BindingDB Reactant_set_id	Ligand SMILES	Ligand InChI	Ligand InChI Key	BindingDB MonomerID	BindingDB Ligand Name	Target Name	Target Source Organism According to Curator or DataSource	Ki (nM)	IC50 (nM)	Kd (nM)	EC50 (nM)	kon (M-1-s-1)	koff (s-1)	pH	Temp (C)	Curation/DataSource	Article DOI	BindingDB Entry DOI	PMID	PubChem AID	Patent Number	Authors	Date of publication	Date in BindingDB	Institution	Link to Ligand in BindingDB	Link to Target in BindingDB	Link to Ligand-Target Pair in BindingDB	Ligand HET ID in PDB	PDB ID(s) for Ligand-Target Complex	PubChem CID	PubChem SID	ChEBI ID of Ligand	ChEMBL ID of Ligand	DrugBank ID of Ligand	IUPHAR_GRAC ID of Ligand	KEGG ID of Ligand	ZINC ID of Ligand	Number of Protein Chains in Target (>1 implies a multichain complex)	BindingDB Target Chain Sequence 1	PDB ID(s) of Target Chain 1	UniProt (SwissProt) Recommended Name of Target Chain 1	UniProt (SwissProt) Entry Name of Target Chain 1	UniProt (SwissProt) Primary ID of Target Chain 1	UniProt (SwissProt) Secondary ID(s) of Target Chain 1	UniProt (SwissProt) Alternative ID(s) of Target Chain 1	UniProt (TrEMBL) Submitted Name of Target Chain 1	UniProt (TrEMBL) Entry Name of Target Chain 1	UniProt (TrEMBL) Primary ID of Target Chain 1	UniProt (TrEMBL) Secondary ID(s) of Target Chain 1	UniProt (TrEMBL) Alternative ID(s) of Target Chain 1	BindingDB Target Chain Sequence 2	PDB ID(s) of Target Chain 2	UniProt (SwissProt) Recommended Name of Target Chain 2	UniProt (SwissProt) Entry Name of Target Chain 2	UniProt (SwissProt) Primary ID of Target Chain 2	UniProt (SwissProt) Secondary ID(s) of Target Chain 2	UniProt (SwissProt) Alternative ID(s) of Target Chain 2	UniProt (TrEMBL) Submitted Name of Target Chain 2	UniProt (TrEMBL) Entry Name of Target Chain 2	UniProt (TrEMBL) Primary ID of Target Chain 2	UniProt (TrEMBL) Secondary ID(s) of Target Chain 2	UniProt (TrEMBL) Alternative ID(s) of Target Chain 2	BindingDB Target Chain Sequence 3	PDB ID(s) of Target Chain 3	UniProt (SwissProt) Recommended Name of Target Chain 3	UniProt (SwissProt) Entry Name of Target Chain 3	UniProt (SwissProt) Primary ID of Target Chain 3	UniProt (SwissProt) Secondary ID(s) of Target Chain 3	UniProt (SwissProt) Alternative ID(s) of Target Chain 3	UniProt (TrEMBL) Submitted Name of Target Chain 3	UniProt (TrEMBL) Entry Name of Target Chain 3	UniProt (TrEMBL) Primary ID of Target Chain 3	UniProt (TrEMBL) Secondary ID(s) of Target Chain 3	UniProt (TrEMBL) Alternative ID(s) of Target Chain 3	BindingDB Target Chain Sequence 4	PDB ID(s) of Target Chain 4	UniProt (SwissProt) Recommended Name of Target Chain 4	UniProt (SwissProt) Entry Name of Target Chain 4	UniProt (SwissProt) Primary ID of Target Chain 4	UniProt (SwissProt) Secondary ID(s) of Target Chain 4	UniProt (SwissProt) Alternative ID(s) of Target Chain 4	UniProt (TrEMBL) Submitted Name of Target Chain 4	UniProt (TrEMBL) Entry Name of Target Chain 4	UniProt (TrEMBL) Primary ID of Target Chain 4	UniProt (TrEMBL) Secondary ID(s) of Target Chain 4	UniProt (TrEMBL) Alternative ID(s) of Target Chain 4	BindingDB Target Chain Sequence 5	PDB ID(s) of Target Chain 5	UniProt (SwissProt) Recommended Name of Target Chain 5	UniProt (SwissProt) Entry Name of Target Chain 5	UniProt (SwissProt) Primary ID of Target Chain 5	UniProt (SwissProt) Secondary ID(s) of Target Chain 5	UniProt (SwissProt) Alternative ID(s) of Target Chain 5	UniProt (TrEMBL) Submitted Name of Target Chain 5	UniProt (TrEMBL) Entry Name of Target Chain 5	UniProt (TrEMBL) Primary ID of Target Chain 5	UniProt (TrEMBL) Secondary ID(s) of Target Chain 5	UniProt (TrEMBL) Alternative ID(s) of Target Chain 5	BindingDB Target Chain Sequence 6	PDB ID(s) of Target Chain 6	UniProt (SwissProt) Recommended Name of Target Chain 6	UniProt (SwissProt) Entry Name of Target Chain 6	UniProt (SwissProt) Primary ID of Target Chain 6	UniProt (SwissProt) Secondary ID(s) of Target Chain 6	UniProt (SwissProt) Alternative ID(s) of Target Chain 6	UniProt (TrEMBL) Submitted Name of Target Chain 6	UniProt (TrEMBL) Entry Name of Target Chain 6	UniProt (TrEMBL) Primary ID of Target Chain 6	UniProt (TrEMBL) Secondary ID(s) of Target Chain 6	UniProt (TrEMBL) Alternative ID(s) of Target Chain 6	BindingDB Target Chain Sequence 7	PDB ID(s) of Target Chain 7	UniProt (SwissProt) Recommended Name of Target Chain 7	UniProt (SwissProt) Entry Name of Target Chain 7	UniProt (SwissProt) Primary ID of Target Chain 7	UniProt (SwissProt) Secondary ID(s) of Target Chain 7	UniProt (SwissProt) Alternative ID(s) of Target Chain 7	UniProt (TrEMBL) Submitted Name of Target Chain 7	UniProt (TrEMBL) Entry Name of Target Chain 7	UniProt (TrEMBL) Primary ID of Target Chain 7	UniProt (TrEMBL) Secondary ID(s) of Target Chain 7	UniProt (TrEMBL) Alternative ID(s) of Target Chain 7	BindingDB Target Chain Sequence 8	PDB ID(s) of Target Chain 8	UniProt (SwissProt) Recommended Name of Target Chain 8	UniProt (SwissProt) Entry Name of Target Chain 8	UniProt (SwissProt) Primary ID of Target Chain 8	UniProt (SwissProt) Secondary ID(s) of Target Chain 8	UniProt (SwissProt) Alternative ID(s) of Target Chain 8	UniProt (TrEMBL) Submitted Name of Target Chain 8	UniProt (TrEMBL) Entry Name of Target Chain 8	UniProt (TrEMBL) Primary ID of Target Chain 8	UniProt (TrEMBL) Secondary ID(s) of Target Chain 8	UniProt (TrEMBL) Alternative ID(s) of Target Chain 8	BindingDB Target Chain Sequence 9	PDB ID(s) of Target Chain 9	UniProt (SwissProt) Recommended Name of Target Chain 9	UniProt (SwissProt) Entry Name of Target Chain 9	UniProt (SwissProt) Primary ID of Target Chain 9	UniProt (SwissProt) Secondary ID(s) of Target Chain 9	UniProt (SwissProt) Alternative ID(s) of Target Chain 9	UniProt (TrEMBL) Submitted Name of Target Chain 9	UniProt (TrEMBL) Entry Name of Target Chain 9	UniProt (TrEMBL) Primary ID of Target Chain 9	UniProt (TrEMBL) Secondary ID(s) of Target Chain 9	UniProt (TrEMBL) Alternative ID(s) of Target Chain 9	BindingDB Target Chain Sequence 10	PDB ID(s) of Target Chain 10	UniProt (SwissProt) Recommended Name of Target Chain 10	UniProt (SwissProt) Entry Name of Target Chain 10	UniProt (SwissProt) Primary ID of Target Chain 10	UniProt (SwissProt) Secondary ID(s) of Target Chain 10	UniProt (SwissProt) Alternative ID(s) of Target Chain 10	UniProt (TrEMBL) Submitted Name of Target Chain 10	UniProt (TrEMBL) Entry Name of Target Chain 10	UniProt (TrEMBL) Primary ID of Target Chain 10	UniProt (TrEMBL) Secondary ID(s) of Target Chain 10	UniProt (TrEMBL) Alternative ID(s) of Target Chain 10	BindingDB Target Chain Sequence 11	PDB ID(s) of Target Chain 11	UniProt (SwissProt) Recommended Name of Target Chain 11	UniProt (SwissProt) Entry Name of Target Chain 11	UniProt (SwissProt) Primary ID of Target Chain 11	UniProt (SwissProt) Secondary ID(s) of Target Chain 11	UniProt (SwissProt) Alternative ID(s) of Target Chain 11	UniProt (TrEMBL) Submitted Name of Target Chain 11	UniProt (TrEMBL) Entry Name of Target Chain 11	UniProt (TrEMBL) Primary ID of Target Chain 11	UniProt (TrEMBL) Secondary ID(s) of Target Chain 11	UniProt (TrEMBL) Alternative ID(s) of Target Chain 11	BindingDB Target Chain Sequence 12	PDB ID(s) of Target Chain 12	UniProt (SwissProt) Recommended Name of Target Chain 12	UniProt (SwissProt) Entry Name of Target Chain 12	UniProt (SwissProt) Primary ID of Target Chain 12	UniProt (SwissProt) Secondary ID(s) of Target Chain 12	UniProt (SwissProt) Alternative ID(s) of Target Chain 12	UniProt (TrEMBL) Submitted Name of Target Chain 12	UniProt (TrEMBL) Entry Name of Target Chain 12	UniProt (TrEMBL) Primary ID of Target Chain 12	UniProt (TrEMBL) Secondary ID(s) of Target Chain 12	UniProt (TrEMBL) Alternative ID(s) of Target Chain 12	BindingDB Target Chain Sequence 13	PDB ID(s) of Target Chain 13	UniProt (SwissProt) Recommended Name of Target Chain 13	UniProt (SwissProt) Entry Name of Target Chain 13	UniProt (SwissProt) Primary ID of Target Chain 13	UniProt (SwissProt) Secondary ID(s) of Target Chain 13	UniProt (SwissProt) Alternative ID(s) of Target Chain 13	UniProt (TrEMBL) Submitted Name of Target Chain 13	UniProt (TrEMBL) Entry Name of Target Chain 13	UniProt (TrEMBL) Primary ID of Target Chain 13	UniProt (TrEMBL) Secondary ID(s) of Target Chain 13	UniProt (TrEMBL) Alternative ID(s) of Target Chain 13	BindingDB Target Chain Sequence 14	PDB ID(s) of Target Chain 14	UniProt (SwissProt) Recommended Name of Target Chain 14	UniProt (SwissProt) Entry Name of Target Chain 14	UniProt (SwissProt) Primary ID of Target Chain 14	UniProt (SwissProt) Secondary ID(s) of Target Chain 14	UniProt (SwissProt) Alternative ID(s) of Target Chain 14	UniProt (TrEMBL) Submitted Name of Target Chain 14	UniProt (TrEMBL) Entry Name of Target Chain 14	UniProt (TrEMBL) Primary ID of Target Chain 14	UniProt (TrEMBL) Secondary ID(s) of Target Chain 14	UniProt (TrEMBL) Alternative ID(s) of Target Chain 14	BindingDB Target Chain Sequence 15	PDB ID(s) of Target Chain 15	UniProt (SwissProt) Recommended Name of Target Chain 15	UniProt (SwissProt) Entry Name of Target Chain 15	UniProt (SwissProt) Primary ID of Target Chain 15	UniProt (SwissProt) Secondary ID(s) of Target Chain 15	UniProt (SwissProt) Alternative ID(s) of Target Chain 15	UniProt (TrEMBL) Submitted Name of Target Chain 15	UniProt (TrEMBL) Entry Name of Target Chain 15	UniProt (TrEMBL) Primary ID of Target Chain 15	UniProt (TrEMBL) Secondary ID(s) of Target Chain 15	UniProt (TrEMBL) Alternative ID(s) of Target Chain 15	BindingDB Target Chain Sequence 16	PDB ID(s) of Target Chain 16	UniProt (SwissProt) Recommended Name of Target Chain 16	UniProt (SwissProt) Entry Name of Target Chain 16	UniProt (SwissProt) Primary ID of Target Chain 16	UniProt (SwissProt) Secondary ID(s) of Target Chain 16	UniProt (SwissProt) Alternative ID(s) of Target Chain 16	UniProt (TrEMBL) Submitted Name of Target Chain 16	UniProt (TrEMBL) Entry Name of Target Chain 16	UniProt (TrEMBL) Primary ID of Target Chain 16	UniProt (TrEMBL) Secondary ID(s) of Target Chain 16	UniProt (TrEMBL) Alternative ID(s) of Target Chain 16	BindingDB Target Chain Sequence 17	PDB ID(s) of Target Chain 17	UniProt (SwissProt) Recommended Name of Target Chain 17	UniProt (SwissProt) Entry Name of Target Chain 17	UniProt (SwissProt) Primary ID of Target Chain 17	UniProt (SwissProt) Secondary ID(s) of Target Chain 17	UniProt (SwissProt) Alternative ID(s) of Target Chain 17	UniProt (TrEMBL) Submitted Name of Target Chain 17	UniProt (TrEMBL) Entry Name of Target Chain 17	UniProt (TrEMBL) Primary ID of Target Chain 17	UniProt (TrEMBL) Secondary ID(s) of Target Chain 17	UniProt (TrEMBL) Alternative ID(s) of Target Chain 17	BindingDB Target Chain Sequence 18	PDB ID(s) of Target Chain 18	UniProt (SwissProt) Recommended Name of Target Chain 18	UniProt (SwissProt) Entry Name of Target Chain 18	UniProt (SwissProt) Primary ID of Target Chain 18	UniProt (SwissProt) Secondary ID(s) of Target Chain 18	UniProt (SwissProt) Alternative ID(s) of Target Chain 18	UniProt (TrEMBL) Submitted Name of Target Chain 18	UniProt (TrEMBL) Entry Name of Target Chain 18	UniProt (TrEMBL) Primary ID of Target Chain 18	UniProt (TrEMBL) Secondary ID(s) of Target Chain 18	UniProt (TrEMBL) Alternative ID(s) of Target Chain 18	BindingDB Target Chain Sequence 19	PDB ID(s) of Target Chain 19	UniProt (SwissProt) Recommended Name of Target Chain 19	UniProt (SwissProt) Entry Name of Target Chain 19	UniProt (SwissProt) Primary ID of Target Chain 19	UniProt (SwissProt) Secondary ID(s) of Target Chain 19	UniProt (SwissProt) Alternative ID(s) of Target Chain 19	UniProt (TrEMBL) Submitted Name of Target Chain 19	UniProt (TrEMBL) Entry Name of Target Chain 19	UniProt (TrEMBL) Primary ID of Target Chain 19	UniProt (TrEMBL) Secondary ID(s) of Target Chain 19	UniProt (TrEMBL) Alternative ID(s) of Target Chain 19	BindingDB Target Chain Sequence 20	PDB ID(s) of Target Chain 20	UniProt (SwissProt) Recommended Name of Target Chain 20	UniProt (SwissProt) Entry Name of Target Chain 20	UniProt (SwissProt) Primary ID of Target Chain 20	UniProt (SwissProt) Secondary ID(s) of Target Chain 20	UniProt (SwissProt) Alternative ID(s) of Target Chain 20	UniProt (TrEMBL) Submitted Name of Target Chain 20	UniProt (TrEMBL) Entry Name of Target Chain 20	UniProt (TrEMBL) Primary ID of Target Chain 20	UniProt (TrEMBL) Secondary ID(s) of Target Chain 20	UniProt (TrEMBL) Alternative ID(s) of Target Chain 20	BindingDB Target Chain Sequence 21	PDB ID(s) of Target Chain 21	UniProt (SwissProt) Recommended Name of Target Chain 21	UniProt (SwissProt) Entry Name of Target Chain 21	UniProt (SwissProt) Primary ID of Target Chain 21	UniProt (SwissProt) Secondary ID(s) of Target Chain 21	UniProt (SwissProt) Alternative ID(s) of Target Chain 21	UniProt (TrEMBL) Submitted Name of Target Chain 21	UniProt (TrEMBL) Entry Name of Target Chain 21	UniProt (TrEMBL) Primary ID of Target Chain 21	UniProt (TrEMBL) Secondary ID(s) of Target Chain 21	UniProt (TrEMBL) Alternative ID(s) of Target Chain 21	BindingDB Target Chain Sequence 22	PDB ID(s) of Target Chain 22	UniProt (SwissProt) Recommended Name of Target Chain 22	UniProt (SwissProt) Entry Name of Target Chain 22	UniProt (SwissProt) Primary ID of Target Chain 22	UniProt (SwissProt) Secondary ID(s) of Target Chain 22	UniProt (SwissProt) Alternative ID(s) of Target Chain 22	UniProt (TrEMBL) Submitted Name of Target Chain 22	UniProt (TrEMBL) Entry Name of Target Chain 22	UniProt (TrEMBL) Primary ID of Target Chain 22	UniProt (TrEMBL) Secondary ID(s) of Target Chain 22	UniProt (TrEMBL) Alternative ID(s) of Target Chain 22	BindingDB Target Chain Sequence 23	PDB ID(s) of Target Chain 23	UniProt (SwissProt) Recommended Name of Target Chain 23	UniProt (SwissProt) Entry Name of Target Chain 23	UniProt (SwissProt) Primary ID of Target Chain 23	UniProt (SwissProt) Secondary ID(s) of Target Chain 23	UniProt (SwissProt) Alternative ID(s) of Target Chain 23	UniProt (TrEMBL) Submitted Name of Target Chain 23	UniProt (TrEMBL) Entry Name of Target Chain 23	UniProt (TrEMBL) Primary ID of Target Chain 23	UniProt (TrEMBL) Secondary ID(s) of Target Chain 23	UniProt (TrEMBL) Alternative ID(s) of Target Chain 23	BindingDB Target Chain Sequence 24	PDB ID(s) of Target Chain 24	UniProt (SwissProt) Recommended Name of Target Chain 24	UniProt (SwissProt) Entry Name of Target Chain 24	UniProt (SwissProt) Primary ID of Target Chain 24	UniProt (SwissProt) Secondary ID(s) of Target Chain 24	UniProt (SwissProt) Alternative ID(s) of Target Chain 24	UniProt (TrEMBL) Submitted Name of Target Chain 24	UniProt (TrEMBL) Entry Name of Target Chain 24	UniProt (TrEMBL) Primary ID of Target Chain 24	UniProt (TrEMBL) Secondary ID(s) of Target Chain 24	UniProt (TrEMBL) Alternative ID(s) of Target Chain 24	BindingDB Target Chain Sequence 25	PDB ID(s) of Target Chain 25	UniProt (SwissProt) Recommended Name of Target Chain 25	UniProt (SwissProt) Entry Name of Target Chain 25	UniProt (SwissProt) Primary ID of Target Chain 25	UniProt (SwissProt) Secondary ID(s) of Target Chain 25	UniProt (SwissProt) Alternative ID(s) of Target Chain 25	UniProt (TrEMBL) Submitted Name of Target Chain 25	UniProt (TrEMBL) Entry Name of Target Chain 25	UniProt (TrEMBL) Primary ID of Target Chain 25	UniProt (TrEMBL) Secondary ID(s) of Target Chain 25	UniProt (TrEMBL) Alternative ID(s) of Target Chain 25	BindingDB Target Chain Sequence 26	PDB ID(s) of Target Chain 26	UniProt (SwissProt) Recommended Name of Target Chain 26	UniProt (SwissProt) Entry Name of Target Chain 26	UniProt (SwissProt) Primary ID of Target Chain 26	UniProt (SwissProt) Secondary ID(s) of Target Chain 26	UniProt (SwissProt) Alternative ID(s) of Target Chain 26	UniProt (TrEMBL) Submitted Name of Target Chain 26	UniProt (TrEMBL) Entry Name of Target Chain 26	UniProt (TrEMBL) Primary ID of Target Chain 26	UniProt (TrEMBL) Secondary ID(s) of Target Chain 26	UniProt (TrEMBL) Alternative ID(s) of Target Chain 26	BindingDB Target Chain Sequence 27	PDB ID(s) of Target Chain 27	UniProt (SwissProt) Recommended Name of Target Chain 27	UniProt (SwissProt) Entry Name of Target Chain 27	UniProt (SwissProt) Primary ID of Target Chain 27	UniProt (SwissProt) Secondary ID(s) of Target Chain 27	UniProt (SwissProt) Alternative ID(s) of Target Chain 27	UniProt (TrEMBL) Submitted Name of Target Chain 27	UniProt (TrEMBL) Entry Name of Target Chain 27	UniProt (TrEMBL) Primary ID of Target Chain 27	UniProt (TrEMBL) Secondary ID(s) of Target Chain 27	UniProt (TrEMBL) Alternative ID(s) of Target Chain 27	BindingDB Target Chain Sequence 28	PDB ID(s) of Target Chain 28	UniProt (SwissProt) Recommended Name of Target Chain 28	UniProt (SwissProt) Entry Name of Target Chain 28	UniProt (SwissProt) Primary ID of Target Chain 28	UniProt (SwissProt) Secondary ID(s) of Target Chain 28	UniProt (SwissProt) Alternative ID(s) of Target Chain 28	UniProt (TrEMBL) Submitted Name of Target Chain 28	UniProt (TrEMBL) Entry Name of Target Chain 28	UniProt (TrEMBL) Primary ID of Target Chain 28	UniProt (TrEMBL) Secondary ID(s) of Target Chain 28	UniProt (TrEMBL) Alternative ID(s) of Target Chain 28	BindingDB Target Chain Sequence 29	PDB ID(s) of Target Chain 29	UniProt (SwissProt) Recommended Name of Target Chain 29	UniProt (SwissProt) Entry Name of Target Chain 29	UniProt (SwissProt) Primary ID of Target Chain 29	UniProt (SwissProt) Secondary ID(s) of Target Chain 29	UniProt (SwissProt) Alternative ID(s) of Target Chain 29	UniProt (TrEMBL) Submitted Name of Target Chain 29	UniProt (TrEMBL) Entry Name of Target Chain 29	UniProt (TrEMBL) Primary ID of Target Chain 29	UniProt (TrEMBL) Secondary ID(s) of Target Chain 29	UniProt (TrEMBL) Alternative ID(s) of Target Chain 29	BindingDB Target Chain Sequence 30	PDB ID(s) of Target Chain 30	UniProt (SwissProt) Recommended Name of Target Chain 30	UniProt (SwissProt) Entry Name of Target Chain 30	UniProt (SwissProt) Primary ID of Target Chain 30	UniProt (SwissProt) Secondary ID(s) of Target Chain 30	UniProt (SwissProt) Alternative ID(s) of Target Chain 30	UniProt (TrEMBL) Submitted Name of Target Chain 30	UniProt (TrEMBL) Entry Name of Target Chain 30	UniProt (TrEMBL) Primary ID of Target Chain 30	UniProt (TrEMBL) Secondary ID(s) of Target Chain 30	UniProt (TrEMBL) Alternative ID(s) of Target Chain 30	BindingDB Target Chain Sequence 31	PDB ID(s) of Target Chain 31	UniProt (SwissProt) Recommended Name of Target Chain 31	UniProt (SwissProt) Entry Name of Target Chain 31	UniProt (SwissProt) Primary ID of Target Chain 31	UniProt (SwissProt) Secondary ID(s) of Target Chain 31	UniProt (SwissProt) Alternative ID(s) of Target Chain 31	UniProt (TrEMBL) Submitted Name of Target Chain 31	UniProt (TrEMBL) Entry Name of Target Chain 31	UniProt (TrEMBL) Primary ID of Target Chain 31	UniProt (TrEMBL) Secondary ID(s) of Target Chain 31	UniProt (TrEMBL) Alternative ID(s) of Target Chain 31	BindingDB Target Chain Sequence 32	PDB ID(s) of Target Chain 32	UniProt (SwissProt) Recommended Name of Target Chain 32	UniProt (SwissProt) Entry Name of Target Chain 32	UniProt (SwissProt) Primary ID of Target Chain 32	UniProt (SwissProt) Secondary ID(s) of Target Chain 32	UniProt (SwissProt) Alternative ID(s) of Target Chain 32	UniProt (TrEMBL) Submitted Name of Target Chain 32	UniProt (TrEMBL) Entry Name of Target Chain 32	UniProt (TrEMBL) Primary ID of Target Chain 32	UniProt (TrEMBL) Secondary ID(s) of Target Chain 32	UniProt (TrEMBL) Alternative ID(s) of Target Chain 32	BindingDB Target Chain Sequence 33	PDB ID(s) of Target Chain 33	UniProt (SwissProt) Recommended Name of Target Chain 33	UniProt (SwissProt) Entry Name of Target Chain 33	UniProt (SwissProt) Primary ID of Target Chain 33	UniProt (SwissProt) Secondary ID(s) of Target Chain 33	UniProt (SwissProt) Alternative ID(s) of Target Chain 33	UniProt (TrEMBL) Submitted Name of Target Chain 33	UniProt (TrEMBL) Entry Name of Target Chain 33	UniProt (TrEMBL) Primary ID of Target Chain 33	UniProt (TrEMBL) Secondary ID(s) of Target Chain 33	UniProt (TrEMBL) Alternative ID(s) of Target Chain 33	BindingDB Target Chain Sequence 34	PDB ID(s) of Target Chain 34	UniProt (SwissProt) Recommended Name of Target Chain 34	UniProt (SwissProt) Entry Name of Target Chain 34	UniProt (SwissProt) Primary ID of Target Chain 34	UniProt (SwissProt) Secondary ID(s) of Target Chain 34	UniProt (SwissProt) Alternative ID(s) of Target Chain 34	UniProt (TrEMBL) Submitted Name of Target Chain 34	UniProt (TrEMBL) Entry Name of Target Chain 34	UniProt (TrEMBL) Primary ID of Target Chain 34	UniProt (TrEMBL) Secondary ID(s) of Target Chain 34	UniProt (TrEMBL) Alternative ID(s) of Target Chain 34	BindingDB Target Chain Sequence 35	PDB ID(s) of Target Chain 35	UniProt (SwissProt) Recommended Name of Target Chain 35	UniProt (SwissProt) Entry Name of Target Chain 35	UniProt (SwissProt) Primary ID of Target Chain 35	UniProt (SwissProt) Secondary ID(s) of Target Chain 35	UniProt (SwissProt) Alternative ID(s) of Target Chain 35	UniProt (TrEMBL) Submitted Name of Target Chain 35	UniProt (TrEMBL) Entry Name of Target Chain 35	UniProt (TrEMBL) Primary ID of Target Chain 35	UniProt (TrEMBL) Secondary ID(s) of Target Chain 35	UniProt (TrEMBL) Alternative ID(s) of Target Chain 35	BindingDB Target Chain Sequence 36	PDB ID(s) of Target Chain 36	UniProt (SwissProt) Recommended Name of Target Chain 36	UniProt (SwissProt) Entry Name of Target Chain 36	UniProt (SwissProt) Primary ID of Target Chain 36	UniProt (SwissProt) Secondary ID(s) of Target Chain 36	UniProt (SwissProt) Alternative ID(s) of Target Chain 36	UniProt (TrEMBL) Submitted Name of Target Chain 36	UniProt (TrEMBL) Entry Name of Target Chain 36	UniProt (TrEMBL) Primary ID of Target Chain 36	UniProt (TrEMBL) Secondary ID(s) of Target Chain 36	UniProt (TrEMBL) Alternative ID(s) of Target Chain 36	BindingDB Target Chain Sequence 37	PDB ID(s) of Target Chain 37	UniProt (SwissProt) Recommended Name of Target Chain 37	UniProt (SwissProt) Entry Name of Target Chain 37	UniProt (SwissProt) Primary ID of Target Chain 37	UniProt (SwissProt) Secondary ID(s) of Target Chain 37	UniProt (SwissProt) Alternative ID(s) of Target Chain 37	UniProt (TrEMBL) Submitted Name of Target Chain 37	UniProt (TrEMBL) Entry Name of Target Chain 37	UniProt (TrEMBL) Primary ID of Target Chain 37	UniProt (TrEMBL) Secondary ID(s) of Target Chain 37	UniProt (TrEMBL) Alternative ID(s) of Target Chain 37	BindingDB Target Chain Sequence 38	PDB ID(s) of Target Chain 38	UniProt (SwissProt) Recommended Name of Target Chain 38	UniProt (SwissProt) Entry Name of Target Chain 38	UniProt (SwissProt) Primary ID of Target Chain 38	UniProt (SwissProt) Secondary ID(s) of Target Chain 38	UniProt (SwissProt) Alternative ID(s) of Target Chain 38	UniProt (TrEMBL) Submitted Name of Target Chain 38	UniProt (TrEMBL) Entry Name of Target Chain 38	UniProt (TrEMBL) Primary ID of Target Chain 38	UniProt (TrEMBL) Secondary ID(s) of Target Chain 38	UniProt (TrEMBL) Alternative ID(s) of Target Chain 38	BindingDB Target Chain Sequence 39	PDB ID(s) of Target Chain 39	UniProt (SwissProt) Recommended Name of Target Chain 39	UniProt (SwissProt) Entry Name of Target Chain 39	UniProt (SwissProt) Primary ID of Target Chain 39	UniProt (SwissProt) Secondary ID(s) of Target Chain 39	UniProt (SwissProt) Alternative ID(s) of Target Chain 39	UniProt (TrEMBL) Submitted Name of Target Chain 39	UniProt (TrEMBL) Entry Name of Target Chain 39	UniProt (TrEMBL) Primary ID of Target Chain 39	UniProt (TrEMBL) Secondary ID(s) of Target Chain 39	UniProt (TrEMBL) Alternative ID(s) of Target Chain 39	BindingDB Target Chain Sequence 40	PDB ID(s) of Target Chain 40	UniProt (SwissProt) Recommended Name of Target Chain 40	UniProt (SwissProt) Entry Name of Target Chain 40	UniProt (SwissProt) Primary ID of Target Chain 40	UniProt (SwissProt) Secondary ID(s) of Target Chain 40	UniProt (SwissProt) Alternative ID(s) of Target Chain 40	UniProt (TrEMBL) Submitted Name of Target Chain 40	UniProt (TrEMBL) Entry Name of Target Chain 40	UniProt (TrEMBL) Primary ID of Target Chain 40	UniProt (TrEMBL) Secondary ID(s) of Target Chain 40	UniProt (TrEMBL) Alternative ID(s) of Target Chain 40	BindingDB Target Chain Sequence 41	PDB ID(s) of Target Chain 41	UniProt (SwissProt) Recommended Name of Target Chain 41	UniProt (SwissProt) Entry Name of Target Chain 41	UniProt (SwissProt) Primary ID of Target Chain 41	UniProt (SwissProt) Secondary ID(s) of Target Chain 41	UniProt (SwissProt) Alternative ID(s) of Target Chain 41	UniProt (TrEMBL) Submitted Name of Target Chain 41	UniProt (TrEMBL) Entry Name of Target Chain 41	UniProt (TrEMBL) Primary ID of Target Chain 41	UniProt (TrEMBL) Secondary ID(s) of Target Chain 41	UniProt (TrEMBL) Alternative ID(s) of Target Chain 41	BindingDB Target Chain Sequence 42	PDB ID(s) of Target Chain 42	UniProt (SwissProt) Recommended Name of Target Chain 42	UniProt (SwissProt) Entry Name of Target Chain 42	UniProt (SwissProt) Primary ID of Target Chain 42	UniProt (SwissProt) Secondary ID(s) of Target Chain 42	UniProt (SwissProt) Alternative ID(s) of Target Chain 42	UniProt (TrEMBL) Submitted Name of Target Chain 42	UniProt (TrEMBL) Entry Name of Target Chain 42	UniProt (TrEMBL) Primary ID of Target Chain 42	UniProt (TrEMBL) Secondary ID(s) of Target Chain 42	UniProt (TrEMBL) Alternative ID(s) of Target Chain 42	BindingDB Target Chain Sequence 43	PDB ID(s) of Target Chain 43	UniProt (SwissProt) Recommended Name of Target Chain 43	UniProt (SwissProt) Entry Name of Target Chain 43	UniProt (SwissProt) Primary ID of Target Chain 43	UniProt (SwissProt) Secondary ID(s) of Target Chain 43	UniProt (SwissProt) Alternative ID(s) of Target Chain 43	UniProt (TrEMBL) Submitted Name of Target Chain 43	UniProt (TrEMBL) Entry Name of Target Chain 43	UniProt (TrEMBL) Primary ID of Target Chain 43	UniProt (TrEMBL) Secondary ID(s) of Target Chain 43	UniProt (TrEMBL) Alternative ID(s) of Target Chain 43	BindingDB Target Chain Sequence 44	PDB ID(s) of Target Chain 44	UniProt (SwissProt) Recommended Name of Target Chain 44	UniProt (SwissProt) Entry Name of Target Chain 44	UniProt (SwissProt) Primary ID of Target Chain 44	UniProt (SwissProt) Secondary ID(s) of Target Chain 44	UniProt (SwissProt) Alternative ID(s) of Target Chain 44	UniProt (TrEMBL) Submitted Name of Target Chain 44	UniProt (TrEMBL) Entry Name of Target Chain 44	UniProt (TrEMBL) Primary ID of Target Chain 44	UniProt (TrEMBL) Secondary ID(s) of Target Chain 44	UniProt (TrEMBL) Alternative ID(s) of Target Chain 44	BindingDB Target Chain Sequence 45	PDB ID(s) of Target Chain 45	UniProt (SwissProt) Recommended Name of Target Chain 45	UniProt (SwissProt) Entry Name of Target Chain 45	UniProt (SwissProt) Primary ID of Target Chain 45	UniProt (SwissProt) Secondary ID(s) of Target Chain 45	UniProt (SwissProt) Alternative ID(s) of Target Chain 45	UniProt (TrEMBL) Submitted Name of Target Chain 45	UniProt (TrEMBL) Entry Name of Target Chain 45	UniProt (TrEMBL) Primary ID of Target Chain 45	UniProt (TrEMBL) Secondary ID(s) of Target Chain 45	UniProt (TrEMBL) Alternative ID(s) of Target Chain 45	BindingDB Target Chain Sequence 46	PDB ID(s) of Target Chain 46	UniProt (SwissProt) Recommended Name of Target Chain 46	UniProt (SwissProt) Entry Name of Target Chain 46	UniProt (SwissProt) Primary ID of Target Chain 46	UniProt (SwissProt) Secondary ID(s) of Target Chain 46	UniProt (SwissProt) Alternative ID(s) of Target Chain 46	UniProt (TrEMBL) Submitted Name of Target Chain 46	UniProt (TrEMBL) Entry Name of Target Chain 46	UniProt (TrEMBL) Primary ID of Target Chain 46	UniProt (TrEMBL) Secondary ID(s) of Target Chain 46	UniProt (TrEMBL) Alternative ID(s) of Target Chain 46	BindingDB Target Chain Sequence 47	PDB ID(s) of Target Chain 47	UniProt (SwissProt) Recommended Name of Target Chain 47	UniProt (SwissProt) Entry Name of Target Chain 47	UniProt (SwissProt) Primary ID of Target Chain 47	UniProt (SwissProt) Secondary ID(s) of Target Chain 47	UniProt (SwissProt) Alternative ID(s) of Target Chain 47	UniProt (TrEMBL) Submitted Name of Target Chain 47	UniProt (TrEMBL) Entry Name of Target Chain 47	UniProt (TrEMBL) Primary ID of Target Chain 47	UniProt (TrEMBL) Secondary ID(s) of Target Chain 47	UniProt (TrEMBL) Alternative ID(s) of Target Chain 47	BindingDB Target Chain Sequence 48	PDB ID(s) of Target Chain 48	UniProt (SwissProt) Recommended Name of Target Chain 48	UniProt (SwissProt) Entry Name of Target Chain 48	UniProt (SwissProt) Primary ID of Target Chain 48	UniProt (SwissProt) Secondary ID(s) of Target Chain 48	UniProt (SwissProt) Alternative ID(s) of Target Chain 48	UniProt (TrEMBL) Submitted Name of Target Chain 48	UniProt (TrEMBL) Entry Name of Target Chain 48	UniProt (TrEMBL) Primary ID of Target Chain 48	UniProt (TrEMBL) Secondary ID(s) of Target Chain 48	UniProt (TrEMBL) Alternative ID(s) of Target Chain 48	BindingDB Target Chain Sequence 49	PDB ID(s) of Target Chain 49	UniProt (SwissProt) Recommended Name of Target Chain 49	UniProt (SwissProt) Entry Name of Target Chain 49	UniProt (SwissProt) Primary ID of Target Chain 49	UniProt (SwissProt) Secondary ID(s) of Target Chain 49	UniProt (SwissProt) Alternative ID(s) of Target Chain 49	UniProt (TrEMBL) Submitted Name of Target Chain 49	UniProt (TrEMBL) Entry Name of Target Chain 49	UniProt (TrEMBL) Primary ID of Target Chain 49	UniProt (TrEMBL) Secondary ID(s) of Target Chain 49	UniProt (TrEMBL) Alternative ID(s) of Target Chain 49	BindingDB Target Chain Sequence 50	PDB ID(s) of Target Chain 50	UniProt (SwissProt) Recommended Name of Target Chain 50	UniProt (SwissProt) Entry Name of Target Chain 50	UniProt (SwissProt) Primary ID of Target Chain 50	UniProt (SwissProt) Secondary ID(s) of Target Chain 50	UniProt (SwissProt) Alternative ID(s) of Target Chain 50	UniProt (TrEMBL) Submitted Name of Target Chain 50	UniProt (TrEMBL) Entry Name of Target Chain 50	UniProt (TrEMBL) Primary ID of Target Chain 50	UniProt (TrEMBL) Secondary ID(s) of Target Chain 50	UniProt (TrEMBL) Alternative ID(s) of Target Chain 50
192689	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccccc1C(F)(F)F	InChI=1S/C21H18F3N3O3/c1-29-18-8-12(14-9-19(28)26-20-15(14)10-25-27-20)6-7-17(18)30-11-13-4-2-3-5-16(13)21(22,23)24/h2-8,10,14H,9,11H2,1H3,(H2,25,26,27,28)	MUMZZCYJPMFJKK-UHFFFAOYSA-N	368764	4-(3-methoxy-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 1	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368764	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368764&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			73389132	402365564							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192690	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccccc1Cl	InChI=1S/C20H18ClN3O3/c1-26-18-8-12(14-9-19(25)23-20-15(14)10-22-24-20)6-7-17(18)27-11-13-4-2-3-5-16(13)21/h2-8,10,14H,9,11H2,1H3,(H2,22,23,24,25)	JNDNUCRTMNCDPI-UHFFFAOYSA-N	368765	4-{4-[(2-chlorophenyl)methoxy]-3-methoxyphenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 2	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368765	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368765&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114330	402365565							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192691	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccccc1Br	InChI=1S/C20H18BrN3O3/c1-26-18-8-12(14-9-19(25)23-20-15(14)10-22-24-20)6-7-17(18)27-11-13-4-2-3-5-16(13)21/h2-8,10,14H,9,11H2,1H3,(H2,22,23,24,25)	QVVUFUHYCGIKSF-UHFFFAOYSA-N	368766	4-{4-[(2-bromophenyl)methoxy]-3-methoxyphenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 4	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368766	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368766&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115246	402365566							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192692	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(C(F)(F)F)cc1C(F)(F)F	InChI=1S/C22H17F6N3O3/c1-33-18-6-11(14-8-19(32)30-20-15(14)9-29-31-20)3-5-17(18)34-10-12-2-4-13(21(23,24)25)7-16(12)22(26,27)28/h2-7,9,14H,8,10H2,1H3,(H2,29,30,31,32)	STNNMOQNYDRPAH-UHFFFAOYSA-N	368767	4-(4-{[2,4-bis(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 8	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368767	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368767&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114806	402365567							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192693	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(F)cc1C(F)(F)F	InChI=1S/C21H17F4N3O3/c1-30-18-6-11(14-8-19(29)27-20-15(14)9-26-28-20)3-5-17(18)31-10-12-2-4-13(22)7-16(12)21(23,24)25/h2-7,9,14H,8,10H2,1H3,(H2,26,27,28,29)	DVXLZZCOKRXNPO-UHFFFAOYSA-N	368768	4-(4-{[4-fluoro-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 9	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368768	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368768&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114888	402365568							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192694	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1cccc(Br)c1	InChI=1S/C20H18BrN3O3/c1-26-18-8-13(15-9-19(25)23-20-16(15)10-22-24-20)5-6-17(18)27-11-12-3-2-4-14(21)7-12/h2-8,10,15H,9,11H2,1H3,(H2,22,23,24,25)	CXJBAQWSZWMGLZ-UHFFFAOYSA-N	368769	4-{4-[(3-bromophenyl)methoxy]-3-methoxyphenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 11	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368769	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368769&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114865	402365569							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192695	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1cc(C(F)(F)F)ccc1C(F)(F)F	InChI=1S/C22H17F6N3O3/c1-33-18-7-11(14-8-19(32)30-20-15(14)9-29-31-20)2-5-17(18)34-10-12-6-13(21(23,24)25)3-4-16(12)22(26,27)28/h2-7,9,14H,8,10H2,1H3,(H2,29,30,31,32)	SBGABTXRUFYBID-UHFFFAOYSA-N	368770	4-(4-{[2,5-bis(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 14	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368770	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368770&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115491	402365570							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192696	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(Cl)cc1C(F)(F)F	InChI=1S/C21H17ClF3N3O3/c1-30-18-6-11(14-8-19(29)27-20-15(14)9-26-28-20)3-5-17(18)31-10-12-2-4-13(22)7-16(12)21(23,24)25/h2-7,9,14H,8,10H2,1H3,(H2,26,27,28,29)	AOJVPOVPZVUHDF-UHFFFAOYSA-N	368771	4-(4-{[4-chloro-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 15	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368771	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368771&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114426	402365571							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192697	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccccc1OC(F)F	InChI=1S/C21H19F2N3O4/c1-28-18-8-12(14-9-19(27)25-20-15(14)10-24-26-20)6-7-17(18)29-11-13-4-2-3-5-16(13)30-21(22)23/h2-8,10,14,21H,9,11H2,1H3,(H2,24,25,26,27)	NJXAKXSVQHGQHW-UHFFFAOYSA-N	368772	4-(4-{[2-(difluoromethoxy)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 17	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368772	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368772&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115486	402365572							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192698	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccccc1[N+](=O)[O-]	InChI=1S/C20H18N4O5/c1-28-18-8-12(14-9-19(25)22-20-15(14)10-21-23-20)6-7-17(18)29-11-13-4-2-3-5-16(13)24(26)27/h2-8,10,14H,9,11H2,1H3,(H2,21,22,23,25)	VIKGPDQVLNQHEC-UHFFFAOYSA-N	368773	4-{3-methoxy-4-[(2-nitrophenyl)methoxy]phenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 18	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368773	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368773&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90137123	402365573							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192699	COc1ccc(COc2ccc(C3CC(=O)Nc4n[nH]cc43)cc2OC)c(C(F)(F)F)c1	InChI=1S/C22H20F3N3O4/c1-30-14-5-3-13(17(8-14)22(23,24)25)11-32-18-6-4-12(7-19(18)31-2)15-9-20(29)27-21-16(15)10-26-28-21/h3-8,10,15H,9,11H2,1-2H3,(H2,26,27,28,29)	KHTGVXXFEDNKNO-UHFFFAOYSA-N	368774	4-(3-methoxy-4-{[4-methoxy-2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 19	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368774	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368774&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114583	402365574							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192700	N#Cc1ccc(COc2ccc(C3CC(=O)Nc4n[nH]cc43)cc2OC)c(C(F)(F)F)c1	InChI=1S/C22H17F3N4O3/c1-31-19-7-13(15-8-20(30)28-21-16(15)10-27-29-21)4-5-18(19)32-11-14-3-2-12(9-26)6-17(14)22(23,24)25/h2-7,10,15H,8,11H2,1H3,(H2,27,28,29,30)	AEWFFIROLRBWSL-UHFFFAOYSA-N	368775	4-(2-methoxy-4-{6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}phenoxymethyl)-3-(trifluoromethyl)benzonitrile::US12527774, Compound 20	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368775	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368775&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114639	402365575							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192701	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1c(F)cccc1C(F)(F)F	InChI=1S/C21H17F4N3O3/c1-30-18-7-11(12-8-19(29)27-20-13(12)9-26-28-20)5-6-17(18)31-10-14-15(21(23,24)25)3-2-4-16(14)22/h2-7,9,12H,8,10H2,1H3,(H2,26,27,28,29)	QGYGJGJIMPJQDI-UHFFFAOYSA-N	368776	4-(4-{[2-fluoro-6-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 21	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368776	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368776&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114556	402365576							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192702	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1cccc(Cl)c1Cl	InChI=1S/C20H17Cl2N3O3/c1-27-17-7-11(13-8-18(26)24-20-14(13)9-23-25-20)5-6-16(17)28-10-12-3-2-4-15(21)19(12)22/h2-7,9,13H,8,10H2,1H3,(H2,23,24,25,26)	DLGXRFVLKXLCKO-UHFFFAOYSA-N	368777	4-{4-[(2,3-dichlorophenyl)methoxy]-3-methoxyphenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 22	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368777	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368777&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114536	402365577							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192703	COc3cc(C2CC(=O)Nc1n[nH]cc12)ccc3OCc4ccccc4I	InChI=1S/C20H18IN3O3/c1-26-18-8-12(14-9-19(25)23-20-15(14)10-22-24-20)6-7-17(18)27-11-13-4-2-3-5-16(13)21/h2-8,10,14H,9,11H2,1H3,(H2,22,23,24,25)	UZXLNROIUDWJQD-UHFFFAOYSA-N	368778	4-{4-[(2-iodophenyl)methoxy]-3-methoxyphenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 23	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368778	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368778&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114626	402365578							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192704	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccccc1OC(F)(F)F	InChI=1S/C21H18F3N3O4/c1-29-18-8-12(14-9-19(28)26-20-15(14)10-25-27-20)6-7-17(18)30-11-13-4-2-3-5-16(13)31-21(22,23)24/h2-8,10,14H,9,11H2,1H3,(H2,25,26,27,28)	QKJCGKWKCSIIFS-UHFFFAOYSA-N	368779	4-(3-methoxy-4-{[2-(trifluoromethoxy)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 24	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368779	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368779&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			73291754	402365579							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192705	COc1ccc([N+](=O)[O-])cc1COc1ccc(C2CC(=O)Nc3n[nH]cc32)cc1OC	InChI=1S/C21H20N4O6/c1-29-17-6-4-14(25(27)28)7-13(17)11-31-18-5-3-12(8-19(18)30-2)15-9-20(26)23-21-16(15)10-22-24-21/h3-8,10,15H,9,11H2,1-2H3,(H2,22,23,24,26)	CAVTUPQIBHIPMD-UHFFFAOYSA-N	368780	4-{3-methoxy-4-[(2-methoxy-5-nitrophenyl)methoxy]phenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 25	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368780	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368780&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			73389131	402365580							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192706	COC(=O)c1ccccc1COc1ccc(C2CC(=O)Nc3n[nH]cc32)cc1OC	InChI=1S/C22H21N3O5/c1-28-19-9-13(16-10-20(26)24-21-17(16)11-23-25-21)7-8-18(19)30-12-14-5-3-4-6-15(14)22(27)29-2/h3-9,11,16H,10,12H2,1-2H3,(H2,23,24,25,26)	PIRISHJEYQDJPH-UHFFFAOYSA-N	368781	methyl 2-(2-methoxy-4-{6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}phenoxymethyl)benzoate::US12527774, Compound 26	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368781	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368781&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114637	402365581							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192707	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1cccc(C(F)(F)F)c1F	InChI=1S/C21H17F4N3O3/c1-30-17-7-11(13-8-18(29)27-20-14(13)9-26-28-20)5-6-16(17)31-10-12-3-2-4-15(19(12)22)21(23,24)25/h2-7,9,13H,8,10H2,1H3,(H2,26,27,28,29)	GTXQPIVTTOOMFK-UHFFFAOYSA-N	368782	4-(4-{[2-fluoro-3-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 28	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368782	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368782&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114348	402365582							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192708	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1cc(Cl)ccc1Cl	InChI=1S/C20H17Cl2N3O3/c1-27-18-7-11(14-8-19(26)24-20-15(14)9-23-25-20)2-5-17(18)28-10-12-6-13(21)3-4-16(12)22/h2-7,9,14H,8,10H2,1H3,(H2,23,24,25,26)	SNOATNAMTCGKEI-UHFFFAOYSA-N	368783	4-{4-[(2,5-dichlorophenyl)methoxy]-3-methoxyphenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 29	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368783	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368783&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114376	402365583							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192709	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccccc1OC(F)(F)F	InChI=1S/C21H18F3N3O4/c1-29-18-8-12(14-9-19(28)26-20-15(14)10-25-27-20)6-7-17(18)30-11-13-4-2-3-5-16(13)31-21(22,23)24/h2-8,10,14H,9,11H2,1H3,(H2,25,26,27,28)	QKJCGKWKCSIIFS-UHFFFAOYSA-N	368784	4-{3-methoxy-4-[(2-methoxyphenyl)methoxy]phenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 30	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368784	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368784&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115114	402365584							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192710	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1cc(Cl)cc(Cl)c1Cl	InChI=1S/C20H16Cl3N3O3/c1-28-17-5-10(13-7-18(27)25-20-14(13)8-24-26-20)2-3-16(17)29-9-11-4-12(21)6-15(22)19(11)23/h2-6,8,13H,7,9H2,1H3,(H2,24,25,26,27)	CJQWIDJITZCKTH-UHFFFAOYSA-N	368785	4-{3-methoxy-4-[(2,3,5-trichlorophenyl)methoxy]phenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 31	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368785	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368785&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114480	402365585							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192711	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1cc(C)ccc1C(F)(F)F	InChI=1S/C22H20F3N3O3/c1-12-3-5-17(22(23,24)25)14(7-12)11-31-18-6-4-13(8-19(18)30-2)15-9-20(29)27-21-16(15)10-26-28-21/h3-8,10,15H,9,11H2,1-2H3,(H2,26,27,28,29)	GXGLHTAMPVULHR-UHFFFAOYSA-N	368786	4-(3-methoxy-4-{[5-methyl-2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 32	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368786	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368786&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114039	402365586							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192712	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(Br)cc1C(F)(F)F	InChI=1S/C21H17BrF3N3O3/c1-30-18-6-11(14-8-19(29)27-20-15(14)9-26-28-20)3-5-17(18)31-10-12-2-4-13(22)7-16(12)21(23,24)25/h2-7,9,14H,8,10H2,1H3,(H2,26,27,28,29)	YFUWRDYQXQGUPH-UHFFFAOYSA-N	368787	4-(4-{[4-bromo-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 33	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368787	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368787&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90113995	402365587							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192713	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc([N+](=O)[O-])cc1C(F)(F)F	InChI=1S/C21H17F3N4O5/c1-32-18-6-11(14-8-19(29)26-20-15(14)9-25-27-20)3-5-17(18)33-10-12-2-4-13(28(30)31)7-16(12)21(22,23)24/h2-7,9,14H,8,10H2,1H3,(H2,25,26,27,29)	TUODFIZRAZWMET-UHFFFAOYSA-N	368788	4-(3-methoxy-4-{[4-nitro-2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 34	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368788	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368788&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115286	402365588							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192714	COc1ccc(C(F)(F)F)c(COc2ccc(C3CC(=O)Nc4n[nH]cc43)cc2OC)c1	InChI=1S/C22H20F3N3O4/c1-30-14-4-5-17(22(23,24)25)13(7-14)11-32-18-6-3-12(8-19(18)31-2)15-9-20(29)27-21-16(15)10-26-28-21/h3-8,10,15H,9,11H2,1-2H3,(H2,26,27,28,29)	MGBLYHOLNQYUSM-UHFFFAOYSA-N	368789	4-(3-methoxy-4-{[5-methoxy-2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 35	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368789	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368789&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114759	402365589							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192715	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1cccc(OC)c1C(F)(F)F	InChI=1S/C22H20F3N3O4/c1-30-17-5-3-4-13(20(17)22(23,24)25)11-32-16-7-6-12(8-18(16)31-2)14-9-19(29)27-21-15(14)10-26-28-21/h3-8,10,14H,9,11H2,1-2H3,(H2,26,27,28,29)	KHSCHICIEDRROJ-UHFFFAOYSA-N	368790	4-(3-methoxy-4-{[3-methoxy-2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 36	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368790	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368790&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115466	402365590							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192716	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(S(C)(=O)=O)cc1C(F)(F)F	InChI=1S/C22H20F3N3O5S/c1-32-19-7-12(15-9-20(29)27-21-16(15)10-26-28-21)4-6-18(19)33-11-13-3-5-14(34(2,30)31)8-17(13)22(23,24)25/h3-8,10,15H,9,11H2,1-2H3,(H2,26,27,28,29)	LOEQLWSTPBCJMO-UHFFFAOYSA-N	368791	4-(4-{[4-methanesulfonyl-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 37	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368791	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368791&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114733	402365591							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192717	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1cccc(OC)c1OC	InChI=1S/C22H23N3O5/c1-27-18-6-4-5-14(21(18)29-3)12-30-17-8-7-13(9-19(17)28-2)15-10-20(26)24-22-16(15)11-23-25-22/h4-9,11,15H,10,12H2,1-3H3,(H2,23,24,25,26)	YLHXCJFVYMORRB-UHFFFAOYSA-N	368792	4-{4-[(2,3-dimethoxyphenyl)methoxy]-3-methoxyphenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 39	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368792	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368792&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115203	402365592							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192718	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccccc1C(C)(C)C	InChI=1S/C24H27N3O3/c1-24(2,3)19-8-6-5-7-16(19)14-30-20-10-9-15(11-21(20)29-4)17-12-22(28)26-23-18(17)13-25-27-23/h5-11,13,17H,12,14H2,1-4H3,(H2,25,26,27,28)	UQMPGCJHAFZIHO-UHFFFAOYSA-N	368793	4-{4-[(2-tert-butylphenyl)methoxy]-3-methoxyphenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 40	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368793	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368793&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114794	402365593							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192719	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(C(C)=O)cc1C(F)(F)F	InChI=1S/C23H20F3N3O4/c1-12(30)13-3-4-15(18(7-13)23(24,25)26)11-33-19-6-5-14(8-20(19)32-2)16-9-21(31)28-22-17(16)10-27-29-22/h3-8,10,16H,9,11H2,1-2H3,(H2,27,28,29,31)	RQNAGACDVZRQDN-UHFFFAOYSA-N	368794	4-(4-{[4-acetyl-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 41	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368794	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368794&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114185	402365594							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192720	COC(=O)c1ccc(COc2ccc(C3CC(=O)Nc4n[nH]cc43)cc2OC)c(C(F)(F)F)c1	InChI=1S/C23H20F3N3O5/c1-32-19-8-12(15-9-20(30)28-21-16(15)10-27-29-21)5-6-18(19)34-11-14-4-3-13(22(31)33-2)7-17(14)23(24,25)26/h3-8,10,15H,9,11H2,1-2H3,(H2,27,28,29,30)	NOULXOMUJGKWCD-UHFFFAOYSA-N	368795	methyl 4-[(2-methoxy-4-{6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}phenoxy)methyl]-3-(trifluoromethyl)benzoate::US12527774, Compound 42	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368795	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368795&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114439	402365595							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192721	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1cc2c(cc1Br)OCO2	InChI=1S/C21H18BrN3O5/c1-27-17-4-11(13-6-20(26)24-21-14(13)8-23-25-21)2-3-16(17)28-9-12-5-18-19(7-15(12)22)30-10-29-18/h2-5,7-8,13H,6,9-10H2,1H3,(H2,23,24,25,26)	UNJREMKJQSBTCZ-UHFFFAOYSA-N	368796	4-{4-[(6-bromo-2H-1,3-benzodioxol-5-yl)methoxy]-3-methoxyphenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 43	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368796	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368796&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115172	402365596							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192722	C#Cc1ccccc1COc1ccc(C2CC(=O)Nc3n[nH]cc32)cc1OC	InChI=1S/C22H19N3O3/c1-3-14-6-4-5-7-16(14)13-28-19-9-8-15(10-20(19)27-2)17-11-21(26)24-22-18(17)12-23-25-22/h1,4-10,12,17H,11,13H2,2H3,(H2,23,24,25,26)	RQADNILNPQUWKW-UHFFFAOYSA-N	368797	4-{4-[(2-ethynylphenyl)methoxy]-3-methoxyphenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 44	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368797	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368797&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115083	402365597							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192723	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1cccc2ccsc12	InChI=1S/C22H19N3O3S/c1-27-19-9-14(16-10-20(26)24-22-17(16)11-23-25-22)5-6-18(19)28-12-15-4-2-3-13-7-8-29-21(13)15/h2-9,11,16H,10,12H2,1H3,(H2,23,24,25,26)	FIMDEMYKGIKCGZ-UHFFFAOYSA-N	368798	4-{4-[(1-benzothiophen-7-yl)methoxy]-3-methoxyphenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 45	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368798	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368798&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115041	402365598							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192724	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1cccc2c1OC(C)(C)C2	InChI=1S/C24H25N3O4/c1-24(2)11-15-5-4-6-16(22(15)31-24)13-30-19-8-7-14(9-20(19)29-3)17-10-21(28)26-23-18(17)12-25-27-23/h4-9,12,17H,10-11,13H2,1-3H3,(H2,25,26,27,28)	HSFJUCKYKRLAIR-UHFFFAOYSA-N	368799	4-{4-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-7-yl)methoxy]-3-methoxyphenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 46	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368799	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368799&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90137115	402365599							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192725	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1cccc2cccnc12	InChI=1S/C23H20N4O3/c1-29-20-10-15(17-11-21(28)26-23-18(17)12-25-27-23)7-8-19(20)30-13-16-5-2-4-14-6-3-9-24-22(14)16/h2-10,12,17H,11,13H2,1H3,(H2,25,26,27,28)	WQPHWUBSDYNCCI-UHFFFAOYSA-N	368800	4-{3-methoxy-4-[(quinolin-8-yl)methoxy]phenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 47	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368800	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368800&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90134696	402365600							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192726	CCOC(=O)c1ccccc1COc1ccc(C2CC(=O)Nc3n[nH]cc32)cc1OC	InChI=1S/C23H23N3O5/c1-3-30-23(28)16-7-5-4-6-15(16)13-31-19-9-8-14(10-20(19)29-2)17-11-21(27)25-22-18(17)12-24-26-22/h4-10,12,17H,3,11,13H2,1-2H3,(H2,24,25,26,27)	IFLRRGDVGAGLEA-UHFFFAOYSA-N	368801	ethyl 2-[(2-methoxy-4-{6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}phenoxy)methyl]benzoate::US12527774, Compound 48	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368801	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368801&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			89993979	402365601							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192727	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccccc1C(F)F	InChI=1S/C21H19F2N3O3/c1-28-18-8-12(15-9-19(27)25-21-16(15)10-24-26-21)6-7-17(18)29-11-13-4-2-3-5-14(13)20(22)23/h2-8,10,15,20H,9,11H2,1H3,(H2,24,25,26,27)	MGHLGRXJXKYGSJ-UHFFFAOYSA-N	368802	4-(4-{[2-(difluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 49	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368802	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368802&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			89993980	402365602							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192728	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccncc1C(F)F	InChI=1S/C20H18F2N4O3/c1-28-17-6-11(13-7-18(27)25-20-15(13)9-24-26-20)2-3-16(17)29-10-12-4-5-23-8-14(12)19(21)22/h2-6,8-9,13,19H,7,10H2,1H3,(H2,24,25,26,27)	ARRZLZHZWFNZKT-UHFFFAOYSA-N	368803	4-(3-methoxy-4-{[3-(trifluoromethyl)pyridin-4-yl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 50	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368803	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368803&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115403	402365603							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192729	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1cccc2c1OCCCO2	InChI=1S/C23H23N3O5/c1-28-20-10-14(16-11-21(27)25-23-17(16)12-24-26-23)6-7-18(20)31-13-15-4-2-5-19-22(15)30-9-3-8-29-19/h2,4-7,10,12,16H,3,8-9,11,13H2,1H3,(H2,24,25,26,27)	KAKDPFHGMJCVJW-UHFFFAOYSA-N	368804	4-{4-[(3,4-dihydro-2H-1,5-benzodioxepin-6-yl)methoxy]-3-methoxyphenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 51	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368804	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368804&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114384	402365604							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192730	O=C1CC(c2ccc(OCc3ccccc3Br)cc2)c2c[nH]nc2N1	InChI=1S/C19H16BrN3O2/c20-17-4-2-1-3-13(17)11-25-14-7-5-12(6-8-14)15-9-18(24)22-19-16(15)10-21-23-19/h1-8,10,15H,9,11H2,(H2,21,22,23,24)	ZEYAFIDUUQDKIM-UHFFFAOYSA-N	368805	4-{4-[(2-bromophenyl)methoxy]phenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 58	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368805	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368805&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			89993984	402365605							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192731	O=C1CC(c2ccc(OCc3ccccc3C(F)(F)F)cc2)c2c[nH]nc2N1	InChI=1S/C20H16F3N3O2/c21-20(22,23)17-4-2-1-3-13(17)11-28-14-7-5-12(6-8-14)15-9-18(27)25-19-16(15)10-24-26-19/h1-8,10,15H,9,11H2,(H2,24,25,26,27)	ILXRESZABULSEO-UHFFFAOYSA-N	368806	4-(4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 59	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368806	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368806&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115038	402365606							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192732	O=C1CC(c2ccc(OCc3ccccc3Cl)cc2)c2c[nH]nc2N1	InChI=1S/C19H16ClN3O2/c20-17-4-2-1-3-13(17)11-25-14-7-5-12(6-8-14)15-9-18(24)22-19-16(15)10-21-23-19/h1-8,10,15H,9,11H2,(H2,21,22,23,24)	MDEWARWDVLDPJR-UHFFFAOYSA-N	368807	4-{4-[(2-chlorophenyl)methoxy]phenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 60	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368807	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368807&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114523	402365607							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192733	CCOc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccccc1C(F)(F)F	InChI=1S/C22H20F3N3O3/c1-2-30-19-9-13(15-10-20(29)27-21-16(15)11-26-28-21)7-8-18(19)31-12-14-5-3-4-6-17(14)22(23,24)25/h3-9,11,15H,2,10,12H2,1H3,(H2,26,27,28,29)	NXVBGSOYUDWPJJ-UHFFFAOYSA-N	368808	4-(3-ethoxy-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 62	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368808	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368808&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90137113	402365608							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192734	O=C1CC(c2ccc(OCc3ccccc3C(F)(F)F)cn2)c2c[nH]nc2N1	InChI=1S/C19H15F3N4O2/c20-19(21,22)15-4-2-1-3-11(15)10-28-12-5-6-16(23-8-12)13-7-17(27)25-18-14(13)9-24-26-18/h1-6,8-9,13H,7,10H2,(H2,24,25,26,27)	DRZARSINLGOEFV-UHFFFAOYSA-N	368809	4-(5-{[2-(trifluoromethyl)phenyl]methoxy}pyridin-2-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 63	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368809	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368809&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114233	402365609							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192735	COc1cc(OCc2ccccc2C(F)(F)F)ccc1C1CC(=O)Nc2n[nH]cc21	InChI=1S/C21H18F3N3O3/c1-29-18-8-13(30-11-12-4-2-3-5-17(12)21(22,23)24)6-7-14(18)15-9-19(28)26-20-16(15)10-25-27-20/h2-8,10,15H,9,11H2,1H3,(H2,25,26,27,28)	PTOLPNQGIQFRKZ-UHFFFAOYSA-N	368810	4-(2-methoxy-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 64	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368810	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368810&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114996	402365610							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192736	COC(=O)c1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccccc1C(F)(F)F	InChI=1S/C22H18F3N3O4/c1-31-21(30)15-8-12(14-9-19(29)27-20-16(14)10-26-28-20)6-7-18(15)32-11-13-4-2-3-5-17(13)22(23,24)25/h2-8,10,14H,9,11H2,1H3,(H2,26,27,28,29)	VTWMAGAMMKNDCP-UHFFFAOYSA-N	368811	methyl 5-{6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}-2-{[2-(trifluoromethyl)phenyl]methoxy}benzoate::US12527774, Compound 65	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368811	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368811&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115321	402365611							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192737	O=C1CC(c2ccc(OCc3ccccc3C(F)(F)F)cc2F)c2c[nH]nc2N1	InChI=1S/C20H15F4N3O2/c21-17-7-12(29-10-11-3-1-2-4-16(11)20(22,23)24)5-6-13(17)14-8-18(28)26-19-15(14)9-25-27-19/h1-7,9,14H,8,10H2,(H2,25,26,27,28)	GDDBUONCMPBFHT-UHFFFAOYSA-N	368812	4-(2-fluoro-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 66	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368812	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368812&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114689	402365612							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192738	O=C1CC(c2ccc(OCc3ccccc3C(F)(F)F)c([N+](=O)[O-])c2)c2c[nH]nc2N1	InChI=1S/C20H15F3N4O4/c21-20(22,23)15-4-2-1-3-12(15)10-31-17-6-5-11(7-16(17)27(29)30)13-8-18(28)25-19-14(13)9-24-26-19/h1-7,9,13H,8,10H2,(H2,24,25,26,28)	BXDYISCGYYKRBI-UHFFFAOYSA-N	368813	4-(3-nitro-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 67	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368813	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368813&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114662	402365613							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192739	O=C1CC(c2ccc(OCc3ccccc3C(F)(F)F)c(OC(F)F)c2)c2c[nH]nc2N1	InChI=1S/C21H16F5N3O3/c22-20(23)32-17-7-11(13-8-18(30)28-19-14(13)9-27-29-19)5-6-16(17)31-10-12-3-1-2-4-15(12)21(24,25)26/h1-7,9,13,20H,8,10H2,(H2,27,28,29,30)	UJPVMDWFNKLYQU-UHFFFAOYSA-N	368814	4-[3-(difluoromethoxy)-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 68	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368814	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368814&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114851	402365614							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192740	O=C1CC(c2ccc(OCc3ccccc3C(F)(F)F)c(OC(F)(F)F)c2)c2c[nH]nc2N1	InChI=1S/C21H15F6N3O3/c22-20(23,24)15-4-2-1-3-12(15)10-32-16-6-5-11(7-17(16)33-21(25,26)27)13-8-18(31)29-19-14(13)9-28-30-19/h1-7,9,13H,8,10H2,(H2,28,29,30,31)	FRBANJUUHFTQTG-UHFFFAOYSA-N	368815	4-[3-(trifluoromethoxy)-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 69	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368815	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368815&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114250	402365615							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192741	O=C1CC(c2ccc(OCc3ccccc3C(F)(F)F)c(Br)c2)c2c[nH]nc2N1	InChI=1S/C20H15BrF3N3O2/c21-16-7-11(13-8-18(28)26-19-14(13)9-25-27-19)5-6-17(16)29-10-12-3-1-2-4-15(12)20(22,23)24/h1-7,9,13H,8,10H2,(H2,25,26,27,28)	AFUWOSXGAVCGMI-UHFFFAOYSA-N	368816	4-(3-bromo-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 70	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368816	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368816&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115427	402365616							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192742	CCc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccccc1C(F)(F)F	InChI=1S/C22H20F3N3O2/c1-2-13-9-14(16-10-20(29)27-21-17(16)11-26-28-21)7-8-19(13)30-12-15-5-3-4-6-18(15)22(23,24)25/h3-9,11,16H,2,10,12H2,1H3,(H2,26,27,28,29)	CEMJOHIIAFQSRN-UHFFFAOYSA-N	368817	4-(3-ethyl-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 71	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368817	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368817&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114483	402365617							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192743	O=C1CC(c2ccc(OCc3ccccc3C(F)(F)F)c(Cl)c2)c2c[nH]nc2N1	InChI=1S/C20H15ClF3N3O2/c21-16-7-11(13-8-18(28)26-19-14(13)9-25-27-19)5-6-17(16)29-10-12-3-1-2-4-15(12)20(22,23)24/h1-7,9,13H,8,10H2,(H2,25,26,27,28)	HOLQCKANGDPGNB-UHFFFAOYSA-N	368818	4-(3-chloro-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 72	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368818	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368818&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114464	402365618							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192744	Cc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccccc1C(F)(F)F	InChI=1S/C21H18F3N3O2/c1-12-8-13(15-9-19(28)26-20-16(15)10-25-27-20)6-7-18(12)29-11-14-4-2-3-5-17(14)21(22,23)24/h2-8,10,15H,9,11H2,1H3,(H2,25,26,27,28)	UHFXJMGNJMWKOM-UHFFFAOYSA-N	368819	4-(3-methyl-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 73	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368819	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368819&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115035	402365619							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192745	O=C1CC(c2ccc(OCc3ccccc3C(F)(F)F)c(F)c2)c2c[nH]nc2N1	InChI=1S/C20H15F4N3O2/c21-16-7-11(13-8-18(28)26-19-14(13)9-25-27-19)5-6-17(16)29-10-12-3-1-2-4-15(12)20(22,23)24/h1-7,9,13H,8,10H2,(H2,25,26,27,28)	XLDPJYJYZBZMMS-UHFFFAOYSA-N	368820	4-(3-fluoro-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 74	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368820	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368820&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114248	402365620							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192746	COc1cc(C2CC(=O)Nc3n[nH]cc32)c(F)cc1OCc1ccccc1C(F)(F)F	InChI=1S/C21H17F4N3O3/c1-30-17-6-13(12-7-19(29)27-20-14(12)9-26-28-20)16(22)8-18(17)31-10-11-4-2-3-5-15(11)21(23,24)25/h2-6,8-9,12H,7,10H2,1H3,(H2,26,27,28,29)	LTKSPLFLDAQEKL-UHFFFAOYSA-N	368821	4-(2-fluoro-5-methoxy-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 75	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368821	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368821&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115085	402365621							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192747	O=C1CC(c2ccc(OCc3ccccc3C(F)(F)F)c(C(F)(F)F)c2)c2c[nH]nc2N1	InChI=1S/C21H15F6N3O2/c22-20(23,24)15-4-2-1-3-12(15)10-32-17-6-5-11(7-16(17)21(25,26)27)13-8-18(31)29-19-14(13)9-28-30-19/h1-7,9,13H,8,10H2,(H2,28,29,30,31)	YMLIUXJAGIJTFX-UHFFFAOYSA-N	368822	4-[3-(trifluoromethyl)-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 76	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368822	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368822&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114867	402365622							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192748	COc1cc(C2CC(=O)Nc3n[nH]cc32)c(F)cc1OCc1cccc(F)c1C(F)(F)F	InChI=1S/C21H16F5N3O3/c1-31-16-5-12(11-6-18(30)28-20-13(11)8-27-29-20)15(23)7-17(16)32-9-10-3-2-4-14(22)19(10)21(24,25)26/h2-5,7-8,11H,6,9H2,1H3,(H2,27,28,29,30)	UVGFMVOXAUVDPP-UHFFFAOYSA-N	368823	4-(2-fluoro-4-{[3-fluoro-2-(trifluoromethyl)phenyl]methoxy}-5-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 77	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368823	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368823&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115181	402365623							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192749	COc1cc(C2CC(=O)Nc3n[nH]cc32)cc(F)c1OCc1ccccc1C(F)(F)F	InChI=1S/C21H17F4N3O3/c1-30-17-7-12(13-8-18(29)27-20-14(13)9-26-28-20)6-16(22)19(17)31-10-11-4-2-3-5-15(11)21(23,24)25/h2-7,9,13H,8,10H2,1H3,(H2,26,27,28,29)	NEUGSKDNWPMWCU-UHFFFAOYSA-N	368824	4-(3-fluoro-5-methoxy-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 78	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368824	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368824&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114287	402365624							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192750	COc1cc(C2CC(=O)Nc3ccsc32)ccc1OCc1ccccc1Cl	InChI=1S/C21H18ClNO3S/c1-25-19-10-13(15-11-20(24)23-17-8-9-27-21(15)17)6-7-18(19)26-12-14-4-2-3-5-16(14)22/h2-10,15H,11-12H2,1H3,(H,23,24)	FXIZLQUMKIUDLF-UHFFFAOYSA-N	368825	7-{4-[(2-chlorophenyl)methoxy]-3-methoxyphenyl}-4H,5H,6H,7H-thieno[3,2-b]pyridin-5-one::US12527774, Compound 79	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368825	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368825&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90001310	402365625							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192751	COc1cc(C2CC(=O)Nc3nn(C)cc32)ccc1OCc1ccccc1C(F)(F)F	InChI=1S/C22H20F3N3O3/c1-28-11-16-15(10-20(29)26-21(16)27-28)13-7-8-18(19(9-13)30-2)31-12-14-5-3-4-6-17(14)22(23,24)25/h3-9,11,15H,10,12H2,1-2H3,(H,26,27,29)	NUECYLRARMGKNA-UHFFFAOYSA-N	368826	4-(3-methoxy-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-2-methyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 80	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368826	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368826&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90137096	402365626							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192752	COc1cc(C2CC(=O)Nc3n[nH]c(C)c32)ccc1OCc1ccccc1C(F)(F)F	InChI=1S/C22H20F3N3O3/c1-12-20-15(10-19(29)26-21(20)28-27-12)13-7-8-17(18(9-13)30-2)31-11-14-5-3-4-6-16(14)22(23,24)25/h3-9,15H,10-11H2,1-2H3,(H2,26,27,28,29)	JJPNJCGNJMBNBB-UHFFFAOYSA-N	368827	4-(3-methoxy-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-3-methyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 82	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368827	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368827&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114685	402365627							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192753	COc1cc(C2CC(=O)Nc3ccsc32)ccc1OCc1ccccc1C(F)(F)F	InChI=1S/C22H18F3NO3S/c1-28-19-10-13(15-11-20(27)26-17-8-9-30-21(15)17)6-7-18(19)29-12-14-4-2-3-5-16(14)22(23,24)25/h2-10,15H,11-12H2,1H3,(H,26,27)	QEEYFYRLRINARM-UHFFFAOYSA-N	368828	7-(3-methoxy-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-4H,5H,6H,7H-thieno[3,2-b]pyridin-5-one::US12527774, Compound 85	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368828	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368828&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90137118	402365628							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192754	COc1cc(C2CC(=O)N(C)c3n[nH]cc32)ccc1OCc1ccccc1C(F)(F)F	InChI=1S/C22H20F3N3O3/c1-28-20(29)10-15(16-11-26-27-21(16)28)13-7-8-18(19(9-13)30-2)31-12-14-5-3-4-6-17(14)22(23,24)25/h3-9,11,15H,10,12H2,1-2H3,(H,26,27)	NCIGGCUUGRZBQT-UHFFFAOYSA-N	368829	4-(3-methoxy-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-7-methyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 86	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368829	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368829&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114046	402365629							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192755	COc1cc(C2CC(=O)Nc3c[nH]nc32)ccc1OCc1ccccc1C(F)(F)F	InChI=1S/C21H18F3N3O3/c1-29-18-8-12(14-9-19(28)26-16-10-25-27-20(14)16)6-7-17(18)30-11-13-4-2-3-5-15(13)21(22,23)24/h2-8,10,14H,9,11H2,1H3,(H,25,27)(H,26,28)	DKQNWOFYMVQIAM-UHFFFAOYSA-N	368830	7-(3-methoxy-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[4,3-b]pyridin-5-one::US12527774, Compound 87	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368830	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368830&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90001219	402365630							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192756	COc1cc(C2CC(=O)Nc3ncsc32)ccc1OCc1ccccc1C(F)(F)F	InChI=1S/C21H17F3N2O3S/c1-28-17-8-12(14-9-18(27)26-20-19(14)30-11-25-20)6-7-16(17)29-10-13-4-2-3-5-15(13)21(22,23)24/h2-8,11,14H,9-10H2,1H3,(H,26,27)	SIUIIPLNTYYPNY-UHFFFAOYSA-N	368831	7-(3-methoxy-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-4H,5H,6H,7H-[1,3]thiazolo[4,5-b]pyridin-5-one::US12527774, Compound 88	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368831	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368831&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115099	402365631							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192757	COc1cc(C2CC(=O)Nc3[nH]cnc32)ccc1OCc1ccccc1C(F)(F)F	InChI=1S/C21H18F3N3O3/c1-29-17-8-12(14-9-18(28)27-20-19(14)25-11-26-20)6-7-16(17)30-10-13-4-2-3-5-15(13)21(22,23)24/h2-8,11,14H,9-10H2,1H3,(H,25,26)(H,27,28)	PXNGWIMLSGBOSY-UHFFFAOYSA-N	368832	7-(3-methoxy-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-3H,4H,5H,6H,7H-imidazo[4,5-b]pyridin-5-one::US12527774, Compound 89	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368832	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368832&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90137142	402365632							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192758	COc1cc(C2CC(=O)Nc3[nH]nnc32)ccc1OCc1ccccc1C(F)(F)F	InChI=1S/C20H17F3N4O3/c1-29-16-8-11(13-9-17(28)24-19-18(13)25-27-26-19)6-7-15(16)30-10-12-4-2-3-5-14(12)20(21,22)23/h2-8,13H,9-10H2,1H3,(H2,24,25,26,27,28)	MZEAZJQJXOKAAG-UHFFFAOYSA-N	368833	7-(3-methoxy-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-3H,4H,5H,6H,7H-[1,2,3]triazolo[4,5-b]pyridin-5-one::US12527774, Compound 90	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368833	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368833&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114236	402365633							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192759	COc1ccc(COc2ccc(C3CC(=O)Nc4[nH]nnc43)cc2OC)c(C(F)(F)F)c1	InChI=1S/C21H19F3N4O4/c1-30-13-5-3-12(15(8-13)21(22,23)24)10-32-16-6-4-11(7-17(16)31-2)14-9-18(29)25-20-19(14)26-28-27-20/h3-8,14H,9-10H2,1-2H3,(H2,25,26,27,28,29)	SKBLBYIJPKZRTP-UHFFFAOYSA-N	368834	7-(3-methoxy-4-{[4-methoxy-2-(trifluoromethyl)phenyl]methoxy}phenyl)-3H,4H,5H,6H,7H-[1,2,3]triazolo[4,5-b]pyridin-5-one::US12527774, Compound 91	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368834	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368834&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114598	402365634							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192760	COc1ccc(COc2ccc(C3CC(=O)Nc4c[nH]nc43)cc2OC)c(C(F)(F)F)c1	InChI=1S/C22H20F3N3O4/c1-30-14-5-3-13(16(8-14)22(23,24)25)11-32-18-6-4-12(7-19(18)31-2)15-9-20(29)27-17-10-26-28-21(15)17/h3-8,10,15H,9,11H2,1-2H3,(H,26,28)(H,27,29)	OUAINVRKAGNCIS-UHFFFAOYSA-N	368835	7-(3-methoxy-4-{[4-methoxy-2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[4,3-b]pyridin-5-one::US12527774, Compound 92	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368835	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368835&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114933	402365635							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192761	COc1cc(C2CC(=O)Nc3n[nH]nc32)ccc1OCc1ccc(C(C)=O)cc1C(F)(F)F	InChI=1S/C22H19F3N4O4/c1-11(30)12-3-4-14(16(7-12)22(23,24)25)10-33-17-6-5-13(8-18(17)32-2)15-9-19(31)26-21-20(15)27-29-28-21/h3-8,15H,9-10H2,1-2H3,(H2,26,27,28,29,31)	MWLDUZMULUXZRA-UHFFFAOYSA-N	368836	7-(4-{[4-acetyl-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-[1,2,3]triazolo[4,5-b]pyridin-5-one::US12527774, Compound 93	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368836	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368836&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114803	402365636							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192762	COc1cc(C2CC(=O)Nc3c[nH]nc32)ccc1OCc1ccc(C(C)=O)cc1C(F)(F)F	InChI=1S/C23H20F3N3O4/c1-12(30)13-3-4-15(17(7-13)23(24,25)26)11-33-19-6-5-14(8-20(19)32-2)16-9-21(31)28-18-10-27-29-22(16)18/h3-8,10,16H,9,11H2,1-2H3,(H,27,29)(H,28,31)	UFKZTNQJFPJUFD-UHFFFAOYSA-N	368837	7-(4-{[4-acetyl-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[4,3-b]pyridin-5-one::US12527774, Compound 94	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368837	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368837&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115042	402365637							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192763	COc1cc(C2CC(=O)Nc3n[nH]c(F)c32)ccc1OCc1ccccc1C(F)(F)F	InChI=1S/C21H17F4N3O3/c1-30-16-8-11(13-9-17(29)26-20-18(13)19(22)27-28-20)6-7-15(16)31-10-12-4-2-3-5-14(12)21(23,24)25/h2-8,13H,9-10H2,1H3,(H2,26,27,28,29)	MASCOAWOKTYXKC-UHFFFAOYSA-N	368838	3-fluoro-4-(3-methoxy-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 95	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368838	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368838&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114672	402365638							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192764	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(Br)cc1C(F)(F)F	InChI=1S/C21H17BrF3N3O3/c1-30-18-6-11(14-8-19(29)27-20-15(14)9-26-28-20)3-5-17(18)31-10-12-2-4-13(22)7-16(12)21(23,24)25/h2-7,9,14H,8,10H2,1H3,(H2,26,27,28,29)	YFUWRDYQXQGUPH-UHFFFAOYSA-N	368839	4-(4-{[4-bromo-2-(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 96	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368839	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368839&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115186	402365639							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192765	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(CCO)cc1C(F)(F)F	InChI=1S/C23H22F3N3O4/c1-32-20-9-14(16-10-21(31)28-22-17(16)11-27-29-22)4-5-19(20)33-12-15-3-2-13(6-7-30)8-18(15)23(24,25)26/h2-5,8-9,11,16,30H,6-7,10,12H2,1H3,(H2,27,28,29,31)	XPBRKGFBHXVFIE-UHFFFAOYSA-N	368840	4-(4-{[4-(2-hydroxyethyl)-2-(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 97	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368840	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368840&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115461	402365640							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192766	COc1ccc(COc2ccc(C3CC(=O)Nc4n[nH]cc43)cc2OC)c(C(F)(F)F)c1	InChI=1S/C22H20F3N3O4/c1-30-14-5-3-13(17(8-14)22(23,24)25)11-32-18-6-4-12(7-19(18)31-2)15-9-20(29)27-21-16(15)10-26-28-21/h3-8,10,15H,9,11H2,1-2H3,(H2,26,27,28,29)	KHTGVXXFEDNKNO-UHFFFAOYSA-N	368841	4-(3-methoxy-4-{[4-methoxy-2-(trifluoromethyl)phenoxy]methyl}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 98	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368841	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368841&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114848	402365641							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192767	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(Cl)cc1C(F)(F)F	InChI=1S/C21H17ClF3N3O3/c1-30-18-6-11(14-8-19(29)27-20-15(14)9-26-28-20)3-5-17(18)31-10-12-2-4-13(22)7-16(12)21(23,24)25/h2-7,9,14H,8,10H2,1H3,(H2,26,27,28,29)	AOJVPOVPZVUHDF-UHFFFAOYSA-N	368842	4-(4-{[4-chloro-2-(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 99	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368842	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368842&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114084	402365642							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192768	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(C(F)(F)F)cc1C(F)(F)F	InChI=1S/C22H17F6N3O3/c1-33-18-6-11(14-8-19(32)30-20-15(14)9-29-31-20)3-5-17(18)34-10-12-2-4-13(21(23,24)25)7-16(12)22(26,27)28/h2-7,9,14H,8,10H2,1H3,(H2,29,30,31,32)	STNNMOQNYDRPAH-UHFFFAOYSA-N	368843	4-(4-{[2,4-bis(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 100	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368843	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368843&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114516	402365643							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192769	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccccc1S(F)(F)(F)(F)F	InChI=1S/C20H18F5N3O3S/c1-30-17-8-12(14-9-19(29)27-20-15(14)10-26-28-20)6-7-16(17)31-11-13-4-2-3-5-18(13)32(21,22,23,24)25/h2-8,10,14H,9,11H2,1H3,(H2,26,27,28,29)	YJDDHQLKJVCQLR-UHFFFAOYSA-N	368844	4-(3-methoxy-4-{[2-(pentafluoro-&#x3bb;<sup>6</sup>-sulfanyl)phenoxy]methyl}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 101	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368844	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368844&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115104	402365644							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192770	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccccc1C(F)(F)F	InChI=1S/C21H18F3N3O3/c1-29-18-8-12(14-9-19(28)26-20-15(14)10-25-27-20)6-7-17(18)30-11-13-4-2-3-5-16(13)21(22,23)24/h2-8,10,14H,9,11H2,1H3,(H2,25,26,27,28)	MUMZZCYJPMFJKK-UHFFFAOYSA-N	368845	4-(3-methoxy-4-{[2-(trifluoromethyl)phenoxy]methyl}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 102	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368845	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368845&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114799	402365645							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192771	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(C(C)=O)cc1C(F)(F)F	InChI=1S/C23H20F3N3O4/c1-12(30)13-3-4-15(18(7-13)23(24,25)26)11-33-19-6-5-14(8-20(19)32-2)16-9-21(31)28-22-17(16)10-27-29-22/h3-8,10,16H,9,11H2,1-2H3,(H2,27,28,29,31)	RQNAGACDVZRQDN-UHFFFAOYSA-N	368846	4-(4-{[4-acetyl-2-(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 103	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368846	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368846&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114229	402365646							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192772	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(F)cc1C(F)(F)F	InChI=1S/C21H17F4N3O3/c1-30-18-6-11(14-8-19(29)27-20-15(14)9-26-28-20)3-5-17(18)31-10-12-2-4-13(22)7-16(12)21(23,24)25/h2-7,9,14H,8,10H2,1H3,(H2,26,27,28,29)	DVXLZZCOKRXNPO-UHFFFAOYSA-N	368847	4-(4-{[4-fluoro-2-(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 104	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368847	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368847&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114481	402365647							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192773	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(C#N)cc1C(F)(F)F	InChI=1S/C22H17F3N4O3/c1-31-19-7-13(15-8-20(30)28-21-16(15)10-27-29-21)4-5-18(19)32-11-14-3-2-12(9-26)6-17(14)22(23,24)25/h2-7,10,15H,8,11H2,1H3,(H2,27,28,29,30)	AEWFFIROLRBWSL-UHFFFAOYSA-N	368848	4-[(2-methoxy-4-{6-oxo-2H,4H,55H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}phenyl)methoxy]-3-(trifluoromethyl)benzonitrile::US12527774, Compound 105	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368848	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368848&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114596	402365648							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192774	O=C1CC(c2ccc(COc3ccc(Br)cc3C(F)(F)F)c(OC(F)(F)F)c2)c2c[nH]nc2N1	InChI=1S/C21H14BrF6N3O3/c22-12-3-4-16(15(6-12)20(23,24)25)33-9-11-2-1-10(5-17(11)34-21(26,27)28)13-7-18(32)30-19-14(13)8-29-31-19/h1-6,8,13H,7,9H2,(H2,29,30,31,32)	PTDNUOSEFJKOJH-UHFFFAOYSA-N	368849	4-(4-{[4-bromo-2-(trifluoromethyl)phenoxy]methyl}-3-(trifluoromethoxy)phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 106	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368849	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368849&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114699	402365649							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192775	O=C1CC(c2ccc(COc3ccccc3S(F)(F)(F)(F)F)c(OC(F)(F)F)c2)c2c[nH]nc2N1	InChI=1S/C20H15F8N3O3S/c21-20(22,23)34-16-7-11(13-8-18(32)30-19-14(13)9-29-31-19)5-6-12(16)10-33-15-3-1-2-4-17(15)35(24,25,26,27)28/h1-7,9,13H,8,10H2,(H2,29,30,31,32)	APJONUCKDLHFHM-UHFFFAOYSA-N	368850	4-(4-{[2-(pentafluoro-&#x3bb;<sup>6</sup>-sulfanyl)phenoxy]methyl}-3-(trifluoromethoxy)phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 107	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368850	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368850&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114879	402365650							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192776	O=C1CC(c2ccc(COc3ccccc3C(F)(F)F)c(OC(F)(F)F)c2)c2c[nH]nc2N1	InChI=1S/C21H15F6N3O3/c22-20(23,24)15-3-1-2-4-16(15)32-10-12-6-5-11(7-17(12)33-21(25,26)27)13-8-18(31)29-19-14(13)9-28-30-19/h1-7,9,13H,8,10H2,(H2,28,29,30,31)	MVHHYBOMUBDTQU-UHFFFAOYSA-N	368851	4-[3-(trifluoromethoxy)-4-{[2-(trifluoromethyl)phenoxy]methyl}phenyl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 108	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368851	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368851&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114941	402365651							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192777	O=C1CC(c2ccc(COc3ccc(C(F)(F)F)cc3C(F)(F)F)c(OC(F)(F)F)c2)c2c[nH]nc2N1	InChI=1S/C22H14F9N3O3/c23-20(24,25)12-3-4-16(15(6-12)21(26,27)28)36-9-11-2-1-10(5-17(11)37-22(29,30)31)13-7-18(35)33-19-14(13)8-32-34-19/h1-6,8,13H,7,9H2,(H2,32,33,34,35)	DJHAKAOAAJMHMU-UHFFFAOYSA-N	368852	4-(4-{[2,4-bis(trifluoromethyl)phenoxy]methyl}-3-(trifluoromethoxy)phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 109	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368852	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368852&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114737	402365652							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192778	O=C1CC(c2ccc(COc3ccc(F)cc3C(F)(F)F)c(OC(F)(F)F)c2)c2c[nH]nc2N1	InChI=1S/C21H14F7N3O3/c22-12-3-4-16(15(6-12)20(23,24)25)33-9-11-2-1-10(5-17(11)34-21(26,27)28)13-7-18(32)30-19-14(13)8-29-31-19/h1-6,8,13H,7,9H2,(H2,29,30,31,32)	MBOOTTWFDOKIED-UHFFFAOYSA-N	368853	4-(4-{[4-fluoro-2-(trifluoromethyl)phenoxy]methyl}-3-(trifluoromethoxy)phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 110	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368853	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368853&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114433	402365653							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192779	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1COc1ccc(C)cc1C	InChI=1S/C22H23N3O3/c1-13-4-7-19(14(2)8-13)28-12-16-6-5-15(9-20(16)27-3)17-10-21(26)24-22-18(17)11-23-25-22/h4-9,11,17H,10,12H2,1-3H3,(H2,23,24,25,26)	KXGSQIASWGEKCI-UHFFFAOYSA-N	368854	4-{4-[(2,4-dimethylphenoxy)methyl]-3-methoxyphenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 111	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368854	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368854&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114405	402365654							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192780	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1COc1ccc(C(F)(F)F)cc1C	InChI=1S/C22H20F3N3O3/c1-12-7-15(22(23,24)25)5-6-18(12)31-11-14-4-3-13(8-19(14)30-2)16-9-20(29)27-21-17(16)10-26-28-21/h3-8,10,16H,9,11H2,1-2H3,(H2,26,27,28,29)	UUSKBVDHAVEMMX-UHFFFAOYSA-N	368855	4-(3-methoxy-4-{[2-methyl-4-(trifluoromethyl)phenoxy]methyl}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 112	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368855	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368855&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114487	402365655							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192781	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1COc1cc(C)cc(C)c1	InChI=1S/C22H23N3O3/c1-13-6-14(2)8-17(7-13)28-12-16-5-4-15(9-20(16)27-3)18-10-21(26)24-22-19(18)11-23-25-22/h4-9,11,18H,10,12H2,1-3H3,(H2,23,24,25,26)	UODMPVCPBGCVJZ-UHFFFAOYSA-N	368856	4-{4-[(3,5-dimethylphenoxy)methyl]-3-methoxyphenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 113	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368856	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368856&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114796	402365656							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192782	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1COc1cc(C)cc(C(F)(F)F)c1	InChI=1S/C22H20F3N3O3/c1-12-5-15(22(23,24)25)8-16(6-12)31-11-14-4-3-13(7-19(14)30-2)17-9-20(29)27-21-18(17)10-26-28-21/h3-8,10,17H,9,11H2,1-2H3,(H2,26,27,28,29)	HTJBNDUEZXQMQI-UHFFFAOYSA-N	368857	4-(3-methoxy-4-{[3-methyl-5-(trifluoromethyl)phenoxy]methyl}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 114	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368857	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368857&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114294	402365657							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192783	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1COc1ccc(C(F)F)cc1C(F)(F)F	InChI=1S/C22H18F5N3O3/c1-32-18-7-11(14-8-19(31)29-21-15(14)9-28-30-21)2-3-13(18)10-33-17-5-4-12(20(23)24)6-16(17)22(25,26)27/h2-7,9,14,20H,8,10H2,1H3,(H2,28,29,30,31)	RQABYVUYGPHALF-UHFFFAOYSA-N	368858	4-(4-{[4-(difluoromethyl)-2-(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 115	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368858	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368858&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114110	402365658							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192784	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1COc1ccc(C(F)F)cc1C(F)F	InChI=1S/C22H19F4N3O3/c1-31-18-7-11(14-8-19(30)28-22-16(14)9-27-29-22)2-3-13(18)10-32-17-5-4-12(20(23)24)6-15(17)21(25)26/h2-7,9,14,20-21H,8,10H2,1H3,(H2,27,28,29,30)	PARYEBOXSLXGBR-UHFFFAOYSA-N	368859	4-(4-{[2,4-bis(difluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 116	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368859	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368859&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114681	402365659							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192785	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1COc1ccc(C(F)(F)F)cc1C(F)F	InChI=1S/C22H18F5N3O3/c1-32-18-6-11(14-8-19(31)29-21-16(14)9-28-30-21)2-3-12(18)10-33-17-5-4-13(22(25,26)27)7-15(17)20(23)24/h2-7,9,14,20H,8,10H2,1H3,(H2,28,29,30,31)	VDTPXOYKXZICNI-UHFFFAOYSA-N	368860	4-(4-{[2-(difluoromethyl)-4-(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 117	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368860	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368860&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114939	402365660							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192786	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1COc1cc(C(F)F)cc(C(F)(F)F)c1	InChI=1S/C22H18F5N3O3/c1-32-18-6-11(16-8-19(31)29-21-17(16)9-28-30-21)2-3-12(18)10-33-15-5-13(20(23)24)4-14(7-15)22(25,26)27/h2-7,9,16,20H,8,10H2,1H3,(H2,28,29,30,31)	UWPYMAGAJZXUJS-UHFFFAOYSA-N	368861	4-(4-{[3-(difluoromethyl)-5-(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 118	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368861	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368861&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115366	402365661							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192787	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1COc1ccc(C#CCO)cc1C(F)(F)F	InChI=1S/C24H20F3N3O4/c1-33-21-10-15(17-11-22(32)29-23-18(17)12-28-30-23)5-6-16(21)13-34-20-7-4-14(3-2-8-31)9-19(20)24(25,26)27/h4-7,9-10,12,17,31H,8,11,13H2,1H3,(H2,28,29,30,32)	MXURCGOTUIGNFJ-UHFFFAOYSA-N	368862	4-(4-{[4-(3-hydroxyprop-1-yn-1-yl)-2-(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 119	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368862	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368862&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115420	402365662							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192788	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(C(=O)O)cc1C(F)(F)F	InChI=1S/C22H18F3N3O5/c1-32-18-7-11(14-8-19(29)27-20-15(14)9-26-28-20)4-5-17(18)33-10-13-3-2-12(21(30)31)6-16(13)22(23,24)25/h2-7,9,14H,8,10H2,1H3,(H,30,31)(H2,26,27,28,29)	DCZQWYKUUWGDMO-UHFFFAOYSA-N	368863	4-(2-methoxy-4-{6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}phenoxymethyl)-3-(trifluoromethyl)benzoic acid::US12527774, Compound 120	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368863	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368863&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115077	402365663							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192789	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(C(N)=O)cc1C(F)(F)F	InChI=1S/C22H19F3N4O4/c1-32-18-7-11(14-8-19(30)28-21-15(14)9-27-29-21)4-5-17(18)33-10-13-3-2-12(20(26)31)6-16(13)22(23,24)25/h2-7,9,14H,8,10H2,1H3,(H2,26,31)(H2,27,28,29,30)	MIZMQFCUBBSYSS-UHFFFAOYSA-N	368864	4-(2-methoxy-4-{6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}phenoxymethyl)-3-(trifluoromethyl)benzamide::US12527774, Compound 121	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368864	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368864&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115039	402365664							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192790	CCCOC(=O)c1ccccc1COc1ccc(C2CC(=O)Nc3n[nH]cc32)cc1OC	InChI=1S/C24H25N3O5/c1-3-10-31-24(29)17-7-5-4-6-16(17)14-32-20-9-8-15(11-21(20)30-2)18-12-22(28)26-23-19(18)13-25-27-23/h4-9,11,13,18H,3,10,12,14H2,1-2H3,(H2,25,26,27,28)	UXPFMXYVLVEAJV-UHFFFAOYSA-N	368865	propyl 2-(2-methoxy-4-{6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}phenoxymethyl)benzoate::US12527774, Compound 125	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368865	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368865&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114641	402365665							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192791	CCCCOC(=O)c1ccccc1COc1ccc(C2CC(=O)Nc3n[nH]cc32)cc1OC	InChI=1S/C25H27N3O5/c1-3-4-11-32-25(30)18-8-6-5-7-17(18)15-33-21-10-9-16(12-22(21)31-2)19-13-23(29)27-24-20(19)14-26-28-24/h5-10,12,14,19H,3-4,11,13,15H2,1-2H3,(H2,26,27,28,29)	ASRKUQUANBAJEV-UHFFFAOYSA-N	368866	butyl 2-(2-methoxy-4-{6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}phenoxymethyl)benzoate::US12527774, Compound 126	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368866	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368866&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114564	402365666							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192792	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccccc1C(=O)OC(C)C	InChI=1S/C24H25N3O5/c1-14(2)32-24(29)17-7-5-4-6-16(17)13-31-20-9-8-15(10-21(20)30-3)18-11-22(28)26-23-19(18)12-25-27-23/h4-10,12,14,18H,11,13H2,1-3H3,(H2,25,26,27,28)	MDUGIQQOTQCWLG-UHFFFAOYSA-N	368867	propan-2-yl 2-(2-methoxy-4-{6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}phenoxymethyl)benzoate::US12527774, Compound 127	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368867	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368867&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114840	402365667							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192793	CCOC(=O)c1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccccc1C(F)(F)F	InChI=1S/C23H20F3N3O4/c1-2-32-22(31)16-9-13(15-10-20(30)28-21-17(15)11-27-29-21)7-8-19(16)33-12-14-5-3-4-6-18(14)23(24,25)26/h3-9,11,15H,2,10,12H2,1H3,(H2,27,28,29,30)	ADFIAUJTQKCVCY-UHFFFAOYSA-N	368868	ethyl 5-{6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}-2-{[2-(trifluoromethyl)phenyl]methoxy}benzoate::US12527774, Compound 128	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368868	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368868&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115115	402365668							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192794	NC(=O)c1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccccc1C(F)(F)F	InChI=1S/C21H17F3N4O3/c22-21(23,24)16-4-2-1-3-12(16)10-31-17-6-5-11(7-14(17)19(25)30)13-8-18(29)27-20-15(13)9-26-28-20/h1-7,9,13H,8,10H2,(H2,25,30)(H2,26,27,28,29)	DPKXSYIJZOJTDW-UHFFFAOYSA-N	368869	5-{6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}-2-{[2-(trifluoromethyl)phenyl]methoxy}benzamide::US12527774, Compound 130	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368869	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368869&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114540	402365669							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192795	O=C1CC(c2ccc(OCc3ccccc3C(F)(F)F)c(C(=O)Nc3nnc[nH]3)c2)c2c[nH]nc2N1	InChI=1S/C23H18F3N7O3/c24-23(25,26)17-4-2-1-3-13(17)10-36-18-6-5-12(7-15(18)21(35)31-22-27-11-29-33-22)14-8-19(34)30-20-16(14)9-28-32-20/h1-7,9,11,14H,8,10H2,(H2,28,30,32,34)(H2,27,29,31,33,35)	BVLWLVMSKACVOJ-UHFFFAOYSA-N	368870	5-{6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}-N-(4H-1,2,4-triazol-3-yl)-2-{[2-(trifluoromethyl)phenyl]methoxy}benzamide::US12527774, Compound 131	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368870	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368870&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114846	402365670							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192796	O=C1CC(c2ccc(OCc3ccccc3C(F)(F)F)c(C(=O)OCCO)c2)c2c[nH]nc2N1	InChI=1S/C23H20F3N3O5/c24-23(25,26)18-4-2-1-3-14(18)12-34-19-6-5-13(9-16(19)22(32)33-8-7-30)15-10-20(31)28-21-17(15)11-27-29-21/h1-6,9,11,15,30H,7-8,10,12H2,(H2,27,28,29,31)	UUHDDPVZYLVZAY-UHFFFAOYSA-N	368871	2-hydroxyethyl 5-{6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}-2-{[2-(trifluoromethyl)phenyl]methoxy}benzoate::US12527774, Compound 132	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368871	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368871&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115010	402365671							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192797	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(N)cc1C(F)(F)F	InChI=1S/C21H19F3N4O3/c1-30-18-6-11(14-8-19(29)27-20-15(14)9-26-28-20)3-5-17(18)31-10-12-2-4-13(25)7-16(12)21(22,23)24/h2-7,9,14H,8,10,25H2,1H3,(H2,26,27,28,29)	WIGNHPDBLRQOKM-UHFFFAOYSA-N	368872	4-(4-{[4-amino-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 135	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368872	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368872&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114335	402365672							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192798	COc1cc(C2CC(=O)Nc3n[nH]nc32)ccc1OCc1ccc(N)cc1C(F)(F)F	InChI=1S/C20H18F3N5O3/c1-30-16-6-10(13-8-17(29)25-19-18(13)26-28-27-19)3-5-15(16)31-9-11-2-4-12(24)7-14(11)20(21,22)23/h2-7,13H,8-9,24H2,1H3,(H2,25,26,27,28,29)	CICJFXSZKQVJRM-UHFFFAOYSA-N	368873	7-(4-{[4-amino-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-[1,2,3]triazolo[4,5-b]pyridin-5-one::US12527774, Compound 136	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368873	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368873&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90001401	402365673							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192799	COc1cc(C2CC(=O)Nc3c[nH]nc32)ccc1OCc1ccc(N)cc1C(F)(F)F	InChI=1S/C21H19F3N4O3/c1-30-18-6-11(14-8-19(29)27-16-9-26-28-20(14)16)3-5-17(18)31-10-12-2-4-13(25)7-15(12)21(22,23)24/h2-7,9,14H,8,10,25H2,1H3,(H,26,28)(H,27,29)	SYVSECVDHVGBEW-UHFFFAOYSA-N	368874	7-(4-{[4-amino-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[4,3-b]pyridin-5-one::US12527774, Compound 137	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368874	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368874&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114902	402365674							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192800	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(N(C)C)cc1C(F)(F)F	InChI=1S/C23H23F3N4O3/c1-30(2)15-6-4-14(18(9-15)23(24,25)26)12-33-19-7-5-13(8-20(19)32-3)16-10-21(31)28-22-17(16)11-27-29-22/h4-9,11,16H,10,12H2,1-3H3,(H2,27,28,29,31)	FOEUQPUCDDKZIN-UHFFFAOYSA-N	368875	4-(4-{[4-(dimethylamino)-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 138	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368875	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368875&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114752	402365675							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192801	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(NC(C)=O)cc1C(F)(F)F	InChI=1S/C23H21F3N4O4/c1-12(31)28-15-5-3-14(18(8-15)23(24,25)26)11-34-19-6-4-13(7-20(19)33-2)16-9-21(32)29-22-17(16)10-27-30-22/h3-8,10,16H,9,11H2,1-2H3,(H,28,31)(H2,27,29,30,32)	MJLLELLNVRMZMI-UHFFFAOYSA-N	368876	N-{4-[(2-methoxy-4-{6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}phenoxy)methyl]-3-(trifluoromethyl)phenyl}acetamide::US12527774, Compound 139	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368876	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368876&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115508	402365676							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192802	CCC(=O)Nc1ccc(COc2ccc(C3CC(=O)Nc4n[nH]cc43)cc2OC)c(C(F)(F)F)c1	InChI=1S/C24H23F3N4O4/c1-3-21(32)29-15-6-4-14(18(9-15)24(25,26)27)12-35-19-7-5-13(8-20(19)34-2)16-10-22(33)30-23-17(16)11-28-31-23/h4-9,11,16H,3,10,12H2,1-2H3,(H,29,32)(H2,28,30,31,33)	HZLQZMODTDUPOL-UHFFFAOYSA-N	368877	2-amino-N-{4-[(2-methoxy-4-{6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}phenoxy)methyl]-3-(trifluoromethyl)phenyl}acetamide::US12527774, Compound 140	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368877	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368877&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114687	402365677							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192803	CNc1ccc(COc2ccc(C3CC(=O)Nc4n[nH]cc43)cc2OC)c(C(F)(F)F)c1	InChI=1S/C22H21F3N4O3/c1-26-14-5-3-13(17(8-14)22(23,24)25)11-32-18-6-4-12(7-19(18)31-2)15-9-20(30)28-21-16(15)10-27-29-21/h3-8,10,15,26H,9,11H2,1-2H3,(H2,27,28,29,30)	VMKFGSGVOKMYKW-UHFFFAOYSA-N	368878	4-(3-methoxy-4-{[4-(methylamino)-2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 141	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368878	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368878&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115043	402365678							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192804	C=CCc1ccc(COc2ccc(C3CC(=O)Nc4n[nH]cc43)cc2OC)c(C(F)(F)F)c1	InChI=1S/C24H22F3N3O3/c1-3-4-14-5-6-16(19(9-14)24(25,26)27)13-33-20-8-7-15(10-21(20)32-2)17-11-22(31)29-23-18(17)12-28-30-23/h3,5-10,12,17H,1,4,11,13H2,2H3,(H2,28,29,30,31)	DDXIZVCVZDMWOZ-UHFFFAOYSA-N	368879	4-(3-methoxy-4-{[4-(prop-2-en-1-yl)-2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 142	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368879	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368879&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114824	402365679							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192805	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(CC(O)CO)cc1C(F)(F)F	InChI=1S/C24H24F3N3O5/c1-34-21-8-14(17-9-22(33)29-23-18(17)10-28-30-23)4-5-20(21)35-12-15-3-2-13(6-16(32)11-31)7-19(15)24(25,26)27/h2-5,7-8,10,16-17,31-32H,6,9,11-12H2,1H3,(H2,28,29,30,33)	KIKICEUTXVSKJA-UHFFFAOYSA-N	368880	4-(4-{[4-(2,3-dihydroxypropyl)-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 143	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368880	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368880&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115174	402365680							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192806	CCc1ccc(COc2ccc(C3CC(=O)Nc4n[nH]cc43)cc2OC)c(C(F)(F)F)c1	InChI=1S/C23H22F3N3O3/c1-3-13-4-5-15(18(8-13)23(24,25)26)12-32-19-7-6-14(9-20(19)31-2)16-10-21(30)28-22-17(16)11-27-29-22/h4-9,11,16H,3,10,12H2,1-2H3,(H2,27,28,29,30)	RONFEIXXSAWJBE-UHFFFAOYSA-N	368881	4-(4-{[4-ethyl-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 144	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368881	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368881&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114308	402365681							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192807	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(C2CC2)cc1C(F)(F)F	InChI=1S/C24H22F3N3O3/c1-32-21-9-15(17-10-22(31)29-23-18(17)11-28-30-23)6-7-20(21)33-12-16-5-4-14(13-2-3-13)8-19(16)24(25,26)27/h4-9,11,13,17H,2-3,10,12H2,1H3,(H2,28,29,30,31)	VYYAGJHTERXCLF-UHFFFAOYSA-N	368882	4-(4-{[4-cyclopropyl-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 145	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368882	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368882&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115029	402365682							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192808	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(C#CCO)cc1C(F)(F)F	InChI=1S/C24H20F3N3O4/c1-33-21-10-15(17-11-22(32)29-23-18(17)12-28-30-23)6-7-20(21)34-13-16-5-4-14(3-2-8-31)9-19(16)24(25,26)27/h4-7,9-10,12,17,31H,8,11,13H2,1H3,(H2,28,29,30,32)	WWEBRKPFDCFPPC-UHFFFAOYSA-N	368883	4-(4-{[4-(3-hydroxyprop-1-yn-1-yl)-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 146	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368883	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368883&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114915	402365683							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192809	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(CC#N)cc1C(F)(F)F	InChI=1S/C23H19F3N4O3/c1-32-20-9-14(16-10-21(31)29-22-17(16)11-28-30-22)4-5-19(20)33-12-15-3-2-13(6-7-27)8-18(15)23(24,25)26/h2-5,8-9,11,16H,6,10,12H2,1H3,(H2,28,29,30,31)	UELPTGHWGGVHKI-UHFFFAOYSA-N	368884	2-[4-(2-methoxy-4-{6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}phenoxymethyl)-3-(trifluoromethyl)phenyl]acetonitrile::US12527774, Compound 147	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368884	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368884&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114864	402365684							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192810	COC(=O)Cc1ccc(COc2ccc(C3CC(=O)Nc4n[nH]cc43)cc2OC)c(C(F)(F)F)c1	InChI=1S/C24H22F3N3O5/c1-33-20-9-14(16-10-21(31)29-23-17(16)11-28-30-23)5-6-19(20)35-12-15-4-3-13(8-22(32)34-2)7-18(15)24(25,26)27/h3-7,9,11,16H,8,10,12H2,1-2H3,(H2,28,29,30,31)	QSYOSZHELRPOSG-UHFFFAOYSA-N	368885	methyl 2-[4-(2-methoxy-4-{6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}phenoxymethyl)-3-(trifluoromethyl)phenyl]acetate::US12527774, Compound 148	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368885	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368885&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114432	402365685							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192811	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(CCCO)cc1C(F)(F)F	InChI=1S/C24H24F3N3O4/c1-33-21-10-15(17-11-22(32)29-23-18(17)12-28-30-23)6-7-20(21)34-13-16-5-4-14(3-2-8-31)9-19(16)24(25,26)27/h4-7,9-10,12,17,31H,2-3,8,11,13H2,1H3,(H2,28,29,30,32)	KWCOFNAOHPZSNF-UHFFFAOYSA-N	368886	4-(4-{[4-(3-hydroxypropyl)-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 149	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368886	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368886&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114444	402365686							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192812	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(CCN)cc1C(F)(F)F	InChI=1S/C23H23F3N4O3/c1-32-20-9-14(16-10-21(31)29-22-17(16)11-28-30-22)4-5-19(20)33-12-15-3-2-13(6-7-27)8-18(15)23(24,25)26/h2-5,8-9,11,16H,6-7,10,12,27H2,1H3,(H2,28,29,30,31)	QWPAGTOUSFCFSO-UHFFFAOYSA-N	368887	4-(4-{[4-(2-aminoethyl)-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 150	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368887	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368887&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114581	402365687							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192813	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(CC(=O)O)cc1C(F)(F)F	InChI=1S/C23H20F3N3O5/c1-33-19-8-13(15-9-20(30)28-22-16(15)10-27-29-22)4-5-18(19)34-11-14-3-2-12(7-21(31)32)6-17(14)23(24,25)26/h2-6,8,10,15H,7,9,11H2,1H3,(H,31,32)(H2,27,28,29,30)	DWMWXIFONZLSTF-UHFFFAOYSA-N	368888	2-{4-[(2-methoxy-4-{6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}phenoxy)methyl]-3-(trifluoromethyl)phenyl}acetic acid::US12527774, Compound 151	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368888	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368888&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114764	402365688							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192814	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(C(C)(C)CO)cc1C(F)(F)F	InChI=1S/C25H26F3N3O4/c1-24(2,13-32)16-6-4-15(19(9-16)25(26,27)28)12-35-20-7-5-14(8-21(20)34-3)17-10-22(33)30-23-18(17)11-29-31-23/h4-9,11,17,32H,10,12-13H2,1-3H3,(H2,29,30,31,33)	YYJHVJIBYSPIGD-UHFFFAOYSA-N	368889	4-(4-{[4-(1-hydroxy-2-methylpropan-2-yl)-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 152	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368889	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368889&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114706	402365689							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192815	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(CC(C)(C)O)cc1C(F)(F)F	InChI=1S/C25H26F3N3O4/c1-24(2,33)11-14-4-5-16(19(8-14)25(26,27)28)13-35-20-7-6-15(9-21(20)34-3)17-10-22(32)30-23-18(17)12-29-31-23/h4-9,12,17,33H,10-11,13H2,1-3H3,(H2,29,30,31,32)	WCHNAEDDSAXBPG-UHFFFAOYSA-N	368890	4-(4-{[4-(2-hydroxy-2-methylpropyl)-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 153	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368890	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368890&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114841	402365690							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192816	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(O)cc1C(F)(F)F	InChI=1S/C21H18F3N3O4/c1-30-18-6-11(14-8-19(29)26-20-15(14)9-25-27-20)3-5-17(18)31-10-12-2-4-13(28)7-16(12)21(22,23)24/h2-7,9,14,28H,8,10H2,1H3,(H2,25,26,27,29)	SJMTUKSJDISFGT-UHFFFAOYSA-N	368891	4-(4-{[4-hydroxy-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 154	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368891	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368891&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114834	402365691							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192817	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(CCO)cc1C(F)(F)F	InChI=1S/C23H22F3N3O4/c1-32-20-9-14(16-10-21(31)28-22-17(16)11-27-29-22)4-5-19(20)33-12-15-3-2-13(6-7-30)8-18(15)23(24,25)26/h2-5,8-9,11,16,30H,6-7,10,12H2,1H3,(H2,27,28,29,31)	XPBRKGFBHXVFIE-UHFFFAOYSA-N	368893	4-(4-{[4-(2-hydroxyethyl)-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 155	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368893	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368893&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90134757	402365692							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192818	COc1cc(C2CC(=O)Nc3c[nH]nc32)ccc1OCc1ccc(CCO)cc1C(F)(F)F	InChI=1S/C23H22F3N3O4/c1-32-20-9-14(16-10-21(31)28-18-11-27-29-22(16)18)4-5-19(20)33-12-15-3-2-13(6-7-30)8-17(15)23(24,25)26/h2-5,8-9,11,16,30H,6-7,10,12H2,1H3,(H,27,29)(H,28,31)	ZOHMVHXWCKYAHL-UHFFFAOYSA-N	368894	7-(4-{[4-(2-hydroxyethyl)-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[4,3-b]pyridin-5-one::US12527774, Compound 156	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368894	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368894&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115003	402365693							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192819	COc1cc(C2CC(=O)Nc3n[nH]nc32)ccc1OCc1ccc(CCO)cc1C(F)(F)F	InChI=1S/C22H21F3N4O4/c1-32-18-9-13(15-10-19(31)26-21-20(15)27-29-28-21)4-5-17(18)33-11-14-3-2-12(6-7-30)8-16(14)22(23,24)25/h2-5,8-9,15,30H,6-7,10-11H2,1H3,(H2,26,27,28,29,31)	NFYCKXAHPFHZSE-UHFFFAOYSA-N	368895	7-(4-{[4-(2-hydroxyethyl)-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-[1,2,3]triazolo[4,5-b]pyridin-5-one::US12527774, Compound 157	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368895	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368895&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90137117	402365694							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192820	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(C=O)cc1C(F)(F)F	InChI=1S/C22H18F3N3O4/c1-31-19-7-13(15-8-20(30)27-21-16(15)9-26-28-21)4-5-18(19)32-11-14-3-2-12(10-29)6-17(14)22(23,24)25/h2-7,9-10,15H,8,11H2,1H3,(H2,26,27,28,30)	PGXHWCIFYFOKNS-UHFFFAOYSA-N	368896	4-[(2-methoxy-4-{6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}phenoxy)methyl]-3-(trifluoromethyl)benzaldehyde::US12527774, Compound 159	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368896	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368896&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114557	402365695							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192821	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1cccc(OCCO)c1C(F)(F)F	InChI=1S/C23H22F3N3O5/c1-32-19-9-13(15-10-20(31)28-22-16(15)11-27-29-22)5-6-17(19)34-12-14-3-2-4-18(33-8-7-30)21(14)23(24,25)26/h2-6,9,11,15,30H,7-8,10,12H2,1H3,(H2,27,28,29,31)	OHPLOERGUJBWKB-UHFFFAOYSA-N	368897	4-(4-{[3-(2-hydroxyethoxy)-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 160	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368897	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368897&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90137122	402365696							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192822	Nc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccccc1C(F)(F)F	InChI=1S/C20H17F3N4O2/c21-20(22,23)15-4-2-1-3-12(15)10-29-17-6-5-11(7-16(17)24)13-8-18(28)26-19-14(13)9-25-27-19/h1-7,9,13H,8,10,24H2,(H2,25,26,27,28)	BNZWZJHGUFTKNT-UHFFFAOYSA-N	368898	4-(3-amino-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 161	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368898	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368898&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114705	402365697							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192823	CN(C)c1cc(OCc2ccccc2C(F)(F)F)ccc1C1CC(=O)Nc2n[nH]cc21	InChI=1S/C22H21F3N4O2/c1-29(2)19-9-14(31-12-13-5-3-4-6-18(13)22(23,24)25)7-8-15(19)16-10-20(30)27-21-17(16)11-26-28-21/h3-9,11,16H,10,12H2,1-2H3,(H2,26,27,28,30)	KRPFEDCBQDGQMV-UHFFFAOYSA-N	368899	4-[2-(dimethylamino)-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 162	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368899	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368899&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114793	402365698							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192824	COCCCOc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccccc1C(F)(F)F	InChI=1S/C24H24F3N3O4/c1-32-9-4-10-33-21-11-15(17-12-22(31)29-23-18(17)13-28-30-23)7-8-20(21)34-14-16-5-2-3-6-19(16)24(25,26)27/h2-3,5-8,11,13,17H,4,9-10,12,14H2,1H3,(H2,28,29,30,31)	KLVMZGSTHRMFNO-UHFFFAOYSA-N	368900	4-[3-(3-methoxypropoxy)-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 163	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368900	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368900&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114307	402365699							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192825	COCCOc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccccc1C(F)(F)F	InChI=1S/C23H22F3N3O4/c1-31-8-9-32-20-10-14(16-11-21(30)28-22-17(16)12-27-29-22)6-7-19(20)33-13-15-4-2-3-5-18(15)23(24,25)26/h2-7,10,12,16H,8-9,11,13H2,1H3,(H2,27,28,29,30)	JXCFBXJBOHJVAQ-UHFFFAOYSA-N	368901	4-[3-(2-methoxyethoxy)-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 164	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368901	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368901&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114935	402365700							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192826	O=C1CC(c2cnc(OCc3ccccc3C(F)(F)F)nc2)c2c[nH]nc2N1	InChI=1S/C18H14F3N5O2/c19-18(20,21)14-4-2-1-3-10(14)9-28-17-22-6-11(7-23-17)12-5-15(27)25-16-13(12)8-24-26-16/h1-4,6-8,12H,5,9H2,(H2,24,25,26,27)	NPTUEUQNLQMIQC-UHFFFAOYSA-N	368902	4-(2-{[2-(trifluoromethyl)phenyl]methoxy}pyrimidin-5-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 165	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368902	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368902&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114862	402365701							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192827	COc1cc(C2CC(=S)Nc3n[nH]cc32)ccc1OCc1ccccc1C(F)(F)F	InChI=1S/C21H18F3N3O2S/c1-28-18-8-12(14-9-19(30)26-20-15(14)10-25-27-20)6-7-17(18)29-11-13-4-2-3-5-16(13)21(22,23)24/h2-8,10,14H,9,11H2,1H3,(H2,25,26,27,30)	WPTSNEFFNSFXGU-UHFFFAOYSA-N	368903	4-(3-methoxy-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-6-thione::US12527774, Compound 166	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368903	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368903&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114835	402365702							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192828	COc1cc(C2CC(=N)Nc3n[nH]cc32)ccc1OCc1ccccc1C(F)(F)F	InChI=1S/C21H19F3N4O2/c1-29-18-8-12(14-9-19(25)27-20-15(14)10-26-28-20)6-7-17(18)30-11-13-4-2-3-5-16(13)21(22,23)24/h2-8,10,14H,9,11H2,1H3,(H3,25,26,27,28)	SUYMWAAZOFZTGS-UHFFFAOYSA-N	368904	4-(3-methoxy-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-imine::US12527774, Compound 167	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368904	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368904&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114215	402365703							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192829	COc1cc(-c2cc(=O)[nH]c3[nH]ccc23)ccc1OCc1ccccc1C(F)(F)F	InChI=1S/C22H17F3N2O3/c1-29-19-10-13(16-11-20(28)27-21-15(16)8-9-26-21)6-7-18(19)30-12-14-4-2-3-5-17(14)22(23,24)25/h2-11H,12H2,1H3,(H2,26,27,28)	OQIFDOAYUWKEFP-UHFFFAOYSA-N	368905	4-(3-methoxy-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-1H,6H,7H-pyrrolo[2,3-b]pyridin-6-one::US12527774, Compound 168	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368905	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368905&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114521	402365704							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192830	COc1cc(-c2cc(=O)[nH]c3n[nH]cc23)ccc1OCc1ccccc1C(F)(F)F	InChI=1S/C21H16F3N3O3/c1-29-18-8-12(14-9-19(28)26-20-15(14)10-25-27-20)6-7-17(18)30-11-13-4-2-3-5-16(13)21(22,23)24/h2-10H,11H2,1H3,(H2,25,26,27,28)	HOCLGQXOQQVOGI-UHFFFAOYSA-N	368906	4-(3-methoxy-4-{[2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 169	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368906	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368906&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115084	402365705							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192831	COc1ccc(COc2ccc(-c3cc(=O)[nH]c4n[nH]cc34)cc2OC)c(C(F)(F)F)c1	InChI=1S/C22H18F3N3O4/c1-30-14-5-3-13(17(8-14)22(23,24)25)11-32-18-6-4-12(7-19(18)31-2)15-9-20(29)27-21-16(15)10-26-28-21/h3-10H,11H2,1-2H3,(H2,26,27,28,29)	WZHLSZAYAOLYJL-UHFFFAOYSA-N	368907	4-(3-methoxy-4-{[4-methoxy-2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 170	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368907	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368907&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114725	402365706							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192832	COc1ccccc1COc1ccc(-c2cc(=O)[nH]c3n[nH]cc23)cc1OC	InChI=1S/C21H19N3O4/c1-26-17-6-4-3-5-14(17)12-28-18-8-7-13(9-19(18)27-2)15-10-20(25)23-21-16(15)11-22-24-21/h3-11H,12H2,1-2H3,(H2,22,23,24,25)	FBVXFBWVHSNNSW-UHFFFAOYSA-N	368908	4-{3-methoxy-4-[(2-methoxyphenyl)methoxy]phenyl}-2H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 171	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368908	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368908&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115464	402365707							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192833	COc1cc(-c2cc(=O)[nH]c3n[nH]cc23)ccc1OCc1ccncc1C(F)(F)F	InChI=1S/C20H15F3N4O3/c1-29-17-6-11(13-7-18(28)26-19-14(13)8-25-27-19)2-3-16(17)30-10-12-4-5-24-9-15(12)20(21,22)23/h2-9H,10H2,1H3,(H2,25,26,27,28)	ZJQUHGLRYQLKBQ-UHFFFAOYSA-N	368909	4-(3-methoxy-4-{[3-(trifluoromethyl)pyridin-4-yl]methoxy}phenyl)-2H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 172	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368909	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368909&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114693	402365708							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192834	COc1cc(-c2cc(=O)[nH]c3n[nH]cc23)ccc1OCc1ccc(N)cc1C(F)(F)F	InChI=1S/C21H17F3N4O3/c1-30-18-6-11(14-8-19(29)27-20-15(14)9-26-28-20)3-5-17(18)31-10-12-2-4-13(25)7-16(12)21(22,23)24/h2-9H,10,25H2,1H3,(H2,26,27,28,29)	RQXRDWDTRLYIOL-UHFFFAOYSA-N	368910	4-(4-{[4-amino-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 173	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368910	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368910&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114302	402365709							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192835	COc1cc(-c2cc(=O)[nH]c3n[nH]cc23)ccc1OCc1ccc(C(C)=O)cc1C(F)(F)F	InChI=1S/C23H18F3N3O4/c1-12(30)13-3-4-15(18(7-13)23(24,25)26)11-33-19-6-5-14(8-20(19)32-2)16-9-21(31)28-22-17(16)10-27-29-22/h3-10H,11H2,1-2H3,(H2,27,28,29,31)	ZUZBOIYEHUOBLT-UHFFFAOYSA-N	368911	4-(4-{[4-acetyl-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 174	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368911	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368911&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115238	402365710							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192836	CCc1ccc(COc2ccc(-c3cc(=O)[nH]c4n[nH]cc34)cc2OC)c(C(F)(F)F)c1	InChI=1S/C23H20F3N3O3/c1-3-13-4-5-15(18(8-13)23(24,25)26)12-32-19-7-6-14(9-20(19)31-2)16-10-21(30)28-22-17(16)11-27-29-22/h4-11H,3,12H2,1-2H3,(H2,27,28,29,30)	DYUWXUMHYKIDQN-UHFFFAOYSA-N	368912	4-(4-{[4-ethyl-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 175	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368912	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368912&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114884	402365711							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192837	COc1cc(-c2cc(=O)[nH]c3n[nH]cc23)ccc1OCc1ccc(CCO)cc1C(F)(F)F	InChI=1S/C23H20F3N3O4/c1-32-20-9-14(16-10-21(31)28-22-17(16)11-27-29-22)4-5-19(20)33-12-15-3-2-13(6-7-30)8-18(15)23(24,25)26/h2-5,8-11,30H,6-7,12H2,1H3,(H2,27,28,29,31)	DHDSGRKNJXPMJP-UHFFFAOYSA-N	368913	4-(4-{[4-(2-hydroxyethyl)-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 176	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368913	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368913&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90003402	402365712							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192838	COc1cc(-c2cc(=O)[nH]c3n[nH]cc23)ccc1OCc1cccc(OC)c1C(F)(F)F	InChI=1S/C22H18F3N3O4/c1-30-17-5-3-4-13(20(17)22(23,24)25)11-32-16-7-6-12(8-18(16)31-2)14-9-19(29)27-21-15(14)10-26-28-21/h3-10H,11H2,1-2H3,(H2,26,27,28,29)	ZLGCTRMHGNXWNN-UHFFFAOYSA-N	368914	4-(3-methoxy-4-{[3-methoxy-2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 177	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368914	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368914&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90004125	402365713							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192839	COc1ccc(C(F)(F)F)c(COc2ccc(-c3cc(=O)[nH]c4n[nH]cc34)cc2OC)c1	InChI=1S/C22H18F3N3O4/c1-30-14-4-5-17(22(23,24)25)13(7-14)11-32-18-6-3-12(8-19(18)31-2)15-9-20(29)27-21-16(15)10-26-28-21/h3-10H,11H2,1-2H3,(H2,26,27,28,29)	WOMIDBZVHGFFEJ-UHFFFAOYSA-N	368915	4-(3-methoxy-4-{[5-methoxy-2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 178	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368915	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368915&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90001821	402365714							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192840	COc1cc(-c2cc(=O)[nH]c3n[nH]cc23)ccc1OCc1ccc(F)cc1C(F)(F)F	InChI=1S/C21H15F4N3O3/c1-30-18-6-11(14-8-19(29)27-20-15(14)9-26-28-20)3-5-17(18)31-10-12-2-4-13(22)7-16(12)21(23,24)25/h2-9H,10H2,1H3,(H2,26,27,28,29)	SIENXVGMZFJJRI-UHFFFAOYSA-N	368916	4-(4-{[4-fluoro-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 179	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368916	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368916&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114195	402365715							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192841	COc1cc(-c2cc(=O)[nH]c3n[nH]cc23)ccc1OCc1ccccc1OC(F)F	InChI=1S/C21H17F2N3O4/c1-28-18-8-12(14-9-19(27)25-20-15(14)10-24-26-20)6-7-17(18)29-11-13-4-2-3-5-16(13)30-21(22)23/h2-10,21H,11H2,1H3,(H2,24,25,26,27)	AAAHZJAFKCBHEI-UHFFFAOYSA-N	368917	4-(4-{[2-(difluoromethoxy)phenyl]methoxy}-3-methoxyphenyl)-2H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 180	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368917	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368917&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90001125	402365716							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192842	COc1cc(-c2cc(=O)[nH]c3n[nH]cc23)ccc1OCc1ccc(C#N)cc1C(F)(F)F	InChI=1S/C22H15F3N4O3/c1-31-19-7-13(15-8-20(30)28-21-16(15)10-27-29-21)4-5-18(19)32-11-14-3-2-12(9-26)6-17(14)22(23,24)25/h2-8,10H,11H2,1H3,(H2,27,28,29,30)	LLFVWKWFVVLTOT-UHFFFAOYSA-N	368918	4-[(2-methoxy-4-{6-oxo-2H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}phenoxy)methyl]-3-(trifluoromethyl)benzonitrile::US12527774, Compound 181	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368918	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368918&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90001362	402365717							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192843	COc1ccc([N+](=O)[O-])cc1COc1ccc(-c2cc(=O)[nH]c3n[nH]cc23)cc1OC	InChI=1S/C21H18N4O6/c1-29-17-6-4-14(25(27)28)7-13(17)11-31-18-5-3-12(8-19(18)30-2)15-9-20(26)23-21-16(15)10-22-24-21/h3-10H,11H2,1-2H3,(H2,22,23,24,26)	CWALSPKZCVXDBZ-UHFFFAOYSA-N	368919	4-{3-methoxy-4-[(2-methoxy-5-nitrophenyl)methoxy]phenyl}-2H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 182	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368919	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368919&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114660	402365718							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192844	COc1cc(-c2cc(=O)[nH]c3n[nH]cc23)ccc1OCc1ccccc1	InChI=1S/C20H17N3O3/c1-25-18-9-14(15-10-19(24)22-20-16(15)11-21-23-20)7-8-17(18)26-12-13-5-3-2-4-6-13/h2-11H,12H2,1H3,(H2,21,22,23,24)	CERSJRSXEJRLSF-UHFFFAOYSA-N	368920	4-[4-(benzyloxy)-3-methoxyphenyl]-2H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 183	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368920	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368920&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114944	402365719							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192845	COc1cc(Br)c(COc2ccc(-c3cc(=O)[nH]c4n[nH]cc34)cc2OC)cc1OC	InChI=1S/C22H20BrN3O5/c1-28-18-6-12(14-8-21(27)25-22-15(14)10-24-26-22)4-5-17(18)31-11-13-7-19(29-2)20(30-3)9-16(13)23/h4-10H,11H2,1-3H3,(H2,24,25,26,27)	KEKKEPDILSDWFJ-UHFFFAOYSA-N	368921	4-{4-[(2-bromo-4,5-dimethoxyphenyl)methoxy]-3-methoxyphenyl}-2H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 184	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368921	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368921&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114850	402365720							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192846	COc1cc(-c2cc(=O)[nH]c3n[nH]cc23)ccc1OCc1ccc(C(F)(F)F)cc1C(F)(F)F	InChI=1S/C22H15F6N3O3/c1-33-18-6-11(14-8-19(32)30-20-15(14)9-29-31-20)3-5-17(18)34-10-12-2-4-13(21(23,24)25)7-16(12)22(26,27)28/h2-9H,10H2,1H3,(H2,29,30,31,32)	XXVKCVQXNLETAF-UHFFFAOYSA-N	368922	4-(4-{[2,4-bis(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 186	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368922	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368922&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114505	402365721							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192847	COC(=O)C1C(=O)Nc2n[nH]cc2C1c1ccc(COc2ccc(C(F)(F)F)cc2C(F)(F)F)c(OC)c1	InChI=1S/C24H19F6N3O5/c1-36-17-7-11(18-14-9-31-33-20(14)32-21(34)19(18)22(35)37-2)3-4-12(17)10-38-16-6-5-13(23(25,26)27)8-15(16)24(28,29)30/h3-9,18-19H,10H2,1-2H3,(H2,31,32,33,34)	NRPNEGNGSJTKTF-UHFFFAOYSA-N	368923	methyl 4-(4-{[2,4-bis(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-5-carboxylate::US12527774, Compound 187	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368923	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368923&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			73389456	402365722							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192848	COc1cc(C2c3c[nH]nc3NC(=O)C2C(=O)N(C)C)ccc1OCc1ccc(C(F)(F)F)cc1C(F)(F)F	InChI=1S/C25H22F6N4O4/c1-35(2)23(37)20-19(15-10-32-34-21(15)33-22(20)36)12-5-7-17(18(8-12)38-3)39-11-13-4-6-14(24(26,27)28)9-16(13)25(29,30)31/h4-10,19-20H,11H2,1-3H3,(H2,32,33,34,36)	DPXNTCCYRIPMAW-UHFFFAOYSA-N	368924	4-(4-{[2,4-bis(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-N,N-dimethyl-6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-5-carboxamide::US12527774, Compound 188	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368924	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368924&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114860	402365723							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192849	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(C)cc1C(F)(F)F	InChI=1S/C22H20F3N3O3/c1-12-3-4-14(17(7-12)22(23,24)25)11-31-18-6-5-13(8-19(18)30-2)15-9-20(29)27-21-16(15)10-26-28-21/h3-8,10,15H,9,11H2,1-2H3,(H2,26,27,28,29)	AABUOCUSIGKCCP-UHFFFAOYSA-N	368925	4-(3-methoxy-4-{[4-methyl-2-(trifluoromethyl)phenoxy]methyl}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 189	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368925	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368925&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114871	402365724							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192850	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(C(F)(F)F)cc1C(F)(F)F	InChI=1S/C22H17F6N3O3/c1-33-18-6-11(14-8-19(32)30-20-15(14)9-29-31-20)3-5-17(18)34-10-12-2-4-13(21(23,24)25)7-16(12)22(26,27)28/h2-7,9,14H,8,10H2,1H3,(H2,29,30,31,32)	STNNMOQNYDRPAH-UHFFFAOYSA-N	368926	4-(4-{[2,4-bis(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-1H,2H,3H,4H,6H-pyrrolo[3,4-b]pyridin-2-one::US12527774, Compound 190	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368926	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368926&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115023	402365725							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192851	COc1cc([C@@H]2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(C(F)(F)F)cc1C(F)(F)F	InChI=1S/C22H17F6N3O3/c1-33-18-6-11(14-8-19(32)30-20-15(14)9-29-31-20)3-5-17(18)34-10-12-2-4-13(21(23,24)25)7-16(12)22(26,27)28/h2-7,9,14H,8,10H2,1H3,(H2,29,30,31,32)	STNNMOQNYDRPAH-UHFFFAOYSA-N	368927	(4R)-4-(4-{[2,4-bis(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one [(+)-4-(4-{[2,4-bis(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one]::US12527774, Compound 191	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368927	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368927&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114401	402365726							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192852	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(C(F)(F)F)cc1C(F)(F)F	InChI=1S/C22H17F6N3O3/c1-33-18-6-11(14-8-19(32)30-20-15(14)9-29-31-20)3-5-17(18)34-10-12-2-4-13(21(23,24)25)7-16(12)22(26,27)28/h2-7,9,14H,8,10H2,1H3,(H2,29,30,31,32)	STNNMOQNYDRPAH-UHFFFAOYSA-N	368928	(4S)-4-(4-{[2,4-bis(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one [(-)4-(4-{[2,4-bis(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one]::US12527774, Compound 192	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368928	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368928&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114524	402365727							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192853	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1COc1ccc(Cl)cc1C(F)(F)F	InChI=1S/C21H17ClF3N3O3/c1-30-18-6-11(14-8-19(29)27-20-15(14)9-26-28-20)2-3-12(18)10-31-17-5-4-13(22)7-16(17)21(23,24)25/h2-7,9,14H,8,10H2,1H3,(H2,26,27,28,29)	XYFBPARNBAOCKV-UHFFFAOYSA-N	368929	(+)-4-(4-{[4-chloro-2-(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 193	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368929	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368929&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114779	402365728							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192854	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1COc1ccc(Cl)cc1C(F)(F)F	InChI=1S/C21H17ClF3N3O3/c1-30-18-6-11(14-8-19(29)27-20-15(14)9-26-28-20)2-3-12(18)10-31-17-5-4-13(22)7-16(17)21(23,24)25/h2-7,9,14H,8,10H2,1H3,(H2,26,27,28,29)	XYFBPARNBAOCKV-UHFFFAOYSA-N	368930	(−)-4-(4-{[4-chloro-2-(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::(−)-4-(4-{[4-chloro-2-(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 194	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368930	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368930&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114349	402365729							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192855	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1COc1ccc(C(F)F)cc1C(F)(F)F	InChI=1S/C22H18F5N3O3/c1-32-18-7-11(14-8-19(31)29-21-15(14)9-28-30-21)2-3-13(18)10-33-17-5-4-12(20(23)24)6-16(17)22(25,26)27/h2-7,9,14,20H,8,10H2,1H3,(H2,28,29,30,31)	RQABYVUYGPHALF-UHFFFAOYSA-N	368931	(+)-4-(4-{[4-(difluoromethyl)-2-(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 195	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368931	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368931&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114551	402365730							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192856	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1COc1ccc(C(F)F)cc1C(F)(F)F	InChI=1S/C22H18F5N3O3/c1-32-18-7-11(14-8-19(31)29-21-15(14)9-28-30-21)2-3-13(18)10-33-17-5-4-12(20(23)24)6-16(17)22(25,26)27/h2-7,9,14,20H,8,10H2,1H3,(H2,28,29,30,31)	RQABYVUYGPHALF-UHFFFAOYSA-N	368932	(−)-4-(4-{[4-(difluoromethyl)-2-(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::(−)-4-(4-{[4-(difluoromethyl)-2-(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 196	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368932	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368932&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114548	402365731							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192857	COc1ccc(COc2ccc(C3CC(=O)Nc4n[nH]cc43)cc2OC)c(C(F)(F)F)c1	InChI=1S/C22H20F3N3O4/c1-30-14-5-3-13(17(8-14)22(23,24)25)11-32-18-6-4-12(7-19(18)31-2)15-9-20(29)27-21-16(15)10-26-28-21/h3-8,10,15H,9,11H2,1-2H3,(H2,26,27,28,29)	KHTGVXXFEDNKNO-UHFFFAOYSA-N	368933	(+)-4-(3-methoxy-4-{[4-methoxy-2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 197	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368933	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368933&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114228	402365732							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192858	COc1ccc(COc2ccc(C3CC(=O)Nc4n[nH]cc43)cc2OC)c(C(F)(F)F)c1	InChI=1S/C22H20F3N3O4/c1-30-14-5-3-13(17(8-14)22(23,24)25)11-32-18-6-4-12(7-19(18)31-2)15-9-20(29)27-21-16(15)10-26-28-21/h3-8,10,15H,9,11H2,1-2H3,(H2,26,27,28,29)	KHTGVXXFEDNKNO-UHFFFAOYSA-N	368934	(−)-4-(3-methoxy-4-{[4-methoxy-2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::(−)-4-(3-methoxy-4-{[4-methoxy-2-(trifluoromethyl)phenyl]methoxy}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 198	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368934	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368934&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114690	402365733							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192859	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(C(C)=O)cc1C(F)(F)F	InChI=1S/C23H20F3N3O4/c1-12(30)13-3-4-15(18(7-13)23(24,25)26)11-33-19-6-5-14(8-20(19)32-2)16-9-21(31)28-22-17(16)10-27-29-22/h3-8,10,16H,9,11H2,1-2H3,(H2,27,28,29,31)	RQNAGACDVZRQDN-UHFFFAOYSA-N	368935	(+)-4-(4-{[4-acetyl-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 199	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368935	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368935&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114485	402365734							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192860	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(C(C)=O)cc1C(F)(F)F	InChI=1S/C23H20F3N3O4/c1-12(30)13-3-4-15(18(7-13)23(24,25)26)11-33-19-6-5-14(8-20(19)32-2)16-9-21(31)28-22-17(16)10-27-29-22/h3-8,10,16H,9,11H2,1-2H3,(H2,27,28,29,31)	RQNAGACDVZRQDN-UHFFFAOYSA-N	368936	(−)-4-(4-{[4-acetyl-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::(−)-4-(4-{[4-acetyl-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 200	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368936	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368936&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114469	402365735							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192861	COc1ccc(COc2ccc(C3CC(=O)Nc4[nH]nnc43)cc2OC)c(C(F)(F)F)c1	InChI=1S/C21H19F3N4O4/c1-30-13-5-3-12(15(8-13)21(22,23)24)10-32-16-6-4-11(7-17(16)31-2)14-9-18(29)25-20-19(14)26-28-27-20/h3-8,14H,9-10H2,1-2H3,(H2,25,26,27,28,29)	SKBLBYIJPKZRTP-UHFFFAOYSA-N	368937	(+)-7-(3-methoxy-4-{[4-methoxy-2-(trifluoromethyl)phenyl]methoxy}phenyl)-3H,4H,5H,6H,7H-[1,2,3]triazolo[4,5-b]pyridin-5-one::US12527774, Compound 201	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368937	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368937&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114085	402365736							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192862	COc1ccc(COc2ccc(C3CC(=O)Nc4[nH]nnc43)cc2OC)c(C(F)(F)F)c1	InChI=1S/C21H19F3N4O4/c1-30-13-5-3-12(15(8-13)21(22,23)24)10-32-16-6-4-11(7-17(16)31-2)14-9-18(29)25-20-19(14)26-28-27-20/h3-8,14H,9-10H2,1-2H3,(H2,25,26,27,28,29)	SKBLBYIJPKZRTP-UHFFFAOYSA-N	368938	(−)-7-(3-methoxy-4-{[4-methoxy-2-(trifluoromethyl)phenyl]methoxy}phenyl)-3H,4H,5H,6H,7H-[1,2,3]triazolo[4,5-b]pyridin-5-one::(−)-7-(3-methoxy-4-{[4-methoxy-2-(trifluoromethyl)phenyl]methoxy}phenyl)-3H,4H,5H,6H,7H-[1,2,3]triazolo[4,5-b]pyridin-5-one::US12527774, Compound 202	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368938	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368938&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114216	402365737							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192863	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(N)cc1C(F)(F)F	InChI=1S/C21H19F3N4O3/c1-30-18-6-11(14-8-19(29)27-20-15(14)9-26-28-20)3-5-17(18)31-10-12-2-4-13(25)7-16(12)21(22,23)24/h2-7,9,14H,8,10,25H2,1H3,(H2,26,27,28,29)	WIGNHPDBLRQOKM-UHFFFAOYSA-N	368939	(+)-4-(4-{[4-amino-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 203	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368939	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368939&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114684	402365738							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192864	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(N)cc1C(F)(F)F	InChI=1S/C21H19F3N4O3/c1-30-18-6-11(14-8-19(29)27-20-15(14)9-26-28-20)3-5-17(18)31-10-12-2-4-13(25)7-16(12)21(22,23)24/h2-7,9,14H,8,10,25H2,1H3,(H2,26,27,28,29)	WIGNHPDBLRQOKM-UHFFFAOYSA-N	368940	(−)-4-(4-{[4-amino-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::(−)-4-(4-{[4-amino-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 204	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368940	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368940&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114820	402365739							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192865	COc1cc(C2CC(=O)Nc3n[nH]nc32)ccc1OCc1ccc(N)cc1C(F)(F)F	InChI=1S/C20H18F3N5O3/c1-30-16-6-10(13-8-17(29)25-19-18(13)26-28-27-19)3-5-15(16)31-9-11-2-4-12(24)7-14(11)20(21,22)23/h2-7,13H,8-9,24H2,1H3,(H2,25,26,27,28,29)	CICJFXSZKQVJRM-UHFFFAOYSA-N	368941	(+)-7-(4-{[4-amino-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-[1,2,3]triazolo[4,5-b]pyridin-5-one::US12527774, Compound 205	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368941	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368941&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115034	402365740							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192866	COc1cc(C2CC(=O)Nc3n[nH]nc32)ccc1OCc1ccc(N)cc1C(F)(F)F	InChI=1S/C20H18F3N5O3/c1-30-16-6-10(13-8-17(29)25-19-18(13)26-28-27-19)3-5-15(16)31-9-11-2-4-12(24)7-14(11)20(21,22)23/h2-7,13H,8-9,24H2,1H3,(H2,25,26,27,28,29)	CICJFXSZKQVJRM-UHFFFAOYSA-N	368942	(−)-7-(4-{[4-amino-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-[1,2,3]triazolo[4,5-b]pyridin-5-one::(−)-7-(4-{[4-amino-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-[1,2,3]triazolo[4,5-b]pyridin-5-one::US12527774, Compound 206	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368942	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368942&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115152	402365741							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192867	CCc1ccc(COc2ccc(C3CC(=O)Nc4n[nH]cc43)cc2OC)c(C(F)(F)F)c1	InChI=1S/C23H22F3N3O3/c1-3-13-4-5-15(18(8-13)23(24,25)26)12-32-19-7-6-14(9-20(19)31-2)16-10-21(30)28-22-17(16)11-27-29-22/h4-9,11,16H,3,10,12H2,1-2H3,(H2,27,28,29,30)	RONFEIXXSAWJBE-UHFFFAOYSA-N	368943	(+)-4-(4-{[4-ethyl-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 207	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368943	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368943&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114775	402365742							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192868	CCc1ccc(COc2ccc(C3CC(=O)Nc4n[nH]cc43)cc2OC)c(C(F)(F)F)c1	InChI=1S/C23H22F3N3O3/c1-3-13-4-5-15(18(8-13)23(24,25)26)12-32-19-7-6-14(9-20(19)31-2)16-10-21(30)28-22-17(16)11-27-29-22/h4-9,11,16H,3,10,12H2,1-2H3,(H2,27,28,29,30)	RONFEIXXSAWJBE-UHFFFAOYSA-N	368944	(−)-4-(4-{[4-ethyl-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::(−)-4-(4-{[4-ethyl-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 208	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368944	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368944&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114653	402365743							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192869	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(O)cc1C(F)(F)F	InChI=1S/C21H18F3N3O4/c1-30-18-6-11(14-8-19(29)26-20-15(14)9-25-27-20)3-5-17(18)31-10-12-2-4-13(28)7-16(12)21(22,23)24/h2-7,9,14,28H,8,10H2,1H3,(H2,25,26,27,29)	SJMTUKSJDISFGT-UHFFFAOYSA-N	368945	(+)-4-(4-{[4-hydroxy-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 209	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368945	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368945&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114723	402365744							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192870	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(O)cc1C(F)(F)F	InChI=1S/C21H18F3N3O4/c1-30-18-6-11(14-8-19(29)26-20-15(14)9-25-27-20)3-5-17(18)31-10-12-2-4-13(28)7-16(12)21(22,23)24/h2-7,9,14,28H,8,10H2,1H3,(H2,25,26,27,29)	SJMTUKSJDISFGT-UHFFFAOYSA-N	368946	(−)-4-(4-{[4-hydroxy-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::(−)-4-(4-{[4-hydroxy-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 210	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368946	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368946&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115096	402365745							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192871	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(CCO)cc1C(F)(F)F	InChI=1S/C23H22F3N3O4/c1-32-20-9-14(16-10-21(31)28-22-17(16)11-27-29-22)4-5-19(20)33-12-15-3-2-13(6-7-30)8-18(15)23(24,25)26/h2-5,8-9,11,16,30H,6-7,10,12H2,1H3,(H2,27,28,29,31)	XPBRKGFBHXVFIE-UHFFFAOYSA-N	368947	(+)-4-(4-{[4-(2-hydroxyethyl)-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 211	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368947	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368947&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114420	402365746							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192872	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1OCc1ccc(CCO)cc1C(F)(F)F	InChI=1S/C23H22F3N3O4/c1-32-20-9-14(16-10-21(31)28-22-17(16)11-27-29-22)4-5-19(20)33-12-15-3-2-13(6-7-30)8-18(15)23(24,25)26/h2-5,8-9,11,16,30H,6-7,10,12H2,1H3,(H2,27,28,29,31)	XPBRKGFBHXVFIE-UHFFFAOYSA-N	368948	(−)-4-(4-{[4-(2-hydroxyethyl)-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::(−)-4-(4-{[4-(2-hydroxyethyl)-2-(trifluoromethyl)phenyl]methoxy}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 212	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368948	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368948&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114276	402365747							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192873	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1COc1ccc(C)cc1C(F)(F)F	InChI=1S/C22H20F3N3O3/c1-12-3-6-18(17(7-12)22(23,24)25)31-11-14-5-4-13(8-19(14)30-2)15-9-20(29)27-21-16(15)10-26-28-21/h3-8,10,15H,9,11H2,1-2H3,(H2,26,27,28,29)	STVRWCYGPGAZFP-UHFFFAOYSA-N	368949	(+)-4-(3-methoxy-4-{[4-methyl-2-(trifluoromethyl)phenoxy]methyl}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 213	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368949	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368949&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90001602	402365748							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192874	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1COc1ccc(C)cc1C(F)(F)F	InChI=1S/C22H20F3N3O3/c1-12-3-6-18(17(7-12)22(23,24)25)31-11-14-5-4-13(8-19(14)30-2)15-9-20(29)27-21-16(15)10-26-28-21/h3-8,10,15H,9,11H2,1-2H3,(H2,26,27,28,29)	STVRWCYGPGAZFP-UHFFFAOYSA-N	368950	(−)-4-(3-methoxy-4-{[4-methyl-2-(trifluoromethyl)phenoxy]methyl}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::(−)-4-(3-methoxy-4-{[4-methyl-2-(trifluoromethyl)phenoxy]methyl}phenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 214	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368950	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368950&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90001962	402365749							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192875	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1COc1ccc(C(F)(F)F)cc1C(F)F	InChI=1S/C22H18F5N3O3/c1-32-18-6-11(14-8-19(31)29-21-16(14)9-28-30-21)2-3-12(18)10-33-17-5-4-13(22(25,26)27)7-15(17)20(23)24/h2-7,9,14,20H,8,10H2,1H3,(H2,28,29,30,31)	VDTPXOYKXZICNI-UHFFFAOYSA-N	368951	(+)-4-(4-{[2-(difluoromethyl)-4-(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 215	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368951	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368951&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114231	402365750							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192876	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1COc1ccc(C(F)(F)F)cc1C(F)F	InChI=1S/C22H18F5N3O3/c1-32-18-6-11(14-8-19(31)29-21-16(14)9-28-30-21)2-3-12(18)10-33-17-5-4-13(22(25,26)27)7-15(17)20(23)24/h2-7,9,14,20H,8,10H2,1H3,(H2,28,29,30,31)	VDTPXOYKXZICNI-UHFFFAOYSA-N	368952	(−)-4-(4-{[2-(difluoromethyl)-4-(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::(−)-4-(4-{[2-(difluoromethyl)-4-(trifluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 216	Steroid hormone receptor ERR1 [181-423]			 55.0							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368952	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368952&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115275	402365751							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192877	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1COc1ccc(C(F)F)cc1C(F)F	InChI=1S/C22H19F4N3O3/c1-31-18-7-11(14-8-19(30)28-22-16(14)9-27-29-22)2-3-13(18)10-32-17-5-4-12(20(23)24)6-15(17)21(25)26/h2-7,9,14,20-21H,8,10H2,1H3,(H2,27,28,29,30)	PARYEBOXSLXGBR-UHFFFAOYSA-N	368953	(+)-4-(4-{[2,4-bis(difluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 217	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368953	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368953&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114625	402365752							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192878	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1COc1ccc(C(F)F)cc1C(F)F	InChI=1S/C22H19F4N3O3/c1-31-18-7-11(14-8-19(30)28-22-16(14)9-27-29-22)2-3-13(18)10-32-17-5-4-12(20(23)24)6-15(17)21(25)26/h2-7,9,14,20-21H,8,10H2,1H3,(H2,27,28,29,30)	PARYEBOXSLXGBR-UHFFFAOYSA-N	368954	(−)-4-(4-{[2,4-bis(difluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::(−)-4-(4-{[2,4-bis(difluoromethyl)phenoxy]methyl}-3-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 218	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368954	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368954&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90114357	402365753							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192879	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1COc1ccc(C)cc1C	InChI=1S/C22H23N3O3/c1-13-4-7-19(14(2)8-13)28-12-16-6-5-15(9-20(16)27-3)17-10-21(26)24-22-18(17)11-23-25-22/h4-9,11,17H,10,12H2,1-3H3,(H2,23,24,25,26)	KXGSQIASWGEKCI-UHFFFAOYSA-N	368955	(+)-4-{4-[(2,4-dimethylphenoxy)methyl]-3-methoxyphenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 219	Steroid hormone receptor ERR1 [181-423]			 550							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368955	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368955&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90115198	402365754							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
192880	COc1cc(C2CC(=O)Nc3n[nH]cc32)ccc1COc1ccc(C)cc1C	InChI=1S/C22H23N3O3/c1-13-4-7-19(14(2)8-13)28-12-16-6-5-15(9-20(16)27-3)17-10-21(26)24-22-18(17)11-23-25-22/h4-9,11,17H,10,12H2,1-3H3,(H2,23,24,25,26)	KXGSQIASWGEKCI-UHFFFAOYSA-N	368956	(−)-4-{4-[(2,4-dimethylphenoxy)methyl]-3-methoxyphenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::(−)-4-{4-[(2,4-dimethylphenoxy)methyl]-3-methoxyphenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one::US12527774, Compound 220	Steroid hormone receptor ERR1 [181-423]			<10.00							US Patent		10.7270/Q23201PM			US12527774	Lemmers, JG; Deretey, E; Klomp, JP; Cals, JM; Oubrie, A	1/20/2026	6/1/2026	Lead Pharma Holding	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=368956	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=2090&target=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=368956&enzyme=Steroid+hormone+receptor+ERR1+%5B181-423%5D&column=ki&startPg=0&Increment=50&submit=Search			90137126	402365755							1	LAVAGGPRKTAAPVNALVSHLLVVEPEKLYAMPDPAGPDGHLPAVATLCDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRAGPGGGAERRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAMMD	3D24,3K6P,1XB7,7E2E	Steroid hormone receptor ERR1	ERR1_HUMAN	P11474	Q14514