10.71,;-5.61,-9.94,;-4.28,-12.25,;-2.94,-13.02,;-1.61,-12.25,;-.28,-13.02,;1.06,-12.25,;1.46,-10.76,;2.94,-11.16,;2.55,-12.65,;4.28,-10.39,;5.61,-11.16,;4.28,-8.85,;-1.61,-10.71,;-.28,-9.94,;-.2,-8.26,;.83,-7.11,;3.14,-3.11,;2.37,-1.78,;4.68,-3.11,;3.91,-1.78,)|	InChI=1S/C23H20Cl2F3NO3/c1-11-5-13(23(26,27)28)8-19-16(11)9-14(29(19)2)10-17-18(24)3-4-20(21(17)25)32-15-6-12(7-15)22(30)31/h3-5,8-9,12,15H,6-7,10H2,1-2H3,(H,30,31)	IBHMOGYCBQRDRE-UHFFFAOYSA-N	293061	trans-4-(2,4-dichloro-3-((1,4-dimethyl-6-(trifluoromethyl)-1H-indol-2-yl)methyl)phenoxy)cyclohexanecarboxylic acid::US10106501, Example AI	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293061	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293061&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124124917	381613345							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558774	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(O[C@H]4C[C@H](C4)C(O)=O)c3Cl)cc12)C(F)(F)F |r,wU:17.16,19.21,(3.14,-8.45,;2.37,-7.11,;3.14,-5.78,;2.37,-4.45,;.83,-4.45,;.06,-5.78,;-1.45,-6.1,;-2.59,-5.07,;-1.61,-7.63,;-2.94,-8.4,;-2.94,-9.94,;-4.28,-10.71,;-5.61,-9.94,;-4.28,-12.25,;-2.94,-13.02,;-1.61,-12.25,;-.28,-13.02,;1.06,-12.25,;1.46,-10.76,;2.94,-11.16,;2.55,-12.65,;4.28,-10.39,;5.61,-11.16,;4.28,-8.85,;-1.61,-10.71,;-.28,-9.94,;-.2,-8.26,;.83,-7.11,;3.14,-3.11,;2.37,-1.78,;4.68,-3.11,;3.91,-1.78,)|	InChI=1S/C23H20Cl2F3NO3/c1-11-5-13(23(26,27)28)8-19-16(11)9-14(29(19)2)10-17-18(24)3-4-20(21(17)25)32-15-6-12(7-15)22(30)31/h3-5,8-9,12,15H,6-7,10H2,1-2H3,(H,30,31)	IBHMOGYCBQRDRE-UHFFFAOYSA-N	293062	cis-4-(2,4-dichloro-3-((1,4-dimethyl-6-(trifluoromethyl)-1H-indol-2-yl)methyl)phenoxy)cyclohexanecarboxylic acid::US10106501, Example AI1	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293062	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293062&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124124917	381613346							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558775	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(O[C@H]4C[C@@H](C4)C(O)=O)c3Cl)cc12)C(F)(F)F |r,wU:17.16,wD:19.21,(3.14,-8.01,;2.37,-6.67,;3.14,-5.34,;2.37,-4,;.83,-4,;.06,-5.34,;-1.45,-5.66,;-2.54,-4.57,;-1.61,-7.19,;-2.94,-7.96,;-2.94,-9.5,;-4.28,-10.27,;-5.61,-9.5,;-4.28,-11.81,;-2.94,-12.58,;-1.61,-11.81,;-.28,-12.58,;1.06,-11.81,;1.46,-10.32,;2.94,-10.72,;2.55,-12.21,;4.28,-9.95,;5.61,-10.72,;4.28,-8.41,;-1.61,-10.27,;-.28,-9.5,;-.2,-7.82,;.83,-6.67,;3.14,-2.67,;2.37,-1.34,;4.68,-2.67,;3.91,-1.34,)|	InChI=1S/C23H20Cl2F3NO3/c1-11-5-13(23(26,27)28)8-19-16(11)9-14(29(19)2)10-17-18(24)3-4-20(21(17)25)32-15-6-12(7-15)22(30)31/h3-5,8-9,12,15H,6-7,10H2,1-2H3,(H,30,31)	IBHMOGYCBQRDRE-UHFFFAOYSA-N	293063	trans-4-(2,4-dichloro-3-((1,4-dimethyl-6-(trifluoromethyl)-1H-indol-2-yl)methyl)phenoxy)cyclohexanecarboxylic acid::US10106501, Example AJ	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293063	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293063&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124124917	381613347							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558776	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(O[C@H]4C[C@H](C4)C(O)=O)c3Cl)cc12)C(F)(F)F |r,wU:17.16,19.21,(3.14,-8.01,;2.37,-6.67,;3.14,-5.34,;2.37,-4,;.83,-4,;.06,-5.34,;-1.45,-5.66,;-2.54,-4.57,;-1.61,-7.19,;-2.94,-7.96,;-2.94,-9.5,;-4.28,-10.27,;-5.61,-9.5,;-4.28,-11.81,;-2.94,-12.58,;-1.61,-11.81,;-.28,-12.58,;1.06,-11.81,;1.46,-10.32,;2.94,-10.72,;2.55,-12.21,;4.28,-9.95,;5.61,-10.72,;4.28,-8.41,;-1.61,-10.27,;-.28,-9.5,;-.2,-7.82,;.83,-6.67,;3.14,-2.67,;2.37,-1.34,;4.68,-2.67,;3.91,-1.34,)|	InChI=1S/C23H20Cl2F3NO3/c1-11-5-13(23(26,27)28)8-19-16(11)9-14(29(19)2)10-17-18(24)3-4-20(21(17)25)32-15-6-12(7-15)22(30)31/h3-5,8-9,12,15H,6-7,10H2,1-2H3,(H,30,31)	IBHMOGYCBQRDRE-UHFFFAOYSA-N	293064	cis-4-(2,4-dichloro-3-((1,4-dimethyl-6-(trifluoromethyl)-1H-indol-2-yl)methyl)phenoxy)cyclohexanecarboxylic acid::US10106501, Example AJ1	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293064	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293064&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124124917	381613348							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558777	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(O[C@H]4CC[C@@H](C4)C(O)=O)c3Cl)cc12)C(F)(F)F |r|	InChI=1S/C24H22Cl2F3NO3/c1-12-7-14(24(27,28)29)9-20-17(12)10-15(30(20)2)11-18-19(25)5-6-21(22(18)26)33-16-4-3-13(8-16)23(31)32/h5-7,9-10,13,16H,3-4,8,11H2,1-2H3,(H,31,32)	RSHWJPYRFKGROC-UHFFFAOYSA-N	293065	trans-3-(2,4-dichloro-3-((1,4-dimethyl-6-(trifluoromethyl)-1H-indol-2-yl)methyl)phenoxy)cyclopentanecarboxylic acid::US10106501, Example AK	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293065	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293065&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123098	381613349							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558778	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(O[C@H]4CC[C@H](C4)C(O)=O)c3Cl)cc12)C(F)(F)F |r|	InChI=1S/C24H22Cl2F3NO3/c1-12-7-14(24(27,28)29)9-20-17(12)10-15(30(20)2)11-18-19(25)5-6-21(22(18)26)33-16-4-3-13(8-16)23(31)32/h5-7,9-10,13,16H,3-4,8,11H2,1-2H3,(H,31,32)	RSHWJPYRFKGROC-UHFFFAOYSA-N	293066	cis-3-(2,4-dichloro-3-((1,4-dimethyl-6-(trifluoromethyl)-1H-indol-2-yl)methyl)phenoxy)cyclopentanecarboxylic acid::US10106501, Example AK1	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293066	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293066&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123666	381613350							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558779	Cc1cc(cc2n(C)c(Cc3c(Cl)cnc(OCC4CCOCC4)c3Cl)cc12)C(F)(F)F	InChI=1S/C23H23Cl2F3N2O2/c1-13-7-15(23(26,27)28)8-20-17(13)9-16(30(20)2)10-18-19(24)11-29-22(21(18)25)32-12-14-3-5-31-6-4-14/h7-9,11,14H,3-6,10,12H2,1-2H3	IUPIYUOPSIEAAH-UHFFFAOYSA-N	293067	US10106501, Example AL1::US10106501, Example AL	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293067	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293067&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122984	381613351							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558780	Cc1cc(cc2n(C)c(Cc3c(Cl)cnc(OCC4CCOCC4)c3Cl)cc12)C(F)(F)F	InChI=1S/C23H23Cl2F3N2O2/c1-13-7-15(23(26,27)28)8-20-17(13)9-16(30(20)2)10-18-19(24)11-29-22(21(18)25)32-12-14-3-5-31-6-4-14/h7-9,11,14H,3-6,10,12H2,1-2H3	IUPIYUOPSIEAAH-UHFFFAOYSA-N	293067	US10106501, Example AL1::US10106501, Example AL	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293067	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293067&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122984	381613351							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558781	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC4)OCC(O)=O)c3Cl)cc12)C#N	InChI=1S/C26H25Cl2N3O4/c1-15-9-16(13-29)10-23-20(15)11-17(30(23)2)12-21-22(27)4-3-19(25(21)28)26(34)31-7-5-18(6-8-31)35-14-24(32)33/h3-4,9-11,18H,5-8,12,14H2,1-2H3,(H,32,33)	WJOFEEQULDYRBB-UHFFFAOYSA-N	293069	US10106501, Example AM	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293069	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293069&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123719	381613352							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558782	CC1CN(CCC1C(O)=O)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C#N)c1Cl	InChI=1S/C26H25Cl2N3O3/c1-14-8-16(12-29)9-23-20(14)10-17(30(23)3)11-21-22(27)5-4-19(24(21)28)25(32)31-7-6-18(26(33)34)15(2)13-31/h4-5,8-10,15,18H,6-7,11,13H2,1-3H3,(H,33,34)	RSSJTDJNWSGFPR-UHFFFAOYSA-N	293070	US10106501, Example AM-1	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293070	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293070&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123888	381613353							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558783	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC4)C(O)=O)c3Cl)cc12)C#N	InChI=1S/C25H23Cl2N3O3/c1-14-9-15(13-28)10-22-19(14)11-17(29(22)2)12-20-21(26)4-3-18(23(20)27)24(31)30-7-5-16(6-8-30)25(32)33/h3-4,9-11,16H,5-8,12H2,1-2H3,(H,32,33)	HNOAGEJJZOAAHF-UHFFFAOYSA-N	293071	US10106501, Example AM-2	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293071	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293071&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123837	381613354							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558784	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)cc12)C#N	InChI=1S/C26H25Cl2N3O3/c1-15-9-17(14-29)10-23-20(15)12-18(30(23)2)13-21-22(27)4-3-19(25(21)28)26(34)31-7-5-16(6-8-31)11-24(32)33/h3-4,9-10,12,16H,5-8,11,13H2,1-2H3,(H,32,33)	QRRCVXOTQGTEJX-UHFFFAOYSA-N	293072	US10106501, Example AM-3	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293072	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293072&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122858	381613355							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558785	Cc1cc(cc2n(C)c(cc12)C(=O)c1c(Cl)ccc(C(=O)N2CCC(O)CC2)c1Cl)C#N	InChI=1S/C24H21Cl2N3O3/c1-13-9-14(12-27)10-19-17(13)11-20(28(19)2)23(31)21-18(25)4-3-16(22(21)26)24(32)29-7-5-15(30)6-8-29/h3-4,9-11,15,30H,5-8H2,1-2H3	SKKQMWZUEAPRPB-UHFFFAOYSA-N	293073	US10106501, Example AN	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293073	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293073&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123007	381613356							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558786	Cc1cc(cc2n(C)c(cc12)C(=O)c1c(Cl)ccc(C(=O)N2CC(O)C2)c1Cl)C#N	InChI=1S/C22H17Cl2N3O3/c1-11-5-12(8-25)6-17-15(11)7-18(26(17)2)21(29)19-16(23)4-3-14(20(19)24)22(30)27-9-13(28)10-27/h3-7,13,28H,9-10H2,1-2H3	AEROWLUUGPUIKD-UHFFFAOYSA-N	293074	US10106501, Example AN-1	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293074	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293074&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123264	381613357							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558787	Cc1cc(cc2n(C)c(cc12)C(=O)c1c(Cl)ccc(C(=O)N2CCN(CC2)C2COC2)c1Cl)C#N	InChI=1S/C26H24Cl2N4O3/c1-15-9-16(12-29)10-21-19(15)11-22(30(21)2)25(33)23-20(27)4-3-18(24(23)28)26(34)32-7-5-31(6-8-32)17-13-35-14-17/h3-4,9-11,17H,5-8,13-14H2,1-2H3	PDHCIMBXCDKIOB-UHFFFAOYSA-N	293075	US10106501, Example AN-2	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293075	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293075&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123742	381613358							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558788	Cc1cc(cc2n(C)c(cc12)C(=O)c1c(Cl)ccc(C(=O)N2CCC(CC2)C(C)(C)CO)c1Cl)C#N	InChI=1S/C28H29Cl2N3O3/c1-16-11-17(14-31)12-22-20(16)13-23(32(22)4)26(35)24-21(29)6-5-19(25(24)30)27(36)33-9-7-18(8-10-33)28(2,3)15-34/h5-6,11-13,18,34H,7-10,15H2,1-4H3	CYYKUQBHCNEBJV-UHFFFAOYSA-N	293076	US10106501, Example AN-3	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293076	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293076&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123386	381613359							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558789	COCCC1CCN(CC1)C(=O)c1ccc(Cl)c(C(=O)c2cc3c(C)cc(cc3n2C)C#N)c1Cl	InChI=1S/C27H27Cl2N3O3/c1-16-12-18(15-30)13-22-20(16)14-23(31(22)2)26(33)24-21(28)5-4-19(25(24)29)27(34)32-9-6-17(7-10-32)8-11-35-3/h4-5,12-14,17H,6-11H2,1-3H3	DALBUJFAYIEZFC-UHFFFAOYSA-N	293077	US10106501, Example AN-4	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293077	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293077&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123636	381613360							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558790	Cc1cc(cc2n(C)c(cc12)C(=O)c1c(Cl)ccc(C(=O)N2CCC(CCO)CC2)c1Cl)C#N	InChI=1S/C26H25Cl2N3O3/c1-15-11-17(14-29)12-21-19(15)13-22(30(21)2)25(33)23-20(27)4-3-18(24(23)28)26(34)31-8-5-16(6-9-31)7-10-32/h3-4,11-13,16,32H,5-10H2,1-2H3	BELMUMMRQQQGGH-UHFFFAOYSA-N	293078	US10106501, Example AN-5	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293078	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293078&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123578	381613361							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558791	Cc1cc(cc2n(C)c(cc12)C(=O)c1c(Cl)ccc(C(=O)N2CCC(CC(O)=O)CC2)c1Cl)C#N	InChI=1S/C26H23Cl2N3O4/c1-14-9-16(13-29)10-20-18(14)12-21(30(20)2)25(34)23-19(27)4-3-17(24(23)28)26(35)31-7-5-15(6-8-31)11-22(32)33/h3-4,9-10,12,15H,5-8,11H2,1-2H3,(H,32,33)	QRBFSTGSULUIQC-UHFFFAOYSA-N	293079	US10106501, Example AO	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293079	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293079&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123341	381613362							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558792	Cc1cc(cc2n(C)c(cc12)C(=O)c1c(Cl)ccc(C(=O)N2CCOCC2)c1Cl)C(F)(F)F	InChI=1S/C23H19Cl2F3N2O3/c1-12-9-13(23(26,27)28)10-17-15(12)11-18(29(17)2)21(31)19-16(24)4-3-14(20(19)25)22(32)30-5-7-33-8-6-30/h3-4,9-11H,5-8H2,1-2H3	UJHSFGXZPKVGOI-UHFFFAOYSA-N	293080	US10106501, Example AP	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293080	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293080&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123104	381613363							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558793	Cc1cc(cc2n(C)c(cc12)C(=O)c1c(Cl)ccc(C(=O)N2CCN(CC2)C2COC2)c1Cl)C(F)(F)F	InChI=1S/C26H24Cl2F3N3O3/c1-14-9-15(26(29,30)31)10-20-18(14)11-21(32(20)2)24(35)22-19(27)4-3-17(23(22)28)25(36)34-7-5-33(6-8-34)16-12-37-13-16/h3-4,9-11,16H,5-8,12-13H2,1-2H3	YONVQCJWEMILRR-UHFFFAOYSA-N	293081	US10106501, Example AP-1	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293081	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293081&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123438	381613364							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558794	Cc1cc(cc2n(C)c(cc12)C(=O)c1c(Cl)ccc(C(=O)N2CCC(CC(O)=O)CC2)c1Cl)C(F)(F)F	InChI=1S/C26H23Cl2F3N2O4/c1-13-9-15(26(29,30)31)11-19-17(13)12-20(32(19)2)24(36)22-18(27)4-3-16(23(22)28)25(37)33-7-5-14(6-8-33)10-21(34)35/h3-4,9,11-12,14H,5-8,10H2,1-2H3,(H,34,35)	MQPIAMQRLSAESP-UHFFFAOYSA-N	293082	US10106501, Example AQ	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293082	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293082&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123299	381613365							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558795	Cc1cc(cc2n(C)c(cc12)C(=O)c1c(Cl)ccc(C(=O)N2CCN(CC(O)=O)CC2)c1Cl)C(F)(F)F	InChI=1S/C25H22Cl2F3N3O4/c1-13-9-14(25(28,29)30)10-18-16(13)11-19(31(18)2)23(36)21-17(26)4-3-15(22(21)27)24(37)33-7-5-32(6-8-33)12-20(34)35/h3-4,9-11H,5-8,12H2,1-2H3,(H,34,35)	QATBTZSKMWYGPP-UHFFFAOYSA-N	293083	US10106501, Example AQ-1	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293083	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293083&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123827	381613366							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558796	Cc1cc(cc2n(C)c(cc12)C(=O)c1c(Cl)ccc(C(=O)N2C[C@H]3[C@@H](C2)[C@@H]3C(O)=O)c1Cl)C(F)(F)F |r|	InChI=1S/C25H19Cl2F3N2O4/c1-10-5-11(25(28,29)30)6-17-13(10)7-18(31(17)2)22(33)20-16(26)4-3-12(21(20)27)23(34)32-8-14-15(9-32)19(14)24(35)36/h3-7,14-15,19H,8-9H2,1-2H3,(H,35,36)	PSDZBDQEWLUOLB-UHFFFAOYSA-N	293084	US10106501, Example AQ-2	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293084	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293084&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123197	381613367							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558797	Cc1cc(cc2n(C)c(cc12)C(=O)c1c(Cl)ccc(CO)c1Cl)C(F)(F)F	InChI=1S/C19H14Cl2F3NO2/c1-9-5-11(19(22,23)24)6-14-12(9)7-15(25(14)2)18(27)16-13(20)4-3-10(8-26)17(16)21/h3-7,26H,8H2,1-2H3	LQCVEAQAASUZIP-UHFFFAOYSA-N	293085	US10106501, Example AR	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293085	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293085&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122950	381613368							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558798	Cc1cc(cc2cc(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)[nH]c12)C(F)(F)F	InChI=1S/C22H19Cl2F3N2O2/c1-12-8-14(22(25,26)27)9-13-10-15(28-20(12)13)11-17-18(23)3-2-16(19(17)24)21(30)29-4-6-31-7-5-29/h2-3,8-10,28H,4-7,11H2,1H3	RYUJXJBNDFIZCO-UHFFFAOYSA-N	293086	US10106501, Example AS	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293086	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293086&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123813	381613369							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558799	Cc1cc(cc2cc(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)n(C)c12)C(F)(F)F	InChI=1S/C23H21Cl2F3N2O2/c1-13-9-15(23(26,27)28)10-14-11-16(29(2)21(13)14)12-18-19(24)4-3-17(20(18)25)22(31)30-5-7-32-8-6-30/h3-4,9-11H,5-8,12H2,1-2H3	GCUPNCWAGFMVKZ-UHFFFAOYSA-N	293087	US10106501, Example AT	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293087	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293087&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123437	381613370							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558800	Cc1cc(cc2n(C)c(cc12)C(=O)c1c(Cl)ccc(CN2CCOCC2=O)c1Cl)C#N	InChI=1S/C23H19Cl2N3O3/c1-13-7-14(10-26)8-18-16(13)9-19(27(18)2)23(30)21-17(24)4-3-15(22(21)25)11-28-5-6-31-12-20(28)29/h3-4,7-9H,5-6,11-12H2,1-2H3	MDIGTDCINFNART-UHFFFAOYSA-N	293088	2-(2,6-dichloro-3-((3-oxomorpholino)methyl)benzyl)-1,4-dimethyl-1H-indole-6-carbonitrile Example AU1: 2-(2,6-dichloro-3-((3-oxomorpholino)methyl)benzoyl)-1,4-dimethyl-1H-indole-6-carbonitrile::US10106501, Example AU	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293088	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293088&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123906	381613371							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558801	CCOC(=O)CN1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C27H28Cl2F3N3O3/c1-4-38-24(36)15-34-7-9-35(10-8-34)26(37)19-5-6-22(28)21(25(19)29)14-18-13-20-16(2)11-17(27(30,31)32)12-23(20)33(18)3/h5-6,11-13H,4,7-10,14-15H2,1-3H3	TURPRYBOJNARRI-UHFFFAOYSA-N	293089	US10106501, Example AV	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293089	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293089&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123936	381613372							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558802	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCN(CC(O)=O)CC4)c3Cl)cc12)C(F)(F)F	InChI=1S/C25H24Cl2F3N3O3/c1-14-9-15(25(28,29)30)10-21-18(14)11-16(31(21)2)12-19-20(26)4-3-17(23(19)27)24(36)33-7-5-32(6-8-33)13-22(34)35/h3-4,9-11H,5-8,12-13H2,1-2H3,(H,34,35)	LOMUCQIYJUEZKU-UHFFFAOYSA-N	293090	US10106501, Example AW	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293090	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293090&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122871	381613373							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558803	Cc1cc(Br)cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)cc12	InChI=1S/C22H21BrCl2N2O2/c1-13-9-14(23)10-20-17(13)11-15(26(20)2)12-18-19(24)4-3-16(21(18)25)22(28)27-5-7-29-8-6-27/h3-4,9-11H,5-8,12H2,1-2H3	IKNSPBUPYSEYDB-UHFFFAOYSA-N	293091	US10106501, Example AX	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293091	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293091&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123279	381613374							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558804	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)cc12)N1CCOCC1	InChI=1S/C26H29Cl2N3O3/c1-17-13-19(30-5-9-33-10-6-30)16-24-21(17)14-18(29(24)2)15-22-23(27)4-3-20(25(22)28)26(32)31-7-11-34-12-8-31/h3-4,13-14,16H,5-12,15H2,1-2H3	RSUARCRRMQGSTB-UHFFFAOYSA-N	293092	US10106501, Example AY	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293092	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293092&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123262	381613375							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558805	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(C(O)=O)C(F)(F)C4)c3Cl)cc12)C(F)(F)F	InChI=1S/C25H21Cl2F5N2O3/c1-12-7-13(25(30,31)32)8-20-16(12)9-14(33(20)2)10-17-19(26)4-3-15(21(17)27)22(35)34-6-5-18(23(36)37)24(28,29)11-34/h3-4,7-9,18H,5-6,10-11H2,1-2H3,(H,36,37)	CBJJWNRCCNZDHX-UHFFFAOYSA-N	293093	US10106501, Example AZ	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293093	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293093&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123389	381613376							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558806	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(C(F)C4)C(O)=O)c3Cl)cc12)C(F)(F)F	InChI=1S/C25H22Cl2F4N2O3/c1-12-7-13(25(29,30)31)8-21-17(12)9-14(32(21)2)10-18-19(26)4-3-16(22(18)27)23(34)33-6-5-15(24(35)36)20(28)11-33/h3-4,7-9,15,20H,5-6,10-11H2,1-2H3,(H,35,36)	BQBHMJCGEDPJJD-UHFFFAOYSA-N	293094	US10106501, Example BA	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293094	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293094&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123387	381613377							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558807	Cc1cc(cc2n(C)c(Cc3c(C)ncc(C(=O)N4CCOCC4)c3C)cc12)C(F)(F)F	InChI=1S/C24H26F3N3O2/c1-14-9-17(24(25,26)27)10-22-19(14)11-18(29(22)4)12-20-15(2)21(13-28-16(20)3)23(31)30-5-7-32-8-6-30/h9-11,13H,5-8,12H2,1-4H3	YWDCSIHDIRXRMA-UHFFFAOYSA-N	293095	US10106501, Example BB	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293095	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293095&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123835	381613378							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558808	Cc1ncc(C(=O)N2CCC(CC(O)=O)CC2)c(C)c1Cc1cc2c(C)cc(cc2n1C)C(F)(F)F	InChI=1S/C27H30F3N3O3/c1-15-9-19(27(28,29)30)11-24-21(15)12-20(32(24)4)13-22-16(2)23(14-31-17(22)3)26(36)33-7-5-18(6-8-33)10-25(34)35/h9,11-12,14,18H,5-8,10,13H2,1-4H3,(H,34,35)	RSPHZVYRXMNQLW-UHFFFAOYSA-N	293096	US10106501, Example BC	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293096	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293096&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123179	381613379							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558809	Cc1ncc(C(=O)N2CCC(CC2)C2COC2)c(C)c1C(=O)c1cc2c(C)cc(cc2n1C)C#N	InChI=1S/C28H30N4O3/c1-16-9-19(12-29)10-24-22(16)11-25(31(24)4)27(33)26-17(2)23(13-30-18(26)3)28(34)32-7-5-20(6-8-32)21-14-35-15-21/h9-11,13,20-21H,5-8,14-15H2,1-4H3	INUCSKCQPLJRDP-UHFFFAOYSA-N	293097	US10106501, Example BD	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293097	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293097&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123537	381613380							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558810	Cc1cc(cc2n(C)c(Cc3c(Cl)cnc(C(=O)N4CCOCC4)c3Cl)cc12)C(F)(F)F	InChI=1S/C22H20Cl2F3N3O2/c1-12-7-13(22(25,26)27)8-18-15(12)9-14(29(18)2)10-16-17(23)11-28-20(19(16)24)21(31)30-3-5-32-6-4-30/h7-9,11H,3-6,10H2,1-2H3	HMTHCBLYDBRGJR-UHFFFAOYSA-N	293098	US10106501, Example BE	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293098	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293098&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122934	381613381							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558811	Cc1cc(cc2n(C)c(Cc3c(Cl)cnc(C(=O)N4CCOCC4)c3Cl)cc12)C#N	InChI=1S/C22H20Cl2N4O2/c1-13-7-14(11-25)8-19-16(13)9-15(27(19)2)10-17-18(23)12-26-21(20(17)24)22(29)28-3-5-30-6-4-28/h7-9,12H,3-6,10H2,1-2H3	IEQANPCSJIDGPV-UHFFFAOYSA-N	293099	US10106501, Example BF	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293099	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293099&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123376	381613382							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558812	Cc1cc(cc2n(C)c(Cc3c(Cl)cnc(C(=O)N4CCC(CC4)C4COC4)c3Cl)cc12)C#N	InChI=1S/C26H26Cl2N4O2/c1-15-7-16(11-29)8-23-20(15)9-19(31(23)2)10-21-22(27)12-30-25(24(21)28)26(33)32-5-3-17(4-6-32)18-13-34-14-18/h7-9,12,17-18H,3-6,10,13-14H2,1-2H3	AMUURDPUDWOJRY-UHFFFAOYSA-N	293100	US10106501, Example BF-1	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293100	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293100&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123741	381613383							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558813	Cc1cc(cc2n(C)c(Cc3c(Cl)cnc(C(=O)N4CCC(O)CC4)c3Cl)cc12)C#N	InChI=1S/C23H22Cl2N4O2/c1-13-7-14(11-26)8-20-17(13)9-15(28(20)2)10-18-19(24)12-27-22(21(18)25)23(31)29-5-3-16(30)4-6-29/h7-9,12,16,30H,3-6,10H2,1-2H3	ZPSUSHXJUFDHDO-UHFFFAOYSA-N	293101	US10106501, Example BF-2	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293101	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293101&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123702	381613384							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558814	Cc1cc(cc2n(C)c(Cc3c(Cl)cnc(C(=O)N4CC(O)C4)c3Cl)cc12)C#N	InChI=1S/C21H18Cl2N4O2/c1-11-3-12(7-24)4-18-15(11)5-13(26(18)2)6-16-17(22)8-25-20(19(16)23)21(29)27-9-14(28)10-27/h3-5,8,14,28H,6,9-10H2,1-2H3	JWTOLFOPXGMWCD-UHFFFAOYSA-N	293102	US10106501, Example BF-3	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293102	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293102&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123783	381613385							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558815	Cc1cc(cc2n(C)c(Cc3c(Cl)cnc(C(=O)N4CCN(CC4)C4COC4)c3Cl)cc12)C#N	InChI=1S/C25H25Cl2N5O2/c1-15-7-16(11-28)8-22-19(15)9-17(30(22)2)10-20-21(26)12-29-24(23(20)27)25(33)32-5-3-31(4-6-32)18-13-34-14-18/h7-9,12,18H,3-6,10,13-14H2,1-2H3	ZAXHIRPHCFNTJJ-UHFFFAOYSA-N	293103	US10106501, Example BF-4	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293103	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293103&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123821	381613386							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558816	Cc1cc(cc2n(C)c(Cc3c(Cl)cnc(C(=O)N4CCC(O)C4)c3Cl)cc12)C#N	InChI=1S/C22H20Cl2N4O2/c1-12-5-13(9-25)6-19-16(12)7-14(27(19)2)8-17-18(23)10-26-21(20(17)24)22(30)28-4-3-15(29)11-28/h5-7,10,15,29H,3-4,8,11H2,1-2H3	VAZSYFCYUZPVOS-UHFFFAOYSA-N	293104	US10106501, Example BF-5	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293104	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293104&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123334	381613387							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558817	Cc1cc(cc2n(C)c(Cc3c(Cl)cnc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)cc12)C#N	InChI=1S/C25H24Cl2N4O3/c1-14-7-16(12-28)8-21-18(14)10-17(30(21)2)11-19-20(26)13-29-24(23(19)27)25(34)31-5-3-15(4-6-31)9-22(32)33/h7-8,10,13,15H,3-6,9,11H2,1-2H3,(H,32,33)	AYZSVVGFDBZATN-UHFFFAOYSA-N	293105	US10106501, Example BG	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293105	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293105&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123260	381613388							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558818	Cc1cc(cc2n(C)c(Cc3c(Cl)ncc(C(=O)N4CCOCC4)c3Cl)cc12)C#N	InChI=1S/C22H20Cl2N4O2/c1-13-7-14(11-25)8-19-16(13)9-15(27(19)2)10-17-20(23)18(12-26-21(17)24)22(29)28-3-5-30-6-4-28/h7-9,12H,3-6,10H2,1-2H3	PNNOLRDZSGKNLW-UHFFFAOYSA-N	293106	US10106501, Example BH	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293106	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293106&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124129579	381613389							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558819	Cc1cc(cc2n(C)c(Cc3c(Cl)cn(CCC(O)=O)c(=O)c3Cl)cc12)C(F)(F)F	InChI=1S/C20H17Cl2F3N2O3/c1-10-5-11(20(23,24)25)6-16-13(10)7-12(26(16)2)8-14-15(21)9-27(4-3-17(28)29)19(30)18(14)22/h5-7,9H,3-4,8H2,1-2H3,(H,28,29)	WGHHJTGRXQGJPQ-UHFFFAOYSA-N	293107	US10106501, Example BI	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293107	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293107&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123004	381613390							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558820	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C22H20Cl2F3N3O2/c1-12-9-13(22(25,26)27)10-17-20(12)28-18(29(17)2)11-15-16(23)4-3-14(19(15)24)21(31)30-5-7-32-8-6-30/h3-4,9-10H,5-8,11H2,1-2H3	ZGXLAYSVWJNCTN-UHFFFAOYSA-N	293108	US10106501, Example BJ	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293108	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293108&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123467	381613391							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558821	CNC(=O)[C@@H]1CCCN1C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl |r|	InChI=1S/C24H23Cl2F3N4O2/c1-12-9-13(24(27,28)29)10-18-21(12)31-19(32(18)3)11-15-16(25)7-6-14(20(15)26)23(35)33-8-4-5-17(33)22(34)30-2/h6-7,9-10,17H,4-5,8,11H2,1-3H3,(H,30,34)	HWTXVAQAZPBEMY-UHFFFAOYSA-N	293109	US10106501, Example BJ-1	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293109	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293109&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123580	381613392							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558822	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CC(CCO)C4)c3Cl)nc12)C(F)(F)F	InChI=1S/C23H22Cl2F3N3O2/c1-12-7-14(23(26,27)28)8-18-21(12)29-19(30(18)2)9-16-17(24)4-3-15(20(16)25)22(33)31-10-13(11-31)5-6-32/h3-4,7-8,13,32H,5-6,9-11H2,1-2H3	CPZQNYOJUZYOCW-UHFFFAOYSA-N	293110	US10106501, Example BJ-2	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293110	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293110&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123256	381613393							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558823	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CC(O)C4)c3Cl)nc12)C(F)(F)F	InChI=1S/C21H18Cl2F3N3O2/c1-10-5-11(21(24,25)26)6-16-19(10)27-17(28(16)2)7-14-15(22)4-3-13(18(14)23)20(31)29-8-12(30)9-29/h3-6,12,30H,7-9H2,1-2H3	JENNBNIJQFIDIC-UHFFFAOYSA-N	293111	US10106501, Example BJ-3	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293111	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293111&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122878	381613394							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558824	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CCO)C4)c3Cl)nc12)C(F)(F)F	InChI=1S/C24H24Cl2F3N3O2/c1-13-9-15(24(27,28)29)10-19-22(13)30-20(31(19)2)11-17-18(25)4-3-16(21(17)26)23(34)32-7-5-14(12-32)6-8-33/h3-4,9-10,14,33H,5-8,11-12H2,1-2H3	BSYZCJXDMGOKSV-UHFFFAOYSA-N	293112	US10106501, Example BJ-4	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293112	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293112&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123270	381613395							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558825	COCC1CCN(C1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C24H24Cl2F3N3O2/c1-13-8-15(24(27,28)29)9-19-22(13)30-20(31(19)2)10-17-18(25)5-4-16(21(17)26)23(33)32-7-6-14(11-32)12-34-3/h4-5,8-9,14H,6-7,10-12H2,1-3H3	ZCBLQANBDSGQDV-UHFFFAOYSA-N	293113	US10106501, Example BJ-5	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293113	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293113&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123959	381613396							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558826	COC1CCN(C1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C23H22Cl2F3N3O2/c1-12-8-13(23(26,27)28)9-18-21(12)29-19(30(18)2)10-16-17(24)5-4-15(20(16)25)22(32)31-7-6-14(11-31)33-3/h4-5,8-9,14H,6-7,10-11H2,1-3H3	CZRPREOUAIODEV-UHFFFAOYSA-N	293114	US10106501, Example BJ-6	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293114	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293114&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122968	381613397							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558827	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(O)C4)c3Cl)nc12)C(F)(F)F	InChI=1S/C22H20Cl2F3N3O2/c1-11-7-12(22(25,26)27)8-17-20(11)28-18(29(17)2)9-15-16(23)4-3-14(19(15)24)21(32)30-6-5-13(31)10-30/h3-4,7-8,13,31H,5-6,9-10H2,1-2H3	MMTUGXRFMKCSCA-UHFFFAOYSA-N	293115	US10106501, Example BJ-7	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293115	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293115&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123828	381613398							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558828	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC5(CCOC5)CC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C26H26Cl2F3N3O2/c1-15-11-16(26(29,30)31)12-20-23(15)32-21(33(20)2)13-18-19(27)4-3-17(22(18)28)24(35)34-8-5-25(6-9-34)7-10-36-14-25/h3-4,11-12H,5-10,13-14H2,1-2H3	ASPQITBAIOKZIR-UHFFFAOYSA-N	293116	US10106501, Example BJ-8	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293116	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293116&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123919	381613399							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558829	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC4)C(C)(C)O)c3Cl)nc12)C(F)(F)F	InChI=1S/C26H28Cl2F3N3O2/c1-14-11-16(26(29,30)31)12-20-23(14)32-21(33(20)4)13-18-19(27)6-5-17(22(18)28)24(35)34-9-7-15(8-10-34)25(2,3)36/h5-6,11-12,15,36H,7-10,13H2,1-4H3	INIUADKEXBVJOJ-UHFFFAOYSA-N	293117	US10106501, Example BJ-9	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293117	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293117&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123358	381613400							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558830	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC4)C(C)(C)CO)c3Cl)nc12)C(F)(F)F	InChI=1S/C27H30Cl2F3N3O2/c1-15-11-17(27(30,31)32)12-21-24(15)33-22(34(21)4)13-19-20(28)6-5-18(23(19)29)25(37)35-9-7-16(8-10-35)26(2,3)14-36/h5-6,11-12,16,36H,7-10,13-14H2,1-4H3	KRGXRXGWAFOAEV-UHFFFAOYSA-N	293118	US10106501, Example BJ-10	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293118	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293118&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123046	381613401							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558831	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CO)CC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C24H24Cl2F3N3O2/c1-13-9-15(24(27,28)29)10-19-22(13)30-20(31(19)2)11-17-18(25)4-3-16(21(17)26)23(34)32-7-5-14(12-33)6-8-32/h3-4,9-10,14,33H,5-8,11-12H2,1-2H3	FEYSSOZBEFZKFR-UHFFFAOYSA-N	293119	US10106501, Example BJ-11	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293119	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293119&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123905	381613402							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558832	CC(O)C1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C25H26Cl2F3N3O2/c1-13-10-16(25(28,29)30)11-20-23(13)31-21(32(20)3)12-18-19(26)5-4-17(22(18)27)24(35)33-8-6-15(7-9-33)14(2)34/h4-5,10-11,14-15,34H,6-9,12H2,1-3H3	GBXYDFKQBBXVQD-UHFFFAOYSA-N	293120	US10106501, Example BJ-12	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293120	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293120&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123931	381613403							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558833	COCC1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C25H26Cl2F3N3O2/c1-14-10-16(25(28,29)30)11-20-23(14)31-21(32(20)2)12-18-19(26)5-4-17(22(18)27)24(34)33-8-6-15(7-9-33)13-35-3/h4-5,10-11,15H,6-9,12-13H2,1-3H3	SJNFSZLWMULYHD-UHFFFAOYSA-N	293121	US10106501, Example BJ-13	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293121	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293121&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123872	381613404							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558834	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC(C)(C)O)CC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C27H30Cl2F3N3O2/c1-15-11-17(27(30,31)32)12-21-24(15)33-22(34(21)4)13-19-20(28)6-5-18(23(19)29)25(36)35-9-7-16(8-10-35)14-26(2,3)37/h5-6,11-12,16,37H,7-10,13-14H2,1-4H3	YILVIKMCFQFKNJ-UHFFFAOYSA-N	293122	US10106501, Example BJ-14	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293122	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293122&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123687	381613405							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558835	COC1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C24H24Cl2F3N3O2/c1-13-10-14(24(27,28)29)11-19-22(13)30-20(31(19)2)12-17-18(25)5-4-16(21(17)26)23(33)32-8-6-15(34-3)7-9-32/h4-5,10-11,15H,6-9,12H2,1-3H3	XWEHQAXZQSUIMP-UHFFFAOYSA-N	293123	US10106501, Example BJ-15	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293123	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293123&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123520	381613406							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558836	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CCO)CC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C25H26Cl2F3N3O2/c1-14-11-16(25(28,29)30)12-20-23(14)31-21(32(20)2)13-18-19(26)4-3-17(22(18)27)24(35)33-8-5-15(6-9-33)7-10-34/h3-4,11-12,15,34H,5-10,13H2,1-2H3	FVSAMDGBBNIVSG-UHFFFAOYSA-N	293124	US10106501, Example BJ-16	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293124	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293124&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123545	381613407							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558837	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC4)C4COC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C26H26Cl2F3N3O2/c1-14-9-17(26(29,30)31)10-21-24(14)32-22(33(21)2)11-19-20(27)4-3-18(23(19)28)25(35)34-7-5-15(6-8-34)16-12-36-13-16/h3-4,9-10,15-16H,5-8,11-13H2,1-2H3	XOMKPRVKZPSGCT-UHFFFAOYSA-N	293125	US10106501, Example BJ-17	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293125	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293125&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123681	381613408							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558838	COCCC1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C26H28Cl2F3N3O2/c1-15-12-17(26(29,30)31)13-21-24(15)32-22(33(21)2)14-19-20(27)5-4-18(23(19)28)25(35)34-9-6-16(7-10-34)8-11-36-3/h4-5,12-13,16H,6-11,14H2,1-3H3	RYVCVAARTVUMGP-UHFFFAOYSA-N	293126	US10106501, Example BJ-18	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293126	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293126&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122866	381613409							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558839	CC(O)CC1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C26H28Cl2F3N3O2/c1-14-10-17(26(29,30)31)12-21-24(14)32-22(33(21)3)13-19-20(27)5-4-18(23(19)28)25(36)34-8-6-16(7-9-34)11-15(2)35/h4-5,10,12,15-16,35H,6-9,11,13H2,1-3H3	ZJUSJCVXICYMRE-UHFFFAOYSA-N	293127	US10106501, Example BJ-19	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293127	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293127&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123696	381613410							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558840	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)NC4COC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C21H18Cl2F3N3O2/c1-10-5-11(21(24,25)26)6-16-19(10)28-17(29(16)2)7-14-15(22)4-3-13(18(14)23)20(30)27-12-8-31-9-12/h3-6,12H,7-9H2,1-2H3,(H,27,30)	UZKFYJMPKIUAQS-UHFFFAOYSA-N	293128	US10106501, Example BJ-20	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293128	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293128&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123803	381613411							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558841	COCCC1CN(C1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C24H24Cl2F3N3O2/c1-13-8-15(24(27,28)29)9-19-22(13)30-20(31(19)2)10-17-18(25)5-4-16(21(17)26)23(33)32-11-14(12-32)6-7-34-3/h4-5,8-9,14H,6-7,10-12H2,1-3H3	KURTYLJOFJVKET-UHFFFAOYSA-N	293129	US10106501, Example BJ-21	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293129	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293129&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123266	381613412							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558842	COC1CCC(CC1)NC(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl |(6.67,-6.01,;5.33,-6.78,;4,-6.01,;2.67,-6.78,;1.33,-6.01,;1.33,-4.47,;2.67,-3.7,;4,-4.47,;,-3.7,;-1.33,-4.47,;-1.33,-6.01,;-2.67,-3.7,;-4,-4.47,;-5.33,-3.7,;-5.33,-2.16,;-6.67,-1.39,;-4,-1.39,;-4,.15,;-2.67,.92,;-1.26,.3,;-.23,1.44,;1.31,1.44,;2.08,.11,;2.08,2.78,;1.31,4.11,;-.23,4.11,;-1,2.78,;-2.51,2.46,;-3.6,3.54,;2.08,5.44,;.75,6.21,;3.41,4.67,;2.85,6.78,;-2.67,-2.16,;-1.33,-1.39,)|	InChI=1S/C25H26Cl2F3N3O2/c1-13-10-14(25(28,29)30)11-20-23(13)32-21(33(20)2)12-18-19(26)9-8-17(22(18)27)24(34)31-15-4-6-16(35-3)7-5-15/h8-11,15-16H,4-7,12H2,1-3H3,(H,31,34)	ZHVPGMBFIGOXOT-UHFFFAOYSA-N	293130	US10106501, Example BJ-22	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293130	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293130&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123120	381613413							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558843	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)NC4CCC(O)CC4)c3Cl)nc12)C(F)(F)F |(2.75,.11,;1.98,1.44,;2.75,2.78,;1.98,4.11,;.44,4.11,;-.33,2.78,;-1.84,2.46,;-2.93,3.54,;-2,.92,;-3.33,.15,;-3.33,-1.39,;-4.67,-2.16,;-6,-1.39,;-4.67,-3.7,;-3.33,-4.47,;-2,-3.7,;-.67,-4.47,;-.67,-6.01,;.67,-3.7,;2,-4.47,;2,-6.01,;3.33,-6.78,;4.67,-6.01,;6,-6.78,;4.67,-4.47,;3.33,-3.7,;-2,-2.16,;-.67,-1.39,;-.59,.3,;.44,1.44,;2.75,5.44,;1.98,6.78,;4.29,5.44,;3.52,6.78,)|	InChI=1S/C24H24Cl2F3N3O2/c1-12-9-13(24(27,28)29)10-19-22(12)31-20(32(19)2)11-17-18(25)8-7-16(21(17)26)23(34)30-14-3-5-15(33)6-4-14/h7-10,14-15,33H,3-6,11H2,1-2H3,(H,30,34)	KQODVWLJPSGJGD-UHFFFAOYSA-N	293131	US10106501, Example BJ-24	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293131	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293131&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123899	381613414							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558844	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC5(COC5)CC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C25H24Cl2F3N3O2/c1-14-9-15(25(28,29)30)10-19-22(14)31-20(32(19)2)11-17-18(26)4-3-16(21(17)27)23(34)33-7-5-24(6-8-33)12-35-13-24/h3-4,9-10H,5-8,11-13H2,1-2H3	ZVMOBKCNWUDOII-UHFFFAOYSA-N	293132	US10106501, Example BJ-25	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293132	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293132&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123055	381613415							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558845	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)NCC4CCCO4)c3Cl)nc12)C(F)(F)F	InChI=1S/C23H22Cl2F3N3O2/c1-12-8-13(23(26,27)28)9-18-21(12)30-19(31(18)2)10-16-17(24)6-5-15(20(16)25)22(32)29-11-14-4-3-7-33-14/h5-6,8-9,14H,3-4,7,10-11H2,1-2H3,(H,29,32)	SBNCNMHYMMTSIW-UHFFFAOYSA-N	293133	US10106501, Example BJ-26	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293133	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293133&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123807	381613416							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558846	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CC(CO)C4)c3Cl)nc12)C(F)(F)F	InChI=1S/C22H20Cl2F3N3O2/c1-11-5-13(22(25,26)27)6-17-20(11)28-18(29(17)2)7-15-16(23)4-3-14(19(15)24)21(32)30-8-12(9-30)10-31/h3-6,12,31H,7-10H2,1-2H3	UCIVLZWQFNSMKV-UHFFFAOYSA-N	293134	US10106501, Example BJ-27	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293134	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293134&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123238	381613417							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558847	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CC5(COC5)C4)c3Cl)nc12)C(F)(F)F	InChI=1S/C23H20Cl2F3N3O2/c1-12-5-13(23(26,27)28)6-17-20(12)29-18(30(17)2)7-15-16(24)4-3-14(19(15)25)21(32)31-8-22(9-31)10-33-11-22/h3-6H,7-11H2,1-2H3	QQHFQWQIFNHAIY-UHFFFAOYSA-N	293135	US10106501, Example BJ-28	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293135	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293135&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123161	381613418							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558848	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCCC(O)C4)c3Cl)nc12)C(F)(F)F	InChI=1S/C23H22Cl2F3N3O2/c1-12-8-13(23(26,27)28)9-18-21(12)29-19(30(18)2)10-16-17(24)6-5-15(20(16)25)22(33)31-7-3-4-14(32)11-31/h5-6,8-9,14,32H,3-4,7,10-11H2,1-2H3	DTIKZBNBNLWWJX-UHFFFAOYSA-N	293136	US10106501, Example BJ-29	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293136	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293136&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122886	381613419							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558849	CN(C)C1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C25H27Cl2F3N4O/c1-14-11-15(25(28,29)30)12-20-23(14)31-21(33(20)4)13-18-19(26)6-5-17(22(18)27)24(35)34-9-7-16(8-10-34)32(2)3/h5-6,11-12,16H,7-10,13H2,1-4H3	CPDIYNBCDGHCMB-UHFFFAOYSA-N	293137	US10106501, Example BJ-30	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293137	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293137&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123922	381613420							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558850	CC1CN(CCN1C)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C24H25Cl2F3N4O/c1-13-9-15(24(27,28)29)10-19-22(13)30-20(32(19)4)11-17-18(25)6-5-16(21(17)26)23(34)33-8-7-31(3)14(2)12-33/h5-6,9-10,14H,7-8,11-12H2,1-4H3	YAHFXWNPNDVLIY-UHFFFAOYSA-N	293138	US10106501, Example BJ-31	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293138	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293138&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123697	381613421							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558851	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCN(CCO)CC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C24H25Cl2F3N4O2/c1-14-11-15(24(27,28)29)12-19-22(14)30-20(31(19)2)13-17-18(25)4-3-16(21(17)26)23(35)33-7-5-32(6-8-33)9-10-34/h3-4,11-12,34H,5-10,13H2,1-2H3	WXHOBHVEAONADY-UHFFFAOYSA-N	293139	US10106501, Example BJ-32	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293139	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293139&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123677	381613422							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558852	CC(O)CN1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C25H27Cl2F3N4O2/c1-14-10-16(25(28,29)30)11-20-23(14)31-21(32(20)3)12-18-19(26)5-4-17(22(18)27)24(36)34-8-6-33(7-9-34)13-15(2)35/h4-5,10-11,15,35H,6-9,12-13H2,1-3H3	HHHSIACKCWEERS-UHFFFAOYSA-N	293140	US10106501, Example BJ-33	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293140	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293140&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123764	381613423							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558853	CN(C)C1CN(C1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C23H23Cl2F3N4O/c1-12-7-13(23(26,27)28)8-18-21(12)29-19(31(18)4)9-16-17(24)6-5-15(20(16)25)22(33)32-10-14(11-32)30(2)3/h5-8,14H,9-11H2,1-4H3	ZTCBLVNMUVGEIG-UHFFFAOYSA-N	293141	US10106501, Example BJ-34	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293141	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293141&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123350	381613424							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558854	COCCN1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C25H27Cl2F3N4O2/c1-15-12-16(25(28,29)30)13-20-23(15)31-21(32(20)2)14-18-19(26)5-4-17(22(18)27)24(35)34-8-6-33(7-9-34)10-11-36-3/h4-5,12-13H,6-11,14H2,1-3H3	YSSSGXYCEAMDDZ-UHFFFAOYSA-N	293142	US10106501, Example BJ-35	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293142	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293142&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122850	381613425							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558855	CC(F)CN1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C25H26Cl2F4N4O/c1-14-10-16(25(29,30)31)11-20-23(14)32-21(33(20)3)12-18-19(26)5-4-17(22(18)27)24(36)35-8-6-34(7-9-35)13-15(2)28/h4-5,10-11,15H,6-9,12-13H2,1-3H3	PXVWSWYWFOFINC-UHFFFAOYSA-N	293143	US10106501, Example BJ-36	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293143	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293143&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123862	381613426							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558856	COCC1CN(C1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C23H22Cl2F3N3O2/c1-12-6-14(23(26,27)28)7-18-21(12)29-19(30(18)2)8-16-17(24)5-4-15(20(16)25)22(32)31-9-13(10-31)11-33-3/h4-7,13H,8-11H2,1-3H3	JTNMYOADYOOLPU-UHFFFAOYSA-N	293144	US10106501, Example BJ-37	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293144	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293144&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123451	381613427							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558857	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCN(CC4)C4COC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C25H25Cl2F3N4O2/c1-14-9-15(25(28,29)30)10-20-23(14)31-21(32(20)2)11-18-19(26)4-3-17(22(18)27)24(35)34-7-5-33(6-8-34)16-12-36-13-16/h3-4,9-10,16H,5-8,11-13H2,1-2H3	SBKSOZYQQYNDGF-UHFFFAOYSA-N	293145	US10106501, Example BJ-38	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293145	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293145&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123446	381613428							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558858	CN1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C23H23Cl2F3N4O/c1-13-10-14(23(26,27)28)11-18-21(13)29-19(31(18)3)12-16-17(24)5-4-15(20(16)25)22(33)32-8-6-30(2)7-9-32/h4-5,10-11H,6-9,12H2,1-3H3	AZBDLCUUPSJITD-UHFFFAOYSA-N	293146	US10106501, Example BJ-39	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293146	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293146&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123876	381613429							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558859	CC(C)N1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C25H27Cl2F3N4O/c1-14(2)33-7-9-34(10-8-33)24(35)17-5-6-19(26)18(22(17)27)13-21-31-23-15(3)11-16(25(28,29)30)12-20(23)32(21)4/h5-6,11-12,14H,7-10,13H2,1-4H3	CXLRCFVEZBLIAD-UHFFFAOYSA-N	293147	US10106501, Example BJ-40	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293147	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293147&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123473	381613430							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558860	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCN(CC(F)(F)F)CC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C24H22Cl2F6N4O/c1-13-9-14(24(30,31)32)10-18-21(13)33-19(34(18)2)11-16-17(25)4-3-15(20(16)26)22(37)36-7-5-35(6-8-36)12-23(27,28)29/h3-4,9-10H,5-8,11-12H2,1-2H3	QIOCFVDAVXXQAG-UHFFFAOYSA-N	293148	US10106501, Example BJ-41	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293148	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293148&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123201	381613431							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558861	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCN(CC5CC5)CC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C26H27Cl2F3N4O/c1-15-11-17(26(29,30)31)12-21-24(15)32-22(33(21)2)13-19-20(27)6-5-18(23(19)28)25(36)35-9-7-34(8-10-35)14-16-3-4-16/h5-6,11-12,16H,3-4,7-10,13-14H2,1-2H3	XSLHBZNHVOEJRJ-UHFFFAOYSA-N	293149	US10106501, Example BJ-42	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293149	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293149&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123859	381613432							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558862	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCCN(CCO)CC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C25H27Cl2F3N4O2/c1-15-12-16(25(28,29)30)13-20-23(15)31-21(32(20)2)14-18-19(26)5-4-17(22(18)27)24(36)34-7-3-6-33(8-9-34)10-11-35/h4-5,12-13,35H,3,6-11,14H2,1-2H3	ASDMFICMVKQBIO-UHFFFAOYSA-N	293150	US10106501, Example BJ-44::US10106501, Example BJ-43	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293150	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293150&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123658	381613433							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558863	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCCN(CCO)CC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C25H27Cl2F3N4O2/c1-15-12-16(25(28,29)30)13-20-23(15)31-21(32(20)2)14-18-19(26)5-4-17(22(18)27)24(36)34-7-3-6-33(8-9-34)10-11-35/h4-5,12-13,35H,3,6-11,14H2,1-2H3	ASDMFICMVKQBIO-UHFFFAOYSA-N	293150	US10106501, Example BJ-44::US10106501, Example BJ-43	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293150	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293150&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123658	381613433							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558864	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC4)C(O)=O)c3Cl)nc12)C(F)(F)F	InChI=1S/C24H22Cl2F3N3O3/c1-12-9-14(24(27,28)29)10-18-21(12)30-19(31(18)2)11-16-17(25)4-3-15(20(16)26)22(33)32-7-5-13(6-8-32)23(34)35/h3-4,9-10,13H,5-8,11H2,1-2H3,(H,34,35)	DCUQVBICPAMUBW-UHFFFAOYSA-N	293152	US10106501, Example BK	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293152	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293152&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123278	381613434							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558865	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4C[C@H]5[C@@H](C4)[C@@H]5C(O)=O)c3Cl)nc12)C(F)(F)F |r|	InChI=1S/C24H20Cl2F3N3O3/c1-10-5-11(24(27,28)29)6-17-21(10)30-18(31(17)2)7-13-16(25)4-3-12(20(13)26)22(33)32-8-14-15(9-32)19(14)23(34)35/h3-6,14-15,19H,7-9H2,1-2H3,(H,34,35)	UWIISQJFSKTEHJ-UHFFFAOYSA-N	293153	US10106501, Example BL	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293153	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293153&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123181	381613435							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558866	CC1CN(CCC1C(O)=O)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C25H24Cl2F3N3O3/c1-12-8-14(25(28,29)30)9-19-22(12)31-20(32(19)3)10-17-18(26)5-4-16(21(17)27)23(34)33-7-6-15(24(35)36)13(2)11-33/h4-5,8-9,13,15H,6-7,10-11H2,1-3H3,(H,35,36)	SOQSMABJHMKXEW-UHFFFAOYSA-N	293154	US10106501, Example BM	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293154	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293154&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123048	381613436							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558867	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CCO)CC4)c3Cl)nc12)C#N	InChI=1S/C25H26Cl2N4O2/c1-15-11-17(14-28)12-21-24(15)29-22(30(21)2)13-19-20(26)4-3-18(23(19)27)25(33)31-8-5-16(6-9-31)7-10-32/h3-4,11-12,16,32H,5-10,13H2,1-2H3	KAFSTANJQIJXOA-UHFFFAOYSA-N	293155	US10106501, Example BN	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293155	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293155&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123709	381613437							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558868	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N[C@@H]4CC[C@H](O)CC4)c3Cl)nc12)C#N |r,wU:19.18,22.22,(2.75,.11,;1.98,1.44,;2.75,2.78,;1.98,4.11,;.44,4.11,;-.33,2.78,;-1.84,2.46,;-2.93,3.54,;-2,.92,;-3.33,.15,;-3.33,-1.39,;-4.67,-2.16,;-6,-1.39,;-4.67,-3.7,;-3.33,-4.47,;-2,-3.7,;-.67,-4.47,;-.67,-6.01,;.67,-3.7,;2,-4.47,;2,-6.01,;3.33,-6.78,;4.67,-6.01,;6,-6.78,;4.67,-4.47,;3.33,-3.7,;-2,-2.16,;-.67,-1.39,;-.59,.3,;.44,1.44,;2.75,5.44,;3.52,6.78,)|	InChI=1S/C24H24Cl2N4O2/c1-13-9-14(12-27)10-20-23(13)29-21(30(20)2)11-18-19(25)8-7-17(22(18)26)24(32)28-15-3-5-16(31)6-4-15/h7-10,15-16,31H,3-6,11H2,1-2H3,(H,28,32)	NMLCEQVIHKMFLE-UHFFFAOYSA-N	293156	US10106501, Example BN-2	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293156	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293156&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123085	381613438							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558869	COCCC1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C#N)c1Cl	InChI=1S/C26H28Cl2N4O2/c1-16-12-18(15-29)13-22-25(16)30-23(31(22)2)14-20-21(27)5-4-19(24(20)28)26(33)32-9-6-17(7-10-32)8-11-34-3/h4-5,12-13,17H,6-11,14H2,1-3H3	ADOPNMPZHQCNRG-UHFFFAOYSA-N	293157	US10106501, Example BN-3	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293157	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293157&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123020	381613439							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558870	COCC1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C#N)c1Cl	InChI=1S/C25H26Cl2N4O2/c1-15-10-17(13-28)11-21-24(15)29-22(30(21)2)12-19-20(26)5-4-18(23(19)27)25(32)31-8-6-16(7-9-31)14-33-3/h4-5,10-11,16H,6-9,12,14H2,1-3H3	QSXOWPHMYNNBJX-UHFFFAOYSA-N	293158	US10106501, Example BN-4	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293158	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293158&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123921	381613440							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558871	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CO)CC4)c3Cl)nc12)C#N	InChI=1S/C24H24Cl2N4O2/c1-14-9-16(12-27)10-20-23(14)28-21(29(20)2)11-18-19(25)4-3-17(22(18)26)24(32)30-7-5-15(13-31)6-8-30/h3-4,9-10,15,31H,5-8,11,13H2,1-2H3	XMEDWJNGOVPPAY-UHFFFAOYSA-N	293159	US10106501, Example BN-5	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293159	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293159&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122883	381613441							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558872	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC4)C(C)(C)CO)c3Cl)nc12)C#N	InChI=1S/C27H30Cl2N4O2/c1-16-11-17(14-30)12-22-25(16)31-23(32(22)4)13-20-21(28)6-5-19(24(20)29)26(35)33-9-7-18(8-10-33)27(2,3)15-34/h5-6,11-12,18,34H,7-10,13,15H2,1-4H3	XCIJSNXFEHMNJM-UHFFFAOYSA-N	293160	US10106501, Example BN-6	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293160	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293160&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122828	381613442							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558873	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC4)C(C)(C)O)c3Cl)nc12)C#N	InChI=1S/C26H28Cl2N4O2/c1-15-11-16(14-29)12-21-24(15)30-22(31(21)4)13-19-20(27)6-5-18(23(19)28)25(33)32-9-7-17(8-10-32)26(2,3)34/h5-6,11-12,17,34H,7-10,13H2,1-4H3	HCCVRQXXUYETLH-UHFFFAOYSA-N	293161	US10106501, Example BN-7	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293161	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293161&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123319	381613443							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558874	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC5(CCOC5)CC4)c3Cl)nc12)C#N	InChI=1S/C26H26Cl2N4O2/c1-16-11-17(14-29)12-21-24(16)30-22(31(21)2)13-19-20(27)4-3-18(23(19)28)25(33)32-8-5-26(6-9-32)7-10-34-15-26/h3-4,11-12H,5-10,13,15H2,1-2H3	NINLGKAEMQZDCV-UHFFFAOYSA-N	293162	US10106501, Example BN-8	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293162	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293162&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122961	381613444							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558875	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCN(CCO)CC4)c3Cl)nc12)C#N	InChI=1S/C24H25Cl2N5O2/c1-15-11-16(14-27)12-20-23(15)28-21(29(20)2)13-18-19(25)4-3-17(22(18)26)24(33)31-7-5-30(6-8-31)9-10-32/h3-4,11-12,32H,5-10,13H2,1-2H3	NRABOHUHXBHDNX-UHFFFAOYSA-N	293163	US10106501, Example BN-9	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293163	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293163&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123378	381613445							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558876	CC(F)CN1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C#N)c1Cl	InChI=1S/C25H26Cl2FN5O/c1-15-10-17(13-29)11-21-24(15)30-22(31(21)3)12-19-20(26)5-4-18(23(19)27)25(34)33-8-6-32(7-9-33)14-16(2)28/h4-5,10-11,16H,6-9,12,14H2,1-3H3	BYTVOZKBYIOZDV-UHFFFAOYSA-N	293164	US10106501, Example BN-10	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293164	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293164&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123793	381613446							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558877	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCN(CC4)C4COC4)c3Cl)nc12)C#N	InChI=1S/C25H25Cl2N5O2/c1-15-9-16(12-28)10-21-24(15)29-22(30(21)2)11-19-20(26)4-3-18(23(19)27)25(33)32-7-5-31(6-8-32)17-13-34-14-17/h3-4,9-10,17H,5-8,11,13-14H2,1-2H3	UUYDCQBEEACKRA-UHFFFAOYSA-N	293165	US10106501, Example BN-11	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293165	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293165&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122913	381613447							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558878	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC4)C4COC4)c3Cl)nc12)C#N	InChI=1S/C26H26Cl2N4O2/c1-15-9-16(12-29)10-22-25(15)30-23(31(22)2)11-20-21(27)4-3-19(24(20)28)26(33)32-7-5-17(6-8-32)18-13-34-14-18/h3-4,9-10,17-18H,5-8,11,13-14H2,1-2H3	MFPQGYQWOPMFEN-UHFFFAOYSA-N	293166	US10106501, Example BN-12	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293166	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293166&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123282	381613448							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558879	COC1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C#N)c1Cl	InChI=1S/C24H24Cl2N4O2/c1-14-10-15(13-27)11-20-23(14)28-21(29(20)2)12-18-19(25)5-4-17(22(18)26)24(31)30-8-6-16(32-3)7-9-30/h4-5,10-11,16H,6-9,12H2,1-3H3	HWKNDRMXIDSYII-UHFFFAOYSA-N	293167	US10106501, Example BN-13	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293167	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293167&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123900	381613449							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558880	CN(C)C1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C#N)c1Cl	InChI=1S/C25H27Cl2N5O/c1-15-11-16(14-28)12-21-24(15)29-22(31(21)4)13-19-20(26)6-5-18(23(19)27)25(33)32-9-7-17(8-10-32)30(2)3/h5-6,11-12,17H,7-10,13H2,1-4H3	UVHWRXDUABEGKD-UHFFFAOYSA-N	293168	US10106501, Example BN-14	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293168	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293168&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123533	381613450							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558881	COCCN1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C#N)c1Cl	InChI=1S/C25H27Cl2N5O2/c1-16-12-17(15-28)13-21-24(16)29-22(30(21)2)14-19-20(26)5-4-18(23(19)27)25(33)32-8-6-31(7-9-32)10-11-34-3/h4-5,12-13H,6-11,14H2,1-3H3	BKTFREXDGSVDPN-UHFFFAOYSA-N	293169	US10106501, Example BN-15	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293169	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293169&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123337	381613451							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558882	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC(C)(C)O)CC4)c3Cl)nc12)C#N	InChI=1S/C27H30Cl2N4O2/c1-16-11-18(15-30)12-22-25(16)31-23(32(22)4)13-20-21(28)6-5-19(24(20)29)26(34)33-9-7-17(8-10-33)14-27(2,3)35/h5-6,11-12,17,35H,7-10,13-14H2,1-4H3	WXLHVLXAFOLGKR-UHFFFAOYSA-N	293170	US10106501, Example BN-16	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293170	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293170&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123457	381613452							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558883	CN1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C#N)c1Cl	InChI=1S/C23H23Cl2N5O/c1-14-10-15(13-26)11-19-22(14)27-20(29(19)3)12-17-18(24)5-4-16(21(17)25)23(31)30-8-6-28(2)7-9-30/h4-5,10-11H,6-9,12H2,1-3H3	WRVWRSCNWDPPSX-UHFFFAOYSA-N	293171	US10106501, Example BN-17	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293171	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293171&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123230	381613453							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558884	Cc1cc(C)c2nc(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)n(C)c2c1	InChI=1S/C22H23Cl2N3O2/c1-13-10-14(2)21-18(11-13)26(3)19(25-21)12-16-17(23)5-4-15(20(16)24)22(28)27-6-8-29-9-7-27/h4-5,10-11H,6-9,12H2,1-3H3	YAJKHVOHMVJBKR-UHFFFAOYSA-N	293172	US10106501, Example BO	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293172	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293172&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123425	381613454							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558885	Cc1cc(cc2nc(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)n(C)c12)C(F)(F)F	InChI=1S/C22H20Cl2F3N3O2/c1-12-9-13(22(25,26)27)10-17-20(12)29(2)18(28-17)11-15-16(23)4-3-14(19(15)24)21(31)30-5-7-32-8-6-30/h3-4,9-10H,5-8,11H2,1-2H3	IJLCXVFUEMBQHX-UHFFFAOYSA-N	293173	US10106501, Example BP	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293173	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293173&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122827	381613455							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558886	Cc1ccc(C(=O)N2CCOCC2)c(C)c1Cc1nc2c(C)cc(Br)cc2n1C	InChI=1S/C23H26BrN3O2/c1-14-5-6-18(23(28)27-7-9-29-10-8-27)16(3)19(14)13-21-25-22-15(2)11-17(24)12-20(22)26(21)4/h5-6,11-12H,7-10,13H2,1-4H3	PRJMNBFSAUWSPI-UHFFFAOYSA-N	293174	US10106501, Example BR	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293174	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293174&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123539	381613456							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558887	Cc1cc(cc2n(C)c(nc12)C(=O)c1c(Cl)ccc(C(=O)N2CCOCC2)c1Cl)C(F)(F)F	InChI=1S/C22H18Cl2F3N3O3/c1-11-9-12(22(25,26)27)10-15-18(11)28-20(29(15)2)19(31)16-14(23)4-3-13(17(16)24)21(32)30-5-7-33-8-6-30/h3-4,9-10H,5-8H2,1-2H3	IWRMJEWAKRDUPX-UHFFFAOYSA-N	293175	US10106501, Example BS	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293175	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293175&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123251	381613457							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558888	Cc1cc(cc2n(C)c(nc12)C(=O)c1c(Cl)ccc(C(=O)N2CCOCC2)c1Cl)C(N)=O	InChI=1S/C22H20Cl2N4O4/c1-11-9-12(20(25)30)10-15-18(11)26-21(27(15)2)19(29)16-14(23)4-3-13(17(16)24)22(31)28-5-7-32-8-6-28/h3-4,9-10H,5-8H2,1-2H3,(H2,25,30)	PSYSJDIGJNJFQD-UHFFFAOYSA-N	293176	US10106501, Example BT	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293176	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293176&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123076	381613458							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558889	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C25H24Cl2F3N3O3/c1-13-9-15(25(28,29)30)11-19-23(13)31-20(32(19)2)12-17-18(26)4-3-16(22(17)27)24(36)33-7-5-14(6-8-33)10-21(34)35/h3-4,9,11,14H,5-8,10,12H2,1-2H3,(H,34,35)	UUVXZOKBZLDOES-UHFFFAOYSA-N	293177	US10106501, Example BU	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293177	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293177&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123716	381613459							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558890	COCCC1CCN(Cc2ccc(Cl)c(Cc3nc4c(C)cc(cc4n3C)C(F)(F)F)c2Cl)CC1	InChI=1S/C26H30Cl2F3N3O/c1-16-12-19(26(29,30)31)13-22-25(16)32-23(33(22)2)14-20-21(27)5-4-18(24(20)28)15-34-9-6-17(7-10-34)8-11-35-3/h4-5,12-13,17H,6-11,14-15H2,1-3H3	LXSALNYXFFJBBC-UHFFFAOYSA-N	293178	US10106501, Example BW	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293178	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293178&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123910	381613460							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558891	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(CN4CCC(CC4)C4COC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C26H28Cl2F3N3O/c1-15-9-19(26(29,30)31)10-22-25(15)32-23(33(22)2)11-20-21(27)4-3-17(24(20)28)12-34-7-5-16(6-8-34)18-13-35-14-18/h3-4,9-10,16,18H,5-8,11-14H2,1-2H3	RYKZRIOGOSSZGZ-UHFFFAOYSA-N	293179	US10106501, Example BW-1	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293179	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293179&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123090	381613461							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558892	COC1CCN(Cc2ccc(Cl)c(Cc3nc4c(C)cc(cc4n3C)C(F)(F)F)c2Cl)CC1	InChI=1S/C24H26Cl2F3N3O/c1-14-10-16(24(27,28)29)11-20-23(14)30-21(31(20)2)12-18-19(25)5-4-15(22(18)26)13-32-8-6-17(33-3)7-9-32/h4-5,10-11,17H,6-9,12-13H2,1-3H3	NAFHXVFRFWGNOI-UHFFFAOYSA-N	293180	US10106501, Example BW-2	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293180	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293180&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123678	381613462							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558893	COCC1CCN(Cc2ccc(Cl)c(Cc3nc4c(C)cc(cc4n3C)C(F)(F)F)c2Cl)CC1	InChI=1S/C25H28Cl2F3N3O/c1-15-10-18(25(28,29)30)11-21-24(15)31-22(32(21)2)12-19-20(26)5-4-17(23(19)27)13-33-8-6-16(7-9-33)14-34-3/h4-5,10-11,16H,6-9,12-14H2,1-3H3	AXDAJKRREPAQMZ-UHFFFAOYSA-N	293181	US10106501, Example BW-3	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293181	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293181&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123607	381613463							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558894	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(CN4CCC(O)CC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C23H24Cl2F3N3O/c1-13-9-15(23(26,27)28)10-19-22(13)29-20(30(19)2)11-17-18(24)4-3-14(21(17)25)12-31-7-5-16(32)6-8-31/h3-4,9-10,16,32H,5-8,11-12H2,1-2H3	UGZUQOCLPXTMPK-UHFFFAOYSA-N	293182	US10106501, Example BW-4	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293182	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293182&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123325	381613464							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558895	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(CN4CCCC(O)C4)c3Cl)nc12)C(F)(F)F	InChI=1S/C23H24Cl2F3N3O/c1-13-8-15(23(26,27)28)9-19-22(13)29-20(30(19)2)10-17-18(24)6-5-14(21(17)25)11-31-7-3-4-16(32)12-31/h5-6,8-9,16,32H,3-4,7,10-12H2,1-2H3	ACBGZXSDEAQGCV-UHFFFAOYSA-N	293183	US10106501, Example BW-5	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293183	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293183&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123535	381613465							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558896	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(CN4CCC(CC4)C(C)(C)CO)c3Cl)nc12)C(F)(F)F	InChI=1S/C27H32Cl2F3N3O/c1-16-11-19(27(30,31)32)12-22-25(16)33-23(34(22)4)13-20-21(28)6-5-17(24(20)29)14-35-9-7-18(8-10-35)26(2,3)15-36/h5-6,11-12,18,36H,7-10,13-15H2,1-4H3	GLYRVZJFVDBJFC-UHFFFAOYSA-N	293184	US10106501, Example BW-6	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293184	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293184&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123528	381613466							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558897	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(CN4CCC(CC4)C(C)(C)O)c3Cl)nc12)C(F)(F)F	InChI=1S/C26H30Cl2F3N3O/c1-15-11-18(26(29,30)31)12-21-24(15)32-22(33(21)4)13-19-20(27)6-5-16(23(19)28)14-34-9-7-17(8-10-34)25(2,3)35/h5-6,11-12,17,35H,7-10,13-14H2,1-4H3	VCJFXQOJBAGCLA-UHFFFAOYSA-N	293185	US10106501, Example BW-7	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293185	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293185&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123206	381613467							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558898	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(CN4CCC5(CCOC5)CC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C26H28Cl2F3N3O/c1-16-11-18(26(29,30)31)12-21-24(16)32-22(33(21)2)13-19-20(27)4-3-17(23(19)28)14-34-8-5-25(6-9-34)7-10-35-15-25/h3-4,11-12H,5-10,13-15H2,1-2H3	GCVCSQADLKKYAW-UHFFFAOYSA-N	293186	US10106501, Example BW-8	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293186	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293186&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123579	381613468							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558899	COCCN1CCN(Cc2ccc(Cl)c(Cc3nc4c(C)cc(cc4n3C)C(F)(F)F)c2Cl)CC1	InChI=1S/C25H29Cl2F3N4O/c1-16-12-18(25(28,29)30)13-21-24(16)31-22(32(21)2)14-19-20(26)5-4-17(23(19)27)15-34-8-6-33(7-9-34)10-11-35-3/h4-5,12-13H,6-11,14-15H2,1-3H3	BWXYAXNFRWKAQG-UHFFFAOYSA-N	293187	US10106501, Example BW-9	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293187	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293187&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123721	381613469							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558900	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(CN4CCOCC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C22H22Cl2F3N3O/c1-13-9-15(22(25,26)27)10-18-21(13)28-19(29(18)2)11-16-17(23)4-3-14(20(16)24)12-30-5-7-31-8-6-30/h3-4,9-10H,5-8,11-12H2,1-2H3	OEXHQPZFSVCZFX-UHFFFAOYSA-N	293188	US10106501, Example BW-10	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293188	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293188&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122954	381613470							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558901	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(CN4CCC(CCO)CC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C25H28Cl2F3N3O/c1-15-11-18(25(28,29)30)12-21-24(15)31-22(32(21)2)13-19-20(26)4-3-17(23(19)27)14-33-8-5-16(6-9-33)7-10-34/h3-4,11-12,16,34H,5-10,13-14H2,1-2H3	PSYWRHRLZPZMEK-UHFFFAOYSA-N	293189	US10106501, Example BW-11	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293189	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293189&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123374	381613471							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558902	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(CN4CCC(CC(C)(C)O)CC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C27H32Cl2F3N3O/c1-16-11-19(27(30,31)32)12-22-25(16)33-23(34(22)4)13-20-21(28)6-5-18(24(20)29)15-35-9-7-17(8-10-35)14-26(2,3)36/h5-6,11-12,17,36H,7-10,13-15H2,1-4H3	JVJIHJVUDKMTAV-UHFFFAOYSA-N	293190	US10106501, Example BW-12	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293190	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293190&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123205	381613472							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558903	CC(O)C1CCN(Cc2ccc(Cl)c(Cc3nc4c(C)cc(cc4n3C)C(F)(F)F)c2Cl)CC1	InChI=1S/C25H28Cl2F3N3O/c1-14-10-18(25(28,29)30)11-21-24(14)31-22(32(21)3)12-19-20(26)5-4-17(23(19)27)13-33-8-6-16(7-9-33)15(2)34/h4-5,10-11,15-16,34H,6-9,12-13H2,1-3H3	YPSRCPRJHZJGKE-UHFFFAOYSA-N	293191	US10106501, Example BW-13	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293191	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293191&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122912	381613473							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558904	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(CN4CCC(CO)CC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C24H26Cl2F3N3O/c1-14-9-17(24(27,28)29)10-20-23(14)30-21(31(20)2)11-18-19(25)4-3-16(22(18)26)12-32-7-5-15(13-33)6-8-32/h3-4,9-10,15,33H,5-8,11-13H2,1-2H3	PDDFDFRWBPAROI-UHFFFAOYSA-N	293192	US10106501, Example BW-14	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293192	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293192&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123536	381613474							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558905	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(CN4CCN(CC(F)(F)F)CC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C24H24Cl2F6N4/c1-14-9-16(24(30,31)32)10-19-22(14)33-20(34(19)2)11-17-18(25)4-3-15(21(17)26)12-35-5-7-36(8-6-35)13-23(27,28)29/h3-4,9-10H,5-8,11-13H2,1-2H3	GLXROVPBTIMOCP-UHFFFAOYSA-N	293193	US10106501, Example BW-15	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293193	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293193&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122887	381613475							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558906	CN(C)C1CCN(Cc2ccc(Cl)c(Cc3nc4c(C)cc(cc4n3C)C(F)(F)F)c2Cl)CC1	InChI=1S/C25H29Cl2F3N4/c1-15-11-17(25(28,29)30)12-21-24(15)31-22(33(21)4)13-19-20(26)6-5-16(23(19)27)14-34-9-7-18(8-10-34)32(2)3/h5-6,11-12,18H,7-10,13-14H2,1-4H3	OVUGGKPELHAZMI-UHFFFAOYSA-N	293194	US10106501, Example BW-16	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293194	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293194&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123188	381613476							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558907	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(CN4CCCC(C)(O)C4)c3Cl)nc12)C(F)(F)F	InChI=1S/C24H26Cl2F3N3O/c1-14-9-16(24(27,28)29)10-19-22(14)30-20(31(19)3)11-17-18(25)6-5-15(21(17)26)12-32-8-4-7-23(2,33)13-32/h5-6,9-10,33H,4,7-8,11-13H2,1-3H3	GXHAKMWWQHHDGY-UHFFFAOYSA-N	293195	US10106501, Example BW-17	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293195	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293195&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123633	381613477							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558908	CCN(CCO)Cc1ccc(Cl)c(Cc2nc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl	InChI=1S/C22H24Cl2F3N3O/c1-4-30(7-8-31)12-14-5-6-17(23)16(20(14)24)11-19-28-21-13(2)9-15(22(25,26)27)10-18(21)29(19)3/h5-6,9-10,31H,4,7-8,11-12H2,1-3H3	VQCVJSBVIGNDOW-UHFFFAOYSA-N	293196	US10106501, Example BW-18	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293196	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293196&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123434	381613478							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558909	Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(CN4CCOCC4=O)c3Cl)nc12)C(F)(F)F	InChI=1S/C22H20Cl2F3N3O2/c1-12-7-14(22(25,26)27)8-17-21(12)28-18(29(17)2)9-15-16(23)4-3-13(20(15)24)10-30-5-6-32-11-19(30)31/h3-4,7-8H,5-6,9-11H2,1-2H3	SXKBAZMHEBRQJM-UHFFFAOYSA-N	293197	US10106501, Example BX	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293197	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293197&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123445	381613479							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558910	Cc1c(ccc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC4)C(O)=O)c3Cl)nc12)C(F)(F)F	InChI=1S/C24H22Cl2F3N3O3/c1-12-16(24(27,28)29)4-6-18-21(12)30-19(31(18)2)11-15-17(25)5-3-14(20(15)26)22(33)32-9-7-13(8-10-32)23(34)35/h3-6,13H,7-11H2,1-2H3,(H,34,35)	HGEZZZRATSPSMZ-UHFFFAOYSA-N	293198	US10106501, Example BY	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293198	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293198&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123232	381613480							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558911	Cc1c(ccc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C25H24Cl2F3N3O3/c1-13-17(25(28,29)30)4-6-19-23(13)31-20(32(19)2)12-16-18(26)5-3-15(22(16)27)24(36)33-9-7-14(8-10-33)11-21(34)35/h3-6,14H,7-12H2,1-2H3,(H,34,35)	SFZLFIYEDQIZHG-UHFFFAOYSA-N	293199	US10106501, Example BZ	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293199	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293199&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123412	381613481							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558912	Cc1c(ccc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C22H20Cl2F3N3O2/c1-12-15(22(25,26)27)4-6-17-20(12)28-18(29(17)2)11-14-16(23)5-3-13(19(14)24)21(31)30-7-9-32-10-8-30/h3-6H,7-11H2,1-2H3	IBKUVKNKIOBYTP-UHFFFAOYSA-N	293200	US10106501, Example CA	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293200	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293200&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123255	381613482							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558913	Cc1c(Br)ccc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)nc12	InChI=1S/C21H20BrCl2N3O2/c1-12-15(22)4-6-17-20(12)25-18(26(17)2)11-14-16(23)5-3-13(19(14)24)21(28)27-7-9-29-10-8-27/h3-6H,7-11H2,1-2H3	ITNUKDYYDKNPLR-UHFFFAOYSA-N	293201	US10106501, Example CB	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293201	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293201&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123468	381613483							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558914	Cc1c(ccc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)nc12)C#N	InChI=1S/C22H20Cl2N4O2/c1-13-14(12-25)3-6-18-21(13)26-19(27(18)2)11-16-17(23)5-4-15(20(16)24)22(29)28-7-9-30-10-8-28/h3-6H,7-11H2,1-2H3	MIYWOHSINDNTOE-UHFFFAOYSA-N	293202	US10106501, Example CC	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293202	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293202&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123062	381613484							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558915	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)nc2cc(ccc12)C#N	InChI=1S/C21H18Cl2N4O2/c1-26-18-5-2-13(12-24)10-17(18)25-19(26)11-15-16(22)4-3-14(20(15)23)21(28)27-6-8-29-9-7-27/h2-5,10H,6-9,11H2,1H3	TUMSTZSGFRKFPX-UHFFFAOYSA-N	293203	US10106501, Example CD	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293203	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293203&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123671	381613485							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558916	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)nc2c(cc(Br)cc12)C(F)(F)F	InChI=1S/C21H17BrCl2F3N3O2/c1-29-16-9-11(22)8-14(21(25,26)27)19(16)28-17(29)10-13-15(23)3-2-12(18(13)24)20(31)30-4-6-32-7-5-30/h2-3,8-9H,4-7,10H2,1H3	ZKLBSSMXIRDDLB-UHFFFAOYSA-N	293204	US10106501, Example CE	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293204	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293204&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123897	381613486							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558917	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)nc2c(cc(cc12)C#N)C(F)(F)F	InChI=1S/C22H17Cl2F3N4O2/c1-30-17-9-12(11-28)8-15(22(25,26)27)20(17)29-18(30)10-14-16(23)3-2-13(19(14)24)21(32)31-4-6-33-7-5-31/h2-3,8-9H,4-7,10H2,1H3	JAYFOHGGWASJPO-UHFFFAOYSA-N	293205	US10106501, Example CF	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293205	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293205&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123647	381613487							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558918	CCn1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)nc2c(C)cc(cc12)C#N	InChI=1S/C23H22Cl2N4O2/c1-3-29-19-11-15(13-26)10-14(2)22(19)27-20(29)12-17-18(24)5-4-16(21(17)25)23(30)28-6-8-31-9-7-28/h4-5,10-11H,3,6-9,12H2,1-2H3	MAIWWHHNDGNZLL-UHFFFAOYSA-N	293206	US10106501, Example CG	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293206	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293206&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123861	381613488							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558919	CC(C)n1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)nc2c(C)cc(cc12)C#N	InChI=1S/C24H24Cl2N4O2/c1-14(2)30-20-11-16(13-27)10-15(3)23(20)28-21(30)12-18-19(25)5-4-17(22(18)26)24(31)29-6-8-32-9-7-29/h4-5,10-11,14H,6-9,12H2,1-3H3	LHFMVTACAGFRGI-UHFFFAOYSA-N	293207	US10106501, Example CH	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293207	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293207&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123655	381613489							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558920	Cc1cc(nc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)nc12)C#N	InChI=1S/C21H19Cl2N5O2/c1-12-9-13(11-24)25-20-19(12)26-17(27(20)2)10-15-16(22)4-3-14(18(15)23)21(29)28-5-7-30-8-6-28/h3-4,9H,5-8,10H2,1-2H3	CPGUBHMHCOATOV-UHFFFAOYSA-N	293208	US10106501, Example CI	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293208	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293208&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123019	381613490							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558921	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)cc2c(Cl)cc(cc12)C#N	InChI=1S/C22H18Cl3N3O2/c1-27-14(10-16-19(24)8-13(12-26)9-20(16)27)11-17-18(23)3-2-15(21(17)25)22(29)28-4-6-30-7-5-28/h2-3,8-10H,4-7,11H2,1H3	VSWJFOCSQQEDEY-UHFFFAOYSA-N	293209	US10106501, Example DQ::US10106501, Example CJ	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293209	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293209&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123760	381613491							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558922	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)cc2cccnc12	InChI=1S/C20H19Cl2N3O2/c1-24-14(11-13-3-2-6-23-19(13)24)12-16-17(21)5-4-15(18(16)22)20(26)25-7-9-27-10-8-25/h2-6,11H,7-10,12H2,1H3	CPWCXPVWOFYEHD-UHFFFAOYSA-N	293210	US10106501, Example CK	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293210	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293210&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123938	381613492							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558923	Cc1cc(nc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)cc12)C#N	InChI=1S/C22H20Cl2N4O2/c1-13-9-14(12-25)26-21-17(13)10-15(27(21)2)11-18-19(23)4-3-16(20(18)24)22(29)28-5-7-30-8-6-28/h3-4,9-10H,5-8,11H2,1-2H3	LBIZTJSLLMLSJX-UHFFFAOYSA-N	293211	US10106501, Example CL	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293211	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293211&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123258	381613493							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558924	Cc1cc(nc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)cc12)C#N	InChI=1S/C22H20Cl2N4O2/c1-13-9-14(12-25)26-21-17(13)10-15(27(21)2)11-18-19(23)4-3-16(20(18)24)22(29)28-5-7-30-8-6-28/h3-4,9-10H,5-8,11H2,1-2H3	LBIZTJSLLMLSJX-UHFFFAOYSA-N	293211	US10106501, Example CL	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293211	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293211&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123258	381613493							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558925	Cc1cc(nc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(O)CC4)c3Cl)cc12)C#N	InChI=1S/C23H22Cl2N4O2/c1-13-9-14(12-26)27-22-18(13)10-15(28(22)2)11-19-20(24)4-3-17(21(19)25)23(31)29-7-5-16(30)6-8-29/h3-4,9-10,16,30H,5-8,11H2,1-2H3	RMFUNNYCMDHPIJ-UHFFFAOYSA-N	293212	US10106501, Example CL-1	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293212	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293212&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124129603	381613494							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558926	Cc1cc(nc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC4)C4COC4)c3Cl)cc12)C#N	InChI=1S/C26H26Cl2N4O2/c1-15-9-18(12-29)30-25-21(15)10-19(31(25)2)11-22-23(27)4-3-20(24(22)28)26(33)32-7-5-16(6-8-32)17-13-34-14-17/h3-4,9-10,16-17H,5-8,11,13-14H2,1-2H3	ZXFXGPHMMSJHCI-UHFFFAOYSA-N	293213	US10106501, Example CL-2	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293213	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293213&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123180	381613495							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558927	Cc1cc(nc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)cc12)C(F)(F)F	InChI=1S/C22H20Cl2F3N3O2/c1-12-9-18(22(25,26)27)28-20-15(12)10-13(29(20)2)11-16-17(23)4-3-14(19(16)24)21(31)30-5-7-32-8-6-30/h3-4,9-10H,5-8,11H2,1-2H3	WBDSEKJGKSYFQD-UHFFFAOYSA-N	293214	(2,4-dichloro-3-((1,4-dimethyl-6-(trifluoromethyl)-1H-pyrrolo[2,3-b]pyridin-2-yl)methyl)phenyl)(morpholino)methanone::US10106501, Example CM	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293214	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293214&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123674	381613496							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558928	Cc1cc(Cl)nc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)cc12	InChI=1S/C21H20Cl3N3O2/c1-12-9-18(23)25-20-15(12)10-13(26(20)2)11-16-17(22)4-3-14(19(16)24)21(28)27-5-7-29-8-6-27/h3-4,9-10H,5-8,11H2,1-2H3	JEQHMOGNUBLDML-UHFFFAOYSA-N	293215	(2,4-dichloro-3-((6-chloro-1,4-dimethyl-1H-pyrrolo[2,3-b]pyridin-2-yl)methyl)phenyl)(morpholino)methanone::US10106501, Example CM1	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293215	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293215&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122985	381613497							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558929	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)cc2ncc(cc12)C(F)(F)F	InChI=1S/C21H18Cl2F3N3O2/c1-28-13(10-17-18(28)8-12(11-27-17)21(24,25)26)9-15-16(22)3-2-14(19(15)23)20(30)29-4-6-31-7-5-29/h2-3,8,10-11H,4-7,9H2,1H3	BVWUXBJTBOQVOC-UHFFFAOYSA-N	293216	US10106501, Example CO	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293216	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293216&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123639	381613498							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558930	Cn1c(cc2ncc(cc12)C(F)(F)F)C(=O)c1c(Cl)ccc(C(=O)N2CCOCC2)c1Cl	InChI=1S/C21H16Cl2F3N3O3/c1-28-15-8-11(21(24,25)26)10-27-14(15)9-16(28)19(30)17-13(22)3-2-12(18(17)23)20(31)29-4-6-32-7-5-29/h2-3,8-10H,4-7H2,1H3	IUCICEWDGXPGSJ-UHFFFAOYSA-N	293217	US10106501, Example CP	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293217	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293217&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122864	381613499							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558931	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)cc2cnc(cc12)C(F)(F)F	InChI=1S/C21H18Cl2F3N3O2/c1-28-13(8-12-11-27-18(10-17(12)28)21(24,25)26)9-15-16(22)3-2-14(19(15)23)20(30)29-4-6-31-7-5-29/h2-3,8,10-11H,4-7,9H2,1H3	OJNMOZGQTFTHEE-UHFFFAOYSA-N	293218	US10106501, Example CQ	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293218	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293218&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123398	381613500							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558932	Cc1nc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)cc12)C(F)(F)F	InChI=1S/C22H20Cl2F3N3O2/c1-12-15-9-13(29(2)18(15)11-19(28-12)22(25,26)27)10-16-17(23)4-3-14(20(16)24)21(31)30-5-7-32-8-6-30/h3-4,9,11H,5-8,10H2,1-2H3	NEIXIEXKPDYXSQ-UHFFFAOYSA-N	293219	US10106501, Example CR	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293219	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293219&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123121	381613501							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558933	Cc1nc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)cc12)C#N	InChI=1S/C22H20Cl2N4O2/c1-13-17-10-15(27(2)20(17)9-14(12-25)26-13)11-18-19(23)4-3-16(21(18)24)22(29)28-5-7-30-8-6-28/h3-4,9-10H,5-8,11H2,1-2H3	LUOWQKKFXZXLDD-UHFFFAOYSA-N	293220	US10106501, Example CS	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293220	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293220&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123450	381613502							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558934	Cc1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)nc2c(C)cc(cn12)C(F)(F)F	InChI=1S/C22H20Cl2F3N3O2/c1-12-9-14(22(25,26)27)11-30-13(2)18(28-20(12)30)10-16-17(23)4-3-15(19(16)24)21(31)29-5-7-32-8-6-29/h3-4,9,11H,5-8,10H2,1-2H3	TUGNJDIYOPABEH-UHFFFAOYSA-N	293221	US10106501, Example CT	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293221	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293221&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123134	381613503							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558935	Cc1c(Cc2c(Cl)ccc(C(=O)N3CCC(O)CC3)c2Cl)nc2c(C)cc(cn12)C(F)(F)F	InChI=1S/C23H22Cl2F3N3O2/c1-12-9-14(23(26,27)28)11-31-13(2)19(29-21(12)31)10-17-18(24)4-3-16(20(17)25)22(33)30-7-5-15(32)6-8-30/h3-4,9,11,15,32H,5-8,10H2,1-2H3	FYMJCQPHSZVTDR-UHFFFAOYSA-N	293222	US10106501, Example CT-1	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293222	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293222&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123695	381613504							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558936	Cc1c(Cc2c(Cl)ccc(C(=O)N3CCC(CCO)CC3)c2Cl)nc2c(C)cc(cn12)C(F)(F)F	InChI=1S/C25H26Cl2F3N3O2/c1-14-11-17(25(28,29)30)13-33-15(2)21(31-23(14)33)12-19-20(26)4-3-18(22(19)27)24(35)32-8-5-16(6-9-32)7-10-34/h3-4,11,13,16,34H,5-10,12H2,1-2H3	RVZFNPKBBXHSBL-UHFFFAOYSA-N	293223	US10106501, Example CT-2	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293223	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293223&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123462	381613505							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558937	Cc1c(Cc2c(Cl)ccc(C(=O)N3CCC(CC3)C(C)(C)O)c2Cl)nc2c(C)cc(cn12)C(F)(F)F	InChI=1S/C26H28Cl2F3N3O2/c1-14-11-17(26(29,30)31)13-34-15(2)21(32-23(14)34)12-19-20(27)6-5-18(22(19)28)24(35)33-9-7-16(8-10-33)25(3,4)36/h5-6,11,13,16,36H,7-10,12H2,1-4H3	JQOPGYXOSGMDQU-UHFFFAOYSA-N	293224	US10106501, Example CT-3	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293224	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293224&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123679	381613506							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558938	Cc1c(Cc2c(Cl)ccc(C(=O)N3CCC(O)C3)c2Cl)nc2c(C)cc(cn12)C(F)(F)F	InChI=1S/C22H20Cl2F3N3O2/c1-11-7-13(22(25,26)27)9-30-12(2)18(28-20(11)30)8-16-17(23)4-3-15(19(16)24)21(32)29-6-5-14(31)10-29/h3-4,7,9,14,31H,5-6,8,10H2,1-2H3	MMJOAEXKQMJHHG-UHFFFAOYSA-N	293225	US10106501, Example CT-4	Nuclear receptor ROR-gamma	Human		>10000							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293225	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293225&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123008	381613507							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558939	CN(C)C1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cn3c2C)C(F)(F)F)c1Cl	InChI=1S/C25H27Cl2F3N4O/c1-14-11-16(25(28,29)30)13-34-15(2)21(31-23(14)34)12-19-20(26)6-5-18(22(19)27)24(35)33-9-7-17(8-10-33)32(3)4/h5-6,11,13,17H,7-10,12H2,1-4H3	ATRJFKAADWARTK-UHFFFAOYSA-N	293226	US10106501, Example CT-5	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293226	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293226&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123706	381613508							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558940	COC1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cn3c2C)C(F)(F)F)c1Cl	InChI=1S/C24H24Cl2F3N3O2/c1-13-10-15(24(27,28)29)12-32-14(2)20(30-22(13)32)11-18-19(25)5-4-17(21(18)26)23(33)31-8-6-16(34-3)7-9-31/h4-5,10,12,16H,6-9,11H2,1-3H3	GISVNJPOTVYTJF-UHFFFAOYSA-N	293227	US10106501, Example CT-6	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293227	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293227&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123379	381613509							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558941	COCCC1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cn3c2C)C(F)(F)F)c1Cl	InChI=1S/C26H28Cl2F3N3O2/c1-15-12-18(26(29,30)31)14-34-16(2)22(32-24(15)34)13-20-21(27)5-4-19(23(20)28)25(35)33-9-6-17(7-10-33)8-11-36-3/h4-5,12,14,17H,6-11,13H2,1-3H3	CBLLBRDUKYYISJ-UHFFFAOYSA-N	293228	US10106501, Example CT-7	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293228	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293228&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123935	381613510							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558942	Cc1c(Cc2c(Cl)ccc(C(=O)N3CCC(CC3)C3COC3)c2Cl)nc2c(C)cc(cn12)C(F)(F)F	InChI=1S/C26H26Cl2F3N3O2/c1-14-9-18(26(29,30)31)11-34-15(2)22(32-24(14)34)10-20-21(27)4-3-19(23(20)28)25(35)33-7-5-16(6-8-33)17-12-36-13-17/h3-4,9,11,16-17H,5-8,10,12-13H2,1-2H3	JZUSZCCSKHUTQA-UHFFFAOYSA-N	293229	US10106501, Example CT-8	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293229	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293229&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123552	381613511							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558943	Cc1c(Cc2c(Cl)ccc(C(=O)N3CCN(CC3)C3COC3)c2Cl)nc2c(C)cc(cn12)C(F)(F)F	InChI=1S/C25H25Cl2F3N4O2/c1-14-9-16(25(28,29)30)11-34-15(2)21(31-23(14)34)10-19-20(26)4-3-18(22(19)27)24(35)33-7-5-32(6-8-33)17-12-36-13-17/h3-4,9,11,17H,5-8,10,12-13H2,1-2H3	SWZMCQIRVSLOST-UHFFFAOYSA-N	293230	US10106501, Example CT-9	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293230	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293230&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123428	381613512							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558944	Cc1c(Cc2c(Cl)ccc(C(=O)N3CCC(CO)CC3)c2Cl)nc2c(C)cc(cn12)C(F)(F)F	InChI=1S/C24H24Cl2F3N3O2/c1-13-9-16(24(27,28)29)11-32-14(2)20(30-22(13)32)10-18-19(25)4-3-17(21(18)26)23(34)31-7-5-15(12-33)6-8-31/h3-4,9,11,15,33H,5-8,10,12H2,1-2H3	BQSVCZAJGGRVLI-UHFFFAOYSA-N	293231	US10106501, Example CT-10	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293231	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293231&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123223	381613513							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558945	CC(O)C1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cn3c2C)C(F)(F)F)c1Cl	InChI=1S/C25H26Cl2F3N3O2/c1-13-10-17(25(28,29)30)12-33-14(2)21(31-23(13)33)11-19-20(26)5-4-18(22(19)27)24(35)32-8-6-16(7-9-32)15(3)34/h4-5,10,12,15-16,34H,6-9,11H2,1-3H3	WCAZJTAXICSKJV-UHFFFAOYSA-N	293232	US10106501, Example CT-11	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293232	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293232&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123400	381613514							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558946	Cc1c(Cc2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)nc2c(C)cc(cn12)C(F)(F)F	InChI=1S/C25H24Cl2F3N3O3/c1-13-9-16(25(28,29)30)12-33-14(2)20(31-23(13)33)11-18-19(26)4-3-17(22(18)27)24(36)32-7-5-15(6-8-32)10-21(34)35/h3-4,9,12,15H,5-8,10-11H2,1-2H3,(H,34,35)	JARVTLAVEVLNAG-UHFFFAOYSA-N	293233	US10106501, Example CU	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293233	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293233&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123293	381613515							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558947	Cc1c(Cc2c(Cl)ccc(C(=O)N3CCC(CCO)CC3)c2Cl)nc2c(C)cc(cn12)C#N	InChI=1S/C25H26Cl2N4O2/c1-15-11-18(13-28)14-31-16(2)22(29-24(15)31)12-20-21(26)4-3-19(23(20)27)25(33)30-8-5-17(6-9-30)7-10-32/h3-4,11,14,17,32H,5-10,12H2,1-2H3	HAUXRTVNCSGRQH-UHFFFAOYSA-N	293234	US10106501, Example CV	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293234	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293234&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123338	381613516							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558948	Cc1c(Cc2c(Cl)ccc(C(=O)N3CCC(CO)CC3)c2Cl)nc2c(C)cc(cn12)C#N	InChI=1S/C24H24Cl2N4O2/c1-14-9-17(11-27)12-30-15(2)21(28-23(14)30)10-19-20(25)4-3-18(22(19)26)24(32)29-7-5-16(13-31)6-8-29/h3-4,9,12,16,31H,5-8,10,13H2,1-2H3	TZTMHHIYIQMWDH-UHFFFAOYSA-N	293235	US10106501, Example CV-1	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293235	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293235&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123042	381613517							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558949	COC1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cn3c2C)C#N)c1Cl	InChI=1S/C24H24Cl2N4O2/c1-14-10-16(12-27)13-30-15(2)21(28-23(14)30)11-19-20(25)5-4-18(22(19)26)24(31)29-8-6-17(32-3)7-9-29/h4-5,10,13,17H,6-9,11H2,1-3H3	JSZXLQMGIAPASP-UHFFFAOYSA-N	293236	US10106501, Example CV-2	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293236	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293236&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123289	381613518							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558950	Cc1c(Cc2c(Cl)ccc(C(=O)N3CCC(CC3)C(C)(C)O)c2Cl)nc2c(C)cc(cn12)C#N	InChI=1S/C26H28Cl2N4O2/c1-15-11-17(13-29)14-32-16(2)22(30-24(15)32)12-20-21(27)6-5-19(23(20)28)25(33)31-9-7-18(8-10-31)26(3,4)34/h5-6,11,14,18,34H,7-10,12H2,1-4H3	DLJFAOUGGBRFBK-UHFFFAOYSA-N	293237	US10106501, Example CV-3	Nuclear receptor ROR-gamma	Human		 750							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293237	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293237&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123588	381613519							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558951	CC(O)C1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cn3c2C)C#N)c1Cl	InChI=1S/C25H26Cl2N4O2/c1-14-10-17(12-28)13-31-15(2)22(29-24(14)31)11-20-21(26)5-4-19(23(20)27)25(33)30-8-6-18(7-9-30)16(3)32/h4-5,10,13,16,18,32H,6-9,11H2,1-3H3	BGTRKSAQWGFYHH-UHFFFAOYSA-N	293238	US10106501, Example CV-4	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293238	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293238&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123812	381613520							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558952	Cc1c(Cc2c(Cl)ccc(C(=O)N3CCC(CC3)C3COC3)c2Cl)nc2c(C)cc(cn12)C#N	InChI=1S/C26H26Cl2N4O2/c1-15-9-17(11-29)12-32-16(2)23(30-25(15)32)10-21-22(27)4-3-20(24(21)28)26(33)31-7-5-18(6-8-31)19-13-34-14-19/h3-4,9,12,18-19H,5-8,10,13-14H2,1-2H3	VKZRFLWOZWYJNN-UHFFFAOYSA-N	293239	US10106501, Example CV-5	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293239	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293239&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123344	381613521							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558953	COCCC1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cn3c2C)C#N)c1Cl	InChI=1S/C26H28Cl2N4O2/c1-16-12-19(14-29)15-32-17(2)23(30-25(16)32)13-21-22(27)5-4-20(24(21)28)26(33)31-9-6-18(7-10-31)8-11-34-3/h4-5,12,15,18H,6-11,13H2,1-3H3	FZCFTSXWXRDOOZ-UHFFFAOYSA-N	293240	US10106501, Example CV-6	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293240	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293240&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123851	381613522							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558954	Cc1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)nc2c(C)cc(Cl)nn12	InChI=1S/C20H19Cl3N4O2/c1-11-9-17(22)25-27-12(2)16(24-19(11)27)10-14-15(21)4-3-13(18(14)23)20(28)26-5-7-29-8-6-26/h3-4,9H,5-8,10H2,1-2H3	OMKVHTSECCTPDK-UHFFFAOYSA-N	293241	US10106501, Example CW	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293241	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293241&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123969	381613523							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558955	Cc1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)nc2cc(C)c(Cl)nn12	InChI=1S/C20H19Cl3N4O2/c1-11-9-17-24-16(12(2)27(17)25-19(11)23)10-14-15(21)4-3-13(18(14)22)20(28)26-5-7-29-8-6-26/h3-4,9H,5-8,10H2,1-2H3	NESHGUBKGHDLNH-UHFFFAOYSA-N	293242	US10106501, Example CY	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293242	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293242&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123061	381613524							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558956	Cc1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)nc2c(C)cc(nn12)C(F)(F)F	InChI=1S/C21H19Cl2F3N4O2/c1-11-9-17(21(24,25)26)28-30-12(2)16(27-19(11)30)10-14-15(22)4-3-13(18(14)23)20(31)29-5-7-32-8-6-29/h3-4,9H,5-8,10H2,1-2H3	AQDHBLSSOZOWNK-UHFFFAOYSA-N	293243	US10106501, Example CZ	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293243	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293243&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123752	381613525							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558957	Cc1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)nc2c(C)cc(nn12)C#N	InChI=1S/C21H19Cl2N5O2/c1-12-9-14(11-24)26-28-13(2)18(25-20(12)28)10-16-17(22)4-3-15(19(16)23)21(29)27-5-7-30-8-6-27/h3-4,9H,5-8,10H2,1-2H3	IKNLNFBKNSGDPP-UHFFFAOYSA-N	293244	US10106501, Example DA	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293244	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293244&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123651	381613526							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558958	Cc1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)nc2cc(C)c(nn12)C#N	InChI=1S/C21H19Cl2N5O2/c1-12-9-19-25-17(13(2)28(19)26-18(12)11-24)10-15-16(22)4-3-14(20(15)23)21(29)27-5-7-30-8-6-27/h3-4,9H,5-8,10H2,1-2H3	IAIZEIPCCMMUSD-UHFFFAOYSA-N	293245	US10106501, Example DB	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293245	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293245&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123870	381613527							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558959	Cc1cc(nc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)nc12)C(F)(F)F	InChI=1S/C21H19Cl2F3N4O2/c1-11-9-15(21(24,25)26)27-19-18(11)28-16(29(19)2)10-13-14(22)4-3-12(17(13)23)20(31)30-5-7-32-8-6-30/h3-4,9H,5-8,10H2,1-2H3	JAURFPBHZXZXHL-UHFFFAOYSA-N	293246	US10106501, Example DC	Nuclear receptor ROR-gamma	Human		 5500							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293246	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293246&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123495	381613528							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558960	Cc1nn(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)c2c(C)cc(cc12)C(F)(F)F	InChI=1S/C22H20Cl2F3N3O2/c1-12-9-14(22(25,26)27)10-16-13(2)28-30(20(12)16)11-17-18(23)4-3-15(19(17)24)21(31)29-5-7-32-8-6-29/h3-4,9-10H,5-8,11H2,1-2H3	GHCOXHZLABXRDO-UHFFFAOYSA-N	293247	US10106501, Example DD	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293247	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293247&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123917	381613529							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558961	Cc1nn(Cc2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)c2c(C)cc(cc12)C(F)(F)F	InChI=1S/C25H24Cl2F3N3O3/c1-13-9-16(25(28,29)30)11-18-14(2)31-33(23(13)18)12-19-20(26)4-3-17(22(19)27)24(36)32-7-5-15(6-8-32)10-21(34)35/h3-4,9,11,15H,5-8,10,12H2,1-2H3,(H,34,35)	XUVCFBHVGIQRTI-UHFFFAOYSA-N	293248	US10106501, Example DE	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293248	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293248&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123901	381613530							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558962	Cc1n(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)nc2c(C)cc(cc12)C(F)(F)F	InChI=1S/C22H20Cl2F3N3O2/c1-12-9-14(22(25,26)27)10-16-13(2)30(28-20(12)16)11-17-18(23)4-3-15(19(17)24)21(31)29-5-7-32-8-6-29/h3-4,9-10H,5-8,11H2,1-2H3	HTJRVYGNWSEGNE-UHFFFAOYSA-N	293249	US10106501, Example DF	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293249	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293249&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123182	381613531							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558963	Cc1n(Cc2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)nc2c(C)cc(cc12)C(F)(F)F	InChI=1S/C25H24Cl2F3N3O3/c1-13-9-16(25(28,29)30)11-18-14(2)33(31-23(13)18)12-19-20(26)4-3-17(22(19)27)24(36)32-7-5-15(6-8-32)10-21(34)35/h3-4,9,11,15H,5-8,10,12H2,1-2H3,(H,34,35)	PRHDZFOPTCDZJO-UHFFFAOYSA-N	293250	US10106501, Example DG	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293250	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293250&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123728	381613532							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558964	Cc1cn(Cc2c(Cl)ccc(C(=O)N3CCC(CC3)C(O)=O)c2Cl)c2c(C)cc(cc12)C(F)(F)F	InChI=1S/C25H23Cl2F3N2O3/c1-13-9-16(25(28,29)30)10-18-14(2)11-32(22(13)18)12-19-20(26)4-3-17(21(19)27)23(33)31-7-5-15(6-8-31)24(34)35/h3-4,9-11,15H,5-8,12H2,1-2H3,(H,34,35)	KETGHMSOAJNUQG-UHFFFAOYSA-N	293251	US10106501, Example DH	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293251	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293251&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123356	381613533							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558965	Cc1cn(Cc2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)c2c(C)cc(cc12)C(F)(F)F	InChI=1S/C26H25Cl2F3N2O3/c1-14-9-17(26(29,30)31)11-19-15(2)12-33(24(14)19)13-20-21(27)4-3-18(23(20)28)25(36)32-7-5-16(6-8-32)10-22(34)35/h3-4,9,11-12,16H,5-8,10,13H2,1-2H3,(H,34,35)	DJDIOIFNJRXELS-UHFFFAOYSA-N	293252	US10106501, Example DI	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293252	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293252&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122947	381613534							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558966	Cc1cn(C(=O)c2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)c2c(C)cc(cc12)C(F)(F)F	InChI=1S/C26H23Cl2F3N2O4/c1-13-9-16(26(29,30)31)11-18-14(2)12-33(23(13)18)25(37)21-19(27)4-3-17(22(21)28)24(36)32-7-5-15(6-8-32)10-20(34)35/h3-4,9,11-12,15H,5-8,10H2,1-2H3,(H,34,35)	ZNZUPLYRQYEHNH-UHFFFAOYSA-N	293253	US10106501, Example DJ	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293253	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293253&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122979	381613535							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558967	Cc1cn(Cc2c(Cl)ccc(C(=O)N3CCC(O)CC3)c2Cl)c2c(C)cc(cc12)C#N	InChI=1S/C24H23Cl2N3O2/c1-14-9-16(11-27)10-19-15(2)12-29(23(14)19)13-20-21(25)4-3-18(22(20)26)24(31)28-7-5-17(30)6-8-28/h3-4,9-10,12,17,30H,5-8,13H2,1-2H3	UYWYSPYYENKPJP-UHFFFAOYSA-N	293254	US10106501, Example DK	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293254	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293254&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123941	381613536							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558968	Cc1cn(Cc2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)c2c(C)cc(cc12)C#N	InChI=1S/C26H25Cl2N3O3/c1-15-9-18(12-29)10-20-16(2)13-31(25(15)20)14-21-22(27)4-3-19(24(21)28)26(34)30-7-5-17(6-8-30)11-23(32)33/h3-4,9-10,13,17H,5-8,11,14H2,1-2H3,(H,32,33)	OCAABOKMMAXNOT-UHFFFAOYSA-N	293255	US10106501, Example DL	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293255	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293255&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123628	381613537							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558969	Cc1cn(C(=O)c2c(Cl)ccc(C(=O)N3CCC(O)CC3)c2Cl)c2c(C)cc(cc12)C#N	InChI=1S/C24H21Cl2N3O3/c1-13-9-15(11-27)10-18-14(2)12-29(22(13)18)24(32)20-19(25)4-3-17(21(20)26)23(31)28-7-5-16(30)6-8-28/h3-4,9-10,12,16,30H,5-8H2,1-2H3	CWTXXEFWWPOUSJ-UHFFFAOYSA-N	293256	US10106501, Example DM	Nuclear receptor ROR-gamma	Human		 300							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293256	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293256&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123125	381613538							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558970	Cc1cn(C(=O)c2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)c2c(C)cc(cc12)C#N	InChI=1S/C26H23Cl2N3O4/c1-14-9-17(12-29)10-19-15(2)13-31(24(14)19)26(35)22-20(27)4-3-18(23(22)28)25(34)30-7-5-16(6-8-30)11-21(32)33/h3-4,9-10,13,16H,5-8,11H2,1-2H3,(H,32,33)	SWNLFMCVYCIMFG-UHFFFAOYSA-N	293257	US10106501, Example DN	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293257	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293257&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123216	381613539							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558971	Cc1cc(nc2n(C)c(Cc3c(Cl)ncc(C(=O)N4CCC(O)CC4)c3Cl)cc12)C(F)(F)F	InChI=1S/C22H21Cl2F3N4O2/c1-11-7-17(22(25,26)27)29-20-14(11)8-12(30(20)2)9-15-18(23)16(10-28-19(15)24)21(33)31-5-3-13(32)4-6-31/h7-8,10,13,32H,3-6,9H2,1-2H3	QRBJKWUCFGBJGP-UHFFFAOYSA-N	293258	US10106501, Example DT::US10106501, Example DO	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293258	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293258&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123421	381613540							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558972	Cc1cc(OC(F)(F)F)cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)cc12	InChI=1S/C26H25Cl2F3N2O4/c1-14-9-17(37-26(29,30)31)13-22-19(14)11-16(32(22)2)12-20-21(27)4-3-18(24(20)28)25(36)33-7-5-15(6-8-33)10-23(34)35/h3-4,9,11,13,15H,5-8,10,12H2,1-2H3,(H,34,35)	ZPNSNSMHWHPGJR-UHFFFAOYSA-N	293259	US10106501, Example DP	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293259	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293259&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123612	381613541							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558973	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)cc2c(Cl)cc(cc12)C#N	InChI=1S/C22H18Cl3N3O2/c1-27-14(10-16-19(24)8-13(12-26)9-20(16)27)11-17-18(23)3-2-15(21(17)25)22(29)28-4-6-30-7-5-28/h2-3,8-10H,4-7,11H2,1H3	VSWJFOCSQQEDEY-UHFFFAOYSA-N	293209	US10106501, Example DQ::US10106501, Example CJ	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293209	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293209&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123760	381613491							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558974	Cn1c(Cc2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)cc2c(Cl)cc(cc12)C#N	InChI=1S/C25H22Cl3N3O3/c1-30-16(11-18-21(27)8-15(13-29)9-22(18)30)12-19-20(26)3-2-17(24(19)28)25(34)31-6-4-14(5-7-31)10-23(32)33/h2-3,8-9,11,14H,4-7,10,12H2,1H3,(H,32,33)	CMFWAERHCPREOM-UHFFFAOYSA-N	292883	US10106501, Example DR::US10106501, Example R	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292883	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292883&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123405	381613168							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558975	Cc1cc(cc2ccn(Cc3c(Cl)ccc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)c12)C(F)(F)F	InChI=1S/C25H23Cl2F3N2O3/c1-14-10-17(25(28,29)30)12-16-6-9-32(23(14)16)13-19-20(26)3-2-18(22(19)27)24(35)31-7-4-15(5-8-31)11-21(33)34/h2-3,6,9-10,12,15H,4-5,7-8,11,13H2,1H3,(H,33,34)	PGISETOBANJZCF-UHFFFAOYSA-N	292869	US10106501, Example DS::US10106501, Example J	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=292869	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=292869&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124122941	381613154							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
558976	Cc1cc(nc2n(C)c(Cc3c(Cl)ncc(C(=O)N4CCC(O)CC4)c3Cl)cc12)C(F)(F)F	InChI=1S/C22H21Cl2F3N4O2/c1-11-7-17(22(25,26)27)29-20-14(11)8-12(30(20)2)9-15-18(23)16(10-28-19(15)24)21(33)31-5-3-13(32)4-6-31/h7-8,10,13,32H,3-6,9H2,1-2H3	QRBJKWUCFGBJGP-UHFFFAOYSA-N	293258	US10106501, Example DT::US10106501, Example DO	Nuclear receptor ROR-gamma	Human		<100							US Patent		10.7270/Q2G44SBV		aid1795887	US10106501	Argiriadi, MA; Breinlinger, EC; Cusack, KP; Hobson, AD; Potin, D; Barth, M; Amaudrut, J; Poupardin, O; Mounier, L; Kort, ME	10/23/2018	2/24/2019	Abbvie	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=293258	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=738&target=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=293258&enzyme=Nuclear+receptor+ROR-gamma&column=ki&startPg=0&Increment=50&submit=Search			124123421	381613540							1	MDRAPQRQHRASRELLAAKKTHTSQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	6CN5,5EJV,5X8U,5X8S,5AYG,5IZ0,4S14,7QP4,3L0L,4WPF,7W3Q,7W3P,7KCO,4QM0,4NB6,4WQP,4WLB,6E3G,5YP6,6J3N,7JH2,6XFV,6O98,6BN6,9N9L,8XU5,7E3M,6NAD,5YP5,4YPQ,4XT9,3L0J,3KYT,3B0W,6NWT,6SLZ,5K74,5K6E,5K3N,5K3M,5K3L,5K38,7LUK,7KXF,7KXE,7KXD,7KQJ,7JYM,7JTM,6XAE,6W9I,6W9H,6VQF,6U25,6P9F,8GXP,6FGQ,5APK,6NWU,6NWS,6R7K,6R7J,6R7A,5LWP,6ESN,7OFK,7OFI,5G46,5G45,5G44,5G43,5G42,5APJ,5APH,5UHI,5UFR,5UFO,5NIB,5NI8,5NI7,5NI5,6SAL,7NP6,7NP5,7NEC,6TLT,6TLQ,6TLM,6T50,6T4Y,6T4X,6T4K,6T4J,6T4I,6T4G,6VSW,5ZA1,6B31,6CVH,5IXK,4ZOM,4ZJW,4ZJR,6Q2W,5ETH,6B33,6E3E,5W4R,6BR3,6BR2,6B30	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8		RAR-related orphan receptor C	Q6I9R9_HUMAN	Q6I9R9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																														
