BindingDB Reactant_set_id	Ligand SMILES	Ligand InChI	Ligand InChI Key	BindingDB MonomerID	BindingDB Ligand Name	Target Name	Target Source Organism According to Curator or DataSource	Ki (nM)	IC50 (nM)	Kd (nM)	EC50 (nM)	kon (M-1-s-1)	koff (s-1)	pH	Temp (C)	Curation/DataSource	Article DOI	BindingDB Entry DOI	PMID	PubChem AID	Patent Number	Authors	Date of publication	Date in BindingDB	Institution	Link to Ligand in BindingDB	Link to Target in BindingDB	Link to Ligand-Target Pair in BindingDB	Ligand HET ID in PDB	PDB ID(s) for Ligand-Target Complex	PubChem CID	PubChem SID	ChEBI ID of Ligand	ChEMBL ID of Ligand	DrugBank ID of Ligand	IUPHAR_GRAC ID of Ligand	KEGG ID of Ligand	ZINC ID of Ligand	Number of Protein Chains in Target (>1 implies a multichain complex)	BindingDB Target Chain Sequence 1	PDB ID(s) of Target Chain 1	UniProt (SwissProt) Recommended Name of Target Chain 1	UniProt (SwissProt) Entry Name of Target Chain 1	UniProt (SwissProt) Primary ID of Target Chain 1	UniProt (SwissProt) Secondary ID(s) of Target Chain 1	UniProt (SwissProt) Alternative ID(s) of Target Chain 1	UniProt (TrEMBL) Submitted Name of Target Chain 1	UniProt (TrEMBL) Entry Name of Target Chain 1	UniProt (TrEMBL) Primary ID of Target Chain 1	UniProt (TrEMBL) Secondary ID(s) of Target Chain 1	UniProt (TrEMBL) Alternative ID(s) of Target Chain 1	BindingDB Target Chain Sequence 2	PDB ID(s) of Target Chain 2	UniProt (SwissProt) Recommended Name of Target Chain 2	UniProt (SwissProt) Entry Name of Target Chain 2	UniProt (SwissProt) Primary ID of Target Chain 2	UniProt (SwissProt) Secondary ID(s) of Target Chain 2	UniProt (SwissProt) Alternative ID(s) of Target Chain 2	UniProt (TrEMBL) Submitted Name of Target Chain 2	UniProt (TrEMBL) Entry Name of Target Chain 2	UniProt (TrEMBL) Primary ID of Target Chain 2	UniProt (TrEMBL) Secondary ID(s) of Target Chain 2	UniProt (TrEMBL) Alternative ID(s) of Target Chain 2	BindingDB Target Chain Sequence 3	PDB ID(s) of Target Chain 3	UniProt (SwissProt) Recommended Name of Target Chain 3	UniProt (SwissProt) Entry Name of Target Chain 3	UniProt (SwissProt) Primary ID of Target Chain 3	UniProt (SwissProt) Secondary ID(s) of Target Chain 3	UniProt (SwissProt) Alternative ID(s) of Target Chain 3	UniProt (TrEMBL) Submitted Name of Target Chain 3	UniProt (TrEMBL) Entry Name of Target Chain 3	UniProt (TrEMBL) Primary ID of Target Chain 3	UniProt (TrEMBL) Secondary ID(s) of Target Chain 3	UniProt (TrEMBL) Alternative ID(s) of Target Chain 3	BindingDB Target Chain Sequence 4	PDB ID(s) of Target Chain 4	UniProt (SwissProt) Recommended Name of Target Chain 4	UniProt (SwissProt) Entry Name of Target Chain 4	UniProt (SwissProt) Primary ID of Target Chain 4	UniProt (SwissProt) Secondary ID(s) of Target Chain 4	UniProt (SwissProt) Alternative ID(s) of Target Chain 4	UniProt (TrEMBL) Submitted Name of Target Chain 4	UniProt (TrEMBL) Entry Name of Target Chain 4	UniProt (TrEMBL) Primary ID of Target Chain 4	UniProt (TrEMBL) Secondary ID(s) of Target Chain 4	UniProt (TrEMBL) Alternative ID(s) of Target Chain 4	BindingDB Target Chain Sequence 5	PDB ID(s) of Target Chain 5	UniProt (SwissProt) Recommended Name of Target Chain 5	UniProt (SwissProt) Entry Name of Target Chain 5	UniProt (SwissProt) Primary ID of Target Chain 5	UniProt (SwissProt) Secondary ID(s) of Target Chain 5	UniProt (SwissProt) Alternative ID(s) of Target Chain 5	UniProt (TrEMBL) Submitted Name of Target Chain 5	UniProt (TrEMBL) Entry Name of Target Chain 5	UniProt (TrEMBL) Primary ID of Target Chain 5	UniProt (TrEMBL) Secondary ID(s) of Target Chain 5	UniProt (TrEMBL) Alternative ID(s) of Target Chain 5	BindingDB Target Chain Sequence 6	PDB ID(s) of Target Chain 6	UniProt (SwissProt) Recommended Name of Target Chain 6	UniProt (SwissProt) Entry Name of Target Chain 6	UniProt (SwissProt) Primary ID of Target Chain 6	UniProt (SwissProt) Secondary ID(s) of Target Chain 6	UniProt (SwissProt) Alternative ID(s) of Target Chain 6	UniProt (TrEMBL) Submitted Name of Target Chain 6	UniProt (TrEMBL) Entry Name of Target Chain 6	UniProt (TrEMBL) Primary ID of Target Chain 6	UniProt (TrEMBL) Secondary ID(s) of Target Chain 6	UniProt (TrEMBL) Alternative ID(s) of Target Chain 6	BindingDB Target Chain Sequence 7	PDB ID(s) of Target Chain 7	UniProt (SwissProt) Recommended Name of Target Chain 7	UniProt (SwissProt) Entry Name of Target Chain 7	UniProt (SwissProt) Primary ID of Target Chain 7	UniProt (SwissProt) Secondary ID(s) of Target Chain 7	UniProt (SwissProt) Alternative ID(s) of Target Chain 7	UniProt (TrEMBL) Submitted Name of Target Chain 7	UniProt (TrEMBL) Entry Name of Target Chain 7	UniProt (TrEMBL) Primary ID of Target Chain 7	UniProt (TrEMBL) Secondary ID(s) of Target Chain 7	UniProt (TrEMBL) Alternative ID(s) of Target Chain 7	BindingDB Target Chain Sequence 8	PDB ID(s) of Target Chain 8	UniProt (SwissProt) Recommended Name of Target Chain 8	UniProt (SwissProt) Entry Name of Target Chain 8	UniProt (SwissProt) Primary ID of Target Chain 8	UniProt (SwissProt) Secondary ID(s) of Target Chain 8	UniProt (SwissProt) Alternative ID(s) of Target Chain 8	UniProt (TrEMBL) Submitted Name of Target Chain 8	UniProt (TrEMBL) Entry Name of Target Chain 8	UniProt (TrEMBL) Primary ID of Target Chain 8	UniProt (TrEMBL) Secondary ID(s) of Target Chain 8	UniProt (TrEMBL) Alternative ID(s) of Target Chain 8	BindingDB Target Chain Sequence 9	PDB ID(s) of Target Chain 9	UniProt (SwissProt) Recommended Name of Target Chain 9	UniProt (SwissProt) Entry Name of Target Chain 9	UniProt (SwissProt) Primary ID of Target Chain 9	UniProt (SwissProt) Secondary ID(s) of Target Chain 9	UniProt (SwissProt) Alternative ID(s) of Target Chain 9	UniProt (TrEMBL) Submitted Name of Target Chain 9	UniProt (TrEMBL) Entry Name of Target Chain 9	UniProt (TrEMBL) Primary ID of Target Chain 9	UniProt (TrEMBL) Secondary ID(s) of Target Chain 9	UniProt (TrEMBL) Alternative ID(s) of Target Chain 9	BindingDB Target Chain Sequence 10	PDB ID(s) of Target Chain 10	UniProt (SwissProt) Recommended Name of Target Chain 10	UniProt (SwissProt) Entry Name of Target Chain 10	UniProt (SwissProt) Primary ID of Target Chain 10	UniProt (SwissProt) Secondary ID(s) of Target Chain 10	UniProt (SwissProt) Alternative ID(s) of Target Chain 10	UniProt (TrEMBL) Submitted Name of Target Chain 10	UniProt (TrEMBL) Entry Name of Target Chain 10	UniProt (TrEMBL) Primary ID of Target Chain 10	UniProt (TrEMBL) Secondary ID(s) of Target Chain 10	UniProt (TrEMBL) Alternative ID(s) of Target Chain 10	BindingDB Target Chain Sequence 11	PDB ID(s) of Target Chain 11	UniProt (SwissProt) Recommended Name of Target Chain 11	UniProt (SwissProt) Entry Name of Target Chain 11	UniProt (SwissProt) Primary ID of Target Chain 11	UniProt (SwissProt) Secondary ID(s) of Target Chain 11	UniProt (SwissProt) Alternative ID(s) of Target Chain 11	UniProt (TrEMBL) Submitted Name of Target Chain 11	UniProt (TrEMBL) Entry Name of Target Chain 11	UniProt (TrEMBL) Primary ID of Target Chain 11	UniProt (TrEMBL) Secondary ID(s) of Target Chain 11	UniProt (TrEMBL) Alternative ID(s) of Target Chain 11	BindingDB Target Chain Sequence 12	PDB ID(s) of Target Chain 12	UniProt (SwissProt) Recommended Name of Target Chain 12	UniProt (SwissProt) Entry Name of Target Chain 12	UniProt (SwissProt) Primary ID of Target Chain 12	UniProt (SwissProt) Secondary ID(s) of Target Chain 12	UniProt (SwissProt) Alternative ID(s) of Target Chain 12	UniProt (TrEMBL) Submitted Name of Target Chain 12	UniProt (TrEMBL) Entry Name of Target Chain 12	UniProt (TrEMBL) Primary ID of Target Chain 12	UniProt (TrEMBL) Secondary ID(s) of Target Chain 12	UniProt (TrEMBL) Alternative ID(s) of Target Chain 12	BindingDB Target Chain Sequence 13	PDB ID(s) of Target Chain 13	UniProt (SwissProt) Recommended Name of Target Chain 13	UniProt (SwissProt) Entry Name of Target Chain 13	UniProt (SwissProt) Primary ID of Target Chain 13	UniProt (SwissProt) Secondary ID(s) of Target Chain 13	UniProt (SwissProt) Alternative ID(s) of Target Chain 13	UniProt (TrEMBL) Submitted Name of Target Chain 13	UniProt (TrEMBL) Entry Name of Target Chain 13	UniProt (TrEMBL) Primary ID of Target Chain 13	UniProt (TrEMBL) Secondary ID(s) of Target Chain 13	UniProt (TrEMBL) Alternative ID(s) of Target Chain 13	BindingDB Target Chain Sequence 14	PDB ID(s) of Target Chain 14	UniProt (SwissProt) Recommended Name of Target Chain 14	UniProt (SwissProt) Entry Name of Target Chain 14	UniProt (SwissProt) Primary ID of Target Chain 14	UniProt (SwissProt) Secondary ID(s) of Target Chain 14	UniProt (SwissProt) Alternative ID(s) of Target Chain 14	UniProt (TrEMBL) Submitted Name of Target Chain 14	UniProt (TrEMBL) Entry Name of Target Chain 14	UniProt (TrEMBL) Primary ID of Target Chain 14	UniProt (TrEMBL) Secondary ID(s) of Target Chain 14	UniProt (TrEMBL) Alternative ID(s) of Target Chain 14	BindingDB Target Chain Sequence 15	PDB ID(s) of Target Chain 15	UniProt (SwissProt) Recommended Name of Target Chain 15	UniProt (SwissProt) Entry Name of Target Chain 15	UniProt (SwissProt) Primary ID of Target Chain 15	UniProt (SwissProt) Secondary ID(s) of Target Chain 15	UniProt (SwissProt) Alternative ID(s) of Target Chain 15	UniProt (TrEMBL) Submitted Name of Target Chain 15	UniProt (TrEMBL) Entry Name of Target Chain 15	UniProt (TrEMBL) Primary ID of Target Chain 15	UniProt (TrEMBL) Secondary ID(s) of Target Chain 15	UniProt (TrEMBL) Alternative ID(s) of Target Chain 15	BindingDB Target Chain Sequence 16	PDB ID(s) of Target Chain 16	UniProt (SwissProt) Recommended Name of Target Chain 16	UniProt (SwissProt) Entry Name of Target Chain 16	UniProt (SwissProt) Primary ID of Target Chain 16	UniProt (SwissProt) Secondary ID(s) of Target Chain 16	UniProt (SwissProt) Alternative ID(s) of Target Chain 16	UniProt (TrEMBL) Submitted Name of Target Chain 16	UniProt (TrEMBL) Entry Name of Target Chain 16	UniProt (TrEMBL) Primary ID of Target Chain 16	UniProt (TrEMBL) Secondary ID(s) of Target Chain 16	UniProt (TrEMBL) Alternative ID(s) of Target Chain 16	BindingDB Target Chain Sequence 17	PDB ID(s) of Target Chain 17	UniProt (SwissProt) Recommended Name of Target Chain 17	UniProt (SwissProt) Entry Name of Target Chain 17	UniProt (SwissProt) Primary ID of Target Chain 17	UniProt (SwissProt) Secondary ID(s) of Target Chain 17	UniProt (SwissProt) Alternative ID(s) of Target Chain 17	UniProt (TrEMBL) Submitted Name of Target Chain 17	UniProt (TrEMBL) Entry Name of Target Chain 17	UniProt (TrEMBL) Primary ID of Target Chain 17	UniProt (TrEMBL) Secondary ID(s) of Target Chain 17	UniProt (TrEMBL) Alternative ID(s) of Target Chain 17	BindingDB Target Chain Sequence 18	PDB ID(s) of Target Chain 18	UniProt (SwissProt) Recommended Name of Target Chain 18	UniProt (SwissProt) Entry Name of Target Chain 18	UniProt (SwissProt) Primary ID of Target Chain 18	UniProt (SwissProt) Secondary ID(s) of Target Chain 18	UniProt (SwissProt) Alternative ID(s) of Target Chain 18	UniProt (TrEMBL) Submitted Name of Target Chain 18	UniProt (TrEMBL) Entry Name of Target Chain 18	UniProt (TrEMBL) Primary ID of Target Chain 18	UniProt (TrEMBL) Secondary ID(s) of Target Chain 18	UniProt (TrEMBL) Alternative ID(s) of Target Chain 18	BindingDB Target Chain Sequence 19	PDB ID(s) of Target Chain 19	UniProt (SwissProt) Recommended Name of Target Chain 19	UniProt (SwissProt) Entry Name of Target Chain 19	UniProt (SwissProt) Primary ID of Target Chain 19	UniProt (SwissProt) Secondary ID(s) of Target Chain 19	UniProt (SwissProt) Alternative ID(s) of Target Chain 19	UniProt (TrEMBL) Submitted Name of Target Chain 19	UniProt (TrEMBL) Entry Name of Target Chain 19	UniProt (TrEMBL) Primary ID of Target Chain 19	UniProt (TrEMBL) Secondary ID(s) of Target Chain 19	UniProt (TrEMBL) Alternative ID(s) of Target Chain 19	BindingDB Target Chain Sequence 20	PDB ID(s) of Target Chain 20	UniProt (SwissProt) Recommended Name of Target Chain 20	UniProt (SwissProt) Entry Name of Target Chain 20	UniProt (SwissProt) Primary ID of Target Chain 20	UniProt (SwissProt) Secondary ID(s) of Target Chain 20	UniProt (SwissProt) Alternative ID(s) of Target Chain 20	UniProt (TrEMBL) Submitted Name of Target Chain 20	UniProt (TrEMBL) Entry Name of Target Chain 20	UniProt (TrEMBL) Primary ID of Target Chain 20	UniProt (TrEMBL) Secondary ID(s) of Target Chain 20	UniProt (TrEMBL) Alternative ID(s) of Target Chain 20	BindingDB Target Chain Sequence 21	PDB ID(s) of Target Chain 21	UniProt (SwissProt) Recommended Name of Target Chain 21	UniProt (SwissProt) Entry Name of Target Chain 21	UniProt (SwissProt) Primary ID of Target Chain 21	UniProt (SwissProt) Secondary ID(s) of Target Chain 21	UniProt (SwissProt) Alternative ID(s) of Target Chain 21	UniProt (TrEMBL) Submitted Name of Target Chain 21	UniProt (TrEMBL) Entry Name of Target Chain 21	UniProt (TrEMBL) Primary ID of Target Chain 21	UniProt (TrEMBL) Secondary ID(s) of Target Chain 21	UniProt (TrEMBL) Alternative ID(s) of Target Chain 21	BindingDB Target Chain Sequence 22	PDB ID(s) of Target Chain 22	UniProt (SwissProt) Recommended Name of Target Chain 22	UniProt (SwissProt) Entry Name of Target Chain 22	UniProt (SwissProt) Primary ID of Target Chain 22	UniProt (SwissProt) Secondary ID(s) of Target Chain 22	UniProt (SwissProt) Alternative ID(s) of Target Chain 22	UniProt (TrEMBL) Submitted Name of Target Chain 22	UniProt (TrEMBL) Entry Name of Target Chain 22	UniProt (TrEMBL) Primary ID of Target Chain 22	UniProt (TrEMBL) Secondary ID(s) of Target Chain 22	UniProt (TrEMBL) Alternative ID(s) of Target Chain 22	BindingDB Target Chain Sequence 23	PDB ID(s) of Target Chain 23	UniProt (SwissProt) Recommended Name of Target Chain 23	UniProt (SwissProt) Entry Name of Target Chain 23	UniProt (SwissProt) Primary ID of Target Chain 23	UniProt (SwissProt) Secondary ID(s) of Target Chain 23	UniProt (SwissProt) Alternative ID(s) of Target Chain 23	UniProt (TrEMBL) Submitted Name of Target Chain 23	UniProt (TrEMBL) Entry Name of Target Chain 23	UniProt (TrEMBL) Primary ID of Target Chain 23	UniProt (TrEMBL) Secondary ID(s) of Target Chain 23	UniProt (TrEMBL) Alternative ID(s) of Target Chain 23	BindingDB Target Chain Sequence 24	PDB ID(s) of Target Chain 24	UniProt (SwissProt) Recommended Name of Target Chain 24	UniProt (SwissProt) Entry Name of Target Chain 24	UniProt (SwissProt) Primary ID of Target Chain 24	UniProt (SwissProt) Secondary ID(s) of Target Chain 24	UniProt (SwissProt) Alternative ID(s) of Target Chain 24	UniProt (TrEMBL) Submitted Name of Target Chain 24	UniProt (TrEMBL) Entry Name of Target Chain 24	UniProt (TrEMBL) Primary ID of Target Chain 24	UniProt (TrEMBL) Secondary ID(s) of Target Chain 24	UniProt (TrEMBL) Alternative ID(s) of Target Chain 24	BindingDB Target Chain Sequence 25	PDB ID(s) of Target Chain 25	UniProt (SwissProt) Recommended Name of Target Chain 25	UniProt (SwissProt) Entry Name of Target Chain 25	UniProt (SwissProt) Primary ID of Target Chain 25	UniProt (SwissProt) Secondary ID(s) of Target Chain 25	UniProt (SwissProt) Alternative ID(s) of Target Chain 25	UniProt (TrEMBL) Submitted Name of Target Chain 25	UniProt (TrEMBL) Entry Name of Target Chain 25	UniProt (TrEMBL) Primary ID of Target Chain 25	UniProt (TrEMBL) Secondary ID(s) of Target Chain 25	UniProt (TrEMBL) Alternative ID(s) of Target Chain 25	BindingDB Target Chain Sequence 26	PDB ID(s) of Target Chain 26	UniProt (SwissProt) Recommended Name of Target Chain 26	UniProt (SwissProt) Entry Name of Target Chain 26	UniProt (SwissProt) Primary ID of Target Chain 26	UniProt (SwissProt) Secondary ID(s) of Target Chain 26	UniProt (SwissProt) Alternative ID(s) of Target Chain 26	UniProt (TrEMBL) Submitted Name of Target Chain 26	UniProt (TrEMBL) Entry Name of Target Chain 26	UniProt (TrEMBL) Primary ID of Target Chain 26	UniProt (TrEMBL) Secondary ID(s) of Target Chain 26	UniProt (TrEMBL) Alternative ID(s) of Target Chain 26	BindingDB Target Chain Sequence 27	PDB ID(s) of Target Chain 27	UniProt (SwissProt) Recommended Name of Target Chain 27	UniProt (SwissProt) Entry Name of Target Chain 27	UniProt (SwissProt) Primary ID of Target Chain 27	UniProt (SwissProt) Secondary ID(s) of Target Chain 27	UniProt (SwissProt) Alternative ID(s) of Target Chain 27	UniProt (TrEMBL) Submitted Name of Target Chain 27	UniProt (TrEMBL) Entry Name of Target Chain 27	UniProt (TrEMBL) Primary ID of Target Chain 27	UniProt (TrEMBL) Secondary ID(s) of Target Chain 27	UniProt (TrEMBL) Alternative ID(s) of Target Chain 27	BindingDB Target Chain Sequence 28	PDB ID(s) of Target Chain 28	UniProt (SwissProt) Recommended Name of Target Chain 28	UniProt (SwissProt) Entry Name of Target Chain 28	UniProt (SwissProt) Primary ID of Target Chain 28	UniProt (SwissProt) Secondary ID(s) of Target Chain 28	UniProt (SwissProt) Alternative ID(s) of Target Chain 28	UniProt (TrEMBL) Submitted Name of Target Chain 28	UniProt (TrEMBL) Entry Name of Target Chain 28	UniProt (TrEMBL) Primary ID of Target Chain 28	UniProt (TrEMBL) Secondary ID(s) of Target Chain 28	UniProt (TrEMBL) Alternative ID(s) of Target Chain 28	BindingDB Target Chain Sequence 29	PDB ID(s) of Target Chain 29	UniProt (SwissProt) Recommended Name of Target Chain 29	UniProt (SwissProt) Entry Name of Target Chain 29	UniProt (SwissProt) Primary ID of Target Chain 29	UniProt (SwissProt) Secondary ID(s) of Target Chain 29	UniProt (SwissProt) Alternative ID(s) of Target Chain 29	UniProt (TrEMBL) Submitted Name of Target Chain 29	UniProt (TrEMBL) Entry Name of Target Chain 29	UniProt (TrEMBL) Primary ID of Target Chain 29	UniProt (TrEMBL) Secondary ID(s) of Target Chain 29	UniProt (TrEMBL) Alternative ID(s) of Target Chain 29	BindingDB Target Chain Sequence 30	PDB ID(s) of Target Chain 30	UniProt (SwissProt) Recommended Name of Target Chain 30	UniProt (SwissProt) Entry Name of Target Chain 30	UniProt (SwissProt) Primary ID of Target Chain 30	UniProt (SwissProt) Secondary ID(s) of Target Chain 30	UniProt (SwissProt) Alternative ID(s) of Target Chain 30	UniProt (TrEMBL) Submitted Name of Target Chain 30	UniProt (TrEMBL) Entry Name of Target Chain 30	UniProt (TrEMBL) Primary ID of Target Chain 30	UniProt (TrEMBL) Secondary ID(s) of Target Chain 30	UniProt (TrEMBL) Alternative ID(s) of Target Chain 30	BindingDB Target Chain Sequence 31	PDB ID(s) of Target Chain 31	UniProt (SwissProt) Recommended Name of Target Chain 31	UniProt (SwissProt) Entry Name of Target Chain 31	UniProt (SwissProt) Primary ID of Target Chain 31	UniProt (SwissProt) Secondary ID(s) of Target Chain 31	UniProt (SwissProt) Alternative ID(s) of Target Chain 31	UniProt (TrEMBL) Submitted Name of Target Chain 31	UniProt (TrEMBL) Entry Name of Target Chain 31	UniProt (TrEMBL) Primary ID of Target Chain 31	UniProt (TrEMBL) Secondary ID(s) of Target Chain 31	UniProt (TrEMBL) Alternative ID(s) of Target Chain 31	BindingDB Target Chain Sequence 32	PDB ID(s) of Target Chain 32	UniProt (SwissProt) Recommended Name of Target Chain 32	UniProt (SwissProt) Entry Name of Target Chain 32	UniProt (SwissProt) Primary ID of Target Chain 32	UniProt (SwissProt) Secondary ID(s) of Target Chain 32	UniProt (SwissProt) Alternative ID(s) of Target Chain 32	UniProt (TrEMBL) Submitted Name of Target Chain 32	UniProt (TrEMBL) Entry Name of Target Chain 32	UniProt (TrEMBL) Primary ID of Target Chain 32	UniProt (TrEMBL) Secondary ID(s) of Target Chain 32	UniProt (TrEMBL) Alternative ID(s) of Target Chain 32	BindingDB Target Chain Sequence 33	PDB ID(s) of Target Chain 33	UniProt (SwissProt) Recommended Name of Target Chain 33	UniProt (SwissProt) Entry Name of Target Chain 33	UniProt (SwissProt) Primary ID of Target Chain 33	UniProt (SwissProt) Secondary ID(s) of Target Chain 33	UniProt (SwissProt) Alternative ID(s) of Target Chain 33	UniProt (TrEMBL) Submitted Name of Target Chain 33	UniProt (TrEMBL) Entry Name of Target Chain 33	UniProt (TrEMBL) Primary ID of Target Chain 33	UniProt (TrEMBL) Secondary ID(s) of Target Chain 33	UniProt (TrEMBL) Alternative ID(s) of Target Chain 33	BindingDB Target Chain Sequence 34	PDB ID(s) of Target Chain 34	UniProt (SwissProt) Recommended Name of Target Chain 34	UniProt (SwissProt) Entry Name of Target Chain 34	UniProt (SwissProt) Primary ID of Target Chain 34	UniProt (SwissProt) Secondary ID(s) of Target Chain 34	UniProt (SwissProt) Alternative ID(s) of Target Chain 34	UniProt (TrEMBL) Submitted Name of Target Chain 34	UniProt (TrEMBL) Entry Name of Target Chain 34	UniProt (TrEMBL) Primary ID of Target Chain 34	UniProt (TrEMBL) Secondary ID(s) of Target Chain 34	UniProt (TrEMBL) Alternative ID(s) of Target Chain 34	BindingDB Target Chain Sequence 35	PDB ID(s) of Target Chain 35	UniProt (SwissProt) Recommended Name of Target Chain 35	UniProt (SwissProt) Entry Name of Target Chain 35	UniProt (SwissProt) Primary ID of Target Chain 35	UniProt (SwissProt) Secondary ID(s) of Target Chain 35	UniProt (SwissProt) Alternative ID(s) of Target Chain 35	UniProt (TrEMBL) Submitted Name of Target Chain 35	UniProt (TrEMBL) Entry Name of Target Chain 35	UniProt (TrEMBL) Primary ID of Target Chain 35	UniProt (TrEMBL) Secondary ID(s) of Target Chain 35	UniProt (TrEMBL) Alternative ID(s) of Target Chain 35	BindingDB Target Chain Sequence 36	PDB ID(s) of Target Chain 36	UniProt (SwissProt) Recommended Name of Target Chain 36	UniProt (SwissProt) Entry Name of Target Chain 36	UniProt (SwissProt) Primary ID of Target Chain 36	UniProt (SwissProt) Secondary ID(s) of Target Chain 36	UniProt (SwissProt) Alternative ID(s) of Target Chain 36	UniProt (TrEMBL) Submitted Name of Target Chain 36	UniProt (TrEMBL) Entry Name of Target Chain 36	UniProt (TrEMBL) Primary ID of Target Chain 36	UniProt (TrEMBL) Secondary ID(s) of Target Chain 36	UniProt (TrEMBL) Alternative ID(s) of Target Chain 36	BindingDB Target Chain Sequence 37	PDB ID(s) of Target Chain 37	UniProt (SwissProt) Recommended Name of Target Chain 37	UniProt (SwissProt) Entry Name of Target Chain 37	UniProt (SwissProt) Primary ID of Target Chain 37	UniProt (SwissProt) Secondary ID(s) of Target Chain 37	UniProt (SwissProt) Alternative ID(s) of Target Chain 37	UniProt (TrEMBL) Submitted Name of Target Chain 37	UniProt (TrEMBL) Entry Name of Target Chain 37	UniProt (TrEMBL) Primary ID of Target Chain 37	UniProt (TrEMBL) Secondary ID(s) of Target Chain 37	UniProt (TrEMBL) Alternative ID(s) of Target Chain 37	BindingDB Target Chain Sequence 38	PDB ID(s) of Target Chain 38	UniProt (SwissProt) Recommended Name of Target Chain 38	UniProt (SwissProt) Entry Name of Target Chain 38	UniProt (SwissProt) Primary ID of Target Chain 38	UniProt (SwissProt) Secondary ID(s) of Target Chain 38	UniProt (SwissProt) Alternative ID(s) of Target Chain 38	UniProt (TrEMBL) Submitted Name of Target Chain 38	UniProt (TrEMBL) Entry Name of Target Chain 38	UniProt (TrEMBL) Primary ID of Target Chain 38	UniProt (TrEMBL) Secondary ID(s) of Target Chain 38	UniProt (TrEMBL) Alternative ID(s) of Target Chain 38	BindingDB Target Chain Sequence 39	PDB ID(s) of Target Chain 39	UniProt (SwissProt) Recommended Name of Target Chain 39	UniProt (SwissProt) Entry Name of Target Chain 39	UniProt (SwissProt) Primary ID of Target Chain 39	UniProt (SwissProt) Secondary ID(s) of Target Chain 39	UniProt (SwissProt) Alternative ID(s) of Target Chain 39	UniProt (TrEMBL) Submitted Name of Target Chain 39	UniProt (TrEMBL) Entry Name of Target Chain 39	UniProt (TrEMBL) Primary ID of Target Chain 39	UniProt (TrEMBL) Secondary ID(s) of Target Chain 39	UniProt (TrEMBL) Alternative ID(s) of Target Chain 39	BindingDB Target Chain Sequence 40	PDB ID(s) of Target Chain 40	UniProt (SwissProt) Recommended Name of Target Chain 40	UniProt (SwissProt) Entry Name of Target Chain 40	UniProt (SwissProt) Primary ID of Target Chain 40	UniProt (SwissProt) Secondary ID(s) of Target Chain 40	UniProt (SwissProt) Alternative ID(s) of Target Chain 40	UniProt (TrEMBL) Submitted Name of Target Chain 40	UniProt (TrEMBL) Entry Name of Target Chain 40	UniProt (TrEMBL) Primary ID of Target Chain 40	UniProt (TrEMBL) Secondary ID(s) of Target Chain 40	UniProt (TrEMBL) Alternative ID(s) of Target Chain 40	BindingDB Target Chain Sequence 41	PDB ID(s) of Target Chain 41	UniProt (SwissProt) Recommended Name of Target Chain 41	UniProt (SwissProt) Entry Name of Target Chain 41	UniProt (SwissProt) Primary ID of Target Chain 41	UniProt (SwissProt) Secondary ID(s) of Target Chain 41	UniProt (SwissProt) Alternative ID(s) of Target Chain 41	UniProt (TrEMBL) Submitted Name of Target Chain 41	UniProt (TrEMBL) Entry Name of Target Chain 41	UniProt (TrEMBL) Primary ID of Target Chain 41	UniProt (TrEMBL) Secondary ID(s) of Target Chain 41	UniProt (TrEMBL) Alternative ID(s) of Target Chain 41	BindingDB Target Chain Sequence 42	PDB ID(s) of Target Chain 42	UniProt (SwissProt) Recommended Name of Target Chain 42	UniProt (SwissProt) Entry Name of Target Chain 42	UniProt (SwissProt) Primary ID of Target Chain 42	UniProt (SwissProt) Secondary ID(s) of Target Chain 42	UniProt (SwissProt) Alternative ID(s) of Target Chain 42	UniProt (TrEMBL) Submitted Name of Target Chain 42	UniProt (TrEMBL) Entry Name of Target Chain 42	UniProt (TrEMBL) Primary ID of Target Chain 42	UniProt (TrEMBL) Secondary ID(s) of Target Chain 42	UniProt (TrEMBL) Alternative ID(s) of Target Chain 42	BindingDB Target Chain Sequence 43	PDB ID(s) of Target Chain 43	UniProt (SwissProt) Recommended Name of Target Chain 43	UniProt (SwissProt) Entry Name of Target Chain 43	UniProt (SwissProt) Primary ID of Target Chain 43	UniProt (SwissProt) Secondary ID(s) of Target Chain 43	UniProt (SwissProt) Alternative ID(s) of Target Chain 43	UniProt (TrEMBL) Submitted Name of Target Chain 43	UniProt (TrEMBL) Entry Name of Target Chain 43	UniProt (TrEMBL) Primary ID of Target Chain 43	UniProt (TrEMBL) Secondary ID(s) of Target Chain 43	UniProt (TrEMBL) Alternative ID(s) of Target Chain 43	BindingDB Target Chain Sequence 44	PDB ID(s) of Target Chain 44	UniProt (SwissProt) Recommended Name of Target Chain 44	UniProt (SwissProt) Entry Name of Target Chain 44	UniProt (SwissProt) Primary ID of Target Chain 44	UniProt (SwissProt) Secondary ID(s) of Target Chain 44	UniProt (SwissProt) Alternative ID(s) of Target Chain 44	UniProt (TrEMBL) Submitted Name of Target Chain 44	UniProt (TrEMBL) Entry Name of Target Chain 44	UniProt (TrEMBL) Primary ID of Target Chain 44	UniProt (TrEMBL) Secondary ID(s) of Target Chain 44	UniProt (TrEMBL) Alternative ID(s) of Target Chain 44	BindingDB Target Chain Sequence 45	PDB ID(s) of Target Chain 45	UniProt (SwissProt) Recommended Name of Target Chain 45	UniProt (SwissProt) Entry Name of Target Chain 45	UniProt (SwissProt) Primary ID of Target Chain 45	UniProt (SwissProt) Secondary ID(s) of Target Chain 45	UniProt (SwissProt) Alternative ID(s) of Target Chain 45	UniProt (TrEMBL) Submitted Name of Target Chain 45	UniProt (TrEMBL) Entry Name of Target Chain 45	UniProt (TrEMBL) Primary ID of Target Chain 45	UniProt (TrEMBL) Secondary ID(s) of Target Chain 45	UniProt (TrEMBL) Alternative ID(s) of Target Chain 45	BindingDB Target Chain Sequence 46	PDB ID(s) of Target Chain 46	UniProt (SwissProt) Recommended Name of Target Chain 46	UniProt (SwissProt) Entry Name of Target Chain 46	UniProt (SwissProt) Primary ID of Target Chain 46	UniProt (SwissProt) Secondary ID(s) of Target Chain 46	UniProt (SwissProt) Alternative ID(s) of Target Chain 46	UniProt (TrEMBL) Submitted Name of Target Chain 46	UniProt (TrEMBL) Entry Name of Target Chain 46	UniProt (TrEMBL) Primary ID of Target Chain 46	UniProt (TrEMBL) Secondary ID(s) of Target Chain 46	UniProt (TrEMBL) Alternative ID(s) of Target Chain 46	BindingDB Target Chain Sequence 47	PDB ID(s) of Target Chain 47	UniProt (SwissProt) Recommended Name of Target Chain 47	UniProt (SwissProt) Entry Name of Target Chain 47	UniProt (SwissProt) Primary ID of Target Chain 47	UniProt (SwissProt) Secondary ID(s) of Target Chain 47	UniProt (SwissProt) Alternative ID(s) of Target Chain 47	UniProt (TrEMBL) Submitted Name of Target Chain 47	UniProt (TrEMBL) Entry Name of Target Chain 47	UniProt (TrEMBL) Primary ID of Target Chain 47	UniProt (TrEMBL) Secondary ID(s) of Target Chain 47	UniProt (TrEMBL) Alternative ID(s) of Target Chain 47	BindingDB Target Chain Sequence 48	PDB ID(s) of Target Chain 48	UniProt (SwissProt) Recommended Name of Target Chain 48	UniProt (SwissProt) Entry Name of Target Chain 48	UniProt (SwissProt) Primary ID of Target Chain 48	UniProt (SwissProt) Secondary ID(s) of Target Chain 48	UniProt (SwissProt) Alternative ID(s) of Target Chain 48	UniProt (TrEMBL) Submitted Name of Target Chain 48	UniProt (TrEMBL) Entry Name of Target Chain 48	UniProt (TrEMBL) Primary ID of Target Chain 48	UniProt (TrEMBL) Secondary ID(s) of Target Chain 48	UniProt (TrEMBL) Alternative ID(s) of Target Chain 48	BindingDB Target Chain Sequence 49	PDB ID(s) of Target Chain 49	UniProt (SwissProt) Recommended Name of Target Chain 49	UniProt (SwissProt) Entry Name of Target Chain 49	UniProt (SwissProt) Primary ID of Target Chain 49	UniProt (SwissProt) Secondary ID(s) of Target Chain 49	UniProt (SwissProt) Alternative ID(s) of Target Chain 49	UniProt (TrEMBL) Submitted Name of Target Chain 49	UniProt (TrEMBL) Entry Name of Target Chain 49	UniProt (TrEMBL) Primary ID of Target Chain 49	UniProt (TrEMBL) Secondary ID(s) of Target Chain 49	UniProt (TrEMBL) Alternative ID(s) of Target Chain 49	BindingDB Target Chain Sequence 50	PDB ID(s) of Target Chain 50	UniProt (SwissProt) Recommended Name of Target Chain 50	UniProt (SwissProt) Entry Name of Target Chain 50	UniProt (SwissProt) Primary ID of Target Chain 50	UniProt (SwissProt) Secondary ID(s) of Target Chain 50	UniProt (SwissProt) Alternative ID(s) of Target Chain 50	UniProt (TrEMBL) Submitted Name of Target Chain 50	UniProt (TrEMBL) Entry Name of Target Chain 50	UniProt (TrEMBL) Primary ID of Target Chain 50	UniProt (TrEMBL) Secondary ID(s) of Target Chain 50	UniProt (TrEMBL) Alternative ID(s) of Target Chain 50
238165	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2ccccc2s1	InChI=1S/C25H20N2O4S/c1-15-6-8-18(26-24(28)17-7-9-20-21(12-17)31-11-10-30-20)14-19(15)27-25(29)23-13-16-4-2-3-5-22(16)32-23/h2-9,12-14H,10-11H2,1H3,(H,26,28)(H,27,29)	LBQVSHNCMINYRK-UHFFFAOYSA-N	536036	US20260028334, Example 1	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=536036	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=536036&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			153283935	464921214							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238166	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2cc(Cl)ccc2o1	InChI=1S/C25H19ClN2O5/c1-14-2-5-18(27-24(29)15-3-6-21-22(11-15)32-9-8-31-21)13-19(14)28-25(30)23-12-16-10-17(26)4-7-20(16)33-23/h2-7,10-13H,8-9H2,1H3,(H,27,29)(H,28,30)	HXIWUYAUNYTRMH-UHFFFAOYSA-N	536037	US20260028334, Example 1/1	L-lactate dehydrogenase A chain	Homo sapiens		 550							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=536037	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=536037&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			138491408	464921215							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238167	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2ccccc2o1	InChI=1S/C25H20N2O5/c1-15-6-8-18(26-24(28)17-7-9-21-22(13-17)31-11-10-30-21)14-19(15)27-25(29)23-12-16-4-2-3-5-20(16)32-23/h2-9,12-14H,10-11H2,1H3,(H,26,28)(H,27,29)	GYJUNEDJRWRDQX-UHFFFAOYSA-N	536038	US20260028334, Example 1/2	L-lactate dehydrogenase A chain	Homo sapiens		 5500							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=536038	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=536038&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			153283921	464921216							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238168	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2cc(C(F)(F)F)ccc2[nH]1	InChI=1S/C26H20F3N3O4/c1-14-2-5-18(30-24(33)15-3-7-22-23(12-15)36-9-8-35-22)13-20(14)32-25(34)21-11-16-10-17(26(27,28)29)4-6-19(16)31-21/h2-7,10-13,31H,8-9H2,1H3,(H,30,33)(H,32,34)	YUEHDVFPJHKLEU-UHFFFAOYSA-N	540097	US20260028334, Example 1/3	L-lactate dehydrogenase A chain	Homo sapiens		 550							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540097	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540097&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447213	464925083							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238169	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2cccnc2[nH]1	InChI=1S/C24H20N4O4/c1-14-4-6-17(26-23(29)16-5-7-20-21(12-16)32-10-9-31-20)13-18(14)28-24(30)19-11-15-3-2-8-25-22(15)27-19/h2-8,11-13H,9-10H2,1H3,(H,25,27)(H,26,29)(H,28,30)	VTSVWYZDTZUDIQ-UHFFFAOYSA-N	540098	US20260028334, Example 1/4	L-lactate dehydrogenase A chain	Homo sapiens		 550							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540098	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540098&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121446917	464925084							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238170	COc1ccc2[nH]c(C(=O)Nc3cc(NC(=O)c4ccc5c(c4)OCCO5)ccc3C)cc2c1	InChI=1S/C26H23N3O5/c1-15-3-5-18(27-25(30)16-4-8-23-24(13-16)34-10-9-33-23)14-21(15)29-26(31)22-12-17-11-19(32-2)6-7-20(17)28-22/h3-8,11-14,28H,9-10H2,1-2H3,(H,27,30)(H,29,31)	UVOQSYODOLRDQV-UHFFFAOYSA-N	540099	US20260028334, Example 1/5	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540099	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540099&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121446980	464925085							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238171	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2cc(Cl)ccc2[nH]1	InChI=1S/C25H20ClN3O4/c1-14-2-5-18(27-24(30)15-3-7-22-23(12-15)33-9-8-32-22)13-20(14)29-25(31)21-11-16-10-17(26)4-6-19(16)28-21/h2-7,10-13,28H,8-9H2,1H3,(H,27,30)(H,29,31)	VFBGZMCMRXXDBC-UHFFFAOYSA-N	540100	US20260028334, Example 1/6	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540100	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540100&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447019	464925086							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238172	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2cc(Cl)cnc2[nH]1	InChI=1S/C24H19ClN4O4/c1-13-2-4-17(27-23(30)14-3-5-20-21(10-14)33-7-6-32-20)11-18(13)29-24(31)19-9-15-8-16(25)12-26-22(15)28-19/h2-5,8-12H,6-7H2,1H3,(H,26,28)(H,27,30)(H,29,31)	USRBYWNFWRXLSN-UHFFFAOYSA-N	540101	US20260028334, Example 1/7	L-lactate dehydrogenase A chain	Homo sapiens		 550							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540101	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540101&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121446981	464925087							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238173	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2ccccc2[nH]1	InChI=1S/C25H21N3O4/c1-15-6-8-18(26-24(29)17-7-9-22-23(13-17)32-11-10-31-22)14-20(15)28-25(30)21-12-16-4-2-3-5-19(16)27-21/h2-9,12-14,27H,10-11H2,1H3,(H,26,29)(H,28,30)	MCLKVLDUNICMGV-UHFFFAOYSA-N	540102	US20260028334, Example 1/8	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540102	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540102&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447095	464925088							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238174	O=C(Nc1ccc(F)c(NC(=O)c2cc3ccccc3[nH]2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C24H18FN3O4/c25-17-7-6-16(26-23(29)15-5-8-21-22(12-15)32-10-9-31-21)13-19(17)28-24(30)20-11-14-3-1-2-4-18(14)27-20/h1-8,11-13,27H,9-10H2,(H,26,29)(H,28,30)	ALYVRQROONSTAD-UHFFFAOYSA-N	540103	US20260028334, Example 1/9	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540103	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540103&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121446998	464925089							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238175	O=C(Nc1ccc(Cl)c(NC(=O)c2cc3ccccc3[nH]2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C24H18ClN3O4/c25-17-7-6-16(26-23(29)15-5-8-21-22(12-15)32-10-9-31-21)13-19(17)28-24(30)20-11-14-3-1-2-4-18(14)27-20/h1-8,11-13,27H,9-10H2,(H,26,29)(H,28,30)	OBPYNKVVJCVHLG-UHFFFAOYSA-N	540104	US20260028334, Example 1/10	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540104	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540104&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447022	464925090							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238176	Cc1ccc2sc(C(=O)Nc3cc(NC(=O)c4ccc5c(c4)OCCO5)ccc3C)cc2c1	InChI=1S/C26H22N2O4S/c1-15-3-8-23-18(11-15)13-24(33-23)26(30)28-20-14-19(6-4-16(20)2)27-25(29)17-5-7-21-22(12-17)32-10-9-31-21/h3-8,11-14H,9-10H2,1-2H3,(H,27,29)(H,28,30)	VQXRPSZUIJCUJH-UHFFFAOYSA-N	540105	US20260028334, Example 1/11	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540105	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540105&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447108	464925091							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238177	COc1ccc2cc(C(=O)Nc3cc(NC(=O)c4ccc5c(c4)OCCO5)ccc3C)sc2c1	InChI=1S/C26H22N2O5S/c1-15-3-6-18(27-25(29)17-5-8-21-22(11-17)33-10-9-32-21)13-20(15)28-26(30)24-12-16-4-7-19(31-2)14-23(16)34-24/h3-8,11-14H,9-10H2,1-2H3,(H,27,29)(H,28,30)	LBQDSOILIYVSLF-UHFFFAOYSA-N	540106	US20260028334, Example 1/12	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540106	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540106&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447116	464925092							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238178	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2cc(C(F)(F)F)ccc2s1	InChI=1S/C26H19F3N2O4S/c1-14-2-5-18(30-24(32)15-3-6-20-21(11-15)35-9-8-34-20)13-19(14)31-25(33)23-12-16-10-17(26(27,28)29)4-7-22(16)36-23/h2-7,10-13H,8-9H2,1H3,(H,30,32)(H,31,33)	RKBOEUKOLSGUGR-UHFFFAOYSA-N	540107	US20260028334, Example 1/13	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540107	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540107&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121446987	464925093							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238179	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2cc(F)ccc2s1	InChI=1S/C25H19FN2O4S/c1-14-2-5-18(27-24(29)15-3-6-20-21(11-15)32-9-8-31-20)13-19(14)28-25(30)23-12-16-10-17(26)4-7-22(16)33-23/h2-7,10-13H,8-9H2,1H3,(H,27,29)(H,28,30)	BYMNOUXLNCIIQU-UHFFFAOYSA-N	540108	US20260028334, Example 1/14	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540108	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540108&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447032	464925094							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238180	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2ccc(C(F)(F)F)cc2s1	InChI=1S/C26H19F3N2O4S/c1-14-2-6-18(30-24(32)16-4-7-20-21(10-16)35-9-8-34-20)13-19(14)31-25(33)23-11-15-3-5-17(26(27,28)29)12-22(15)36-23/h2-7,10-13H,8-9H2,1H3,(H,30,32)(H,31,33)	YSLTXSDGOQUTFH-UHFFFAOYSA-N	540109	US20260028334, Example 1/15	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540109	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540109&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447035	464925095							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238181	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1sc2cc(F)ccc2c1Cl	InChI=1S/C25H18ClFN2O4S/c1-13-2-5-16(28-24(30)14-3-7-19-20(10-14)33-9-8-32-19)12-18(13)29-25(31)23-22(26)17-6-4-15(27)11-21(17)34-23/h2-7,10-12H,8-9H2,1H3,(H,28,30)(H,29,31)	JKFSMRXMGCVHNH-UHFFFAOYSA-N	540110	US20260028334, Example 1/16	L-lactate dehydrogenase A chain	Homo sapiens		 5500							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540110	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540110&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447037	464925096							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238182	O=C(Nc1ccc(F)c(NC(=O)c2cc3ccccc3s2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C24H17FN2O4S/c25-17-7-6-16(26-23(28)15-5-8-19-20(11-15)31-10-9-30-19)13-18(17)27-24(29)22-12-14-3-1-2-4-21(14)32-22/h1-8,11-13H,9-10H2,(H,26,28)(H,27,29)	UJQJRRNTHQRHDM-UHFFFAOYSA-N	540111	US20260028334, Example 1/17	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540111	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540111&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447040	464925097							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238183	O=C(Nc1ccc(Cl)c(NC(=O)c2cc3ccccc3s2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C24H17ClN2O4S/c25-17-7-6-16(26-23(28)15-5-8-19-20(11-15)31-10-9-30-19)13-18(17)27-24(29)22-12-14-3-1-2-4-21(14)32-22/h1-8,11-13H,9-10H2,(H,26,28)(H,27,29)	SOYXJUJBANQUPI-UHFFFAOYSA-N	540112	US20260028334, Example 1/18	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540112	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540112&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447000	464925098							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238184	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1sc2ccccc2c1Cl	InChI=1S/C25H19ClN2O4S/c1-14-6-8-16(27-24(29)15-7-9-19-20(12-15)32-11-10-31-19)13-18(14)28-25(30)23-22(26)17-4-2-3-5-21(17)33-23/h2-9,12-13H,10-11H2,1H3,(H,27,29)(H,28,30)	JCKXYDQFOIAAKR-UHFFFAOYSA-N	540113	US20260028334, Example 1/19	L-lactate dehydrogenase A chain	Homo sapiens		 5500							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540113	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540113&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447141	464925099							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238185	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2ccc(O)cc2[nH]1	InChI=1S/C25H21N3O5/c1-14-2-5-17(26-24(30)16-4-7-22-23(11-16)33-9-8-32-22)12-19(14)28-25(31)21-10-15-3-6-18(29)13-20(15)27-21/h2-7,10-13,27,29H,8-9H2,1H3,(H,26,30)(H,28,31)	LBFDTVCLGXGBLX-UHFFFAOYSA-N	540114	US20260028334, Example 2	L-lactate dehydrogenase A chain	Homo sapiens		 550							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540114	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540114&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121446924	464925100							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238186	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2ccc(O)cc2[nH]1	InChI=1S/C25H21N3O5/c1-14-2-5-17(26-24(30)16-4-7-22-23(11-16)33-9-8-32-22)12-19(14)28-25(31)21-10-15-3-6-18(29)13-20(15)27-21/h2-7,10-13,27,29H,8-9H2,1H3,(H,26,30)(H,28,31)	LBFDTVCLGXGBLX-UHFFFAOYSA-N	540115	US20260028334, Example 2/1	L-lactate dehydrogenase A chain	Homo sapiens		 550							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540115	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540115&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447001	464925101							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238187	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2ccc(OCc3ccccn3)cc2s1	InChI=1S/C31H25N3O5S/c1-19-5-8-22(33-30(35)21-7-10-26-27(14-21)38-13-12-37-26)16-25(19)34-31(36)29-15-20-6-9-24(17-28(20)40-29)39-18-23-4-2-3-11-32-23/h2-11,14-17H,12-13,18H2,1H3,(H,33,35)(H,34,36)	FXSVMBHRXBRKGI-UHFFFAOYSA-N	540116	US20260028334, Example 3	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540116	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540116&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447298	464925102							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238188	O=C(Nc1ccc(F)c(NC(=O)c2cc3ccc(OCc4ccccn4)cc3s2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C30H22FN3O5S/c31-23-8-6-20(33-29(35)19-5-9-25-26(13-19)38-12-11-37-25)15-24(23)34-30(36)28-14-18-4-7-22(16-27(18)40-28)39-17-21-3-1-2-10-32-21/h1-10,13-16H,11-12,17H2,(H,33,35)(H,34,36)	CZBQSNPQWZRPFG-UHFFFAOYSA-N	540117	US20260028334, Example 3/1	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540117	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540117&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447144	464925103							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238189	O=C(Nc1ccc(Cl)c(NC(=O)c2cc3ccc(OCc4ccccn4)cc3s2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C30H22ClN3O5S/c31-23-8-6-20(33-29(35)19-5-9-25-26(13-19)38-12-11-37-25)15-24(23)34-30(36)28-14-18-4-7-22(16-27(18)40-28)39-17-21-3-1-2-10-32-21/h1-10,13-16H,11-12,17H2,(H,33,35)(H,34,36)	TYNPMVOTJKBUNB-UHFFFAOYSA-N	540118	US20260028334, Example 3/2	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540118	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540118&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121446923	464925104							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238190	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2ccc(OCCc3ccccn3)cc2s1	InChI=1S/C32H27N3O5S/c1-20-5-8-24(34-31(36)22-7-10-27-28(16-22)40-15-14-39-27)18-26(20)35-32(37)30-17-21-6-9-25(19-29(21)41-30)38-13-11-23-4-2-3-12-33-23/h2-10,12,16-19H,11,13-15H2,1H3,(H,34,36)(H,35,37)	YRPBKWOATFKTDP-UHFFFAOYSA-N	540119	US20260028334, Example 3/3	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540119	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540119&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121446925	464925105							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238191	O=C(Nc1ccc(F)c(NC(=O)c2cc3ccc(OCCc4ccccn4)cc3s2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C31H24FN3O5S/c32-24-8-6-22(34-30(36)20-5-9-26-27(15-20)40-14-13-39-26)17-25(24)35-31(37)29-16-19-4-7-23(18-28(19)41-29)38-12-10-21-3-1-2-11-33-21/h1-9,11,15-18H,10,12-14H2,(H,34,36)(H,35,37)	KPWZAPYZKOPQHY-UHFFFAOYSA-N	540120	US20260028334, Example 3/4	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540120	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540120&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447257	464925106							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238192	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2cc(OCCCN3CCCC3)ccc2s1	InChI=1S/C32H33N3O5S/c1-21-5-7-24(33-31(36)22-6-9-27-28(18-22)40-16-15-39-27)20-26(21)34-32(37)30-19-23-17-25(8-10-29(23)41-30)38-14-4-13-35-11-2-3-12-35/h5-10,17-20H,2-4,11-16H2,1H3,(H,33,36)(H,34,37)	SZFKYFNWPKAIOL-UHFFFAOYSA-N	540121	US20260028334, Example 3/5	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540121	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540121&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121446989	464925107							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238193	O=C(Nc1ccc(F)c(NC(=O)c2cc3cc(OCCCN4CCCC4)ccc3s2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C31H30FN3O5S/c32-24-7-5-22(33-30(36)20-4-8-26-27(17-20)40-15-14-39-26)19-25(24)34-31(37)29-18-21-16-23(6-9-28(21)41-29)38-13-3-12-35-10-1-2-11-35/h4-9,16-19H,1-3,10-15H2,(H,33,36)(H,34,37)	YBIPRHXMYJIFGN-UHFFFAOYSA-N	540122	US20260028334, Example 3/6	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540122	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540122&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447265	464925108							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238194	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2ccc(OCCCN3CCCC3)cc2s1	InChI=1S/C32H33N3O5S/c1-21-5-8-24(33-31(36)23-7-10-27-28(17-23)40-16-15-39-27)19-26(21)34-32(37)30-18-22-6-9-25(20-29(22)41-30)38-14-4-13-35-11-2-3-12-35/h5-10,17-20H,2-4,11-16H2,1H3,(H,33,36)(H,34,37)	NUGVNKWOFTUQRR-UHFFFAOYSA-N	540123	US20260028334, Example 3/7	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540123	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540123&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447042	464925109							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238195	O=C(Nc1ccc(F)c(NC(=O)c2cc3ccc(OCCCN4CCCC4)cc3s2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C31H30FN3O5S/c32-24-8-6-22(33-30(36)21-5-9-26-27(16-21)40-15-14-39-26)18-25(24)34-31(37)29-17-20-4-7-23(19-28(20)41-29)38-13-3-12-35-10-1-2-11-35/h4-9,16-19H,1-3,10-15H2,(H,33,36)(H,34,37)	RVUFPHWOLGXOFK-UHFFFAOYSA-N	540124	US20260028334, Example 3/8	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540124	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540124&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447044	464925110							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238196	O=C(Nc1ccc(Cl)c(NC(=O)c2cc3ccc(OCCCN4CCCC4)cc3s2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C31H30ClN3O5S/c32-24-8-6-22(33-30(36)21-5-9-26-27(16-21)40-15-14-39-26)18-25(24)34-31(37)29-17-20-4-7-23(19-28(20)41-29)38-13-3-12-35-10-1-2-11-35/h4-9,16-19H,1-3,10-15H2,(H,33,36)(H,34,37)	MNJBIWFSCWQPNF-UHFFFAOYSA-N	540125	US20260028334, Example 3/9	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540125	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540125&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447045	464925111							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238197	O=C(Nc1ccc(F)c(NC(=O)c2cc3ccc(OCCN4CCCC4)cc3s2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C30H28FN3O5S/c31-23-7-5-21(32-29(35)20-4-8-25-26(15-20)39-14-13-38-25)17-24(23)33-30(36)28-16-19-3-6-22(18-27(19)40-28)37-12-11-34-9-1-2-10-34/h3-8,15-18H,1-2,9-14H2,(H,32,35)(H,33,36)	CRPVXPXZZPDDNK-UHFFFAOYSA-N	540126	US20260028334, Example 3/10	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540126	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540126&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121446984	464925112							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238198	COc1ccc2[nH]c(C(=O)Nc3cc(NC(=O)c4ccc5c(c4)OCCO5)ccc3F)cc2c1	InChI=1S/C25H20FN3O5/c1-32-17-4-6-19-15(10-17)11-21(28-19)25(31)29-20-13-16(3-5-18(20)26)27-24(30)14-2-7-22-23(12-14)34-9-8-33-22/h2-7,10-13,28H,8-9H2,1H3,(H,27,30)(H,29,31)	KDMDUCOBLVAVPN-UHFFFAOYSA-N	540127	US20260028334, Example 3/11	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540127	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540127&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447046	464925113							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238199	O=C(Nc1ccc(F)c(NC(=O)c2cc3cc(C(F)(F)F)ccc3s2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C25H16F4N2O4S/c26-17-4-3-16(30-23(32)13-1-5-19-20(10-13)35-8-7-34-19)12-18(17)31-24(33)22-11-14-9-15(25(27,28)29)2-6-21(14)36-22/h1-6,9-12H,7-8H2,(H,30,32)(H,31,33)	LSWDLNDGKMCZDB-UHFFFAOYSA-N	540128	US20260028334, Example 3/12	L-lactate dehydrogenase A chain	Homo sapiens		 550							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540128	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540128&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447262	464925114							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238200	O=C(Nc1ccc(F)c(NC(=O)c2cc3cc(F)ccc3s2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C24H16F2N2O4S/c25-15-2-6-21-14(9-15)11-22(33-21)24(30)28-18-12-16(3-4-17(18)26)27-23(29)13-1-5-19-20(10-13)32-8-7-31-19/h1-6,9-12H,7-8H2,(H,27,29)(H,28,30)	VVQPZEWFWZIJBZ-UHFFFAOYSA-N	540129	US20260028334, Example 3/13	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540129	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540129&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447295	464925115							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238201	COc1ccc2cc(C(=O)Nc3cc(NC(=O)c4ccc5c(c4)OCCO5)ccc3F)sc2c1	InChI=1S/C25H19FN2O5S/c1-31-17-5-2-14-11-23(34-22(14)13-17)25(30)28-19-12-16(4-6-18(19)26)27-24(29)15-3-7-20-21(10-15)33-9-8-32-20/h2-7,10-13H,8-9H2,1H3,(H,27,29)(H,28,30)	SXSKUQCQISDPMM-UHFFFAOYSA-N	540130	US20260028334, Example 3/14	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540130	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540130&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447316	464925116							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238202	O=C(Nc1ccc(F)c(NC(=O)c2cc3cccnc3s2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C23H16FN3O4S/c24-16-5-4-15(26-21(28)13-3-6-18-19(10-13)31-9-8-30-18)12-17(16)27-22(29)20-11-14-2-1-7-25-23(14)32-20/h1-7,10-12H,8-9H2,(H,26,28)(H,27,29)	CWECEOJSRKUFFG-UHFFFAOYSA-N	540131	US20260028334, Example 3/15	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540131	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540131&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447047	464925117							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238203	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2cccnc2s1	InChI=1S/C24H19N3O4S/c1-14-4-6-17(26-22(28)15-5-7-19-20(11-15)31-10-9-30-19)13-18(14)27-23(29)21-12-16-3-2-8-25-24(16)32-21/h2-8,11-13H,9-10H2,1H3,(H,26,28)(H,27,29)	AUCWAITXVFDDRF-UHFFFAOYSA-N	540132	US20260028334, Example 3/16	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540132	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540132&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121446928	464925118							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238204	COc1ccc2nc(C(=O)Nc3cc(NC(=O)c4ccc5c(c4)OCCO5)ccc3C)sc2c1	InChI=1S/C25H21N3O5S/c1-14-3-5-16(26-23(29)15-4-8-20-21(11-15)33-10-9-32-20)12-19(14)27-24(30)25-28-18-7-6-17(31-2)13-22(18)34-25/h3-8,11-13H,9-10H2,1-2H3,(H,26,29)(H,27,30)	BMEIHHVPIXYYSI-UHFFFAOYSA-N	540133	US20260028334, Example 3/17	L-lactate dehydrogenase A chain	Homo sapiens		 550							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540133	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540133&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447293	464925119							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238205	CCN1CCN(Cc2ccc3cc(C(=O)Nc4cc(NC(=O)c5ccc6c(c5)OCCO6)ccc4F)sc3c2)CC1	InChI=1S/C31H31FN4O4S/c1-2-35-9-11-36(12-10-35)19-20-3-4-21-17-29(41-28(21)15-20)31(38)34-25-18-23(6-7-24(25)32)33-30(37)22-5-8-26-27(16-22)40-14-13-39-26/h3-8,15-18H,2,9-14,19H2,1H3,(H,33,37)(H,34,38)	FJXHBPJDZSXCFO-UHFFFAOYSA-N	540134	US20260028334, Example 3/18	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540134	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540134&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447156	464925120							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238206	CCN1CCN(Cc2ccc3cc(C(=O)Nc4cc(NC(=O)c5ccc6c(c5)OCCO6)ccc4F)sc3n2)CC1	InChI=1S/C30H30FN5O4S/c1-2-35-9-11-36(12-10-35)18-22-5-3-20-16-27(41-30(20)33-22)29(38)34-24-17-21(6-7-23(24)31)32-28(37)19-4-8-25-26(15-19)40-14-13-39-25/h3-8,15-17H,2,9-14,18H2,1H3,(H,32,37)(H,34,38)	ZULXJCUIDWKCDT-UHFFFAOYSA-N	540135	US20260028334, Example 3/19	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540135	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540135&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447056	464925121							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238207	O=C(Nc1ccc(F)c(NC(=O)c2cc3ccc(CN4CCOCC4)cc3s2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C29H26FN3O5S/c30-22-5-4-21(31-28(34)20-3-6-24-25(14-20)38-12-11-37-24)16-23(22)32-29(35)27-15-19-2-1-18(13-26(19)39-27)17-33-7-9-36-10-8-33/h1-6,13-16H,7-12,17H2,(H,31,34)(H,32,35)	YQDRRRKKERLKKW-UHFFFAOYSA-N	540136	US20260028334, Example 3/20	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540136	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540136&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			132051683	464925122							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238208	CC(=O)NCCOc1ccc2cc(C(=O)Nc3cc(NC(=O)c4ccc5c(c4)OCCO5)ccc3C)sc2c1	InChI=1S/C29H27N3O6S/c1-17-3-6-21(31-28(34)20-5-8-24-25(13-20)38-12-11-37-24)15-23(17)32-29(35)27-14-19-4-7-22(16-26(19)39-27)36-10-9-30-18(2)33/h3-8,13-16H,9-12H2,1-2H3,(H,30,33)(H,31,34)(H,32,35)	NKPXLXQJSJOTFR-UHFFFAOYSA-N	540137	US20260028334, Example 3/21	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540137	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540137&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447161	464925123							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238209	CCN1C[C@@H]2CN(Cc3ccc4cc(C(=O)Nc5cc(NC(=O)c6ccc7c(c6)OCCO7)ccc5F)sc4n3)C[C@@H]2C1	InChI=1S/C32H32FN5O4S/c1-2-37-14-21-16-38(17-22(21)15-37)18-24-5-3-20-12-29(43-32(20)35-24)31(40)36-26-13-23(6-7-25(26)33)34-30(39)19-4-8-27-28(11-19)42-10-9-41-27/h3-8,11-13,21-22H,2,9-10,14-18H2,1H3,(H,34,39)(H,36,40)	XBZIBQJMKXMXTB-UHFFFAOYSA-N	540138	US20260028334, Example 3/22	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540138	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540138&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447306	464925124							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238210	COC1CN(CCCOc2ccc3cc(C(=O)Nc4cc(NC(=O)c5ccc6c(c5)OCCO6)ccc4C)sc3c2)C1	InChI=1S/C32H33N3O6S/c1-20-4-7-23(33-31(36)22-6-9-27-28(14-22)41-13-12-40-27)16-26(20)34-32(37)30-15-21-5-8-24(17-29(21)42-30)39-11-3-10-35-18-25(19-35)38-2/h4-9,14-17,25H,3,10-13,18-19H2,1-2H3,(H,33,36)(H,34,37)	DKTMXUWQGNGCRV-UHFFFAOYSA-N	540139	US20260028334, Example 3/23	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540139	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540139&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121446929	464925125							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238211	O=C(Nc1ccc(F)c(NC(=O)c2cn3ccnc3s2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C21H15FN4O4S/c22-14-3-2-13(24-19(27)12-1-4-16-17(9-12)30-8-7-29-16)10-15(14)25-20(28)18-11-26-6-5-23-21(26)31-18/h1-6,9-11H,7-8H2,(H,24,27)(H,25,28)	IRHIHKJEEVSZSE-UHFFFAOYSA-N	540140	US20260028334, Example 3/24	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540140	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540140&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121446930	464925126							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238212	O=C(Nc1ccc(F)c(NC(=O)c2cc3sccc3s2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C22H15FN2O4S2/c23-14-3-2-13(24-21(26)12-1-4-16-17(9-12)29-7-6-28-16)10-15(14)25-22(27)20-11-19-18(31-20)5-8-30-19/h1-5,8-11H,6-7H2,(H,24,26)(H,25,27)	WNQNIRWBIRHYRY-UHFFFAOYSA-N	540141	US20260028334, Example 3/25	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540141	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540141&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447163	464925127							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238213	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2ccc(Br)cc2s1	InChI=1S/C25H19BrN2O4S/c1-14-2-6-18(27-24(29)16-4-7-20-21(10-16)32-9-8-31-20)13-19(14)28-25(30)23-11-15-3-5-17(26)12-22(15)33-23/h2-7,10-13H,8-9H2,1H3,(H,27,29)(H,28,30)	KNGHMLMWQLJSMO-UHFFFAOYSA-N	540142	US20260028334, Example 3/26	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540142	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540142&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447055	464925128							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238214	CN1CCN(Cc2ccc3cc(C(=O)Nc4cc(NC(=O)c5ccc6c(c5)OCCO6)ccc4F)sc3c2)CC1	InChI=1S/C30H29FN4O4S/c1-34-8-10-35(11-9-34)18-19-2-3-20-16-28(40-27(20)14-19)30(37)33-24-17-22(5-6-23(24)31)32-29(36)21-4-7-25-26(15-21)39-13-12-38-25/h2-7,14-17H,8-13,18H2,1H3,(H,32,36)(H,33,37)	KMQDSPHIMGWXBM-UHFFFAOYSA-N	540143	US20260028334, Example 3/27	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540143	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540143&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447301	464925129							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238215	O=C(Nc1ccc(F)c(NC(=O)c2cc3ccc(CN4CCN(CC(F)(F)F)CC4)cc3s2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C31H28F4N4O4S/c32-23-5-4-22(36-29(40)21-3-6-25-26(14-21)43-12-11-42-25)16-24(23)37-30(41)28-15-20-2-1-19(13-27(20)44-28)17-38-7-9-39(10-8-38)18-31(33,34)35/h1-6,13-16H,7-12,17-18H2,(H,36,40)(H,37,41)	CLLCTNPBWOTXMO-UHFFFAOYSA-N	540144	US20260028334, Example 3/28	L-lactate dehydrogenase A chain	Homo sapiens		 550							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540144	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540144&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447315	464925130							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238216	CCN1CCN(Cc2ccc3cc(C(=O)Nc4cc(NC(=O)c5ccc6c(c5)OCCO6)ccc4C)sc3n2)CC1	InChI=1S/C31H33N5O4S/c1-3-35-10-12-36(13-11-35)19-24-8-5-22-17-28(41-31(22)33-24)30(38)34-25-18-23(7-4-20(25)2)32-29(37)21-6-9-26-27(16-21)40-15-14-39-26/h4-9,16-18H,3,10-15,19H2,1-2H3,(H,32,37)(H,34,38)	ZVOVASAXKZHXCF-UHFFFAOYSA-N	540145	US20260028334, Example 3/29	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540145	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540145&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447061	464925131							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238217	CCN1CCN(Cc2ccc3cc(C(=O)Nc4cc(NC(=O)c5ccc6c(c5)OCCO6)ccc4Cl)sc3n2)CC1	InChI=1S/C30H30ClN5O4S/c1-2-35-9-11-36(12-10-35)18-22-5-3-20-16-27(41-30(20)33-22)29(38)34-24-17-21(6-7-23(24)31)32-28(37)19-4-8-25-26(15-19)40-14-13-39-25/h3-8,15-17H,2,9-14,18H2,1H3,(H,32,37)(H,34,38)	PMFLUZCWYAKIRL-UHFFFAOYSA-N	540146	US20260028334, Example 3/30	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540146	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540146&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447064	464925132							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238218	CCN1CCC(NCc2ccc3cc(C(=O)Nc4cc(NC(=O)c5ccc6c(c5)OCCO6)ccc4F)sc3n2)CC1	InChI=1S/C31H32FN5O4S/c1-2-37-11-9-21(10-12-37)33-18-23-5-3-20-16-28(42-31(20)35-23)30(39)36-25-17-22(6-7-24(25)32)34-29(38)19-4-8-26-27(15-19)41-14-13-40-26/h3-8,15-17,21,33H,2,9-14,18H2,1H3,(H,34,38)(H,36,39)	RSKMTDRNPMYDFS-UHFFFAOYSA-N	540147	US20260028334, Example 3/31	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540147	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540147&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			163408074	464925133							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238219	CCN1CCN(Cc2ccc3cc(C(=O)Nc4cc(NC(=O)c5ccc6c(c5)OCCO6)ccc4F)sc3n2)CC1(C)C	InChI=1S/C32H34FN5O4S/c1-4-38-12-11-37(19-32(38,2)3)18-23-7-5-21-16-28(43-31(21)35-23)30(40)36-25-17-22(8-9-24(25)33)34-29(39)20-6-10-26-27(15-20)42-14-13-41-26/h5-10,15-17H,4,11-14,18-19H2,1-3H3,(H,34,39)(H,36,40)	OYEUMULHPKRDLS-UHFFFAOYSA-N	540148	US20260028334, Example 3/32	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540148	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540148&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			163408075	464925134							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238220	O=C(Nc1ccc(F)c(NC(=O)c2cc3ccc(CN4CC(F)(F)C4)nc3s2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C27H21F3N4O4S/c28-19-5-4-17(31-24(35)15-2-6-21-22(9-15)38-8-7-37-21)11-20(19)33-25(36)23-10-16-1-3-18(32-26(16)39-23)12-34-13-27(29,30)14-34/h1-6,9-11H,7-8,12-14H2,(H,31,35)(H,33,36)	MWEFAAFYEPDVOD-UHFFFAOYSA-N	540149	US20260028334, Example 3/33	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540149	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540149&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121446933	464925135							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238221	CCN(CC)Cc1ccc2cc(C(=O)Nc3cc(NC(=O)c4ccc5c(c4)OCCO5)ccc3F)sc2n1	InChI=1S/C28H27FN4O4S/c1-3-33(4-2)16-20-7-5-18-14-25(38-28(18)31-20)27(35)32-22-15-19(8-9-21(22)29)30-26(34)17-6-10-23-24(13-17)37-12-11-36-23/h5-10,13-15H,3-4,11-12,16H2,1-2H3,(H,30,34)(H,32,35)	ZVSDBMYBCPXYOX-UHFFFAOYSA-N	540150	US20260028334, Example 3/34	L-lactate dehydrogenase A chain	Homo sapiens		 550							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540150	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540150&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447066	464925136							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238222	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2sccc2s1	InChI=1S/C23H18N2O4S2/c1-13-2-4-15(24-22(26)14-3-5-17-18(10-14)29-8-7-28-17)11-16(13)25-23(27)21-12-20-19(31-21)6-9-30-20/h2-6,9-12H,7-8H2,1H3,(H,24,26)(H,25,27)	LYNXCMXYCYRZFK-UHFFFAOYSA-N	540151	US20260028334, Example 3/37	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540151	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540151&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447072	464925137							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238223	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2ncccc2[nH]1	InChI=1S/C24H20N4O4/c1-14-4-6-16(26-23(29)15-5-7-21-22(11-15)32-10-9-31-21)12-18(14)28-24(30)20-13-19-17(27-20)3-2-8-25-19/h2-8,11-13,27H,9-10H2,1H3,(H,26,29)(H,28,30)	GJERTQYSITVJIB-UHFFFAOYSA-N	540152	US20260028334, Example 3/38	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540152	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540152&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121446935	464925138							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238224	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cn2ccnc2s1	InChI=1S/C22H18N4O4S/c1-13-2-4-15(24-20(27)14-3-5-17-18(10-14)30-9-8-29-17)11-16(13)25-21(28)19-12-26-7-6-23-22(26)31-19/h2-7,10-12H,8-9H2,1H3,(H,24,27)(H,25,28)	RDXJBMCFIUOAJB-UHFFFAOYSA-N	540153	US20260028334, Example 3/39	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540153	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540153&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447341	464925139							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238225	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2occc2[nH]1	InChI=1S/C23H19N3O5/c1-13-2-4-15(24-22(27)14-3-5-19-21(10-14)31-9-8-30-19)11-17(13)26-23(28)18-12-20-16(25-18)6-7-29-20/h2-7,10-12,25H,8-9H2,1H3,(H,24,27)(H,26,28)	CMTCQHXRDVMTAR-UHFFFAOYSA-N	540154	US20260028334, Example 3/40	L-lactate dehydrogenase A chain	Homo sapiens		 550							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540154	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540154&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447331	464925140							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238226	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2sccc2[nH]1	InChI=1S/C23H19N3O4S/c1-13-2-4-15(24-22(27)14-3-5-19-20(10-14)30-8-7-29-19)11-17(13)26-23(28)18-12-21-16(25-18)6-9-31-21/h2-6,9-12,25H,7-8H2,1H3,(H,24,27)(H,26,28)	MQGPFWRLBDXPTN-UHFFFAOYSA-N	540155	US20260028334, Example 3/42	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540155	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540155&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447346	464925141							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238227	O=C(Nc1ccc(F)c(NC(=O)c2cc3cc(OCCN4CCCC4)ccc3[nH]2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C30H29FN4O5/c31-23-6-4-21(32-29(36)19-3-8-27-28(17-19)40-14-13-39-27)18-25(23)34-30(37)26-16-20-15-22(5-7-24(20)33-26)38-12-11-35-9-1-2-10-35/h3-8,15-18,33H,1-2,9-14H2,(H,32,36)(H,34,37)	CMMYYJQBPJHCAL-UHFFFAOYSA-N	540156	US20260028334, Example 3/44	L-lactate dehydrogenase A chain	Homo sapiens		 550							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540156	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540156&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447079	464925142							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238228	CCN1CCN(Cc2ccc3cc(C(=O)Nc4cc(NC(=O)c5cc6c(cc5F)OCCO6)ccc4F)sc3n2)CC1	InChI=1S/C30H29F2N5O4S/c1-2-36-7-9-37(10-8-36)17-20-4-3-18-13-27(42-30(18)34-20)29(39)35-24-14-19(5-6-22(24)31)33-28(38)21-15-25-26(16-23(21)32)41-12-11-40-25/h3-6,13-16H,2,7-12,17H2,1H3,(H,33,38)(H,35,39)	KVOFBLQKZGKFAF-UHFFFAOYSA-N	540157	US20260028334, Example 3/45	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540157	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540157&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121446991	464925143							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238229	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2nccnc2s1	InChI=1S/C23H18N4O4S/c1-13-2-4-15(26-21(28)14-3-5-18-19(10-14)31-9-8-30-18)11-16(13)27-22(29)20-12-17-23(32-20)25-7-6-24-17/h2-7,10-12H,8-9H2,1H3,(H,26,28)(H,27,29)	RINCSPPLJIICFT-UHFFFAOYSA-N	540158	US20260028334, Example 4	L-lactate dehydrogenase A chain	Homo sapiens		 550							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540158	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540158&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447170	464925144							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238230	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2cc(OCC(C)(C)O)ccc2o1	InChI=1S/C29H28N2O7/c1-17-4-6-20(30-27(32)18-5-8-24-25(13-18)36-11-10-35-24)15-22(17)31-28(33)26-14-19-12-21(7-9-23(19)38-26)37-16-29(2,3)34/h4-9,12-15,34H,10-11,16H2,1-3H3,(H,30,32)(H,31,33)	KUVJIYRHXYWYIB-UHFFFAOYSA-N	540159	US20260028334, Example 5	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540159	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540159&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447173	464925145							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238231	Cc3ccc(NC(=O)c2ccc1OCCOc1c2)cc3NC(=O)c5cc4ccc(O)cc4s5	InChI=1S/C25H20N2O5S/c1-14-2-5-17(26-24(29)16-4-7-20-21(10-16)32-9-8-31-20)12-19(14)27-25(30)23-11-15-3-6-18(28)13-22(15)33-23/h2-7,10-13,28H,8-9H2,1H3,(H,26,29)(H,27,30)	YMCUTSMQODXBGQ-UHFFFAOYSA-N	540160	US20260028334, Example 6	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540160	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540160&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447020	464925146							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238232	COCCOc1ccc2cc(C(=O)Nc3cc(NC(=O)c4ccc5c(c4)OCCO5)ccc3C)sc2c1	InChI=1S/C28H26N2O6S/c1-17-3-6-20(29-27(31)19-5-8-23-24(13-19)36-12-11-35-23)15-22(17)30-28(32)26-14-18-4-7-21(16-25(18)37-26)34-10-9-33-2/h3-8,13-16H,9-12H2,1-2H3,(H,29,31)(H,30,32)	NKERBEDEYRTWNJ-UHFFFAOYSA-N	540161	US20260028334, Example 7	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540161	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540161&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			132051842	464925147							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238233	CC(=O)COc1ccc2cc(C(=O)Nc3cc(NC(=O)c4ccc5c(c4)OCCO5)ccc3C)sc2c1	InChI=1S/C28H24N2O6S/c1-16-3-6-20(29-27(32)19-5-8-23-24(11-19)35-10-9-34-23)13-22(16)30-28(33)26-12-18-4-7-21(14-25(18)37-26)36-15-17(2)31/h3-8,11-14H,9-10,15H2,1-2H3,(H,29,32)(H,30,33)	DOAUPDNPUASFOG-UHFFFAOYSA-N	540162	US20260028334, Example 8	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540162	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540162&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447352	464925148							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238234	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2ccc(OCC(C)(C)O)cc2s1	InChI=1S/C29H28N2O6S/c1-17-4-7-20(30-27(32)19-6-9-23-24(12-19)36-11-10-35-23)14-22(17)31-28(33)26-13-18-5-8-21(15-25(18)38-26)37-16-29(2,3)34/h4-9,12-15,34H,10-11,16H2,1-3H3,(H,30,32)(H,31,33)	BDZBUBODEMSYMU-UHFFFAOYSA-N	540163	US20260028334, Example 9	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540163	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540163&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			132051679	464925149							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238235	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2ccc(OCCO)cc2s1	InChI=1S/C27H24N2O6S/c1-16-2-5-19(28-26(31)18-4-7-22-23(12-18)35-11-10-34-22)14-21(16)29-27(32)25-13-17-3-6-20(33-9-8-30)15-24(17)36-25/h2-7,12-15,30H,8-11H2,1H3,(H,28,31)(H,29,32)	KHGKWNADKSUMAC-UHFFFAOYSA-N	540164	US20260028334, Example 10	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540164	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540164&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			132051853	464925150							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238236	CC(=O)COCCOc1ccc2cc(C(=O)Nc3cc(NC(=O)c4ccc5c(c4)OCCO5)ccc3C)sc2c1	InChI=1S/C30H28N2O7S/c1-18-3-6-22(31-29(34)21-5-8-25-26(13-21)39-12-11-38-25)15-24(18)32-30(35)28-14-20-4-7-23(16-27(20)40-28)37-10-9-36-17-19(2)33/h3-8,13-16H,9-12,17H2,1-2H3,(H,31,34)(H,32,35)	UCRYLDCVYGJDDC-UHFFFAOYSA-N	540165	US20260028334, Example 11	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540165	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540165&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			132051672	464925151							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238237	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2ccc(OCCN3CCCC3)cc2s1	InChI=1S/C31H31N3O5S/c1-20-4-7-23(32-30(35)22-6-9-26-27(16-22)39-15-14-38-26)18-25(20)33-31(36)29-17-21-5-8-24(19-28(21)40-29)37-13-12-34-10-2-3-11-34/h4-9,16-19H,2-3,10-15H2,1H3,(H,32,35)(H,33,36)	IOUMTCNIXOSQCN-UHFFFAOYSA-N	540166	US20260028334, Example 12	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540166	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540166&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			132051697	464925152							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238238	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2ccc(OCCCN3CC[C@H](F)C3)cc2s1	InChI=1S/C32H32FN3O5S/c1-20-3-6-24(34-31(37)22-5-8-27-28(15-22)41-14-13-40-27)17-26(20)35-32(38)30-16-21-4-7-25(18-29(21)42-30)39-12-2-10-36-11-9-23(33)19-36/h3-8,15-18,23H,2,9-14,19H2,1H3,(H,34,37)(H,35,38)	ZBRCYEWMFFYLPH-UHFFFAOYSA-N	540167	US20260028334, Example 13	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540167	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540167&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			132051680	464925153							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238239	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2ccc(OCCCN3CC[C@H](F)C3)cc2s1	InChI=1S/C32H32FN3O5S/c1-20-3-6-24(34-31(37)22-5-8-27-28(15-22)41-14-13-40-27)17-26(20)35-32(38)30-16-21-4-7-25(18-29(21)42-30)39-12-2-10-36-11-9-23(33)19-36/h3-8,15-18,23H,2,9-14,19H2,1H3,(H,34,37)(H,35,38)	ZBRCYEWMFFYLPH-UHFFFAOYSA-N	540168	US20260028334, Example 13/1	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540168	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540168&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			132051674	464925154							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238240	Cc3ccc(NC(=O)c2ccc1OCCOc1c2)cc3NC(=O)c6cc5ccc(OCCCN4CCC(F)(F)C4)cc5s6	InChI=1S/C32H31F2N3O5S/c1-20-3-6-23(35-30(38)22-5-8-26-27(15-22)42-14-13-41-26)17-25(20)36-31(39)29-16-21-4-7-24(18-28(21)43-29)40-12-2-10-37-11-9-32(33,34)19-37/h3-8,15-18H,2,9-14,19H2,1H3,(H,35,38)(H,36,39)	RYWCKTQZGHASFI-UHFFFAOYSA-N	540169	US20260028334, Example 13/2	L-lactate dehydrogenase A chain	Homo sapiens		 550							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540169	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540169&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447078	464925155							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238241	Cc3ccc(NC(=O)c2ccc1OCCOc1c2)cc3NC(=O)c6cc5ccc(OCCCN4CC(F)(F)C4)cc5s6	InChI=1S/C31H29F2N3O5S/c1-19-3-6-22(34-29(37)21-5-8-25-26(13-21)41-12-11-40-25)15-24(19)35-30(38)28-14-20-4-7-23(16-27(20)42-28)39-10-2-9-36-17-31(32,33)18-36/h3-8,13-16H,2,9-12,17-18H2,1H3,(H,34,37)(H,35,38)	WLHFFIRWOOENQN-UHFFFAOYSA-N	540170	US20260028334, Example 13/3	L-lactate dehydrogenase A chain	Homo sapiens		 5500							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540170	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540170&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447018	464925156							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238242	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2ccccc2n1C	InChI=1S/C26H23N3O4/c1-16-7-9-19(27-25(30)18-8-10-23-24(14-18)33-12-11-32-23)15-20(16)28-26(31)22-13-17-5-3-4-6-21(17)29(22)2/h3-10,13-15H,11-12H2,1-2H3,(H,27,30)(H,28,31)	SQHYPGHINSZEBE-UHFFFAOYSA-N	540171	US20260028334, Example 14	L-lactate dehydrogenase A chain	Homo sapiens		 550							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540171	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540171&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447188	464925157							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238243	Cc1ccc(NC(=O)c2ccc3c(c2)OCCC3)cc1NC(=O)c1cc2ccccc2s1	InChI=1S/C26H22N2O3S/c1-16-8-11-20(27-25(29)19-10-9-17-6-4-12-31-22(17)13-19)15-21(16)28-26(30)24-14-18-5-2-3-7-23(18)32-24/h2-3,5,7-11,13-15H,4,6,12H2,1H3,(H,27,29)(H,28,30)	WELYJUDQQGKJBL-UHFFFAOYSA-N	540172	US20260028334, Example 15	L-lactate dehydrogenase A chain	Homo sapiens		 5500							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540172	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540172&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121446934	464925158							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238244	CCN1C[C@@H]2C[C@H]1CN2Cc7ccc6cc(C(=O)Nc5cc(NC(=O)c4ccc3OCCOc3c4)ccc5F)sc6c7	InChI=1S/C32H31FN4O4S/c1-2-36-17-24-15-23(36)18-37(24)16-19-3-4-20-13-30(42-29(20)11-19)32(39)35-26-14-22(6-7-25(26)33)34-31(38)21-5-8-27-28(12-21)41-10-9-40-27/h3-8,11-14,23-24H,2,9-10,15-18H2,1H3,(H,34,38)(H,35,39)	BDGXTHKFLNLILE-UHFFFAOYSA-N	540173	US20260028334, Example 16	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540173	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540173&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447084	464925159							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238245	CCN6CCCN(Cc5ccc4cc(C(=O)Nc3cc(NC(=O)c2ccc1OCCOc1c2)ccc3F)sc4c5)CC6	InChI=1S/C32H33FN4O4S/c1-2-36-10-3-11-37(13-12-36)20-21-4-5-22-18-30(42-29(22)16-21)32(39)35-26-19-24(7-8-25(26)33)34-31(38)23-6-9-27-28(17-23)41-15-14-40-27/h4-9,16-19H,2-3,10-15,20H2,1H3,(H,34,38)(H,35,39)	PFVVTWSVSOZHIY-UHFFFAOYSA-N	540174	US20260028334, Example 17	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540174	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540174&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121446941	464925160							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238246	O=C(Nc1ccc(F)c(NC(=O)c2cc3ccc(CN4CC[C@@H](O)C4)nc3s2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C28H25FN4O5S/c29-21-5-4-18(30-26(35)16-2-6-23-24(11-16)38-10-9-37-23)13-22(21)32-27(36)25-12-17-1-3-19(31-28(17)39-25)14-33-8-7-20(34)15-33/h1-6,11-13,20,34H,7-10,14-15H2,(H,30,35)(H,32,36)	OSWSCTYFYGTDFE-UHFFFAOYSA-N	540175	US20260028334, Example 18	L-lactate dehydrogenase A chain	Homo sapiens		 550							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540175	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540175&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447086	464925161							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238247	O=C(Nc1ccc(F)c(NC(=O)c2cc3ccc(CC4CC[C@H](O)C4)nc3s2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C29H26FN3O5S/c30-22-7-5-20(31-27(35)17-3-8-24-25(13-17)38-10-9-37-24)15-23(22)33-28(36)26-14-18-2-4-19(32-29(18)39-26)11-16-1-6-21(34)12-16/h2-5,7-8,13-16,21,34H,1,6,9-12H2,(H,31,35)(H,33,36)	YBMDGDQFBQLROZ-UHFFFAOYSA-N	540176	US20260028334, Example 18/1	L-lactate dehydrogenase A chain	Homo sapiens		 550							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540176	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540176&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447014	464925162							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238248	O=C(Nc1ccc(F)c(NC(=O)c2cc3ccc(CN4CCC(O)CC4)nc3s2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C29H27FN4O5S/c30-22-5-4-19(31-27(36)17-2-6-24-25(13-17)39-12-11-38-24)15-23(22)33-28(37)26-14-18-1-3-20(32-29(18)40-26)16-34-9-7-21(35)8-10-34/h1-6,13-15,21,35H,7-12,16H2,(H,31,36)(H,33,37)	BVKQYQODJNCBMG-UHFFFAOYSA-N	540177	US20260028334, Example 18/2	L-lactate dehydrogenase A chain	Homo sapiens		 550							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540177	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540177&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447373	464925163							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238249	O=C(Nc1ccc(F)c(NC(=O)c2cc3ccc(OCCN4CCCC4)nc3s2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C29H27FN4O5S/c30-21-6-5-20(31-27(35)18-3-7-23-24(15-18)38-14-13-37-23)17-22(21)32-28(36)25-16-19-4-8-26(33-29(19)40-25)39-12-11-34-9-1-2-10-34/h3-8,15-17H,1-2,9-14H2,(H,31,35)(H,32,36)	UJGZDLDOKSAMPV-UHFFFAOYSA-N	540178	US20260028334, Example 19	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540178	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540178&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447088	464925164							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238250	O=C(Nc1ccc(F)c(NC(=O)c2cc3ccc(OCCCN4CCCC4)nc3s2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C30H29FN4O5S/c31-22-7-6-21(32-28(36)19-4-8-24-25(16-19)39-15-14-38-24)18-23(22)33-29(37)26-17-20-5-9-27(34-30(20)41-26)40-13-3-12-35-10-1-2-11-35/h4-9,16-18H,1-3,10-15H2,(H,32,36)(H,33,37)	BCSAKQDCPNOFNY-UHFFFAOYSA-N	540179	US20260028334, Example 19/1	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540179	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540179&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447005	464925165							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238251	CCN1CCN(CCc2ccc3cc(C(=O)Nc4cc(NC(=O)c5ccc6c(c5)OCCO6)ccc4F)sc3n2)CC1	InChI=1S/C31H32FN5O4S/c1-2-36-11-13-37(14-12-36)10-9-22-5-3-21-18-28(42-31(21)34-22)30(39)35-25-19-23(6-7-24(25)32)33-29(38)20-4-8-26-27(17-20)41-16-15-40-26/h3-8,17-19H,2,9-16H2,1H3,(H,33,38)(H,35,39)	ZCSIIRDAWWTYPD-UHFFFAOYSA-N	540180	US20260028334, Example 19/2	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540180	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540180&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121446942	464925166							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238252	CCN1CCC(Cc2ccc3cc(C(=O)Nc4cc(NC(=O)c5ccc6c(c5)OCCO6)ccc4F)sc3n2)CC1	InChI=1S/C31H31FN4O4S/c1-2-36-11-9-19(10-12-36)15-22-5-3-21-17-28(41-31(21)34-22)30(38)35-25-18-23(6-7-24(25)32)33-29(37)20-4-8-26-27(16-20)40-14-13-39-26/h3-8,16-19H,2,9-15H2,1H3,(H,33,37)(H,35,38)	MVCMWLWERKFNPL-UHFFFAOYSA-N	540181	US20260028334, Example 19/3	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540181	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540181&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447089	464925167							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238253	CCN1CCN(Cc2cn3cc(C(=O)Nc4cc(NC(=O)c5ccc6c(c5)OCCO6)ccc4F)sc3n2)CC1	InChI=1S/C28H29FN6O4S/c1-2-33-7-9-34(10-8-33)15-20-16-35-17-25(40-28(35)31-20)27(37)32-22-14-19(4-5-21(22)29)30-26(36)18-3-6-23-24(13-18)39-12-11-38-23/h3-6,13-14,16-17H,2,7-12,15H2,1H3,(H,30,36)(H,32,37)	PGPVPUFQBJPQBO-UHFFFAOYSA-N	540182	US20260028334, Example 20	L-lactate dehydrogenase A chain	Homo sapiens		 5500							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540182	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540182&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447091	464925168							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238254	O=C(Nc1ccc(F)c(NC(=O)c2cc3ccc(COc4ccccn4)cc3s2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C30H22FN3O5S/c31-22-8-7-21(33-29(35)20-6-9-24-25(14-20)38-12-11-37-24)16-23(22)34-30(36)27-15-19-5-4-18(13-26(19)40-27)17-39-28-3-1-2-10-32-28/h1-10,13-16H,11-12,17H2,(H,33,35)(H,34,36)	ZHFKUXPNKLKQEB-UHFFFAOYSA-N	540183	US20260028334, Example 20/1	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540183	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540183&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447106	464925169							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238255	CCN1CCN(C(C)c2ccc3cc(C(=O)Nc4cc(NC(=O)c5ccc6c(c5)OCCO6)ccc4F)sc3c2)CC1	InChI=1S/C32H33FN4O4S/c1-3-36-10-12-37(13-11-36)20(2)21-4-5-22-18-30(42-29(22)17-21)32(39)35-26-19-24(7-8-25(26)33)34-31(38)23-6-9-27-28(16-23)41-15-14-40-27/h4-9,16-20H,3,10-15H2,1-2H3,(H,34,38)(H,35,39)	ABGILFVIGUACDU-UHFFFAOYSA-N	540184	US20260028334, Example 21	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540184	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540184&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447102	464925170							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238256	Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1cc2ccc(OCCN)cc2s1	InChI=1S/C27H25N3O5S/c1-16-2-5-19(29-26(31)18-4-7-22-23(12-18)35-11-10-34-22)14-21(16)30-27(32)25-13-17-3-6-20(33-9-8-28)15-24(17)36-25/h2-7,12-15H,8-11,28H2,1H3,(H,29,31)(H,30,32)	TZZIUOREOBZKOT-UHFFFAOYSA-N	540185	US20260028334, Example 22	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540185	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540185&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447109	464925171							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238257	CC(=O)N1CCN(Cc2ccc3cc(C(=O)Nc4cc(NC(=O)c5ccc6c(c5)OCCO6)ccc4F)sc3n2)CC1	InChI=1S/C30H28FN5O5S/c1-18(37)36-10-8-35(9-11-36)17-22-4-2-20-15-27(42-30(20)33-22)29(39)34-24-16-21(5-6-23(24)31)32-28(38)19-3-7-25-26(14-19)41-13-12-40-25/h2-7,14-16H,8-13,17H2,1H3,(H,32,38)(H,34,39)	GPXBENWDADTFBD-UHFFFAOYSA-N	540186	US20260028334, Example 23	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540186	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540186&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447119	464925172							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238258	CCN1CCN(CCOc2ccc3cc(C(=O)Nc4cc(NC(=O)c5ccc6c(c5)OCCO6)ccc4C)sc3c2)CC1	InChI=1S/C33H36N4O5S/c1-3-36-10-12-37(13-11-36)14-15-40-26-8-5-23-19-31(43-30(23)21-26)33(39)35-27-20-25(7-4-22(27)2)34-32(38)24-6-9-28-29(18-24)42-17-16-41-28/h4-9,18-21H,3,10-17H2,1-2H3,(H,34,38)(H,35,39)	QMVYJEZMQVKULC-UHFFFAOYSA-N	540187	US20260028334, Example 24	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540187	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540187&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447121	464925173							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238259	Cc1ccc(NC(=O)c2ccc3c(c2)OCCCO3)cc1NC(=O)c1cc2ccccc2s1	InChI=1S/C26H22N2O4S/c1-16-7-9-19(27-25(29)18-8-10-21-22(13-18)32-12-4-11-31-21)15-20(16)28-26(30)24-14-17-5-2-3-6-23(17)33-24/h2-3,5-10,13-15H,4,11-12H2,1H3,(H,27,29)(H,28,30)	KUNQFSMVMIRKNI-UHFFFAOYSA-N	540188	US20260028334, Example 25	L-lactate dehydrogenase A chain	Homo sapiens		 550							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540188	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540188&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121446943	464925174							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238260	COC1CN(CCCOc2ccc3cc(C(=O)Nc4cc(NC(=O)c5ccc6c(c5)OCCO6)ccc4C)sc3c2)C1	InChI=1S/C32H33N3O6S/c1-20-4-7-23(33-31(36)22-6-9-27-28(14-22)41-13-12-40-27)16-26(20)34-32(37)30-15-21-5-8-24(17-29(21)42-30)39-11-3-10-35-18-25(19-35)38-2/h4-9,14-17,25H,3,10-13,18-19H2,1-2H3,(H,33,36)(H,34,37)	DKTMXUWQGNGCRV-UHFFFAOYSA-N	540189	US20260028334, Example 26	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540189	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540189&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447233	464925175							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238261	CC(C)N6CCN(Cc5ccc4cc(C(=O)Nc3cc(NC(=O)c2ccc1OCCOc1c2)ccc3F)sc4n5)CC6	InChI=1S/C31H32FN5O4S/c1-19(2)37-11-9-36(10-12-37)18-23-5-3-21-16-28(42-31(21)34-23)30(39)35-25-17-22(6-7-24(25)32)33-29(38)20-4-8-26-27(15-20)41-14-13-40-26/h3-8,15-17,19H,9-14,18H2,1-2H3,(H,33,38)(H,35,39)	UROKJZJZWWYYSH-UHFFFAOYSA-N	540190	US20260028334, Example 27	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540190	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540190&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447380	464925176							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238262	CCN1C[C@H]2C[C@@H]1CN2Cc1ccc2cc(C(=O)Nc3cc(NC(=O)c4ccc5c(c4)OCCO5)ccc3F)sc2n1	InChI=1S/C31H30FN5O4S/c1-2-36-16-23-14-22(36)17-37(23)15-21-5-3-19-12-28(42-31(19)34-21)30(39)35-25-13-20(6-7-24(25)32)33-29(38)18-4-8-26-27(11-18)41-10-9-40-26/h3-8,11-13,22-23H,2,9-10,14-17H2,1H3,(H,33,38)(H,35,39)	PKYULGFPYRJCCR-UHFFFAOYSA-N	540191	US20260028334, Example 27/1	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540191	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540191&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447198	464925177							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238263	CCN1C[C@@H]2C[C@H]1CN2Cc1ccc2cc(C(=O)Nc3cc(NC(=O)c4ccc5c(c4)OCCO5)ccc3F)sc2n1	InChI=1S/C31H30FN5O4S/c1-2-36-16-23-14-22(36)17-37(23)15-21-5-3-19-12-28(42-31(19)34-21)30(39)35-25-13-20(6-7-24(25)32)33-29(38)18-4-8-26-27(11-18)41-10-9-40-26/h3-8,11-13,22-23H,2,9-10,14-17H2,1H3,(H,33,38)(H,35,39)	PKYULGFPYRJCCR-UHFFFAOYSA-N	540192	US20260028334, Example 27/2	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540192	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540192&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447396	464925178							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238264	CCN1CCCN(Cc2ccc3cc(C(=O)Nc4cc(NC(=O)c5ccc6c(c5)OCCO6)ccc4F)sc3n2)CC1	InChI=1S/C31H32FN5O4S/c1-2-36-10-3-11-37(13-12-36)19-23-6-4-21-17-28(42-31(21)34-23)30(39)35-25-18-22(7-8-24(25)32)33-29(38)20-5-9-26-27(16-20)41-15-14-40-26/h4-9,16-18H,2-3,10-15,19H2,1H3,(H,33,38)(H,35,39)	JGDFLEQZHONWEY-UHFFFAOYSA-N	540193	US20260028334, Example 27/3	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540193	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540193&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447132	464925179							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238265	O=C(Nc5ccc(F)c(NC(=O)c4cc3ccc(CN2C[C@H]1CNC[C@H]1C2)cc3s4)c5)c7ccc6OCCOc6c7	InChI=1S/C31H29FN4O4S/c32-24-5-4-23(34-30(37)20-3-6-26-27(10-20)40-8-7-39-26)12-25(24)35-31(38)29-11-19-2-1-18(9-28(19)41-29)15-36-16-21-13-33-14-22(21)17-36/h1-6,9-12,21-22,33H,7-8,13-17H2,(H,34,37)(H,35,38)	HWALKJFAVAHJBR-UHFFFAOYSA-N	540194	US20260028334, Example 28	L-lactate dehydrogenase A chain	Homo sapiens		 550							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540194	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540194&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447202	464925180							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238266	CCN6CCC(C(O)c5ccc4cc(C(=O)Nc3cc(NC(=O)c2ccc1OCCOc1c2)ccc3F)sc4c5)CC6	InChI=1S/C32H32FN3O5S/c1-2-36-11-9-19(10-12-36)30(37)21-4-3-20-16-29(42-28(20)17-21)32(39)35-25-18-23(6-7-24(25)33)34-31(38)22-5-8-26-27(15-22)41-14-13-40-26/h3-8,15-19,30,37H,2,9-14H2,1H3,(H,34,38)(H,35,39)	PZXQDFQWDYWEKZ-UHFFFAOYSA-N	540195	US20260028334, Example 29	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540195	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540195&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447374	464925181							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238267	O=C(Nc1ccc(F)c(NC(=O)c2cc3ccc(OCC(O)CN4CCCC4)cc3s2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C31H30FN3O6S/c32-24-7-5-21(33-30(37)20-4-8-26-27(13-20)40-12-11-39-26)15-25(24)34-31(38)29-14-19-3-6-23(16-28(19)42-29)41-18-22(36)17-35-9-1-2-10-35/h3-8,13-16,22,36H,1-2,9-12,17-18H2,(H,33,37)(H,34,38)	QNUSIQKKHFSRHA-UHFFFAOYSA-N	540196	US20260028334, Example 30	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540196	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540196&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447252	464925182							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238268	O=C(Nc1ccc(F)c(NC(=O)c2cc3ccc(OC[C@@H](O)CN4CCCC4)cc3s2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C31H30FN3O6S/c32-24-7-5-21(33-30(37)20-4-8-26-27(13-20)40-12-11-39-26)15-25(24)34-31(38)29-14-19-3-6-23(16-28(19)42-29)41-18-22(36)17-35-9-1-2-10-35/h3-8,13-16,22,36H,1-2,9-12,17-18H2,(H,33,37)(H,34,38)	QNUSIQKKHFSRHA-UHFFFAOYSA-N	540197	US20260028334, Example 30/1	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540197	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540197&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447135	464925183							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
238269	O=C(Nc1ccc(F)c(NC(=O)c2cc3ccc(OC[C@H](O)CN4CCCC4)cc3s2)c1)c1ccc2c(c1)OCCO2	InChI=1S/C31H30FN3O6S/c32-24-7-5-21(33-30(37)20-4-8-26-27(13-20)40-12-11-39-26)15-25(24)34-31(38)29-14-19-3-6-23(16-28(19)42-29)41-18-22(36)17-35-9-1-2-10-35/h3-8,13-16,22,36H,1-2,9-12,17-18H2,(H,33,37)(H,34,38)	QNUSIQKKHFSRHA-UHFFFAOYSA-N	540198	US20260028334, Example 30/2	L-lactate dehydrogenase A chain	Homo sapiens		<100							US Patent		10.7270/Q22Z1BCB			US20260028334	TARASEWICZ, A; STEENECK, C; LESZCZYNSKI, B; VIEIRA, A; SECHI, S; REID, G; CHARAPITSA, I; FABIAN, J; KROL, H; KREMOSER, C	1/29/2026	6/10/2026	Wmt Aktiengesellschaft	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=540198	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=5051&target=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=540198&enzyme=L-lactate+dehydrogenase+A+chain&column=ki&startPg=0&Increment=50&submit=Search			121447138	464925184							1	MATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF	6Q13,6Q0D,6MVA,6MV8,5W8L,5W8K,5W8J,5W8I,5W8H,4ZVV,8FW6,7M2N,9IOV,9BK3,9BK2,6SBV,6SBU,6BB3,6BB2,6BB1,6BB0,6BAZ,6BAX,6BAG,6BAD,5IXY,5IXS,4RLS,4R69,4R68,4QO8,4QO7,4M49,4JNK,1I10,4L4S,4L4R,6ZZR,5ZJF,5ZJE,5ZJD,4QT0,4QSM,4OKN,4OJN,4AJP,4AJ4	L-lactate dehydrogenase A chain	LDHA_HUMAN	P00338	B4DKQ2 B7Z5E3 D3DQY3 F8W819 Q53G53 Q6IBM7 Q6ZNV1 Q9UDE8 Q9UDE9																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
